Page last updated: 2024-08-24

rhodamine 123 and digoxin

rhodamine 123 has been researched along with digoxin in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's11 (44.00)29.6817
2010's14 (56.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Asano, Y; Fujimura, A; Imai, M; Muto, S; Sugimoto, KI; Tsuruoka, S1
Annaert, PP; Booth, CL; Brouwer, KL; Thakker, DR; Turncliff, RZ1
Ohnishi, N; Takara, K; Tsujimoto, M; Yokoyama, T1
Banide, H; Faivre, L; Farinotti, R; Lacour, B; Soursac, M; Tardivel, S; Veau, C1
Akhtar, S; Barar, J; Campbell, L; Connell, D; Gumbleton, M; Omidi, Y1
Annaert, PP; Brouwer, KL1
Kim, DH; Lee, M; Lee, MW; Lim, SY; Shin, J; Yoo, HH1
Chung, HJ; Kim, DH; Lee, M; Lee, SK; Yoo, HH1
Azuma, J; Hou, XL; Komatsu, K; Qiu, F; Takahashi, K; Tanaka, K; Tougou, K1
Hirano, T; Iseki, K; Itagaki, S; Kobayashi, M; Ochiai, A; Sugawara, M1
Kaku, T; Sato, J; Sato, T; Takahashi, T; Watanabe, K1
Ai, H; Gu, Y; Hao, G; Li, Y; Peng, Y; Sun, J; Wang, G; Wu, X; Zhang, J; Zhang, X; Zheng, Y; Zhou, F1
Fahmi, OA; Kagota, S; Nejime, N; Shinozuka, K; Tada, Y; Umegaki, K; Wakuda, H; Yamada, S1
Bosquillon, C; Cooper, A; Hilgendorf, C; Hutter, V; Pritchard, DI; Zann, V1
Gerk, PM; Hylemon, PB; Liu, X; Pandak, WM; Shi, J; Studer, E; Wang, G; Wang, Y; Xu, W; Zha, BS; Zha, W; Zhao, Q; Zhou, H1
Baum, L; Chanteux, H; Kwan, P; Zhang, C; Zuo, Z1
Al-Jayyoussi, G; Eddershaw, P; Edwards, CD; Francombe, D; Gumbleton, M; Morris, C; Price, DF; Smith, MW; Taylor, G1
Carpini, GD; Ghanem, CI; Luquita, MG; Mottino, AD; Novak, A; Rubio, MC; Ruiz, ML1
Ge, G; Li, N; Liu, Y; Wang, D; Wang, X; Yang, L1
Fan, H; Fawcett, JP; Gu, J; Guo, Y; Liu, J; Ma, W; Sun, Y; Wang, T; Yang, J; Yang, Y; Yang, Z1
Celuch, SM; Ghanem, CI; Godoy, YC; Martinez, SA; Novak, A1
Dolberg, AM; Reichl, S1
Murakami, T; Oda, K1
Bocci, G; Denizot, C; Fardel, O; Moreau, A; Parmentier, Y; Vayer, P1
Hargrove, P; Kim, RB; Lan, LB; Lecureur, V; Schuetz, EG; Schuetz, JD; Sun, D1

Other Studies

25 other study(ies) available for rhodamine 123 and digoxin

ArticleYear
P-glycoprotein-mediated drug secretion in mouse proximal tubule perfused in vitro.
    Journal of the American Society of Nephrology : JASN, 2001, Volume: 12, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; Digoxin; Fluorescent Dyes; Genes, MDR; In Vitro Techniques; Kidney Tubules, Proximal; Male; Mice; Mice, Knockout; Perfusion; Rhodamine 123

2001
P-glycoprotein-mediated in vitro biliary excretion in sandwich-cultured rat hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 2001, Volume: 29, Issue:10

    Topics: Acridines; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biliary Tract; Calcium; Cell Culture Techniques; Culture Media; Dexamethasone; Digoxin; Glucocorticoids; Hepatocytes; Isoquinolines; Male; Metabolic Clearance Rate; Polystyrenes; Rats; Rats, Wistar; Rhodamine 123; Tetrahydroisoquinolines; Time Factors; Tritium

2001
Digoxin up-regulates MDR1 in human colon carcinoma Caco-2 cells.
    Biochemical and biophysical research communications, 2002, Mar-22, Volume: 292, Issue:1

    Topics: Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cell Division; Digoxin; Dose-Response Relationship, Drug; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Kinetics; Paclitaxel; Rhodamine 123; RNA, Messenger; Up-Regulation

2002
Effect of interleukin-2 on intestinal P-glycoprotein expression and functionality in mice.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Digoxin; DNA Primers; Gene Expression Regulation; Interleukin-2; Intestinal Absorption; Kinetics; Male; Mice; Mice, Inbred Strains; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123

