rhodamine 123 has been researched along with daunorubicin in 81 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (2.47) | 18.7374 |
1990's | 39 (48.15) | 18.2507 |
2000's | 33 (40.74) | 29.6817 |
2010's | 6 (7.41) | 24.3611 |
2020's | 1 (1.23) | 2.80 |
Authors | Studies |
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Arias, IM; Gatmaitan, Z; Hsing, S | 1 |
Drach, D; Drach, J; Gattringer, C; Hofmann, J; Huber, H; Ludescher, C; Spitaler, M; Thaler, J | 1 |
Aszalos, A; Currier, SJ; Gottesman, MM; Padmanabhan, R; Pine, PS; Schoenlein, PV; Weaver, JL | 1 |
Drach, J; Grunicke, H; Hofmann, J; Ludescher, C | 1 |
Kessel, D | 1 |
Fourcade, A; Lampidis, TJ; Munck, JN; Tapiero, H | 1 |
Gollapudi, S; Gupta, S; Patel, K; Singh, H | 1 |
Assaraf, YG; Borgnia, MJ | 1 |
Bagrij, T; Broxterman, HJ; Scheper, RJ; Twentyman, PR; Versantvoort, CH | 1 |
Lizard, G; Lizard-Nacol, S; Maynadié, M; Poupon, MF; Roignot, P | 1 |
Broxterman, HJ; Feller, N; Kuiper, CM; Lankelma, J; Pinedo, HM; Ruhdal, JK; Scheper, RJ | 1 |
Aszalos, A; Goldenberg, S; Gottesman, MM; Pine, PS; Szabo, G; Weaver, JL | 1 |
Bailly, JD; Bordier, C; Demur, C; Gassar, G; Jaffrézou, JP; Laurent, G; Muller, C | 1 |
Kessel, D; Woodburn, K | 1 |
Cianfriglia, M; Eisterer, W; Gotwald, M; Hilbe, W; Hofmann, J; Ludescher, C; Thaler, J; Zabernigg, A | 1 |
Carbone, R; Chen, HX; Dannies, PS; Hochberg, RB; Jancis, EM | 1 |
Bailly, JD; Cassar, G; Demur, C; Huynh, A; Jaffrézou, JP; Laredo, J; Laurent, G; Muller, C | 1 |
Arias, IM; Fantappié, O; Gatmaitan, Z; Gentilini, P; Kamimoto, Y; Mazzanti, R | 1 |
Altmayr, F; Andreesen, R; Diddens, H; Rastetter, J; Reichle, A | 1 |
Damjanovich, S; Gaspar, R; Goda, K; Krasznai, Z; Lankelma, J; Szabó, G; Westerhoff, HV | 1 |
Bamberger, U; Esteban, M; Heckel, A; Kasimir-Bauer, S; Müller, MR; Scheulen, ME; Schröder, J; Seeber, S | 1 |
Broxterman, HJ; Eekman, CA; Feller, N; Lankelma, J; Löwenberg, B; Ossenkoppele, GJ; Pinedo, HM; Schoester, M; Schuurhuis, GJ; Sonneveld, P; Währer, DC | 1 |
Colombani, PM; Sola, JE | 1 |
Fernández Puentes, JL; García Grávalos, MD; Quesada, AR | 1 |
Buquen, JJ; Canitrot, D; Canitrot, Y; Lahmy, S; Lautier, D | 1 |
Davey, MW; Davey, RA; Hargrave, RM | 1 |
Bordes, M; Lizard, G; Lizard-Nacol, S; Maynadie, M; Poupon, MF; Roignot, P | 1 |
Cybularz-Kolaczkowska, A; Goffeau, A; Kolaczkowski, M; Konings, WN; Soumillion, JP; van der Rest, M | 1 |
Chiba, P; Cordes, HP; Csöllei, J; Ecker, G; Hitzler, M; Schaper, KJ; Schmid, D; Seydel, JK; Visser, K | 1 |
Altenberg, GA; Castro, AF | 1 |
Rhodes, T; Twentyman, PR; Versantvoort, CH | 1 |
Baccarani, M; Damiani, D; Ermacora, A; Fanin, R; Grimaz, S; Lauria, F; Masolini, P; Michelutti, A; Michieli, M; Raspadori, D; Russo, D | 1 |
Boer, R; Gekeler, V; Haas, S; Ise, W; Schödl, A; Ulrich, WR; Zimmermann, P | 1 |
Ashman, LK; Sincock, PM | 1 |
Ling, V; Shapiro, AB | 1 |
Aszalos, A; Weaver, JL | 1 |
Liu, R; Lu, P; Sharom, FJ; Yu, X | 1 |
Calado, RT; Falcão, RP; Garcia, AB | 1 |
Bechmann, G; Chiba, P; Ecker, G; Hitzler, M; Holzer, W; Landau, M; Lorenz, K; Plagens, B; Richter, E | 1 |
Aszalos, A; Molnár, J; Ocsovszki, I; Szabó, D; Szabó, G | 1 |
Chu, JW; Hose, CD; Liu, R; Lu, P; Monks, A; Müller, M; Sarkadi, B; Seprôdi, J; Sharom, FJ; Szabó, K; Váradi, A; Yu, X | 1 |
