Page last updated: 2024-08-24

rhodamine 123 and daunorubicin

rhodamine 123 has been researched along with daunorubicin in 81 studies

Research

Studies (81)

TimeframeStudies, this research(%)All Research%
pre-19902 (2.47)18.7374
1990's39 (48.15)18.2507
2000's33 (40.74)29.6817
2010's6 (7.41)24.3611
2020's1 (1.23)2.80

Authors

AuthorsStudies
Arias, IM; Gatmaitan, Z; Hsing, S1
Drach, D; Drach, J; Gattringer, C; Hofmann, J; Huber, H; Ludescher, C; Spitaler, M; Thaler, J1
Aszalos, A; Currier, SJ; Gottesman, MM; Padmanabhan, R; Pine, PS; Schoenlein, PV; Weaver, JL1
Drach, J; Grunicke, H; Hofmann, J; Ludescher, C1
Kessel, D1
Fourcade, A; Lampidis, TJ; Munck, JN; Tapiero, H1
Gollapudi, S; Gupta, S; Patel, K; Singh, H1
Assaraf, YG; Borgnia, MJ1
Bagrij, T; Broxterman, HJ; Scheper, RJ; Twentyman, PR; Versantvoort, CH1
Lizard, G; Lizard-Nacol, S; Maynadié, M; Poupon, MF; Roignot, P1
Broxterman, HJ; Feller, N; Kuiper, CM; Lankelma, J; Pinedo, HM; Ruhdal, JK; Scheper, RJ1
Aszalos, A; Goldenberg, S; Gottesman, MM; Pine, PS; Szabo, G; Weaver, JL1
Bailly, JD; Bordier, C; Demur, C; Gassar, G; Jaffrézou, JP; Laurent, G; Muller, C1
Kessel, D; Woodburn, K1
Cianfriglia, M; Eisterer, W; Gotwald, M; Hilbe, W; Hofmann, J; Ludescher, C; Thaler, J; Zabernigg, A1
Carbone, R; Chen, HX; Dannies, PS; Hochberg, RB; Jancis, EM1
Bailly, JD; Cassar, G; Demur, C; Huynh, A; Jaffrézou, JP; Laredo, J; Laurent, G; Muller, C1
Arias, IM; Fantappié, O; Gatmaitan, Z; Gentilini, P; Kamimoto, Y; Mazzanti, R1
Altmayr, F; Andreesen, R; Diddens, H; Rastetter, J; Reichle, A1
Damjanovich, S; Gaspar, R; Goda, K; Krasznai, Z; Lankelma, J; Szabó, G; Westerhoff, HV1
Bamberger, U; Esteban, M; Heckel, A; Kasimir-Bauer, S; Müller, MR; Scheulen, ME; Schröder, J; Seeber, S1
Broxterman, HJ; Eekman, CA; Feller, N; Lankelma, J; Löwenberg, B; Ossenkoppele, GJ; Pinedo, HM; Schoester, M; Schuurhuis, GJ; Sonneveld, P; Währer, DC1
Colombani, PM; Sola, JE1
Fernández Puentes, JL; García Grávalos, MD; Quesada, AR1
Buquen, JJ; Canitrot, D; Canitrot, Y; Lahmy, S; Lautier, D1
Davey, MW; Davey, RA; Hargrave, RM1
Bordes, M; Lizard, G; Lizard-Nacol, S; Maynadie, M; Poupon, MF; Roignot, P1
Cybularz-Kolaczkowska, A; Goffeau, A; Kolaczkowski, M; Konings, WN; Soumillion, JP; van der Rest, M1
Chiba, P; Cordes, HP; Csöllei, J; Ecker, G; Hitzler, M; Schaper, KJ; Schmid, D; Seydel, JK; Visser, K1
Altenberg, GA; Castro, AF1
Rhodes, T; Twentyman, PR; Versantvoort, CH1
Baccarani, M; Damiani, D; Ermacora, A; Fanin, R; Grimaz, S; Lauria, F; Masolini, P; Michelutti, A; Michieli, M; Raspadori, D; Russo, D1
Boer, R; Gekeler, V; Haas, S; Ise, W; Schödl, A; Ulrich, WR; Zimmermann, P1
Ashman, LK; Sincock, PM1
Ling, V; Shapiro, AB1
Aszalos, A; Weaver, JL1
Liu, R; Lu, P; Sharom, FJ; Yu, X1
Calado, RT; Falcão, RP; Garcia, AB1
Bechmann, G; Chiba, P; Ecker, G; Hitzler, M; Holzer, W; Landau, M; Lorenz, K; Plagens, B; Richter, E1
Aszalos, A; Molnár, J; Ocsovszki, I; Szabó, D; Szabó, G1
Chu, JW; Hose, CD; Liu, R; Lu, P; Monks, A; Müller, M; Sarkadi, B; Seprôdi, J; Sharom, FJ; Szabó, K; Váradi, A; Yu, X1
Casciano, CN; Clement, RP; Johnson, WW; Wang, E2
Krishan, A1
Green, LJ; Marder, P; Slapak, CA1
Azevedo, I; Keating, E; Martel, F1
Anagnostopoulos, N; Androutsos, G; Galanopoulos, A; Kalmantis, T; Meletis, J; Paterakis, G; Rombos, Y; Sagriotis, A; Symeonidis, A; Tiniakou, M; Tsimberidou, AM; Yataganas, X; Zoumbos, N1
Cory, JG; Crenshaw, TR1
Barbier, M; Boumendjel, A; Boutonnat, J; Hadjeri, M; Mariotte, AM; Ronot, X1
Garnier-Suillerot, A; Loetchutinat, C; Saengkhae, C1
Lin, QY; Liu, ZM; Luo, HY; Yan, LN; Yang, JY1
Mori, A; Satsu, H; Shimizu, M; Sugita-Konishi, Y; Tsukazaki, M1
Aizawa, K; Hatsugai, Y; Inakuma, T; Konishi, T; Nagasawa, H; Nagata, S; Sakuda, SH; Satsu, H; Shimizu, M1
Balkay, L; Krasznai, Z; Krasznai, ZT; Márián, T; Szabó-Péli, J; Trón, L1
Hamelik, RM; Krishan, A1
Das-Gupta, E; Pallis, M1
Aran, JM; Gottesman, MM; Pétriz, J1
Huang, W; Li, L; Min, T; Xu, J1
Murakami, T; Nagai, J; Patanasethanont, D; Sripanidkulchai, BO; Sutthanut, K; Takano, M; Yenjai, C; Yumoto, R1
Hayashi, M; Idota, Y; Iida, A; Takizawa, Y; Tomita, M1
Emel'yanov, MO; Korystov, YN; Korystova, AF; Kublik, LN; Shaposhnikova, VV1
Kashiwada, Y; Kitagawa, S; Nabekura, T; Nakamura, Y; Takahashi, T1
Chen, SG; Li, GY; Liu, JZ; Wang, CB; Wang, LX; Zhang, B1
Czyzewski, K; Styczynski, J1
Bacsó, Z; Goda, K; Szabó, G1
Baumert, D; Jacobs, A; Möllmann, L; Sterz, K; Wiese, M1
Ha, I; Han, HK; Im, YB; Kang, KW; Lee, MY1
Arnoult, C; Barattin, R; Bourges, K; Boutonnat, J; D'Hardemare, AD; Gerby, B; Hardy, G; Olivares, J; Ronot, X1
Fodor, Z; Galuska, L; Goda, K; Hernádi, Z; Krasznai, ZT; Mikecz, P; Szabó, G; Tóth, A1
Cannon, RD; Gillet, JP; Gottesman, MM; Holmes, AR; Keniya, MV; Lamping, E; Niimi, M1
Huang, W; Jiao, L; Li, Y; Liu, B; Qian, H; Qiu, Q; Zhao, T1
Gorbenko, AS; Olkhovskii, IA1
Jamialahmadi, K; Mosaffa, F; Palizban, A; Valinezhad Sani, F1
Hargrove, P; Kim, RB; Lan, LB; Lecureur, V; Schuetz, EG; Schuetz, JD; Sun, D1
Bates, S; Litman, T; Nagy, Z; Ozvegy, C; Sarkadi, B; Szakács, G; Váradi, A1
Balakrishnan, L; Janvilisri, T; Reuter, G; Shahi, S; van Veen, HW; Venter, H1
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ1
Bauer, KS; Doyle, LA; Fang, HB; Hassel, B; Nakanishi, T; Pumplin, DW; Ross, DD; Wei, Y; Wu, S1
Borchardt, RT; Ouyang, H; Tang, F; Yang, JZ1
Globisch, C; Kassack, MU; Klinkhammer, W; Müller, H; Pajeva, IK; Wiese, M1
Ghosh, I; Manoharlal, R; Prakash, O; Prasad, R; Puri, N; Sharma, M1

