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rhodamine 123 and sdz psc 833

rhodamine 123 has been researched along with sdz psc 833 in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (40.00)18.2507
2000's12 (48.00)29.6817
2010's3 (12.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Didier, AD; Loor, F; Muller, CD; Pourtier-Manzanedo, A1
Boer, R; Haas, S; Schödl, A1
Aracil, M; Barbacid, MM; Márquez, G; Mira, E; Quesada, AR1
Bello-Reuss, E; Ernest, S1
Davey, MW; Davey, RA; Hargrave, RM1
Bertrán, J; García-López, J; Pétriz, J; Sánchez, J1
Altenberg, GA; Castro, AF; Germain, GS; Gowda, GK; Horton, JK; Houghton, PJ; Thimmaiah, KN1
Haberl, I; Hamilton, G; Schaufler, K; Swatonek, H; Thalhammer, T; Theyer, G; Ulsperger, E; Wenzl, E1
Béliveau, R; Jetté, L; Murphy, GF1
Beck, JF; Boer, R; Buchholz, F; Gekeler, V; Niethammer, D; Sanders, KH; Ulrich, WR1
de Vries, EG; Ossenkoppele, GJ; van der Kolk, DM; van Putten, WJ; Vellenga, E; Verdonck, LF; Verhoef, GE1
Beketic-Oreskovic, L; Chen, GK; Durán, GE; Mangili, A; Sikic, BI1
Cho, CW; Henthorn, T; Liu, Y; Ng, KY; Yan, X1
Cohen, D; Uchiyama-Kokubu, N; Watanabe, T1
Ambudkar, SV; Kasir, J; Kimchi-Sarfaty, C; Rahamimoff, H1
Christians, U; Cobb, WN; Lillehei, K; Liu, Y; Ng, KY1
Fendrich, Z; Kopecky, M; Libra, A; Nobilis, M; Novotna, M; Pavek, P; Semecky, V; Sklenarova, H; Staud, F1
Grundy, M; Pallis, M; Russell, N; Seedhouse, C; Turzanski, J1
DeVane, CL; Donovan, JL; Markowitz, JS; Wang, JS; Zhu, HJ1
DeVane, CL; Donovan, JL; Gibson, BB; Jiang, Y; Markowitz, JS; Wang, JS; Zhu, HJ1
Ambudkar, SV; Barnett, D; Bates, SE; Finley, EM; Fojo, T; Oldham, RK; Robey, RW; Shukla, S1
Beghin, D; Claude, N; Delongeas, JL; Farinotti, R; Forestier, F; Gil, S1
Adrián, L; Carlos, L; Guillermo, V; Juan, S; Laura, M; Mariana, B1
Carpini, GD; Ghanem, CI; Luquita, MG; Mottino, AD; Novak, A; Rubio, MC; Ruiz, ML1
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M1

Trials

1 trial(s) available for rhodamine 123 and sdz psc 833

ArticleYear
Inhibition of P-glycoprotein (ABCB1)- and multidrug resistance-associated protein 1 (ABCC1)-mediated transport by the orally administered inhibitor, CBT-1((R)).
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Adenosine Triphosphatases; Alkaloids; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Factors; Biological Transport; Cell Line; Cell Line, Tumor; Cyclosporins; Depsipeptides; Fluorescent Dyes; Fluorouracil; Humans; Insecta; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Prazosin; Quinolines; Rhodamine 123; Verapamil; Vinblastine

2008

Other Studies

24 other study(ies) available for rhodamine 123 and sdz psc 833

ArticleYear
SDZ PSC 833 and SDZ 280-446 are the most active of various resistance-modifying agents in restoring rhodamine-123 retention within multidrug resistant P388 cells.
    Anti-cancer drugs, 1992, Volume: 3, Issue:4