Casciano, CN; Clement, RP; Johnson, WW; Wang, E | 2 |
Krishan, A | 1 |
Green, LJ; Marder, P; Slapak, CA | 1 |
Azevedo, I; Keating, E; Martel, F | 1 |
Anagnostopoulos, N; Androutsos, G; Galanopoulos, A; Kalmantis, T; Meletis, J; Paterakis, G; Rombos, Y; Sagriotis, A; Symeonidis, A; Tiniakou, M; Tsimberidou, AM; Yataganas, X; Zoumbos, N | 1 |
Cory, JG; Crenshaw, TR | 1 |
Barbier, M; Boumendjel, A; Boutonnat, J; Hadjeri, M; Mariotte, AM; Ronot, X | 1 |
Garnier-Suillerot, A; Loetchutinat, C; Saengkhae, C | 1 |
Lin, QY; Liu, ZM; Luo, HY; Yan, LN; Yang, JY | 1 |
Mori, A; Satsu, H; Shimizu, M; Sugita-Konishi, Y; Tsukazaki, M | 1 |
Aizawa, K; Hatsugai, Y; Inakuma, T; Konishi, T; Nagasawa, H; Nagata, S; Sakuda, SH; Satsu, H; Shimizu, M | 1 |
Balkay, L; Krasznai, Z; Krasznai, ZT; Márián, T; Szabó-Péli, J; Trón, L | 1 |
Hamelik, RM; Krishan, A | 1 |
Das-Gupta, E; Pallis, M | 1 |
Aran, JM; Gottesman, MM; Pétriz, J | 1 |
Huang, W; Li, L; Min, T; Xu, J | 1 |
Murakami, T; Nagai, J; Patanasethanont, D; Sripanidkulchai, BO; Sutthanut, K; Takano, M; Yenjai, C; Yumoto, R | 1 |
Hayashi, M; Idota, Y; Iida, A; Takizawa, Y; Tomita, M | 1 |
Emel'yanov, MO; Korystov, YN; Korystova, AF; Kublik, LN; Shaposhnikova, VV | 1 |
Kashiwada, Y; Kitagawa, S; Nabekura, T; Nakamura, Y; Takahashi, T | 1 |
Chen, SG; Li, GY; Liu, JZ; Wang, CB; Wang, LX; Zhang, B | 1 |
Czyzewski, K; Styczynski, J | 1 |
Bacsó, Z; Goda, K; Szabó, G | 1 |
Baumert, D; Jacobs, A; Möllmann, L; Sterz, K; Wiese, M | 1 |
Ha, I; Han, HK; Im, YB; Kang, KW; Lee, MY | 1 |
Arnoult, C; Barattin, R; Bourges, K; Boutonnat, J; D'Hardemare, AD; Gerby, B; Hardy, G; Olivares, J; Ronot, X | 1 |
Fodor, Z; Galuska, L; Goda, K; Hernádi, Z; Krasznai, ZT; Mikecz, P; Szabó, G; Tóth, A | 1 |
Cannon, RD; Gillet, JP; Gottesman, MM; Holmes, AR; Keniya, MV; Lamping, E; Niimi, M | 1 |
Huang, W; Jiao, L; Li, Y; Liu, B; Qian, H; Qiu, Q; Zhao, T | 1 |
Gorbenko, AS; Olkhovskii, IA | 1 |
Jamialahmadi, K; Mosaffa, F; Palizban, A; Valinezhad Sani, F | 1 |
Hargrove, P; Kim, RB; Lan, LB; Lecureur, V; Schuetz, EG; Schuetz, JD; Sun, D | 1 |
Bates, S; Litman, T; Nagy, Z; Ozvegy, C; Sarkadi, B; Szakács, G; Váradi, A | 1 |
Balakrishnan, L; Janvilisri, T; Reuter, G; Shahi, S; van Veen, HW; Venter, H | 1 |
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ | 1 |
Bauer, KS; Doyle, LA; Fang, HB; Hassel, B; Nakanishi, T; Pumplin, DW; Ross, DD; Wei, Y; Wu, S | 1 |
Borchardt, RT; Ouyang, H; Tang, F; Yang, JZ | 1 |
Globisch, C; Kassack, MU; Klinkhammer, W; Müller, H; Pajeva, IK; Wiese, M | 1 |
Ghosh, I; Manoharlal, R; Prakash, O; Prasad, R; Puri, N; Sharma, M | 1 |
1 review(s) available for rhodamine 123 and daunorubicin
Article | Year |
---|---|
Multidrug resistance through the spectacle of P-glycoprotein.
Topics: Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cloning, Molecular; Daunorubicin; Drug Resistance, Multiple; Genes, MDR; Humans; Kinetics; Models, Genetic; Neoplasms; Rhodamine 123 | 2009 |
1 trial(s) available for rhodamine 123 and daunorubicin
Article | Year |
---|---|
Cyclosporine diminishes multidrug resistance in K562/ADM cells and improves complete remission in patients with acute myeloid leukemia.