Reviews

1 review(s) available for rhodamine 123 and daunorubicin

ArticleYear
Multidrug resistance through the spectacle of P-glycoprotein.
    Current cancer drug targets, 2009, Volume: 9, Issue:3

    Topics: Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cloning, Molecular; Daunorubicin; Drug Resistance, Multiple; Genes, MDR; Humans; Kinetics; Models, Genetic; Neoplasms; Rhodamine 123

2009

Trials

1 trial(s) available for rhodamine 123 and daunorubicin

ArticleYear
Cyclosporine diminishes multidrug resistance in K562/ADM cells and improves complete remission in patients with acute myeloid leukemia.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2009, Volume: 63, Issue:8

    Topics: Adult; Antibiotics, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Cyclosporine; Cytarabine; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Fluorescent Dyes; Humans; Idarubicin; Inhibitory Concentration 50; K562 Cells; Leukemia, Myeloid, Acute; Male; Rhodamine 123; Time Factors; Treatment Outcome; Verapamil

2009

Other Studies

79 other study(ies) available for rhodamine 123 and daunorubicin

ArticleYear
The function of Gp170, the multidrug-resistance gene product, in the brush border of rat intestinal mucosa.
    Gastroenterology, 1992, Volume: 102, Issue:3

    Topics: Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Colchicine; Daunorubicin; Diltiazem; Dose-Response Relationship, Drug; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Ileum; In Vitro Techniques; Intestinal Mucosa; Jejunum; Male; Membrane Glycoproteins; Microvilli; Rats; Rats, Inbred Strains; Rhodamine 123; Rhodamines; Temperature; Verapamil

1992
Detection of activity of P-glycoprotein in human tumour samples using rhodamine 123.
    British journal of haematology, 1992, Volume: 82, Issue:1

    Topics: Acute Disease; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Daunorubicin; Drug Resistance; Humans; Leukemia, Myeloid; Membrane Glycoproteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1992
Laser scanning and confocal microscopy of daunorubicin, doxorubicin, and rhodamine 123 in multidrug-resistant cells.
    Experimental cell research, 1991, Volume: 196, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Daunorubicin; Doxorubicin; Drug Resistance; Humans; KB Cells; Lasers; Membrane Glycoproteins; Mice; Microscopy, Fluorescence; Rhodamine 123; Rhodamines; Transfection; Verapamil

1991
Rapid functional assay for the detection of multidrug-resistant cells using the fluorescent dye rhodamine 123.
    Blood, 1991, Sep-01, Volume: 78, Issue:5

    Topics: Cell Line; Daunorubicin; Drug Resistance; Fluorescent Dyes; Rhodamine 123; Rhodamines

