Page last updated: 2024-08-24

rhodamine 123 and prazosin

rhodamine 123 has been researched along with prazosin in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (26.67)18.2507
2000's8 (53.33)29.6817
2010's3 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ambudkar, SV; Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M1
Chen, G; Dumontet, C; Durán, GE; Jaffrézou, JP; Lacayo, NJ; Sikic, BI; Steger, KA1
Béliveau, R; Jetté, L; Murphy, GF1
Fox, K; Lam, P; Ling, V; Shapiro, AB1
Ambudkar, SV; Anuchapreeda, S; Leechanachai, P; Limtrakul, PN; Smith, MM1
Ambudkar, SV; Anuchapreeda, S; Chearwae, W; Limtrakul, P; Nandigama, K1
Chattopadhyay, A; Dey, S; Fong, WF; Shen, XL; Wan, CK; Zhu, GY1
Chmielewski, J; Hrycyna, CA; Pires, MM1
Ambudkar, SV; Barnett, D; Bates, SE; Finley, EM; Fojo, T; Oldham, RK; Robey, RW; Shukla, S1
Chmielewski, J; Emmert, D; Hrycyna, CA; Pires, MM1
Ceckova, M; Cygalova, LH; Hofman, J; Staud, F1
Ambudkar, SV; Limtrakul, P; Ohnuma, S; Pintha, K; Pitchakarn, P; Pompimon, W1
Ambudkar, SV; Chanmahasathien, W; Limtrakul, P; Ohnuma, S1
Desai, TA; Kroetz, DL; Lamson, NG; Levy, ES; Samy, KE; Whitehead, KA1
Bates, S; Litman, T; Nagy, Z; Ozvegy, C; Sarkadi, B; Szakács, G; Váradi, A1

Trials

1 trial(s) available for rhodamine 123 and prazosin

ArticleYear
Inhibition of P-glycoprotein (ABCB1)- and multidrug resistance-associated protein 1 (ABCC1)-mediated transport by the orally administered inhibitor, CBT-1((R)).
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Adenosine Triphosphatases; Alkaloids; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Factors; Biological Transport; Cell Line; Cell Line, Tumor; Cyclosporins; Depsipeptides; Fluorescent Dyes; Fluorouracil; Humans; Insecta; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Prazosin; Quinolines; Rhodamine 123; Verapamil; Vinblastine

2008

Other Studies

14 other study(ies) available for rhodamine 123 and prazosin

ArticleYear
Functional characterization of a glycine 185-to-valine substitution in human P-glycoprotein by using a vaccinia-based transient expression system.
    Molecular biology of the cell, 1996, Volume: 7, Issue:10

    Topics: 3T3 Cells; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Bone Neoplasms; Cell Membrane; Colchicine; Drug Resistance, Multiple; Genetic Vectors; Humans; Mice; Nicardipine; Onium Compounds; Organophosphorus Compounds; Osteosarcoma; Point Mutation; Prazosin; Recombinant Fusion Proteins; Rhodamine 123; Rhodamines; Transfection; Tumor Cells, Cultured; Vaccinia virus; Verapamil; Vinblastine

1996
Multidrug-resistant human sarcoma cells with a mutant P-glycoprotein, altered phenotype, and resistance to cyclosporins.
    The Journal of biological chemistry, 1997, Feb-28, Volume: 272, Issue:9

    Topics: Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Survival; Cyclosporins; Dihydropyridines; DNA Topoisomerases, Type II; Doxorubicin; Drug Resistance, Multiple; Humans; Neoplasm Proteins; Phenotype; Polymerase Chain Reaction; Prazosin; Rhodamine 123; Rhodamines; Sarcoma; Vault Ribonucleoprotein Particles; Verapamil

1997
Drug binding to P-glycoprotein is inhibited in normal tissues following SDZ-PSC 833 treatment.
    International journal of cancer, 1998, May-29, Volume: 76, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Brain; Calcium Channel Blockers; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Fluorescent Dyes; Injections, Subcutaneous; Iodine Radioisotopes; Kidney; Liver; Male; Microvilli; Photoaffinity Labels; Prazosin; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Verapamil; Vinblastine

1998
Stimulation of P-glycoprotein-mediated drug transport by prazosin and progesterone. Evidence for a third drug-binding site.
    European journal of biochemistry, 1999, Volume: 259, Issue:3

    Topics: Allosteric Site; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Membrane; CHO Cells; Cricetinae; Fluorescent Dyes; Flupenthixol; Haloperidol; Molecular Structure; Prazosin; Progesterone; Propranolol; Protein Binding; Rhodamine 123; Spiperone

