Page last updated: 2024-08-24

rhodamine 123 and ketoconazole

rhodamine 123 has been researched along with ketoconazole in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (20.00)18.2507
2000's3 (30.00)29.6817
2010's5 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Clark, FS; Gow, NA; Hitchcock, CA; Parkinson, T1
Fukuda, T; Hasegawa, R; Murakami, T; Nagai, J; Takano, M; Yumoto, R1
Chen, XJ1
Allen, JD; Kota, BP; Roufogalis, BD1
Choi, DH; Choi, JS; Li, C1
Choi, DH; Choi, JS; Lee, CK1
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M1
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ1
Cannon, RD; Holmes, AR; Lamping, E; Nakamura, K; Niimi, K; Niimi, M; Ranchod, A; Tyndall, JD1
Ghosh, I; Manoharlal, R; Prakash, O; Prasad, R; Puri, N; Sharma, M1

Other Studies

10 other study(ies) available for rhodamine 123 and ketoconazole

ArticleYear
Correlation between rhodamine 123 accumulation and azole sensitivity in Candida species: possible role for drug efflux in drug resistance.
    Antimicrobial agents and chemotherapy, 1996, Volume: 40, Issue:2

    Topics: Antifungal Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azoles; Candida; Drug Resistance, Microbial; Fluconazole; Fluorescent Dyes; Itraconazole; Ketoconazole; Microbial Sensitivity Tests; Rhodamine 123; Rhodamines

1996
Interaction with P-glycoprotein and transport of erythromycin, midazolam and ketoconazole in Caco-2 cells.
    European journal of pharmacology, 1998, Oct-09, Volume: 358, Issue:3

    Topics: Anti-Bacterial Agents; Antifungal Agents; Aryl Hydrocarbon Hydroxylases; ATP Binding Cassette Transporter, Subfamily B; Biological Transport; Caco-2 Cells; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Enzyme Inhibitors; Erythromycin; GABA Modulators; Humans; Ketoconazole; Midazolam; Oxidoreductases, N-Demethylating; Rhodamine 123; Substrate Specificity; Vasodilator Agents; Verapamil

1998
Activity of the Kluyveromyces lactis Pdr5 multidrug transporter is modulated by the Sit4 protein phosphatase.
    Journal of bacteriology, 2001, Volume: 183, Issue:13

    Topics: Antifungal Agents; Antimycin A; ATP-Binding Cassette Transporters; Biological Transport, Active; Drug Resistance, Multiple; Econazole; Ketoconazole; Kluyveromyces; Membrane Proteins; Molecular Sequence Data; Mutation; Oligomycins; Phosphoprotein Phosphatases; Protein Phosphatase 2; Protein Processing, Post-Translational; Rhodamine 123; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Transcription, Genetic

2001
The effect of vitamin D3 and ketoconazole combination on VDR-mediated P-gp expression and function in human colon adenocarcinoma cells: implications in drug disposition and resistance.
    Basic & clinical pharmacology & toxicology, 2011, Volume: 109, Issue:2

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcitriol; Cell Line, Tumor; Colchicine; Colonic Neoplasms; Drug Resistance, Neoplasm; Humans; Ketoconazole; Receptors, Calcitriol; Rhodamine 123

2011
Effects of efonidipine on the pharmacokinetics and pharmacodynamics of repaglinide: possible role of CYP3A4 and P-glycoprotein inhibition by efonidipine.
    Journal of pharmacokinetics and pharmacodynamics, 2012, Volume: 39, Issue:1

    Topics: Animals; Antihypertensive Agents; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biocatalysis; Biological Availability; Blood Glucose; Carbamates; Cell Line, Tumor; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dihydropyridines; Drug Interactions; Humans; Hypoglycemic Agents; Ketoconazole; Male; Models, Biological; Nitrophenols; Organophosphorus Compounds; Pharmacological Phenomena; Piperidines; Rats; Rats, Sprague-Dawley; Rhodamine 123

2012
Effects of HMG-CoA reductase inhibitors on the pharmacokinetics of nifedipine in rats: Possible role of P-gp and CYP3A4 inhibition by HMG-CoA reductase inhibitors.
    Pharmacological reports : PR, 2015, Volume: 67, Issue:1

    Topics: Animals; Antifungal Agents; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biotransformation; Calcium Channel Blockers; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Fluorescent Dyes; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Ketoconazole; Male; Nifedipine; Rats; Rats, Sprague-Dawley; Rhodamine 123

2015
Rat precision-cut intestinal slices to study P-gp activity and the potency of its inhibitors ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2015, Volume: 29, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Cyclosporins; In Vitro Techniques; Intestinal Mucosa; Isoquinolines; Ketoconazole; Male; Quinazolines; Quinidine; Rats, Wistar; Rhodamine 123; Verapamil

2015
Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.
    Pharmaceutical research, 2003, Volume: 20, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Binding Sites; Biological Transport, Active; Biomarkers; Cells, Cultured; Drug Interactions; Fluorescent Dyes; Humans

2003
Abc1p is a multidrug efflux transporter that tips the balance in favor of innate azole resistance in Candida krusei.
    Antimicrobial agents and chemotherapy, 2009, Volume: 53, Issue:2

    Topics: Amino Acid Sequence; Animals; Antifungal Agents; ATP-Binding Cassette Transporters; Azoles; Blotting, Northern; Blotting, Southern; Candida; Candidiasis; Cell Membrane; Chromosomes, Fungal; Drug Resistance, Fungal; Endoplasmic Reticulum; Humans; Phenotype; Plasmids; Reverse Transcriptase Polymerase Chain Reaction; Saccharomyces cerevisiae

2009
Analysis of physico-chemical properties of substrates of ABC and MFS multidrug transporters of pathogenic Candida albicans.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Candida albicans; Membrane Transport Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Substrate Specificity

2010