1991
Exploring multidrug resistance using rhodamine 123.
    Cancer communications, 1989, Volume: 1, Issue:3

    Topics: Animals; Daunorubicin; Doxorubicin; Drug Resistance; Fluorescent Dyes; Kinetics; Leukemia P388; Leukemia, Experimental; Mice; Microscopy, Fluorescence; Rhodamine 123; Rhodamines; Spectrometry, Fluorescence; Tumor Cells, Cultured

1989
Cross-resistance to rhodamine 123 in Adriamycin- and daunorubicin-resistant Friend leukemia cell variants.
    Cancer research, 1984, Volume: 44, Issue:12 Pt 1

    Topics: Animals; Biological Transport; Cell Line; Daunorubicin; Doxorubicin; Drug Resistance; Kinetics; Leukemia, Experimental; Mice; Rhodamine 123; Rhodamines; Xanthenes

1984
Effect of Calphostin C (PKC inhibitor) on daunorubicin resistance in P388/ADR and HL60/AR cells: reversal of drug resistance possibly via P-glycoprotein.
    Cancer letters, 1994, Jan-30, Volume: 76, Issue:2-3

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Leukemia P388; Leukemia, Experimental; Leukemia, Myeloid; Membrane Glycoproteins; Mice; Naphthalenes; Polycyclic Compounds; Protein Kinase C; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1994
Probing the interaction of the multidrug-resistance phenotype with the polypeptide ionophore gramicidin D via functional channel formation.
    European journal of biochemistry, 1994, Jun-15, Volume: 222, Issue:3

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cell Line; CHO Cells; Cricetinae; Cricetulus; Daunorubicin; Drug Resistance; Flow Cytometry; Gene Amplification; Gramicidin; Ion Channels; Ionophores; Membrane Glycoproteins; Phenotype; Rhodamine 123; Rhodamines; Rubidium; Sodium-Potassium-Exchanging ATPase

1994
Regulation by glutathione of drug transport in multidrug-resistant human lung tumour cell lines overexpressing multidrug resistance-associated protein.
    British journal of cancer, 1995, Volume: 72, Issue:1

    Topics: Biological Transport; Buthionine Sulfoximine; Daunorubicin; Drug Resistance, Multiple; Glutathione; Humans; Lung Neoplasms; Methionine Sulfoximine; Rhodamine 123; Rhodamines; RNA, Messenger; Tumor Cells, Cultured

1995
Evaluation of multidrug resistant phenotype by flow cytometry with monoclonal antibodies and functional tests.
    Bulletin du cancer, 1995, Volume: 82, Issue:3

    Topics: Antibodies, Monoclonal; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Antibody Technique; Fluorescent Dyes; Humans; Leukemia, Erythroblastic, Acute; Lymphoma, Non-Hodgkin; Phenotype; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Rhodamine 123; Rhodamines

1995
Functional detection of MDR1/P170 and MRP/P190-mediated multidrug resistance in tumour cells by flow cytometry.
    British journal of cancer, 1995, Volume: 72, Issue:3

    Topics: Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluoresceins; Fluorescent Dyes; Humans; KB Cells; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Sensitivity and Specificity

1995
The effect of ion channel blockers, immunosuppressive agents, and other drugs on the activity of the multi-drug transporter.
    International journal of cancer, 1993, May-28, Volume: 54, Issue:3

    Topics: Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzofurans; Biological Transport, Active; Carrier Proteins; Cell Membrane; Daunorubicin; Drug Resistance; Ethers, Cyclic; Flow Cytometry; Fluorescent Dyes; Hydrogen-Ion Concentration; Immunosuppressive Agents; Intracellular Fluid; Ion Channels; Leukemia L5178; Lymphoma, T-Cell; Membrane Glycoproteins; Membrane Potentials; Mice; Molecular Sequence Data; Potassium; Potassium Channels; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1993
Lack of correlation between expression and function of P-glycoprotein in acute myeloid leukemia cell lines.
    Leukemia, 1995, Volume: 9, Issue:5

    Topics: Acute Disease; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Differentiation; Coloring Agents; Daunorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Flow Cytometry; Gene Expression; Humans; Immunohistochemistry; Leukemia, Myeloid; Phenotype; Polymerase Chain Reaction; Rhodamine 123; Rhodamines; Transcription, Genetic; Tumor Cells, Cultured; Vincristine

1995
Selective photodynamic inactivation of a multidrug transporter by a cationic photosensitising agent.
    British journal of cancer, 1995, Volume: 71, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cycloleucine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Leukemia P388; Mice; Microscopy, Fluorescence; Neoplasm Proteins; Oxygen; Photochemotherapy; Radiation-Sensitizing Agents; Rhodamine 123; Rhodamines; Singlet Oxygen; Spectrometry, Fluorescence; Tumor Cells, Cultured

1995
Low frequency of activity of P-glycoprotein (P-170) in acute lymphoblastic leukemia compared to acute myeloid leukemia.
    Leukemia, 1995, Volume: 9, Issue:2

    Topics: Acute Disease; Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow; Bone Marrow Transplantation; Child; Child, Preschool; Cytarabine; Daunorubicin; Drug Resistance, Multiple; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Neoplasm Proteins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prognosis; Remission Induction; Rhodamine 123; Rhodamines; Survival Analysis

1995
Rapid stimulation of rhodamine 123 efflux from multidrug-resistant KB cells by progesterone.
    Biochemical pharmacology, 1993, Nov-02, Volume: 46, Issue:9

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carrier Proteins; Daunorubicin; Drug Resistance; Exocytosis; Fluorescent Dyes; Humans; Membrane Glycoproteins; Membrane Potentials; Mice; Progesterone; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Up-Regulation; Verapamil