1999
Modulation of P-glycoprotein expression and function by curcumin in multidrug-resistant human KB cells.
    Biochemical pharmacology, 2002, Aug-15, Volume: 64, Issue:4

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cell Survival; Curcumin; Down-Regulation; Drug Resistance, Multiple; Fluorescent Dyes; Gene Expression; Humans; KB Cells; Photoaffinity Labels; Prazosin; Rhodamine 123; Tumor Cells, Cultured; Vinblastine

2002
Biochemical mechanism of modulation of human P-glycoprotein (ABCB1) by curcumin I, II, and III purified from Turmeric powder.
    Biochemical pharmacology, 2004, Nov-15, Volume: 68, Issue:10

    Topics: Adenosine Triphosphatases; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Cell Survival; Curcuma; Curcumin; Diarylheptanoids; Drug Combinations; Drug Interactions; Fluoresceins; Humans; Iodine Radioisotopes; KB Cells; Multidrug Resistance-Associated Proteins; Photoaffinity Labels; Plant Extracts; Prazosin; Rhodamine 123; Vinblastine

2004
Gomisin A alters substrate interaction and reverses P-glycoprotein-mediated multidrug resistance in HepG2-DR cells.
    Biochemical pharmacology, 2006, Sep-28, Volume: 72, Issue:7

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Anticarcinogenic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Cell Line, Tumor; Cell Survival; Cyclooctanes; Dioxoles; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Humans; Hydrolysis; Lignans; Prazosin; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Vanadates; Verapamil; Vinblastine

2006
Bivalent probes of the human multidrug transporter P-glycoprotein.
    Biochemistry, 2006, Sep-26, Volume: 45, Issue:38

    Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cross-Linking Reagents; Dimerization; Doxorubicin; Emetine; Flow Cytometry; Humans; Hydrolysis; Inhibitory Concentration 50; Models, Biological; Molecular Probes; Photoaffinity Labels; Prazosin; Rhodamine 123; Substrate Specificity; Tumor Cells, Cultured

2006
Inhibition of P-glycoprotein-mediated paclitaxel resistance by reversibly linked quinine homodimers.
    Molecular pharmacology, 2009, Volume: 75, Issue:1

    Topics: Adenocarcinoma; Adenosine Triphosphatases; Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Cell Line, Tumor; Cell Survival; Dimerization; Dose-Response Relationship, Drug; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Flow Cytometry; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Molecular Structure; Paclitaxel; Prazosin; Quinine; Rhodamine 123; Verapamil

2009
Transplacental pharmacokinetics of glyburide, rhodamine 123, and BODIPY FL prazosin: effect of drug efflux transporters and lipid solubility.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Boron Compounds; Dose-Response Relationship, Drug; Female; Glyburide; In Vitro Techniques; Lipids; Maternal-Fetal Exchange; Perfusion; Placenta; Prazosin; Pregnancy; Rats; Rhodamine 123; Solubility; Substrate Specificity

2009
Kuguacin J isolated from Momordica charantia leaves inhibits P-glycoprotein (ABCB1)-mediated multidrug resistance.
    The Journal of nutritional biochemistry, 2012, Volume: 23, Issue:1

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Fluoresceins; Humans; Molecular Structure; Momordica charantia; Paclitaxel; Plant Leaves; Prazosin; Rhodamine 123; Triterpenes; Uterine Cervical Neoplasms; Vinblastine

2012
Biochemical mechanism of modulation of human P-glycoprotein by stemofoline.
    Planta medica, 2011, Volume: 77, Issue:18

    Topics: Adenosine Triphosphatases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Heterocyclic Compounds, 4 or More Rings; Humans; Insecta; Membranes; Photoaffinity Labels; Plant Roots; Prazosin; Protein Binding; Rhodamine 123; Stemonaceae; Vinblastine

2011
Reversible inhibition of efflux transporters by hydrogel microdevices.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2019, Volume: 145

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; Biological Availability; Biological Transport; Boron Compounds; Caco-2 Cells; Cell Line, Tumor; Humans; Hydrogels; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Mice; Mice, Inbred C57BL; Polyethylene Glycols; Prazosin; Rhodamine 123; Solubility

2019
Functional characterization of the human multidrug transporter, ABCG2, expressed in insect cells.
    Biochemical and biophysical research communications, 2001, Jul-06, Volume: 285, Issue:1

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Membrane; Cloning, Molecular; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Recombinant Proteins; Spodoptera; Tumor Cells, Cultured

2001