Page last updated: 2024-09-04

retrothiorphan and bradykinin

retrothiorphan has been researched along with bradykinin in 5 studies

Compound Research Comparison

Studies
(retrothiorphan)
Trials
(retrothiorphan)
Recent Studies (post-2010)
(retrothiorphan)
Studies
(bradykinin)
Trials
(bradykinin)
Recent Studies (post-2010) (bradykinin)
180214,1953551,520

Protein Interaction Comparison

ProteinTaxonomyretrothiorphan (IC50)bradykinin (IC50)
B2 bradykinin receptorHomo sapiens (human)0.0018

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (80.00)18.2507
2000's1 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Corvol, P; el Amrani, AI; FourniƩ-Zaluski, MC; Michel, JB; Pham, I; Roques, B1
Doucet, J; Fournie-Zaluski, MC; Gonzalez, W; Michel, JB; Pham, I; Roques, BP1
Adam, A; Blais, C; Drapeau, G; Gervais, N; Lamontagne, D; Raymond, P; Venneman, I1
Adam, A; Blais, C; Dumoulin, MJ; Lamontagne, D1
Arbin, V; Claperon, N; FourniƩ-Zaluski, MC; Peyroux, J; Roques, BP1

Other Studies

5 other study(ies) available for retrothiorphan and bradykinin

ArticleYear
Effects of the selective neutral endopeptidase inhibitor, retrothiorphan, on renal function and blood pressure in conscious normotensive Wistar and hypertensive DOCA-salt rats.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:6

    Topics: Animals; Atrial Natriuretic Factor; Blood Pressure; Bradykinin; Cyclic GMP; Desoxycorticosterone; Diuresis; Hypertension; Kidney; Kininogens; Male; Natriuresis; Neprilysin; Rats; Rats, Wistar; Sulfhydryl Compounds; Thiorphan

1992
Effects of angiotensin-converting enzyme and neutral endopeptidase inhibitors: influence of bradykinin.
    European journal of pharmacology, 1996, Feb-05, Volume: 296, Issue:3

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Pressure; Bradykinin; Cyclic GMP; Enalaprilat; Hypertension; Kidney; Male; Neprilysin; Rats; Rats, Wistar; Thiorphan

1996
Contribution of angiotensin-converting enzyme to the cardiac metabolism of bradykinin: an interspecies study.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Amino Acid Sequence; Angiotensin-Converting Enzyme Inhibitors; Animals; Antibodies; Bradykinin; Cross Reactions; Dogs; Enalaprilat; Humans; Kinetics; Losartan; Myocardium; Peptidyl-Dipeptidase A; Protease Inhibitors; Rabbits; Rats; Species Specificity; Substrate Specificity; Thiorphan

1997
Metabolism of bradykinin by the rat coronary vascular bed.
    Cardiovascular research, 1998, Volume: 38, Issue:1

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Bradykinin; Chromatography, High Pressure Liquid; Coronary Circulation; Coronary Vessels; Enalaprilat; Hemodynamics; Immunoenzyme Techniques; In Vitro Techniques; Male; Neprilysin; Perfusion; Protease Inhibitors; Rats; Rats, Sprague-Dawley; Thiorphan; Time Factors

1998
Effects of combined neutral endopeptidase 24-11 and angiotensin-converting enzyme inhibition on femoral vascular conductance in streptozotocin-induced diabetic rats.
    British journal of pharmacology, 2000, Volume: 130, Issue:6

    Topics: 3-Mercaptopropionic Acid; Angiotensin-Converting Enzyme Inhibitors; Animals; Blood Flow Velocity; Blood Pressure; Bradykinin; Bradykinin Receptor Antagonists; Captopril; Diabetes Mellitus, Experimental; Enzyme Inhibitors; Femoral Artery; Hemodynamics; Kininogens; Lysine Carboxypeptidase; Male; Neprilysin; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Peptidyl-Dipeptidase A; Protease Inhibitors; Rats; Rats, Inbred BN; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Thiorphan; Time Factors

2000