    Topics: Animals; Antineoplastic Agents; Cyclosporins; Drug Resistance; Flow Cytometry; Fluorescent Dyes; Microscopy, Fluorescence; Peptides, Cyclic; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1992
Influence of dexniguldipine-HC1 on rhodamine-123 accumulation in a multidrug-resistant leukaemia cell line: comparison with other chemosensitisers.
    European journal of cancer (Oxford, England : 1990), 1994, Volume: 30A, Issue:8

    Topics: Antineoplastic Agents; Cyclosporins; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Humans; Hydrogen-Ion Concentration; Leukemia; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1994
Chemosensitization and drug accumulation assays as complementary methods for the screening of multidrug resistance reversal agents.
    Cancer letters, 1996, Jan-19, Volume: 99, Issue:1

    Topics: Adenocarcinoma; Animals; Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Colonic Neoplasms; Cyclosporins; Doxorubicin; Drug Resistance, Multiple; Drug Screening Assays, Antitumor; Fluorescent Dyes; Humans; Leukemia P388; Mice; Rhodamine 123; Rhodamines; Verapamil

1996
Xenobiotic transport differences in mouse mesangial cell clones expressing mdr1 and mdr3.
    The American journal of physiology, 1996, Volume: 270, Issue:3 Pt 1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport; Calcium; Cell Division; Cell Line; Cell Membrane; Clone Cells; Cyclosporine; Cyclosporins; Doxorubicin; Drug Resistance, Multiple; Gene Expression; Glomerular Mesangium; Kidney Tubules, Proximal; Kinetics; Mice; Mice, Transgenic; Rhodamine 123; Rhodamines; RNA, Messenger; Vinblastine; Xenobiotics

1996
Comparison of drug accumulation in P-glycoprotein-expressing and MRP-expressing human leukaemia cells.
    Leukemia research, 1996, Volume: 20, Issue:8

    Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Buthionine Sulfoximine; Calcium Channel Blockers; Cyclosporins; Daunorubicin; Humans; Idarubicin; Leukemia, T-Cell; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Verapamil

1996
Comparative effect of verapamil, cyclosporin A and SDZ PSC 833 on rhodamine 123 transport and cell cycle in vinblastine-resistant Chinese hamster ovary cells overexpressing P-glycoprotein.
    Anti-cancer drugs, 1997, Volume: 8, Issue:9

    Topics: Animals; Antimetabolites, Antineoplastic; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Cell Cycle; Cell Line; CHO Cells; Cricetinae; Cyclosporine; Cyclosporins; DNA; Drug Resistance, Neoplasm; Flow Cytometry; Immunosuppressive Agents; Rhodamine 123; Rhodamines; Verapamil; Vinblastine

1997
Characterization of a novel bisacridone and comparison with PSC 833 as a potent and poorly reversible modulator of P-glycoprotein.
    Molecular pharmacology, 1997, Volume: 52, Issue:6

    Topics: Acridines; Acridones; Adenosine Triphosphatases; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carcinoma, Squamous Cell; Cyclosporins; Drug Interactions; Drug Resistance, Multiple; Fluorescent Dyes; Humans; KB Cells; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Vinblastine

1997
P-glycoprotein-mediated multidrug resistance is modulated by pretreatment with chemosensitizers in HCT-8 carcinoma cells in vitro.
    International journal of oncology, 1998, Volume: 12, Issue:5

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclosporine; Cyclosporins; Doxorubicin; Drug Resistance, Multiple; Epithelial Cells; Humans; Ileal Neoplasms; Ileocecal Valve; Kinetics; Phosphorylation; Rhodamine 123; Rhodamines; Tamoxifen; Tetradecanoylphorbol Acetate; Time Factors; Tumor Cells, Cultured; Verapamil; Vinblastine

1998
Drug binding to P-glycoprotein is inhibited in normal tissues following SDZ-PSC 833 treatment.
    International journal of cancer, 1998, May-29, Volume: 76, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Brain; Calcium Channel Blockers; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Fluorescent Dyes; Injections, Subcutaneous; Iodine Radioisotopes; Kidney; Liver; Male; Microvilli; Photoaffinity Labels; Prazosin; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Verapamil; Vinblastine