1993
Effect of the protein kinase C inhibitor staurosporine on chemosensitivity to daunorubicin of normal and leukemic fresh myeloid cells.
    Blood, 1994, Jul-01, Volume: 84, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Alkaloids; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Child; Daunorubicin; Hematopoietic Stem Cells; Humans; Leukemia, Myeloid, Acute; Membrane Glycoproteins; Middle Aged; Neoplastic Stem Cells; Protein Kinase C; Rhodamine 123; Rhodamines; Staurosporine; Tumor Cells, Cultured

1994
Bile acid inhibition of P-glycoprotein-mediated transport in multidrug-resistant cells and rat liver canalicular membrane vesicles.
    Hepatology (Baltimore, Md.), 1994, Volume: 20, Issue:1 Pt 1

    Topics: Animals; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bile Acids and Salts; Bile Canaliculi; Biological Transport; Carcinoma, Hepatocellular; Carrier Proteins; Cell Membrane; Daunorubicin; Depression, Chemical; Doxorubicin; Drug Resistance; Liver Neoplasms; Male; Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1994
Chemomodulation of drugs involved in multidrug resistance in chronic lymphatic leukemia of the B-cell type.
    Cancer chemotherapy and pharmacology, 1994, Volume: 34, Issue:4

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Daunorubicin; Drug Resistance; Flow Cytometry; Humans; Immunophenotyping; In Vitro Techniques; Leukemia, Lymphocytic, Chronic, B-Cell; Membrane Glycoproteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Verapamil; Vincristine

1994
Reversal of multidrug resistance by valinomycin is overcome by CCCP.
    Biochemical and biophysical research communications, 1996, Feb-15, Volume: 219, Issue:2

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carbonyl Cyanide m-Chlorophenyl Hydrazone; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Coloring Agents; Daunorubicin; Drug Resistance, Multiple; Humans; Ionophores; KB Cells; Kinetics; Potassium; Rhodamine 123; Rhodamines; Valinomycin; Vinblastine

1996
Modulation of multidrug resistance by BIBW22BS in blasts of de novo or relapsed or persistent acute myeloid leukemia ex vivo.
    Journal of cancer research and clinical oncology, 1996, Volume: 122, Issue:5

    Topics: Antigens, CD34; Daunorubicin; Drug Resistance, Multiple; Humans; Idarubicin; Leukemia, Myeloid, Acute; Morpholines; Rhodamine 123; Rhodamines; Triamterene

1996
Quality control of multidrug resistance assays in adult acute leukemia: correlation between assays for P-glycoprotein expression and activity.
    Blood, 1996, Jun-01, Volume: 87, Issue:11

    Topics: Acute Disease; Adult; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cryopreservation; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Feasibility Studies; Fluorescent Dyes; Humans; Leukemia; Leukemia, Myeloid; Neoplasm Proteins; Neoplastic Stem Cells; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Reproducibility of Results; Rhodamine 123; Rhodamines; Sensitivity and Specificity; Verapamil; Vincristine

1996
Modulation of multidrug resistance with antisense oligodeoxynucleotide to mdr1 mRNA.
    Annals of surgical oncology, 1996, Volume: 3, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Codon; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Humans; Leukemia, Erythroblastic, Acute; Oligonucleotides, Antisense; Rhodamine 123; Rhodamines; RNA, Messenger; Thymidine; Tumor Cells, Cultured

1996
Polyaromatic alkaloids from marine invertebrates as cytotoxic compounds and inhibitors of multidrug resistance caused by P-glycoprotein.
    British journal of cancer, 1996, Volume: 74, Issue:5

    Topics: Adenocarcinoma; Alkaloids; Animals; Antimetabolites, Antineoplastic; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Survival; Colonic Neoplasms; Cricetinae; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Leukemia P388; Lung Neoplasms; Mice; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Verapamil; Vinblastine

1996
Functional study of multidrug resistance with fluorescent dyes. Limits of the assay for low levels of resistance and application in clinical samples.
    Cancer letters, 1996, Aug-23, Volume: 106, Issue:1

    Topics: Animals; Anthracyclines; Benzimidazoles; Cell Survival; Clone Cells; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Leukemia L1210; Mice; Phenotype; Quantum Theory; Reproducibility of Results; Rhodamine 123; Rhodamines; Sensitivity and Specificity; Tumor Cells, Cultured; Vinblastine

1996
Comparison of drug accumulation in P-glycoprotein-expressing and MRP-expressing human leukaemia cells.
    Leukemia research, 1996, Volume: 20, Issue:8

    Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Buthionine Sulfoximine; Calcium Channel Blockers; Cyclosporins; Daunorubicin; Humans; Idarubicin; Leukemia, T-Cell; Multidrug Resistance-Associated Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Verapamil

1996
Flow cytometry evaluation of the multidrug-resistant phenotype with functional tests involving uptake of daunorubicin, Hoechst 33342, or rhodamine 123: a comparative study.
    Cancer detection and prevention, 1995, Volume: 19, Issue:6

    Topics: Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Death; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Hot Temperature; Humans; Phenotype; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1995
Anticancer drugs, ionophoric peptides, and steroids as substrates of the yeast multidrug transporter Pdr5p.
    The Journal of biological chemistry, 1996, Dec-06, Volume: 271, Issue:49

    Topics: Animals; Antineoplastic Agents; ATP-Binding Cassette Transporters; Daunorubicin; Desoxycorticosterone; Doxorubicin; Fungal Proteins; Ionophores; Kinetics; Membrane Proteins; Phenotype; Progesterone; Rhodamine 123; Rhodamines; Saccharomyces cerevisiae Proteins

1996
Structure-activity relationship studies on benzofuran analogs of propafenone-type modulators of tumor cell multidrug resistance.
    Journal of medicinal chemistry, 1996, Nov-22, Volume: 39, Issue:24

