Page last updated: 2024-09-03

renzapride and zacopride

renzapride has been researched along with zacopride in 6 studies

Compound Research Comparison

Studies
(renzapride)
Trials
(renzapride)
Recent Studies (post-2010)
(renzapride)
Studies
(zacopride)
Trials
(zacopride)
Recent Studies (post-2010) (zacopride)
70122180416

Protein Interaction Comparison

ProteinTaxonomyrenzapride (IC50)zacopride (IC50)
Neuronal acetylcholine receptor subunit alpha-7Rattus norvegicus (Norway rat)7.0597

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's0 (0.00)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Delarue, C; Idres, S; Lefebvre, H; Vaudry, H1
Boddeke, HW; Kalkman, HO1
Bockaert, J; Dumuis, A; Sebben, M1
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M1
Akuzawa, S; Ito, H; Kamato, T; Miyata, K; Nagakura, Y; Suzuki, T; Yamaguchi, T1
Chinkwo, KA; Coupar, IM; Grabbe, C; Irving, HR; Li, JG; Pouton, CW; Shapiro, M; Tochon-Danguy, N1

Other Studies

6 other study(ies) available for renzapride and zacopride

ArticleYear
Benzamide derivatives provide evidence for the involvement of a 5-HT4 receptor type in the mechanism of action of serotonin in frog adrenocortical cells.
    Brain research. Molecular brain research, 1991, Volume: 10, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenal Cortex; Adrenal Cortex Hormones; Aldosterone; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Corticosterone; In Vitro Techniques; Kinetics; Methysergide; Piperidines; Rana ridibunda; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Zacopride and BRL 24924 induce an increase in EEG-energy in rats.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electroencephalography; Indoles; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Scopolamine; Serotonin Antagonists; Tropisetron

1990
Pharmacological characterization of 5-hydroxytryptamine4(5-HT4) receptors positively coupled to adenylate cyclase in adult guinea pig hippocampal membranes: effect of substituted benzamide derivatives.
    Molecular pharmacology, 1990, Volume: 37, Issue:3

    Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Activation; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Receptors, Serotonin; Serotonin; Signal Transduction; Spiperone; Structure-Activity Relationship; Tropisetron

1990
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
    European journal of pharmacology, 1996, Sep-05, Volume: 311, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1996
Pharmacological properties of a novel gastrointestinal prokinetic benzamide selective for human 5-HT4 receptor versus human 5-HT3 receptor.
    Pharmacological research, 1999, Volume: 39, Issue:5

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Digestive System; Esophagus; Gastrointestinal Transit; Guinea Pigs; Humans; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxadiazoles; Piperidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists

1999
Investigations into the binding affinities of different human 5-HT4 receptor splice variants.
    Pharmacology, 2010, Volume: 85, Issue:4

    Topics: Aniline Compounds; Animals; Benzamides; Benzimidazoles; Benzofurans; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Chlorocebus aethiops; COS Cells; Cyclic AMP; Dose-Response Relationship, Drug; Humans; Indoles; Kinetics; Ligands; Piperidines; Protein Isoforms; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists

2010