1998
Rhodamine 123 efflux modulation in the presence of low or high serum from CD56+ hematopoietic cells or CD34+ leukemic blasts by B9309-068, a newly designed pyridine derivative.
    Cancer letters, 1998, Jul-17, Volume: 129, Issue:2

    Topics: Acridines; Antigens, CD34; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Blood Proteins; Calcium Channel Blockers; CD56 Antigen; Cyclosporins; Dihydropyridines; Dose-Response Relationship, Drug; Flow Cytometry; Fluorescent Dyes; Gene Expression; Humans; Isoquinolines; Leukemia, Myeloid, Acute; Leukocytes, Mononuclear; Morpholines; Multidrug Resistance-Associated Proteins; Pyrimidines; Rhodamine 123; Rhodamines; Tetrahydroisoquinolines; Verapamil

1998
P-glycoprotein and multidrug resistance protein activities in relation to treatment outcome in acute myeloid leukemia.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2000, Volume: 6, Issue:8

    Topics: Adolescent; Adult; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Cyclosporins; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Glutathione; Humans; Leukemia, Myeloid; Male; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Propionates; Quinolines; Randomized Controlled Trials as Topic; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Survival Analysis; Treatment Outcome; Tumor Cells, Cultured

2000
MDR 1 activation is the predominant resistance mechanism selected by vinblastine in MES-SA cells.
    British journal of cancer, 2000, Volume: 83, Issue:7

    Topics: Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Cyclosporins; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Gene Expression Regulation, Neoplastic; Genes, MDR; Humans; Multidrug Resistance-Associated Proteins; Mutation; Neoplasm Proteins; Paclitaxel; Phenotype; Rhodamine 123; RNA, Messenger; Sarcoma; Tritium; Tumor Cells, Cultured; Uterine Neoplasms; Vault Ribonucleoprotein Particles; Vinblastine

2000
Carrier-mediated uptake of rhodamine 123: implications on its use for MDR research.
    Biochemical and biophysical research communications, 2000, Dec-09, Volume: 279, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporins; Drug Resistance, Multiple; Humans; Rhodamine 123; Tumor Cells, Cultured; Verapamil

2000
Intracellular levels of two cyclosporin derivatives valspodar (PSC 833) and cyclosporin a closely associated with multidrug resistance-modulating activity in sublines of human colorectal adenocarcinoma HCT-15.
    Japanese journal of cancer research : Gann, 2001, Volume: 92, Issue:10

    Topics: Adenocarcinoma; Anticarcinogenic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Division; Colorectal Neoplasms; Cyclosporine; Cyclosporins; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Inhibitory Concentration 50; Intracellular Fluid; Rhodamine 123; Tumor Cells, Cultured; Verapamil

2001
Transport activity and surface expression of the Na+-Ca2+ exchanger NCX1 are inhibited by the immunosuppressive agent cyclosporin A and by the nonimmunosuppressive agent PSC833.
    The Journal of biological chemistry, 2002, Jan-25, Volume: 277, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blotting, Western; Calcium; Cell Line; Cell Separation; Coloring Agents; Cyclosporine; Cyclosporins; Dose-Response Relationship, Drug; Endoplasmic Reticulum; Flow Cytometry; HeLa Cells; Humans; Immunosuppressive Agents; Mutation; Myocardium; Protein Binding; Protein Transport; Rats; Rhodamine 123; Sodium-Calcium Exchanger; Spectrometry, Fluorescence; Transfection

2002
Overcoming MDR by ultrasound-induced hyperthermia and P-glycoprotein modulation.
    Biochemical and biophysical research communications, 2001, Nov-23, Volume: 289, Issue:1

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Division; Cell Survival; Cyclosporins; Doxorubicin; Drug Resistance, Multiple; Hot Temperature; Humans; Rhodamine 123; Tumor Cells, Cultured; Ultrasonics