Topics: Adult; Antibiotics, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Cyclosporine; Cytarabine; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Fluorescent Dyes; Humans; Idarubicin; Inhibitory Concentration 50; K562 Cells; Leukemia, Myeloid, Acute; Male; Rhodamine 123; Time Factors; Treatment Outcome; Verapamil | 2009 |
79 other study(ies) available for rhodamine 123 and daunorubicin
Article | Year |
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The function of Gp170, the multidrug-resistance gene product, in the brush border of rat intestinal mucosa.
Topics: Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Colchicine; Daunorubicin; Diltiazem; Dose-Response Relationship, Drug; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Ileum; In Vitro Techniques; Intestinal Mucosa; Jejunum; Male; Membrane Glycoproteins; Microvilli; Rats; Rats, Inbred Strains; Rhodamine 123; Rhodamines; Temperature; Verapamil | 1992 |
Detection of activity of P-glycoprotein in human tumour samples using rhodamine 123.
Topics: Acute Disease; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Daunorubicin; Drug Resistance; Humans; Leukemia, Myeloid; Membrane Glycoproteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1992 |
Laser scanning and confocal microscopy of daunorubicin, doxorubicin, and rhodamine 123 in multidrug-resistant cells.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Daunorubicin; Doxorubicin; Drug Resistance; Humans; KB Cells; Lasers; Membrane Glycoproteins; Mice; Microscopy, Fluorescence; Rhodamine 123; Rhodamines; Transfection; Verapamil | 1991 |
Rapid functional assay for the detection of multidrug-resistant cells using the fluorescent dye rhodamine 123.
Topics: Cell Line; Daunorubicin; Drug Resistance; Fluorescent Dyes; Rhodamine 123; Rhodamines | 1991 |
Exploring multidrug resistance using rhodamine 123.
Topics: Animals; Daunorubicin; Doxorubicin; Drug Resistance; Fluorescent Dyes; Kinetics; Leukemia P388; Leukemia, Experimental; Mice; Microscopy, Fluorescence; Rhodamine 123; Rhodamines; Spectrometry, Fluorescence; Tumor Cells, Cultured | 1989 |
Cross-resistance to rhodamine 123 in Adriamycin- and daunorubicin-resistant Friend leukemia cell variants.
Topics: Animals; Biological Transport; Cell Line; Daunorubicin; Doxorubicin; Drug Resistance; Kinetics; Leukemia, Experimental; Mice; Rhodamine 123; Rhodamines; Xanthenes | 1984 |
Effect of Calphostin C (PKC inhibitor) on daunorubicin resistance in P388/ADR and HL60/AR cells: reversal of drug resistance possibly via P-glycoprotein.
Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Leukemia P388; Leukemia, Experimental; Leukemia, Myeloid; Membrane Glycoproteins; Mice; Naphthalenes; Polycyclic Compounds; Protein Kinase C; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1994 |
Probing the interaction of the multidrug-resistance phenotype with the polypeptide ionophore gramicidin D via functional channel formation.
Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cell Line; CHO Cells; Cricetinae; Cricetulus; Daunorubicin; Drug Resistance; Flow Cytometry; Gene Amplification; Gramicidin; Ion Channels; Ionophores; Membrane Glycoproteins; Phenotype; Rhodamine 123; Rhodamines; Rubidium; Sodium-Potassium-Exchanging ATPase | 1994 |
Regulation by glutathione of drug transport in multidrug-resistant human lung tumour cell lines overexpressing multidrug resistance-associated protein.
Topics: Biological Transport; Buthionine Sulfoximine; Daunorubicin; Drug Resistance, Multiple; Glutathione; Humans; Lung Neoplasms; Methionine Sulfoximine; Rhodamine 123; Rhodamines; RNA, Messenger; Tumor Cells, Cultured | 1995 |
Evaluation of multidrug resistant phenotype by flow cytometry with monoclonal antibodies and functional tests.
Topics: Antibodies, Monoclonal; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Antibody Technique; Fluorescent Dyes; Humans; Leukemia, Erythroblastic, Acute; Lymphoma, Non-Hodgkin; Phenotype; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Rhodamine 123; Rhodamines | 1995 |
Functional detection of MDR1/P170 and MRP/P190-mediated multidrug resistance in tumour cells by flow cytometry.
Topics: Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; KB Cells; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Sensitivity and Specificity | 1995 |
The effect of ion channel blockers, immunosuppressive agents, and other drugs on the activity of the multi-drug transporter.
Topics: Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzofurans; Biological Transport, Active; Carrier Proteins; Cell Membrane; Daunorubicin; Drug Resistance; Ethers, Cyclic; Flow Cytometry; Fluorescent Dyes; Hydrogen-Ion Concentration; Immunosuppressive Agents; Intracellular Fluid; Ion Channels; Leukemia L5178; Lymphoma, T-Cell; Membrane Glycoproteins; Membrane Potentials; Mice; Molecular Sequence Data; Potassium; Potassium Channels; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1993 |
Lack of correlation between expression and function of P-glycoprotein in acute myeloid leukemia cell lines.