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzofurans; Calorimetry, Differential Scanning; Cells, Cultured; Daunorubicin; Drug Resistance, Multiple; Ethanolamines; Liposomes; Magnetic Resonance Spectroscopy; Membranes, Artificial; Propafenone; Regression Analysis; Rhodamine 123; Rhodamines; Structure-Activity Relationship

1996
Inhibition of drug transport by genistein in multidrug-resistant cells expressing P-glycoprotein.
    Biochemical pharmacology, 1997, Jan-10, Volume: 53, Issue:1

    Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Biological Transport; Daunorubicin; Drug Resistance, Multiple; Enzyme Inhibitors; Genistein; Humans; Isoflavones; Mice; Multidrug Resistance-Associated Proteins; Protein-Tyrosine Kinases; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1997
Acceleration of MRP-associated efflux of rhodamine 123 by genistein and related compounds.
    British journal of cancer, 1996, Volume: 74, Issue:12

    Topics: Antimetabolites, Antineoplastic; Daunorubicin; Drug Resistance, Multiple; Genistein; Humans; Isoflavones; Monosaccharide Transport Proteins; Quercetin; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1996
P-glycoprotein (PGP) and lung resistance-related protein (LRP) expression and function in leukaemic blast cells.
    British journal of haematology, 1997, Volume: 96, Issue:2

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Leukemia; Lymphocytes; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Rhodamine 123; Rhodamines; Vault Ribonucleoprotein Particles

1997
Modulation of P-glycoprotein mediated drug accumulation in multidrug resistant CCRF VCR-1000 cells by chemosensitisers.
    European journal of cancer (Oxford, England : 1990), 1996, Volume: 32A, Issue:5

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Rhodamine 123; Rhodamines; Tumor Cells, Cultured; Vincristine

1996
Expression of c-Kit and functional drug efflux are correlated in de novo acute myeloid leukaemia.
    Leukemia, 1997, Volume: 11, Issue:11

    Topics: Acute Disease; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Fluorescent Antibody Technique, Indirect; Humans; Immunosuppressive Agents; Leukemia, Myeloid; Phenotype; Proto-Oncogene Proteins c-kit; Rhodamine 123; Rhodamines; Tumor Cells, Cultured

1997
Positively cooperative sites for drug transport by P-glycoprotein with distinct drug specificities.
    European journal of biochemistry, 1997, Nov-15, Volume: 250, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Daunorubicin; Doxorubicin; Etoposide; Fluorescence; Fluorescent Dyes; Kinetics; Liposomes; Protein Binding; Quercetin; Rhodamine 123; Rhodamines; Vinblastine

1997
Estimation of drug resistance by flow cytometry.
    Methods in molecular biology (Clifton, N.J.), 1998, Volume: 91

    Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Flow Cytometry; Genistein; Leukemia L5178; Mice; Probenecid; Recombinant Proteins; Rhodamine 123; Rhodamines; Transfection; Tumor Cells, Cultured; Verapamil

1998
Linear and cyclic peptides as substrates and modulators of P-glycoprotein: peptide binding and effects on drug transport and accumulation.
    The Biochemical journal, 1998, Aug-01, Volume: 333 ( Pt 3)

    Topics: Adenosine Triphosphatases; Animals; Antibiotics, Antineoplastic; Antimetabolites, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Membrane; CHO Cells; Cricetinae; Daunorubicin; Drug Resistance, Multiple; Ionophores; Kinetics; Oligopeptides; Peptides, Cyclic; Protein Binding; Rhodamine 123; Rhodamines; Substrate Specificity

1998
Decreased activity of the multidrug resistance P-glycoprotein in acquired aplastic anaemia: possible pathophysiologic implications.
    British journal of haematology, 1998, Volume: 102, Issue:5

    Topics: Adolescent; Adult; Anemia, Aplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Child; Child, Preschool; Daunorubicin; Drug Resistance, Multiple; Female; Fluorescent Dyes; Humans; Male; Rhodamine 123

1998
Substituted 4-acylpyrazoles and 4-acylpyrazolones: synthesis and multidrug resistance-modulating activity.
    Journal of medicinal chemistry, 1998, Oct-08, Volume: 41, Issue:21

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Isomerism; Magnetic Resonance Spectroscopy; Mice; Pyrazoles; Regression Analysis; Rhodamine 123; Structure-Activity Relationship; Tumor Cells, Cultured

1998
Anti-psychotic drugs reverse multidrug resistance of tumor cell lines and human AML cells ex-vivo.
    Cancer letters, 1999, May-03, Volume: 139, Issue:1

    Topics: Antipsychotic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Daunorubicin; Drug Interactions; Drug Resistance, Multiple; Enzyme Inhibitors; Humans; Leukemia, Myeloid; Rhodamine 123; Tumor Cells, Cultured

1999
Interaction of the P-glycoprotein multidrug transporter (MDR1) with high affinity peptide chemosensitizers in isolated membranes, reconstituted systems, and intact cells.
    Biochemical pharmacology, 1999, Aug-15, Volume: 58, Issue:4

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cell Membrane; CHO Cells; Colchicine; Cricetinae; Daunorubicin; Dihydropyridines; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluorescent Dyes; Humans; Oligopeptides; Peptides; Photoaffinity Labels; Rhodamine 123; Tumor Cells, Cultured

1999
Cholesterol interaction with the daunorubicin binding site of P-glycoprotein.
    Biochemical and biophysical research communications, 2000, Oct-05, Volume: 276, Issue:3

    Topics: Adenosine Triphosphate; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Biological Transport, Active; Cell Line; Cell Survival; Cholesterol; Daunorubicin; Flow Cytometry; Fluorescence; Humans; Hydrolysis; Inhibitory Concentration 50; Kinetics; Microsomes; Protein Binding; Rhodamine 123

2000
Monitoring of cellular resistance to cancer chemotherapy: drug retention and efflux.
    Methods in cell biology, 2001, Volume: 64

    Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Calcium Channel Blockers; Cell Membrane Permeability; Chlorpromazine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Dyes; Humans; Mice; Rhodamine 123; Staining and Labeling; Tumor Cells, Cultured; Verapamil

2001
Modulation by LY335979 of P-glycoprotein function in multidrug-resistant cell lines and human natural killer cells.
    Biochemical pharmacology, 2001, Jun-01, Volume: 61, Issue:11

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Daunorubicin; Dibenzocycloheptenes; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance, Multiple; Fluorescent Dyes; HL-60 Cells; Humans; Killer Cells, Natural; Quinolines; Rhodamine 123

2001
Effect of P-glycoprotein modulators on the human extraneuronal monoamine transporter.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: 1-Methyl-4-phenylpyridinium; Arginine; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Carrier Proteins; Cations; Cell Line; Cyclosporine; Daunorubicin; Dose-Response Relationship, Drug; Histidine; Humans; Organic Cation Transport Proteins; Rhodamine 123; Time Factors; Tritium; Tyramine; Verapamil; Vinblastine

2001
The farnesyl protein transferase inhibitor SCH66336 is a potent inhibitor of MDR1 product P-glycoprotein.
    Cancer research, 2001, Oct-15, Volume: 61, Issue:20

    Topics: 3T3 Cells; Adenosine Triphosphate; Alkyl and Aryl Transferases; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport, Active; Cell Line; CHO Cells; Cricetinae; Daunorubicin; Drug Synergism; Enzyme Inhibitors; Farnesyltranstransferase; Genes, MDR; Humans; Hydrolysis; Mice; Paclitaxel; Piperidines; Pyridines; Rhodamine 123; Tamoxifen; Vinblastine

2001
Evaluation of the clinical relevance of the expression and function of P-glycoprotein, multidrug resistance protein and lung resistance protein in patients with primary acute myelogenous leukemia.
    Leukemia research, 2002, Volume: 26, Issue:2

    Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Antineoplastic Combined Chemotherapy Protocols; ATP Binding Cassette Transporter, Subfamily B, Member 1; Bone Marrow Transplantation; Calcium Channel Blockers; Carbocyanines; Combined Modality Therapy; Cytarabine; Daunorubicin; Disease-Free Survival; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Enzyme Inhibitors; Female; Fluoresceins; Fluorescent Dyes; Genistein; Humans; Idarubicin; Immunophenotyping; Leukemia, Myeloid; Male; Middle Aged; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Probenecid; Prognosis; Prospective Studies; Rhodamine 123; Survival Analysis; Tumor Cells, Cultured; Vault Ribonucleoprotein Particles; Verapamil

2002
Overexpression of protein disulfide isomerase-like protein in a mouse leukemia L1210 cell line selected for resistance to 4-methyl-5-amino-1-formylisoquinoline thiosemicarbazone, a ribonucleotide reductase inhibitor.
    Advances in enzyme regulation, 2002, Volume: 42

    Topics: Amino Acid Sequence; Animals; Antibiotics, Antineoplastic; Blotting, Northern; Blotting, Southern; Blotting, Western; Cell Line; Daunorubicin; DNA, Complementary; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Fluorescent Dyes; Isoquinolines; Mice; Molecular Sequence Data; Protein Biosynthesis; Protein Disulfide-Isomerases; Proteins; Rhodamine 123; Ribonucleotide Reductases; RNA, Messenger; Sulfhydryl Compounds

2002
Modulation of P-glycoprotein-mediated multidrug resistance by flavonoid derivatives and analogues.
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Antineoplastic Agents; Apoptosis; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Chromones; Daunorubicin; Drug Resistance, Multiple; Drug Synergism; Flavonoids; Fluorescent Dyes; Humans; Necrosis; Piperazines; Quinolinium Compounds; Rhodamine 123; Thiazoles; Tumor Cells, Cultured

2003
Kinetic analysis of rhodamines efflux mediated by the multidrug resistance protein (MRP1).
    Biophysical journal, 2003, Volume: 85, Issue:3

    Topics: Biophysical Phenomena; Biophysics; Cell Line, Tumor; Chlorine; Daunorubicin; Dose-Response Relationship, Drug; Fluorescent Dyes; Glutathione; Humans; Kinetics; Membrane Potentials; Models, Chemical; Models, Theoretical; Multidrug Resistance-Associated Proteins; Phenotype; Potassium; Rhodamine 123; Rhodamines; Time Factors

2003
[Reversal of multidrug resistance gene MDR1 and MRP of drug-resistant human hepatocellular carcinoma cells SMMC-7721/ADM with antisense phosphorothioate oligonucleotides].
    Zhonghua gan zang bing za zhi = Zhonghua ganzangbing zazhi = Chinese journal of hepatology, 2004, Volume: 12, Issue:2

    Topics: Carcinoma, Hepatocellular; Cell Line, Tumor; Daunorubicin; Doxorubicin; Drug Resistance, Neoplasm; Genes, MDR; Humans; Liver Neoplasms; Multidrug Resistance-Associated Proteins; Oligonucleotides, Antisense; Rhodamine 123

2004
Effects of tributyltin on barrier functions in human intestinal Caco-2 cells.
    Biochemical and biophysical research communications, 2004, Mar-19, Volume: 315, Issue:4

    Topics: Actin Cytoskeleton; Alkaline Phosphatase; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caco-2 Cells; CD13 Antigens; Cell Membrane Permeability; Daunorubicin; Electric Impedance; Epithelium; Humans; Intestinal Absorption; Intestinal Mucosa; Isoquinolines; Rhodamine 123; RNA, Messenger; Tight Junctions; Time Factors; Trialkyltin Compounds

2004
Inhibitory effect of a bitter melon extract on the P-glycoprotein activity in intestinal Caco-2 cells.
    British journal of pharmacology, 2004, Volume: 143, Issue:3