2001
Examination of the functional activity of P-glycoprotein in the rat placental barrier using rhodamine 123.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Chlorpromazine; Cyclosporins; Drug Interactions; Female; Fluorescent Dyes; Placenta; Pregnancy; Quinidine; Rats; Rats, Wistar; Rhodamine 123; Sodium Azide

2003
Resistance to spontaneous apoptosis in acute myeloid leukaemia blasts is associated with p-glycoprotein expression and function, but not with the presence of FLT3 internal tandem duplications.
    British journal of haematology, 2003, Volume: 120, Issue:6

    Topics: Acute Disease; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporins; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; fms-Like Tyrosine Kinase 3; Humans; Leukemia, Myeloid; Proto-Oncogene Proteins; Receptor Protein-Tyrosine Kinases; Recurrence; Remission Induction; Repetitive Sequences, Nucleic Acid; Rhodamine 123; Statistics, Nonparametric; Tumor Cells, Cultured

2003
Evaluation of antipsychotic drugs as inhibitors of multidrug resistance transporter P-glycoprotein.
    Psychopharmacology, 2006, Volume: 187, Issue:4

    Topics: Animals; Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzodiazepines; Chlorpromazine; Clozapine; Cyclosporins; Dibenzothiazepines; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Interactions; Flow Cytometry; Fluorescent Dyes; Haloperidol; Isoxazoles; Kidney; Liver; LLC-PK1 Cells; Olanzapine; Paliperidone Palmitate; Pyrimidines; Quetiapine Fumarate; Rhodamine 123; Risperidone; Swine; Transfection

2006
Interactions of attention-deficit/hyperactivity disorder therapeutic agents with the efflux transporter P-glycoprotein.
    European journal of pharmacology, 2008, Jan-14, Volume: 578, Issue:2-3

    Topics: Adenosine Triphosphate; Amphetamine; Animals; Atomoxetine Hydrochloride; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Attention Deficit Disorder with Hyperactivity; Benzhydryl Compounds; Biological Transport; Central Nervous System Stimulants; Cyclosporins; Dose-Response Relationship, Drug; Doxorubicin; Isomerism; LLC-PK1 Cells; Methylphenidate; Modafinil; Propylamines; Reproducibility of Results; Rhodamine 123; Swine; Transfection

2008
Development and characterisation of a new model of rat trophoblasts.
    Toxicology in vitro : an international journal published in association with BIBRA, 2009, Volume: 23, Issue:1

    Topics: Animal Testing Alternatives; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cell Proliferation; Cell Survival; Cryopreservation; Cyclosporine; Cyclosporins; Drug Evaluation, Preclinical; Female; Fluoresceins; Fluorescent Dyes; Neoplasm Proteins; Organ Culture Techniques; Pregnancy; Rats; Rats, Wistar; Rhodamine 123; Trophoblasts

2009
Gender-related differences on P-glycoprotein-mediated drug intestinal transport in rats.
    The Journal of pharmacy and pharmacology, 2011, Volume: 63, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporins; Female; Ileum; Intestinal Absorption; Intestinal Mucosa; Ivermectin; Jejunum; Male; Rats; Rats, Wistar; Rhodamine 123; Sex Factors

2011
Acetaminophen inhibits intestinal p-glycoprotein transport activity.
    Journal of pharmaceutical sciences, 2013, Volume: 102, Issue:10

    Topics: Acetaminophen; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Line, Tumor; Cyclosporins; Digoxin; Enterocytes; Hep G2 Cells; Humans; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Permeability; Rats; Rats, Wistar; Rhodamine 123; Verapamil

2013
Rat precision-cut intestinal slices to study P-gp activity and the potency of its inhibitors ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2015, Volume: 29, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Cyclosporins; In Vitro Techniques; Intestinal Mucosa; Isoquinolines; Ketoconazole; Male; Quinazolines; Quinidine; Rats, Wistar; Rhodamine 123; Verapamil

2015