Topics: Acute Disease; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Differentiation; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Flow Cytometry; Gene Expression; Humans; Immunohistochemistry; Leukemia, Myeloid; Phenotype; Polymerase Chain Reaction; Rhodamine 123; Rhodamines; Transcription, Genetic; Tumor Cells, Cultured; Vincristine | 1995 |
Selective photodynamic inactivation of a multidrug transporter by a cationic photosensitising agent.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cycloleucine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Leukemia P388; Mice; Microscopy, Fluorescence; Neoplasm Proteins; Oxygen; Photochemotherapy; Radiation-Sensitizing Agents; Rhodamine 123; Rhodamines; Singlet Oxygen; Spectrometry, Fluorescence; Tumor Cells, Cultured | 1995 |
Low frequency of activity of P-glycoprotein (P-170) in acute lymphoblastic leukemia compared to acute myeloid leukemia.
Topics: Acute Disease; Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow; Bone Marrow Transplantation; Child; Child, Preschool; Cytarabine; Daunorubicin; Drug Resistance, Multiple; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Neoplasm Proteins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prognosis; Remission Induction; Rhodamine 123; Rhodamines; Survival Analysis | 1995 |
Rapid stimulation of rhodamine 123 efflux from multidrug-resistant KB cells by progesterone.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carrier Proteins; Daunorubicin; Drug Resistance; Exocytosis; Fluorescent Dyes; Humans; Membrane Glycoproteins; Membrane Potentials; Mice; Progesterone; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Up-Regulation; Verapamil | 1993 |
Effect of the protein kinase C inhibitor staurosporine on chemosensitivity to daunorubicin of normal and leukemic fresh myeloid cells.
Topics: Adult; Aged; Aged, 80 and over; Alkaloids; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Child; Daunorubicin; Hematopoietic Stem Cells; Humans; Leukemia, Myeloid, Acute; Membrane Glycoproteins; Middle Aged; Neoplastic Stem Cells; Protein Kinase C; Rhodamine 123; Rhodamines; Staurosporine; Tumor Cells, Cultured | 1994 |
Bile acid inhibition of P-glycoprotein-mediated transport in multidrug-resistant cells and rat liver canalicular membrane vesicles.
Topics: Animals; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile Acids and Salts; Bile Canaliculi; Biological Transport; Carcinoma, Hepatocellular; Carrier Proteins; Cell Membrane; Daunorubicin; Depression, Chemical; Doxorubicin; Drug Resistance; Liver Neoplasms; Male; Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1994 |
Chemomodulation of drugs involved in multidrug resistance in chronic lymphatic leukemia of the B-cell type.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Daunorubicin; Drug Resistance; Flow Cytometry; Humans; Immunophenotyping; In Vitro Techniques; Leukemia, Lymphocytic, Chronic, B-Cell; Membrane Glycoproteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Verapamil; Vincristine | 1994 |
Reversal of multidrug resistance by valinomycin is overcome by CCCP.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Coloring Agents; Daunorubicin; Drug Resistance, Multiple; Humans; Ionophores; KB Cells; Kinetics; Potassium; Rhodamine 123; Rhodamines; Valinomycin; Vinblastine | 1996 |
Modulation of multidrug resistance by BIBW22BS in blasts of de novo or relapsed or persistent acute myeloid leukemia ex vivo.
Topics: Antigens, CD34; Daunorubicin; Drug Resistance, Multiple; Humans; Idarubicin; Leukemia, Myeloid, Acute; Morpholines; Rhodamine 123; Rhodamines; Triamterene | 1996 |
Quality control of multidrug resistance assays in adult acute leukemia: correlation between assays for P-glycoprotein expression and activity.
Topics: Acute Disease; Adult; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cryopreservation; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Feasibility Studies; Fluorescent Dyes; Humans; Leukemia; Leukemia, Myeloid; Neoplasm Proteins; Neoplastic Stem Cells; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Reproducibility of Results; Rhodamine 123; Rhodamines; Sensitivity and Specificity; Verapamil; Vincristine | 1996 |
Modulation of multidrug resistance with antisense oligodeoxynucleotide to mdr1 mRNA.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Codon; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Humans; Leukemia, Erythroblastic, Acute; Oligonucleotides, Antisense; Rhodamine 123; Rhodamines; RNA, Messenger; Thymidine; Tumor Cells, Cultured | 1996 |
Polyaromatic alkaloids from marine invertebrates as cytotoxic compounds and inhibitors of multidrug resistance caused by P-glycoprotein.
Topics: Adenocarcinoma; Alkaloids; Animals; Antimetabolites, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Survival; Colonic Neoplasms; Cricetinae; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Leukemia P388; Lung Neoplasms; Mice; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Verapamil; Vinblastine | 1996 |
Functional study of multidrug resistance with fluorescent dyes. Limits of the assay for low levels of resistance and application in clinical samples.
