Page last updated: 2024-09-03

rg 12525 and leukotriene d4

rg 12525 has been researched along with leukotriene d4 in 3 studies

Compound Research Comparison

Studies
(rg 12525)
Trials
(rg 12525)
Recent Studies (post-2010)
(rg 12525)
Studies
(leukotriene d4)
Trials
(leukotriene d4)
Recent Studies (post-2010) (leukotriene d4)
14306974297

Protein Interaction Comparison

ProteinTaxonomyrg 12525 (IC50)leukotriene d4 (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.0007
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.0007
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.0007
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.0007
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.0007
Canalicular multispecific organic anion transporter 1Rattus norvegicus (Norway rat)5.48
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.0007
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.0007
Cysteinyl leukotriene receptor 1Homo sapiens (human)0.0039

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Feiss, G; Nelson, HS; Paull, BR; Smith, JA; Tobey, RE; Welch, MJ1
Beys, E; Bonnefoi, MS; Jayyosi, Z; Kelley, MF; Kornbrust, DJ; Langloss, JM; Sanders, JE; Wells, RE1
Carlton, RA; Difeo, TJ; Powner, TH; Santos, I; Thompson, MD1

Trials

1 trial(s) available for rg 12525 and leukotriene d4

ArticleYear
Effect of RG 12525, a new leukotriene antagonist, on pulmonary function of asthmatic adults.
    Annals of allergy, 1994, Volume: 72, Issue:4

    Topics: Adolescent; Adult; Asthma; Double-Blind Method; Female; Humans; Leukotriene D4; Lung; Male; Patient Dropouts; Placebos; Quinolines; Respiratory Function Tests; Tetrazoles

1994

Other Studies

2 other study(ies) available for rg 12525 and leukotriene d4

ArticleYear
Subchronic toxicity studies with the leukotriene D4 antagonist RG 12525.
    Fundamental and applied toxicology : official journal of the Society of Toxicology, 1995, Volume: 28, Issue:1

    Topics: Animals; Corpus Luteum; Eating; Erythrocyte Count; Estrus; Female; Hematocrit; Kidney Diseases; Leukotriene D4; Liver; Macaca mulatta; Male; Mice; Mice, Inbred ICR; Microbodies; Organ Size; Quinolines; Rats; Rats, Sprague-Dawley; Sex Characteristics; Tetrazoles; Weight Gain

1995
Preparation and characterization of polymorphs for an LTD4 antagonist, RG 12525.
    Journal of pharmaceutical sciences, 1996, Volume: 85, Issue:5

    Topics: Calorimetry, Differential Scanning; Chemical Phenomena; Chemistry, Physical; Drug Stability; Heating; Leukotriene D4; Microscopy; Quinolines; Solubility; Tetrazoles; Thermodynamics; X-Ray Diffraction

1996