Page last updated: 2024-08-24

rhodamine 123 and elacridar

rhodamine 123 has been researched along with elacridar in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (30.00)18.2507
2000's5 (50.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
den Ouden, D; Schoester, M; Sonneveld, P; van den Heuvel, M; van Rens, G1
Beck, JF; Boer, R; Buchholz, F; Gekeler, V; Niethammer, D; Sanders, KH; Ulrich, WR1
Dalton, WS; Emerson, DL; Kerr, BM; Lloyd, TL; Wissel, PS; Witherspoon, SM1
Berridge, G; Callaghan, R; Charlton, P; Higgins, CF; Martin, C; Mistry, P1
Alvaro, D; Boyer, JL; Fraioli, F; Gigliozzi, A; Lee, J; Mennone, A; Sundaram, P1
Annaert, PP; Booth, CL; Brouwer, KL; Thakker, DR; Turncliff, RZ1
Biswas, NR; Ghose, S; Saxena, R; Senthilkumari, S; Velpandian, T1
Biswas, NR; Ghose, S; Senthilkumari, S; Sonali, N; Velpandian, T1
Wang, XD; Zeng, S1
Christlieb, M; Marighetti, F; Pajeva, IK; Steggemann, K; Sterz, K; Wiese, M1

Other Studies

10 other study(ies) available for rhodamine 123 and elacridar

ArticleYear
In vitro effect of GF120918, a novel reversal agent of multidrug resistance, on acute leukemia and multiple myeloma cells.
    Leukemia, 1996, Volume: 10, Issue:12

    Topics: Acridines; Acute Disease; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Drug Resistance, Multiple; Humans; Isoquinolines; Kinetics; Leukemia, Myeloid; Multiple Myeloma; Neoplasm Proteins; Polymerase Chain Reaction; Rhodamine 123; Rhodamines; Tetrahydroisoquinolines; Transcription, Genetic; Tumor Cells, Cultured

1996
Rhodamine 123 efflux modulation in the presence of low or high serum from CD56+ hematopoietic cells or CD34+ leukemic blasts by B9309-068, a newly designed pyridine derivative.
    Cancer letters, 1998, Jul-17, Volume: 129, Issue:2

    Topics: Acridines; Antigens, CD34; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Blood Proteins; Calcium Channel Blockers; CD56 Antigen; Cyclosporins; Dihydropyridines; Dose-Response Relationship, Drug; Flow Cytometry; Fluorescent Dyes; Gene Expression; Humans; Isoquinolines; Leukemia, Myeloid, Acute; Leukocytes, Mononuclear; Morpholines; Multidrug Resistance-Associated Proteins; Pyrimidines; Rhodamine 123; Rhodamines; Tetrahydroisoquinolines; Verapamil

1998
Flow cytometric assay of modulation of P-glycoprotein function in whole blood by the multidrug resistance inhibitor GG918.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 1996, Volume: 2, Issue:1

    Topics: Acridines; ATP Binding Cassette Transporter, Subfamily B, Member 1; CD56 Antigen; Drug Resistance, Multiple; Flow Cytometry; Humans; Isoquinolines; Rhodamine 123; Tetrahydroisoquinolines

1996
Communication between multiple drug binding sites on P-glycoprotein.
    Molecular pharmacology, 2000, Volume: 58, Issue:3

    Topics: Acridines; Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Benzylidene Compounds; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Drug Interactions; Isoquinolines; Kinetics; Nicardipine; Paclitaxel; Quinolines; Radioligand Assay; Radiopharmaceuticals; Rhodamine 123; Tetrahydroisoquinolines; Tritium; Vinblastine

2000
Molecular identification and functional characterization of Mdr1a in rat cholangiocytes.
    Gastroenterology, 2000, Volume: 119, Issue:4

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Bile Ducts; Cell Division; Cell Membrane; Cytosol; Drug Resistance, Multiple; In Vitro Techniques; Isoquinolines; Kinetics; Male; Microscopy, Confocal; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Messenger; Tetrahydroisoquinolines; Transcription, Genetic; Vanadates; Verapamil

2000
P-glycoprotein-mediated in vitro biliary excretion in sandwich-cultured rat hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 2001, Volume: 29, Issue:10

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biliary Tract; Calcium; Cell Culture Techniques; Culture Media; Dexamethasone; Digoxin; Glucocorticoids; Hepatocytes; Isoquinolines; Male; Metabolic Clearance Rate; Polystyrenes; Rats; Rats, Wistar; Rhodamine 123; Tetrahydroisoquinolines; Time Factors; Tritium

2001
Evaluation of the modulation of P-glycoprotein (P-gp) on the intraocular disposition of its substrate in rabbits.
    Current eye research, 2008, Volume: 33, Issue:4

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blood-Brain Barrier; Carrier Proteins; Chromatography, High Pressure Liquid; Eye; Fluorescent Dyes; Injections; Injections, Intravenous; Kinetics; Male; Microdialysis; Rabbits; Retina; Rhodamine 123; Rifampin; Tetrahydroisoquinolines; Tissue Distribution; Vitreous Body

2008
Evaluation of the impact of P-glycoprotein (P-gp) drug efflux transporter blockade on the systemic and ocular disposition of P-gp substrate.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2008, Volume: 24, Issue:3

    Topics: Acridines; Animals; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromatography, High Pressure Liquid; Data Interpretation, Statistical; Eye; Female; Fluorescent Dyes; Injections, Intravenous; Male; Pharmaceutical Preparations; Rabbits; Reproducibility of Results; Rhodamine 123; Tetrahydroisoquinolines; Tissue Distribution

2008
The transport of gastrodin in Caco-2 cells and uptake in Bcap37 and Bcap37/MDR1 cells.
    Yao xue xue bao = Acta pharmaceutica Sinica, 2010, Volume: 45, Issue:12

    Topics: Acridines; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzyl Alcohols; Biological Transport; Blood-Brain Barrier; Breast Neoplasms; Caco-2 Cells; Cell Line, Tumor; Drug Resistance, Multiple; Gastrodia; Glucosides; Humans; Plants, Medicinal; Prohibitins; Rhodamine 123; Tetrahydroisoquinolines; Verapamil

2010
Interactions of the multidrug resistance modulators tariquidar and elacridar and their analogues with P-glycoprotein.
    ChemMedChem, 2013, Volume: 8, Issue:10

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Cell Line, Tumor; Drug Resistance, Multiple; Humans; Mice; Molecular Docking Simulation; Protein Binding; Protein Structure, Tertiary; Quinolines; Rhodamine 123; Structure-Activity Relationship; Substrate Specificity; Tetrahydroisoquinolines

2013