Topics: Animals; Anthracyclines; Benzimidazoles; Cell Survival; Clone Cells; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Leukemia L1210; Mice; Phenotype; Quantum Theory; Reproducibility of Results; Rhodamine 123; Rhodamines; Sensitivity and Specificity; Tumor Cells, Cultured; Vinblastine | 1996 |
Comparison of drug accumulation in P-glycoprotein-expressing and MRP-expressing human leukaemia cells.
Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Buthionine Sulfoximine; Calcium Channel Blockers; Cyclosporins; Daunorubicin; Humans; Idarubicin; Leukemia, T-Cell; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Verapamil | 1996 |
Flow cytometry evaluation of the multidrug-resistant phenotype with functional tests involving uptake of daunorubicin, Hoechst 33342, or rhodamine 123: a comparative study.
Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Death; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Hot Temperature; Humans; Phenotype; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1995 |
Anticancer drugs, ionophoric peptides, and steroids as substrates of the yeast multidrug transporter Pdr5p.
Topics: Animals; Antineoplastic Agents; ATP-Binding Cassette Transporters; Daunorubicin; Desoxycorticosterone; Doxorubicin; Fungal Proteins; Ionophores; Kinetics; Membrane Proteins; Phenotype; Progesterone; Rhodamine 123; Rhodamines; Saccharomyces cerevisiae Proteins | 1996 |
Structure-activity relationship studies on benzofuran analogs of propafenone-type modulators of tumor cell multidrug resistance.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzofurans; Calorimetry, Differential Scanning; Cells, Cultured; Daunorubicin; Drug Resistance, Multiple; Ethanolamines; Liposomes; Magnetic Resonance Spectroscopy; Membranes, Artificial; Propafenone; Regression Analysis; Rhodamine 123; Rhodamines; Structure-Activity Relationship | 1996 |
Inhibition of drug transport by genistein in multidrug-resistant cells expressing P-glycoprotein.
Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport; Daunorubicin; Drug Resistance, Multiple; Enzyme Inhibitors; Genistein; Humans; Isoflavones; Mice; Multidrug Resistance-Associated Proteins; Protein-Tyrosine Kinases; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1997 |
Acceleration of MRP-associated efflux of rhodamine 123 by genistein and related compounds.
Topics: Antimetabolites, Antineoplastic; Daunorubicin; Drug Resistance, Multiple; Genistein; Humans; Isoflavones; Monosaccharide Transport Proteins; Quercetin; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1996 |
P-glycoprotein (PGP) and lung resistance-related protein (LRP) expression and function in leukaemic blast cells.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Leukemia; Lymphocytes; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Vault Ribonucleoprotein Particles | 1997 |
Modulation of P-glycoprotein mediated drug accumulation in multidrug resistant CCRF VCR-1000 cells by chemosensitisers.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Vincristine | 1996 |
Expression of c-Kit and functional drug efflux are correlated in de novo acute myeloid leukaemia.
Topics: Acute Disease; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Fluorescent Antibody Technique, Indirect; Humans; Immunosuppressive Agents; Leukemia, Myeloid; Phenotype; Proto-Oncogene Proteins c-kit; Rhodamine 123; Rhodamines; Tumor Cells, Cultured | 1997 |
Positively cooperative sites for drug transport by P-glycoprotein with distinct drug specificities.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Daunorubicin; Doxorubicin; Etoposide; Fluorescence; Fluorescent Dyes; Kinetics; Liposomes; Protein Binding; Quercetin; Rhodamine 123; Rhodamines; Vinblastine | 1997 |
Estimation of drug resistance by flow cytometry.
Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Genistein; Leukemia L5178; Mice; Probenecid; Recombinant Proteins; Rhodamine 123; Rhodamines; Transfection; Tumor Cells, Cultured; Verapamil | 1998 |
Linear and cyclic peptides as substrates and modulators of P-glycoprotein: peptide binding and effects on drug transport and accumulation.
Topics: Adenosine Triphosphatases; Animals; Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Membrane; CHO Cells; Cricetinae; Daunorubicin; Drug Resistance, Multiple; Ionophores; Kinetics; Oligopeptides; Peptides, Cyclic; Protein Binding; Rhodamine 123; Rhodamines; Substrate Specificity | 1998 |
Decreased activity of the multidrug resistance P-glycoprotein in acquired aplastic anaemia: possible pathophysiologic implications.
Topics: Adolescent; Adult; Anemia, Aplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Child; Child, Preschool; Daunorubicin; Drug Resistance, Multiple; Female; Fluorescent Dyes; Humans; Male; Rhodamine 123 | 1998 |
Substituted 4-acylpyrazoles and 4-acylpyrazolones: synthesis and multidrug resistance-modulating activity.
Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Isomerism; Magnetic Resonance Spectroscopy; Mice; Pyrazoles; Regression Analysis; Rhodamine 123; Structure-Activity Relationship; Tumor Cells, Cultured | 1998 |
Anti-psychotic drugs reverse multidrug resistance of tumor cell lines and human AML cells ex-vivo.