    Topics: Adenocarcinoma; Amino Acids; ATP Binding Cassette Transporter, Subfamily B; Biological Transport; Caco-2 Cells; Chromatography, High Pressure Liquid; Colonic Neoplasms; Daunorubicin; Dose-Response Relationship, Drug; Fruit; Glycerides; Hot Temperature; Humans; L-Lactate Dehydrogenase; Mass Spectrometry; Methanol; Momordica charantia; Plant Extracts; Pronase; Rhodamine 123; Vegetables

2004
Effects of miltefosine on membrane permeability and accumulation of [99mTc]-hexakis-2-methoxyisobutyl isonitrile, 2-[18F]fluoro-2-deoxy-D-glucose, daunorubucin and rhodamine123 in multidrug-resistant and sensitive cells.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2005, Volume: 24, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Membrane Permeability; Daunorubicin; Drug Resistance, Multiple; Fluorodeoxyglucose F18; Humans; Membrane Fluidity; Mice; NIH 3T3 Cells; Phosphorylcholine; Rhodamine 123; Technetium Tc 99m Sestamibi; Verapamil

2005
Flow cytometric monitoring of fluorescent drug retention and efflux.
    Methods in molecular medicine, 2005, Volume: 111

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Benzimidazoles; Cell Line, Tumor; Daunorubicin; Drug Monitoring; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Flow Cytometry; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; Phenotype; Rhodamine 123

2005
Flow cytometric measurement of functional and phenotypic P-glycoprotein.
    Methods in molecular medicine, 2005, Volume: 111

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Clinical Trials as Topic; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Humans; Leukemia, Myeloid, Acute; Leukocyte Common Antigens; Microscopy, Fluorescence; Phenotype; Rhodamine 123

2005
An MDR-EGFP gene fusion allows for direct cellular localization, function and stability assessment of P-glycoprotein.
    Current drug delivery, 2004, Volume: 1, Issue:1

    Topics: Amino Acid Sequence; Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Line; Cell Survival; Daunorubicin; DNA Primers; Dogs; Doxorubicin; Drug Resistance, Multiple; Flow Cytometry; Fluorescence; Fluorescent Antibody Technique; Gene Fusion; Genes, MDR; Genetic Vectors; Green Fluorescent Proteins; Humans; Microscopy, Confocal; Molecular Sequence Data; Oligonucleotides; Rhodamine 123; Subcellular Fractions; Transfection

2004
Reversal of MDR1 gene-dependent multidrug resistance using low concentration of endonuclease-prepared small interference RNA.
    European journal of pharmacology, 2006, Apr-24, Volume: 536, Issue:1-2

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Survival; CHO Cells; Cricetinae; Cricetulus; Daunorubicin; Dose-Response Relationship, Drug; Down-Regulation; Drug Resistance, Neoplasm; Green Fluorescent Proteins; Humans; Plasmids; Recombinant Fusion Proteins; Rhodamine 123; Ribonuclease III; RNA Interference; RNA, Messenger; RNA, Small Interfering; Transfection

2006
Effects of Kaempferia parviflora extracts and their flavone constituents on P-glycoprotein function.
    Journal of pharmaceutical sciences, 2007, Volume: 96, Issue:1

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Ethanol; Flavones; Flavonoids; Fluorescent Dyes; Humans; LLC-PK1 Cells; Plant Extracts; Rhizome; Rhodamine 123; Solvents; Swine; Time Factors; Transfection; Water; Zingiberaceae

2007
Improvement of intestinal absorption of P-glycoprotein substrate by D-tartaric acid.
    Drug metabolism and pharmacokinetics, 2006, Volume: 21, Issue:5

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blotting, Western; Cardiovascular Agents; Colon; Daunorubicin; Diffusion Chambers, Culture; Fluorescent Dyes; Ileum; Injections, Intravenous; Intestinal Absorption; Jejunum; Male; Rats; Rats, Wistar; Rhodamine 123; Tartrates; Verapamil

2006
Modification of multidrug resistance of tumor cells by ionizing radiation.
    Cancer chemotherapy and pharmacology, 2008, Volume: 61, Issue:1

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; Cell Count; Cell Line, Tumor; Combined Modality Therapy; Cyclosporine; Daunorubicin; Dose-Response Relationship, Radiation; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Laryngeal Neoplasms; Paclitaxel; Radiation, Ionizing; Reactive Oxygen Species; Rhodamine 123; Time Factors; Vincristine

2008
Inhibition of P-glycoprotein function by tannic acid and pentagalloylglucose.
    The Journal of pharmacy and pharmacology, 2007, Volume: 59, Issue:7

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Daunorubicin; Humans; Hydrolyzable Tannins; KB Cells; Rhodamine 123; Tannins

2007
Imatinib is a substrate for various multidrug resistance proteins.
    Neoplasma, 2009, Volume: 56, Issue:3

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzamides; Daunorubicin; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; K562 Cells; Multidrug Resistance-Associated Proteins; Piperazines; Pyrimidines; Rhodamine 123; Vault Ribonucleoprotein Particles

2009
Activators of P-glycoprotein: Structure-activity relationships and investigation of their mode of action.
    ChemMedChem, 2009, Volume: 4, Issue:11

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Benzothiazoles; Cell Line, Tumor; Daunorubicin; Drug Resistance, Neoplasm; Humans; Imidazoles; Rhodamine 123; Structure-Activity Relationship; Thiazoles

2009
Macelignan: a new modulator of P-glycoprotein in multidrug-resistant cancer cells.
    Nutrition and cancer, 2009, Volume: 61, Issue:4

