retrothiorphan has been researched along with enalaprilat anhydrous in 6 studies
Studies (retrothiorphan) | Trials (retrothiorphan) | Recent Studies (post-2010) (retrothiorphan) | Studies (enalaprilat anhydrous) | Trials (enalaprilat anhydrous) | Recent Studies (post-2010) (enalaprilat anhydrous) |
---|---|---|---|---|---|
18 | 0 | 2 | 846 | 109 | 76 |
Protein | Taxonomy | retrothiorphan (IC50) | enalaprilat anhydrous (IC50) |
---|---|---|---|
Angiotensin-converting enzyme | Mus musculus (house mouse) | 0.0115 | |
Angiotensin-converting enzyme | Homo sapiens (human) | 0.2405 | |
Angiotensin-converting enzyme | Oryctolagus cuniculus (rabbit) | 0.0054 | |
Type-2 angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.0012 | |
Angiotensin-converting enzyme | Rattus norvegicus (Norway rat) | 0.0036 | |
Angiotensin-converting enzyme 2 | Homo sapiens (human) | 0.0024 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Crippen, GM | 1 |
Fournié-Zaluski, MC; Lévy, B; Michel, JB; Pham, I; Poitevin, P; Roques, BP | 1 |
el Amrani, AI; Fournié-Zaluski, MC; Gonzalez, W; Laboulandine, I; Michel, JB; Pham, I; Philippe, M; Roques, BP | 1 |
Doucet, J; Fournie-Zaluski, MC; Gonzalez, W; Michel, JB; Pham, I; Roques, BP | 1 |
Adam, A; Blais, C; Drapeau, G; Gervais, N; Lamontagne, D; Raymond, P; Venneman, I | 1 |
Adam, A; Blais, C; Dumoulin, MJ; Lamontagne, D | 1 |
6 other study(ies) available for retrothiorphan and enalaprilat anhydrous
Article | Year |
---|---|
Validation of EGSITE2, a mixed integer program for deducing objective site models for experimental binding data.
Topics: Algorithms; Animals; Binding Sites; Computer Simulation; Folic Acid Antagonists; Models, Molecular; Peptidyl-Dipeptidase A; Protein Binding; Receptors, Cell Surface; Sex Hormone-Binding Globulin; Steroids; Testosterone; Tetrahydrofolate Dehydrogenase; Transcortin | 1997 |
Acute hemodynamic effects of combined inhibition of neutral endopeptidase and angiotensin converting enzyme in spontaneously hypertensive rats.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Drug Therapy, Combination; Enalaprilat; Heart Rate; Hemodynamics; Hypertension; Kinetics; Neprilysin; Rats; Rats, Inbred SHR; Thiorphan; Time Factors | 1995 |
Effects of converting enzyme inhibitor and neutral endopeptidase inhibitor on blood pressure and renal function in experimental hypertension.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Desoxycorticosterone; Diuresis; Enalaprilat; Hypertension, Renovascular; Kidney; Male; Natriuresis; Neprilysin; Protease Inhibitors; Rats; Rats, Inbred SHR; Rats, Wistar; Sodium Chloride; Sulfhydryl Compounds; Thiorphan | 1993 |
Effects of angiotensin-converting enzyme and neutral endopeptidase inhibitors: influence of bradykinin.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Cyclic GMP; Enalaprilat; Hypertension; Kidney; Male; Neprilysin; Rats; Rats, Wistar; Thiorphan | 1996 |
Contribution of angiotensin-converting enzyme to the cardiac metabolism of bradykinin: an interspecies study.
Topics: Amino Acid Sequence; Angiotensin-Converting Enzyme Inhibitors; Animals; Antibodies; Bradykinin; Cross Reactions; Dogs; Enalaprilat; Humans; Kinetics; Losartan; Myocardium; Peptidyl-Dipeptidase A; Protease Inhibitors; Rabbits; Rats; Species Specificity; Substrate Specificity; Thiorphan | 1997 |
Metabolism of bradykinin by the rat coronary vascular bed.
Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Chromatography, High Pressure Liquid; Coronary Circulation; Coronary Vessels; Enalaprilat; Hemodynamics; Immunoenzyme Techniques; In Vitro Techniques; Male; Neprilysin; Perfusion; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Thiorphan; Time Factors | 1998 |