Topics: Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Interactions; Drug Resistance, Multiple; Enzyme Inhibitors; Humans; Leukemia, Myeloid; Rhodamine 123; Tumor Cells, Cultured | 1999 |
Interaction of the P-glycoprotein multidrug transporter (MDR1) with high affinity peptide chemosensitizers in isolated membranes, reconstituted systems, and intact cells.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cell Membrane; CHO Cells; Colchicine; Cricetinae; Daunorubicin; Dihydropyridines; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Oligopeptides; Peptides; Photoaffinity Labels; Rhodamine 123; Tumor Cells, Cultured | 1999 |
Cholesterol interaction with the daunorubicin binding site of P-glycoprotein.
Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Biological Transport, Active; Cell Line; Cell Survival; Cholesterol; Daunorubicin; Flow Cytometry; Fluorescence; Humans; Hydrolysis; Inhibitory Concentration 50; Kinetics; Microsomes; Protein Binding; Rhodamine 123 | 2000 |
Monitoring of cellular resistance to cancer chemotherapy: drug retention and efflux.
Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Calcium Channel Blockers; Cell Membrane Permeability; Chlorpromazine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Dyes; Humans; Mice; Rhodamine 123; Staining and Labeling; Tumor Cells, Cultured; Verapamil | 2001 |
Modulation by LY335979 of P-glycoprotein function in multidrug-resistant cell lines and human natural killer cells.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Dibenzocycloheptenes; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Fluorescent Dyes; HL-60 Cells; Humans; Killer Cells, Natural; Quinolines; Rhodamine 123 | 2001 |
Effect of P-glycoprotein modulators on the human extraneuronal monoamine transporter.
Topics: 1-Methyl-4-phenylpyridinium; Arginine; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carrier Proteins; Cations; Cell Line; Cyclosporine; Daunorubicin; Dose-Response Relationship, Drug; Histidine; Humans; Organic Cation Transport Proteins; Rhodamine 123; Time Factors; Tritium; Tyramine; Verapamil; Vinblastine | 2001 |
The farnesyl protein transferase inhibitor SCH66336 is a potent inhibitor of MDR1 product P-glycoprotein.
Topics: 3T3 Cells; Adenosine Triphosphate; Alkyl and Aryl Transferases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Line; CHO Cells; Cricetinae; Daunorubicin; Drug Synergism; Enzyme Inhibitors; Farnesyltranstransferase; Genes, MDR; Humans; Hydrolysis; Mice; Paclitaxel; Piperidines; Pyridines; Rhodamine 123; Tamoxifen; Vinblastine | 2001 |
Evaluation of the clinical relevance of the expression and function of P-glycoprotein, multidrug resistance protein and lung resistance protein in patients with primary acute myelogenous leukemia.
Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow Transplantation; Calcium Channel Blockers; Carbocyanines; Combined Modality Therapy; Cytarabine; Daunorubicin; Disease-Free Survival; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Female; Fluoresceins; Fluorescent Dyes; Genistein; Humans; Idarubicin; Immunophenotyping; Leukemia, Myeloid; Male; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; Prognosis; Prospective Studies; Rhodamine 123; Survival Analysis; Tumor Cells, Cultured; Vault Ribonucleoprotein Particles; Verapamil | 2002 |
Overexpression of protein disulfide isomerase-like protein in a mouse leukemia L1210 cell line selected for resistance to 4-methyl-5-amino-1-formylisoquinoline thiosemicarbazone, a ribonucleotide reductase inhibitor.
Topics: Amino Acid Sequence; Animals; Antibiotics, Antineoplastic; Blotting, Northern; Blotting, Southern; Blotting, Western; Cell Line; Daunorubicin; DNA, Complementary; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Fluorescent Dyes; Isoquinolines; Mice; Molecular Sequence Data; Protein Biosynthesis; Protein Disulfide-Isomerases; Proteins; Rhodamine 123; Ribonucleotide Reductases; RNA, Messenger; Sulfhydryl Compounds | 2002 |
Modulation of P-glycoprotein-mediated multidrug resistance by flavonoid derivatives and analogues.
Topics: Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Chromones; Daunorubicin; Drug Resistance, Multiple; Drug Synergism; Flavonoids; Fluorescent Dyes; Humans; Necrosis; Piperazines; Quinolinium Compounds; Rhodamine 123; Thiazoles; Tumor Cells, Cultured | 2003 |
Kinetic analysis of rhodamines efflux mediated by the multidrug resistance protein (MRP1).
Topics: Biophysical Phenomena; Biophysics; Cell Line, Tumor; Chlorine; Daunorubicin; Dose-Response Relationship, Drug; Fluorescent Dyes; Glutathione; Humans; Kinetics; Membrane Potentials; Models, Chemical; Models, Theoretical; Multidrug Resistance-Associated Proteins; Phenotype; Potassium; Rhodamine 123; Rhodamines; Time Factors | 2003 |
[Reversal of multidrug resistance gene MDR1 and MRP of drug-resistant human hepatocellular carcinoma cells SMMC-7721/ADM with antisense phosphorothioate oligonucleotides].