    Topics: Adenocarcinoma; Analysis of Variance; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B; Biological Transport, Active; Breast Neoplasms; Cell Line, Tumor; Cell Survival; Daunorubicin; Dose-Response Relationship, Drug; Drug Design; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Drug Synergism; Female; Fluorescent Dyes; Growth Inhibitors; Humans; Lignans; Phytoestrogens; Phytotherapy; Rhodamine 123; Vinblastine

2009
Iodination increases the activity of verapamil derivatives in reversing PGP multidrug resistance.
    Anticancer research, 2010, Volume: 30, Issue:7

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Calcium Channels, L-Type; Cell Cycle; Cyclosporine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Humans; K562 Cells; Male; Myocytes, Cardiac; Rats; Rats, Wistar; Rhodamine 123; Verapamil

2010
Pgp inhibition by UIC2 antibody can be followed in vitro by using tumor-diagnostic radiotracers, 99mTc-MIBI and 18FDG.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2010, Dec-23, Volume: 41, Issue:5

    Topics: Antibodies, Monoclonal; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Female; Fluorodeoxyglucose F18; Glucose; Humans; Ovarian Neoplasms; Paclitaxel; Protein Binding; Rhodamine 123; Technetium Tc 99m Sestamibi; Tumor Cells, Cultured

2010
Drug resistance is conferred on the model yeast Saccharomyces cerevisiae by expression of full-length melanoma-associated human ATP-binding cassette transporter ABCB5.
    Molecular pharmaceutics, 2014, Oct-06, Volume: 11, Issue:10

    Topics: ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Clorgyline; Daunorubicin; Humans; Melanoma; Rhodamine 123; Rhodamines; Saccharomyces cerevisiae; Tacrolimus

2014
6,7-Dimethoxy-2-{2-[4-(1H-1,2,3-triazol-1-yl)phenyl]ethyl}-1,2,3,4-tetrahydroisoquinolines as superior reversal agents for P-glycoprotein-mediated multidrug resistance.
    ChemMedChem, 2015, Volume: 10, Issue:2

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Benzamides; Cell Survival; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Daunorubicin; Drug Resistance, Neoplasm; Humans; K562 Cells; Paclitaxel; Protein Binding; Rhodamine 123; Structure-Activity Relationship; Tetrahydroisoquinolines; Triazoles; Vincristine

2015
[The study of mechanisms of accumulation of daunorubicin and rodamin-123 in cells of human venous blood using cytometry technique].
    Klinicheskaia laboratornaia diagnostika, 2015, Volume: 60, Issue:2

    Topics: Blood Platelets; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Healthy Volunteers; Humans; Leukocytes; Neoplasms; Rhodamine 123

2015
Glucosamine Reverses P-Glycoprotein-Mediated Multidrug Resistance in the Daunorubicin-Resistant Human Gastric Cancer Cells.
    Nutrition and cancer, 2020, Volume: 72, Issue:3

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Proliferation; Cell Survival; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Glucosamine; Humans; Reverse Transcriptase Polymerase Chain Reaction; Rhodamine 123; RNA, Neoplasm; Stomach Neoplasms

2020
Cloning and expression of murine sister of P-glycoprotein reveals a more discriminating transporter than MDR1/P-glycoprotein.
    Molecular pharmacology, 2000, Volume: 57, Issue:1

    Topics: Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Cells, Cultured; Cloning, Molecular; DNA, Complementary; Humans; Karyotyping; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Sequence Homology, Amino Acid

2000
Functional characterization of the human multidrug transporter, ABCG2, expressed in insect cells.
    Biochemical and biophysical research communications, 2001, Jul-06, Volume: 285, Issue:1

    Topics: Adenosine Triphosphatases; Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Breast Neoplasms; Cell Membrane; Cloning, Molecular; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Neoplasm Proteins; Recombinant Proteins; Spodoptera; Tumor Cells, Cultured

2001
Sterol transport by the human breast cancer resistance protein (ABCG2) expressed in Lactococcus lactis.
    The Journal of biological chemistry, 2003, Jun-06, Volume: 278, Issue:23

    Topics: Antineoplastic Agents, Hormonal; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Cholesterol; Estradiol; Gene Expression; Humans; Lactococcus lactis; Neoplasm Proteins; Progesterone; Sterols; Tamoxifen; Testosterone; Tritium

2003
Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites.
    Pharmaceutical research, 2003, Volume: 20, Issue:4

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Binding Sites; Biological Transport, Active; Biomarkers; Cells, Cultured; Drug Interactions; Fluorescent Dyes; Humans

2003
Functional characterization of human breast cancer resistance protein (BCRP, ABCG2) expressed in the oocytes of Xenopus laevis.
    Molecular pharmacology, 2003, Volume: 64, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Drug Resistance, Neoplasm; Female; Gene Expression Regulation, Neoplastic; Humans; Neoplasm Proteins; Oocytes; Xenopus laevis

2003
Bidirectional transport of rhodamine 123 and Hoechst 33342, fluorescence probes of the binding sites on P-glycoprotein, across MDCK-MDR1 cell monolayers.
    Journal of pharmaceutical sciences, 2004, Volume: 93, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Binding Sites; Biological Transport; Cell Line; Cell Membrane; Dogs; Fluorescent Dyes; Humans; Rhodamine 123

2004
New functional assay of P-glycoprotein activity using Hoechst 33342.
    Bioorganic & medicinal chemistry, 2007, Dec-01, Volume: 15, Issue:23

    Topics: Adenosine Triphosphatases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Cell Line, Tumor; Cell Proliferation; Dose-Response Relationship, Drug; Drug Resistance, Neoplasm; Fluoresceins; Humans; Microscopy, Fluorescence; Molecular Structure; Principal Component Analysis; Time Factors

2007
Analysis of physico-chemical properties of substrates of ABC and MFS multidrug transporters of pathogenic Candida albicans.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Candida albicans; Membrane Transport Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Substrate Specificity

2010