2002
Evaluation of the immortalised mouse brain capillary endothelial cell line, b.End3, as an in vitro blood-brain barrier model for drug uptake and transport studies.
    Brain research, 2003, Nov-14, Volume: 990, Issue:1-2

    Topics: Alkaline Phosphatase; Amino Acid Transport Systems, Neutral; Animals; Biological Transport; Blood-Brain Barrier; Blotting, Western; Brain; Capillaries; Carrier Proteins; Cell Line; Cell Membrane Permeability; Digoxin; Electrophysiology; Endothelial Cells; Fluorescent Dyes; Glucose; Kinetics; Mice; Models, Biological; Pharmaceutical Preparations; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA; Swine; Tight Junctions; Up-Regulation

2003
Assessment of drug interactions in hepatobiliary transport using rhodamine 123 in sandwich-cultured rat hepatocytes.
    Drug metabolism and disposition: the biological fate of chemicals, 2005, Volume: 33, Issue:3

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Culture Techniques; Cells, Cultured; Collagenases; Digoxin; Drug Interactions; Hepatocytes; Male; Progesterone; Quercetin; Quinidine; Rats; Rats, Wistar; Rhodamine 123; Verapamil

2005
Effects of Schisandra lignans on P-glycoprotein-mediated drug efflux in human intestinal Caco-2.
    Planta medica, 2007, Volume: 73, Issue:5

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cyclooctanes; Digoxin; Humans; Lignans; Polycyclic Compounds; Rhodamine 123; Schisandra

2007
Effects of diosmin, a flavonoid glycoside in citrus fruits, on P-glycoprotein-mediated drug efflux in human intestinal Caco-2 cells.
    Journal of agricultural and food chemistry, 2007, Sep-05, Volume: 55, Issue:18

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Citrus; Digoxin; Diosmin; Fruit; Humans; Intestinal Mucosa; Intestines; Rhodamine 123

2007
Curcuma drugs and curcumin regulate the expression and function of P-gp in Caco-2 cells in completely opposite ways.
    International journal of pharmaceutics, 2008, Jun-24, Volume: 358, Issue:1-2

    Topics: ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Caco-2 Cells; Chromatography, High Pressure Liquid; Curcuma; Curcumin; Digoxin; Fluorescent Dyes; Humans; Plant Extracts; Rhodamine 123; RNA

2008
Interaction of coenzyme Q10 with the intestinal drug transporter P-glycoprotein.
    Journal of agricultural and food chemistry, 2008, Aug-27, Volume: 56, Issue:16

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Digoxin; Drug Interactions; Humans; Intestinal Mucosa; Quinidine; Rhodamine 123; Ubiquinone; Vitamins

2008
Effects of Acanthopanax senticosus HARMS extract on drug transport in human intestinal cell line Caco-2.
    Journal of natural medicines, 2010, Volume: 64, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cephalexin; Digoxin; Dose-Response Relationship, Drug; Drug Interactions; Drugs, Chinese Herbal; Eleutherococcus; Humans; Intestinal Absorption; Membrane Transport Proteins; Plant Extracts; Rhodamine 123

2010
20(S)-ginsenoside Rh2 noncompetitively inhibits P-glycoprotein in vitro and in vivo: a case for herb-drug interactions.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Digoxin; Etoposide; Ginsenosides; Herb-Drug Interactions; Humans; Ileum; Male; Rats; Rats, Sprague-Dawley; Rhodamine 123; Terfenadine; Verapamil

2010
A novel method using confocal laser scanning microscopy for sensitive measurement of P-glycoprotein-mediated transport activity in Caco-2 cells.
    The Journal of pharmacy and pharmacology, 2011, Volume: 63, Issue:8

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Digoxin; Drug Interactions; Fluorescent Dyes; Humans; Hypericum; Microscopy, Confocal; Plant Extracts; Rhodamine 123

2011
Evaluation of layers of the rat airway epithelial cell line RL-65 for permeability screening of inhaled drug candidates.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2012, Sep-29, Volume: 47, Issue:2

    Topics: Administration, Inhalation; Animals; Bronchi; Cell Line; Cell Membrane Permeability; Digoxin; Epithelial Cells; Fluorescent Dyes; Gene Expression; Humans; Mannitol; Membrane Transport Proteins; Microscopy, Confocal; Microscopy, Electron, Scanning; Pharmaceutical Preparations; Rats; Rhodamine 123; RNA, Messenger

2012
Inhibition of P-glycoprotein by HIV protease inhibitors increases intracellular accumulation of berberine in murine and human macrophages.
    PloS one, 2013, Volume: 8, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Berberine; Binding, Competitive; Biological Transport; Cell Line; Chromatography, High Pressure Liquid; Digoxin; Dogs; Gene Expression; HIV Protease Inhibitors; Humans; Macrophages; Madin Darby Canine Kidney Cells; Mice; Molecular Docking Simulation; Protein Binding; Rhodamine 123; Ritonavir