Topics: Carcinoma, Hepatocellular; Cell Line, Tumor; Daunorubicin; Doxorubicin; Drug Resistance, Neoplasm; Genes, MDR; Humans; Liver Neoplasms; Multidrug Resistance-Associated Proteins; Oligonucleotides, Antisense; Rhodamine 123 | 2004 |
Effects of tributyltin on barrier functions in human intestinal Caco-2 cells.
Topics: Actin Cytoskeleton; Alkaline Phosphatase; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; CD13 Antigens; Cell Membrane Permeability; Daunorubicin; Electric Impedance; Epithelium; Humans; Intestinal Absorption; Intestinal Mucosa; Isoquinolines; Rhodamine 123; RNA, Messenger; Tight Junctions; Time Factors; Trialkyltin Compounds | 2004 |
Inhibitory effect of a bitter melon extract on the P-glycoprotein activity in intestinal Caco-2 cells.
Topics: Adenocarcinoma; Amino Acids; ATP Binding Cassette Transporter, Subfamily B; Biological Transport; Caco-2 Cells; Chromatography, High Pressure Liquid; Colonic Neoplasms; Daunorubicin; Dose-Response Relationship, Drug; Fruit; Glycerides; Hot Temperature; Humans; L-Lactate Dehydrogenase; Mass Spectrometry; Methanol; Momordica charantia; Plant Extracts; Pronase; Rhodamine 123; Vegetables | 2004 |
Effects of miltefosine on membrane permeability and accumulation of [99mTc]-hexakis-2-methoxyisobutyl isonitrile, 2-[18F]fluoro-2-deoxy-D-glucose, daunorubucin and rhodamine123 in multidrug-resistant and sensitive cells.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Membrane Permeability; Daunorubicin; Drug Resistance, Multiple; Fluorodeoxyglucose F18; Humans; Membrane Fluidity; Mice; NIH 3T3 Cells; Phosphorylcholine; Rhodamine 123; Technetium Tc 99m Sestamibi; Verapamil | 2005 |
Flow cytometric monitoring of fluorescent drug retention and efflux.
Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Daunorubicin; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Flow Cytometry; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; Phenotype; Rhodamine 123 | 2005 |
Flow cytometric measurement of functional and phenotypic P-glycoprotein.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Clinical Trials as Topic; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Leukemia, Myeloid, Acute; Leukocyte Common Antigens; Microscopy, Fluorescence; Phenotype; Rhodamine 123 | 2005 |
An MDR-EGFP gene fusion allows for direct cellular localization, function and stability assessment of P-glycoprotein.
Topics: Amino Acid Sequence; Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Line; Cell Survival; Daunorubicin; DNA Primers; Dogs; Doxorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescence; Fluorescent Antibody Technique; Gene Fusion; Genes, MDR; Genetic Vectors; Green Fluorescent Proteins; Humans; Microscopy, Confocal; Molecular Sequence Data; Oligonucleotides; Rhodamine 123; Subcellular Fractions; Transfection | 2004 |
Reversal of MDR1 gene-dependent multidrug resistance using low concentration of endonuclease-prepared small interference RNA.
Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Survival; CHO Cells; Cricetinae; Cricetulus; Daunorubicin; Dose-Response Relationship, Drug; Down-Regulation; Drug Resistance, Neoplasm; Green Fluorescent Proteins; Humans; Plasmids; Recombinant Fusion Proteins; Rhodamine 123; Ribonuclease III; RNA Interference; RNA, Messenger; RNA, Small Interfering; Transfection | 2006 |
Effects of Kaempferia parviflora extracts and their flavone constituents on P-glycoprotein function.
Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Ethanol; Flavones; Flavonoids; Fluorescent Dyes; Humans; LLC-PK1 Cells; Plant Extracts; Rhizome; Rhodamine 123; Solvents; Swine; Time Factors; Transfection; Water; Zingiberaceae | 2007 |
Improvement of intestinal absorption of P-glycoprotein substrate by D-tartaric acid.
Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blotting, Western; Cardiovascular Agents; Colon; Daunorubicin; Diffusion Chambers, Culture; Fluorescent Dyes; Ileum; Injections, Intravenous; Intestinal Absorption; Jejunum; Male; Rats; Rats, Wistar; Rhodamine 123; Tartrates; Verapamil | 2006 |
Modification of multidrug resistance of tumor cells by ionizing radiation.
Topics: Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; Cell Count; Cell Line, Tumor; Combined Modality Therapy; Cyclosporine; Daunorubicin; Dose-Response Relationship, Radiation; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Laryngeal Neoplasms; Paclitaxel; Radiation, Ionizing; Reactive Oxygen Species; Rhodamine 123; Time Factors; Vincristine | 2008 |
Inhibition of P-glycoprotein function by tannic acid and pentagalloylglucose.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Humans; Hydrolyzable Tannins; KB Cells; Rhodamine 123; Tannins | 2007 |
Imatinib is a substrate for various multidrug resistance proteins.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Daunorubicin; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; K562 Cells; Multidrug Resistance-Associated Proteins; Piperazines; Pyrimidines; Rhodamine 123; Vault Ribonucleoprotein Particles | 2009 |
Activators of P-glycoprotein: Structure-activity relationships and investigation of their mode of action.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Benzothiazoles; Cell Line, Tumor; Daunorubicin; Drug Resistance, Neoplasm; Humans; Imidazoles; Rhodamine 123; Structure-Activity Relationship; Thiazoles | 2009 |
Macelignan: a new modulator of P-glycoprotein in multidrug-resistant cancer cells.
Topics: Adenocarcinoma; Analysis of Variance; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B; Biological Transport, Active; Breast Neoplasms; Cell Line, Tumor; Cell Survival; Daunorubicin; Dose-Response Relationship, Drug; Drug Design; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Female; Fluorescent Dyes; Growth Inhibitors; Humans; Lignans; Phytoestrogens; Phytotherapy; Rhodamine 123; Vinblastine | 2009 |
Iodination increases the activity of verapamil derivatives in reversing PGP multidrug resistance.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Cycle; Cyclosporine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Humans; K562 Cells; Male; Myocytes, Cardiac; Rats; Rats, Wistar; Rhodamine 123; Verapamil | 2010 |
Pgp inhibition by UIC2 antibody can be followed in vitro by using tumor-diagnostic radiotracers, 99mTc-MIBI and 18FDG.
Topics: Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Female; Fluorodeoxyglucose F18; Glucose; Humans; Ovarian Neoplasms; Paclitaxel; Protein Binding; Rhodamine 123; Technetium Tc 99m Sestamibi; Tumor Cells, Cultured | 2010 |
Drug resistance is conferred on the model yeast Saccharomyces cerevisiae by expression of full-length melanoma-associated human ATP-binding cassette transporter ABCB5.
Topics: ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Clorgyline; Daunorubicin; Humans; Melanoma; Rhodamine 123; Rhodamines; Saccharomyces cerevisiae; Tacrolimus | 2014 |
6,7-Dimethoxy-2-{2-[4-(1H-1,2,3-triazol-1-yl)phenyl]ethyl}-1,2,3,4-tetrahydroisoquinolines as superior reversal agents for P-glycoprotein-mediated multidrug resistance.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Benzamides; Cell Survival; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Daunorubicin; Drug Resistance, Neoplasm; Humans; K562 Cells; Paclitaxel; Protein Binding; Rhodamine 123; Structure-Activity Relationship; Tetrahydroisoquinolines; Triazoles; Vincristine | 2015 |
[The study of mechanisms of accumulation of daunorubicin and rodamin-123 in cells of human venous blood using cytometry technique].
Topics: Blood Platelets; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Healthy Volunteers; Humans; Leukocytes; Neoplasms; Rhodamine 123 | 2015 |
Glucosamine Reverses P-Glycoprotein-Mediated Multidrug Resistance in the Daunorubicin-Resistant Human Gastric Cancer Cells.
Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Proliferation; Cell Survival; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Glucosamine; Humans; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Neoplasm; Stomach Neoplasms | 2020 |
Cloning and expression of murine sister of P-glycoprotein reveals a more discriminating transporter than MDR1/P-glycoprotein.
Topics: Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Cells, Cultured; Cloning, Molecular; DNA, Complementary; Humans; Karyotyping; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Sequence Homology, Amino Acid | 2000 |
Functional characterization of the human multidrug transporter, ABCG2, expressed in insect cells.
Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Membrane; Cloning, Molecular; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Recombinant Proteins; Spodoptera; Tumor Cells, Cultured | 2001 |
Sterol transport by the human breast cancer resistance protein (ABCG2) expressed in Lactococcus lactis.
Topics: Antineoplastic Agents, Hormonal; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cholesterol; Estradiol; Gene Expression; Humans; Lactococcus lactis; Neoplasm Proteins; Progesterone; Sterols; Tamoxifen; Testosterone; Tritium | 2003 |
Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.
Topics: ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Binding Sites; Biological Transport, Active; Biomarkers; Cells, Cultured; Drug Interactions; Fluorescent Dyes; Humans | 2003 |
Functional characterization of human breast cancer resistance protein (BCRP, ABCG2) expressed in the oocytes of Xenopus laevis.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Drug Resistance, Neoplasm; Female; Gene Expression Regulation, Neoplastic; Humans; Neoplasm Proteins; Oocytes; Xenopus laevis | 2003 |
Bidirectional transport of rhodamine 123 and Hoechst 33342, fluorescence probes of the binding sites on P-glycoprotein, across MDCK-MDR1 cell monolayers.
Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Dogs; Fluorescent Dyes; Humans; Rhodamine 123 | 2004 |
New functional assay of P-glycoprotein activity using Hoechst 33342.
Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fluoresceins; Humans; Microscopy, Fluorescence; Molecular Structure; Principal Component Analysis; Time Factors | 2007 |
Analysis of physico-chemical properties of substrates of ABC and MFS multidrug transporters of pathogenic Candida albicans.
Topics: Candida albicans; Membrane Transport Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Substrate Specificity | 2010 |