2013
Potential role for human P-glycoprotein in the transport of lacosamide.
    Epilepsia, 2013, Volume: 54, Issue:7

    Topics: Acetamides; Animals; Anticonvulsants; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Calcium Channel Blockers; Cell Line; Digoxin; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; Humans; Lacosamide; Quinolines; Rhodamine 123; RNA, Messenger; Swine; Time Factors; Transfection; Tritium; Verapamil

2013
Selectivity in the impact of P-glycoprotein upon pulmonary absorption of airway-dosed substrates: a study in ex vivo lung models using chemical inhibition and genetic knockout.
    Journal of pharmaceutical sciences, 2013, Volume: 102, Issue:9

    Topics: Animals; Anti-Arrhythmia Agents; Antidiarrheals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Sub-Family B Member 4; Biological Transport; Digoxin; Dogs; Gene Knockout Techniques; HIV Protease Inhibitors; Humans; Loperamide; Lung; Madin Darby Canine Kidney Cells; Male; Mice; Mice, Knockout; Permeability; Rats; Rats, Sprague-Dawley; Rhodamine 123; Saquinavir

2013
Acetaminophen inhibits intestinal p-glycoprotein transport activity.
    Journal of pharmaceutical sciences, 2013, Volume: 102, Issue:10

    Topics: Acetaminophen; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Line, Tumor; Cyclosporins; Digoxin; Enterocytes; Hep G2 Cells; Humans; Intestinal Absorption; Intestinal Mucosa; Intestines; Male; Permeability; Rats; Rats, Wistar; Rhodamine 123; Verapamil

2013
Ginsenoside metabolites inhibit P-glycoprotein in vitro and in situ using three absorption models.
    Planta medica, 2014, Volume: 80, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; Digoxin; Ginsenosides; Herb-Drug Interactions; Humans; Intestinal Absorption; Intestines; Male; Panax; Rats; Rats, Sprague-Dawley; Rhodamine 123

2014
Trantinterol, a novel β2-adrenoceptor agonist, noncompetitively inhibits P-glycoprotein function in vitro and in vivo.
    Molecular pharmaceutics, 2015, Jan-05, Volume: 12, Issue:1

    Topics: Adenosine Triphosphatases; Adrenergic beta-Agonists; Animals; Antibodies, Monoclonal; Area Under Curve; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Biological Transport; Caco-2 Cells; Clenbuterol; Cyclosporine; Digoxin; Dogs; Drug Evaluation, Preclinical; Humans; Madin Darby Canine Kidney Cells; Male; Paclitaxel; Rats; Rats, Wistar; Rhodamine 123

2015
Fructose-induced metabolic syndrome decreases protein expression and activity of intestinal P-glycoprotein.
    Nutrition (Burbank, Los Angeles County, Calif.), 2015, Volume: 31, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Availability; Dietary Carbohydrates; Digoxin; Enzyme Inhibitors; Fructose; Ileum; Intestinal Absorption; Intestinal Mucosa; Male; Membrane Transport Proteins; Metabolic Syndrome; Rats, Sprague-Dawley; Rhodamine 123

2015
Expression of P-glycoprotein in excised human nasal mucosa and optimized models of RPMI 2650 cells.
    International journal of pharmaceutics, 2016, Jul-11, Volume: 508, Issue:1-2

    Topics: ATP Binding Cassette Transporter, Subfamily B; Cell Line; Digoxin; Electric Impedance; Humans; Nasal Mucosa; Rhodamine 123

2016
Pharmacokinetic interaction of green tea beverage containing cyclodextrins and high concentration catechins with P-glycoprotein substrates in LLC-GA5-COL150 cells in vitro and in the small intestine of rats in vivo.
    The Journal of pharmacy and pharmacology, 2017, Volume: 69, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Catechin; Cell Line; Cyclodextrins; Digoxin; Food-Drug Interactions; Intestinal Absorption; Intestine, Small; Male; Quinidine; Rats; Rats, Sprague-Dawley; Rhodamine 123; Solubility; Swine; Tea

2017
New insights in the in vitro characterisation and molecular modelling of the P-glycoprotein inhibitory promiscuity.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2018, 08-30, Volume: 121

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Line, Tumor; Digoxin; Humans; Models, Molecular; Rhodamine 123

2018
Cloning and expression of murine sister of P-glycoprotein reveals a more discriminating transporter than MDR1/P-glycoprotein.
    Molecular pharmacology, 2000, Volume: 57, Issue:1

    Topics: Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Cells, Cultured; Cloning, Molecular; DNA, Complementary; Humans; Karyotyping; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Sequence Homology, Amino Acid

2000