Page last updated: 2024-09-03

renzapride and tropisetron

renzapride has been researched along with tropisetron in 20 studies

Compound Research Comparison

Studies
(renzapride)
Trials
(renzapride)
Recent Studies (post-2010)
(renzapride)
Studies
(tropisetron)
Trials
(tropisetron)
Recent Studies (post-2010) (tropisetron)
70122944218150

Protein Interaction Comparison

ProteinTaxonomyrenzapride (IC50)tropisetron (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)3.1623
Muscarinic acetylcholine receptor M2Homo sapiens (human)3.1623
Muscarinic acetylcholine receptor M5Homo sapiens (human)3.45
Neuronal acetylcholine receptor subunit beta-4Homo sapiens (human)1.8
Sodium-dependent serotonin transporterHomo sapiens (human)0.488
Neuronal acetylcholine receptor subunit alpha-3Homo sapiens (human)1.8

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19903 (15.00)18.7374
1990's17 (85.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ansanay, H; Dumuis, A; Giraldo, E; Gozlan, H; Ladinsky, H; Monferini, E; Rizzi, CA; Schiantarelli, P; Sebben, M; Turconi, M1
Candura, SM; Coccini, T; Manzo, L; Onori, L; Rizzi, CA; Tonini, M1
Clarke, DE; Craig, DA1
Brown, AM; Brown, MJ; Kaumann, AJ; Murray, KJ; Sanders, L1
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N1
Gullikson, GW; Loeffler, RF; Viriña, MA1
Kaumann, AJ1
den Boer, MO; Heiligers, JP; Saxena, PR; Villalón, CM1
Andrade, R; Araneda, RC; Chaput, Y1
Boddeke, HW; Kalkman, HO1
Bockaert, J; Dumuis, A; Sebben, M2
Ito, A; Ito, T; Iwanaga, H; Karasawa, T; Mizumoto, A; Yoshida, N1
Gullikson, GW; Nemeth, PR1
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ1
Galligan, JJ; Pan, H1
Buchheit, KH; Buhl, T1
Hansen, MB; Skadhauge, E1
Hansen, MB; Jaffe, BM1
Flynn, DL; Goldstin, B; Gullikson, GW; Moormann, AE; Yang, DC1

Other Studies

20 other study(ies) available for renzapride and tropisetron

ArticleYear
Characterization of a novel 5-HT4 receptor antagonist of the azabicycloalkyl benzimidazolone class: DAU 6285.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:3

    Topics: Animals; Benzamides; Benzimidazoles; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cyclic AMP; Embryo, Mammalian; Heart Rate; Indoles; Kinetics; Mesencephalon; Mice; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stimulation, Chemical; Tropisetron

1992
The influence of neuronal 5-hydroxytryptamine receptor antagonists on non-cholinergic ganglionic transmission in the guinea-pig enteric excitatory reflex.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Female; Guinea Pigs; Indoles; Intestine, Small; Male; Methiothepin; Muscle Contraction; Ondansetron; Serotonin Antagonists; Synaptic Transmission; Tropisetron

1992
Peristalsis evoked by 5-HT and renzapride: evidence for putative 5-HT4 receptor activation.
    British journal of pharmacology, 1991, Volume: 102, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Guinea Pigs; In Vitro Techniques; Indoles; Male; Peristalsis; Receptors, Serotonin; Serotonin; Tropisetron

1991
A 5-HT4-like receptor in human right atrium.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:2

    Topics: Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Cyclic AMP; Embryo, Mammalian; Female; Heart Atria; Humans; Indoles; Male; Middle Aged; Myocardial Contraction; Piperidines; Protein Kinases; Receptors, Serotonin; Serotonin; Structure-Activity Relationship; Tropisetron

1991
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron

1991
Relationship of serotonin-3 receptor antagonist activity to gastric emptying and motor-stimulating actions of prokinetic drugs in dogs.
    The Journal of pharmacology and experimental therapeutics, 1991, Jul-01, Volume: 258, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Cisplatin; Dogs; Dose-Response Relationship, Drug; Female; Gastric Emptying; Gastrointestinal Motility; Indoles; Injections, Intravenous; Male; Metoclopramide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Tropisetron

1991
Piglet sinoatrial 5-HT receptors resemble human atrial 5-HT4-like receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:5

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cardiotonic Agents; Cisapride; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Indoles; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sinoatrial Node; Swine; Tropisetron

1990
Mediation of 5-hydroxytryptamine-induced tachycardia in the pig by the putative 5-HT4 receptor.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Anesthesia; Animals; Benzamides; Blood Pressure; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Heart; Heart Rate; In Vitro Techniques; Indoles; Isoproterenol; Myocardium; Receptors, Serotonin; Serotonin; Swine; Tropisetron

1990
Pharmacological and functional analysis of a novel serotonin receptor in the rat hippocampus.
    European journal of pharmacology, 1990, Jul-17, Volume: 182, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Hippocampus; In Vitro Techniques; Indoles; Male; Neurons; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron

1990
Zacopride and BRL 24924 induce an increase in EEG-energy in rats.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electroencephalography; Indoles; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Scopolamine; Serotonin Antagonists; Tropisetron

1990
Pharmacological characterization of 5-hydroxytryptamine4(5-HT4) receptors positively coupled to adenylate cyclase in adult guinea pig hippocampal membranes: effect of substituted benzamide derivatives.
    Molecular pharmacology, 1990, Volume: 37, Issue:3

    Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Activation; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Receptors, Serotonin; Serotonin; Signal Transduction; Spiperone; Structure-Activity Relationship; Tropisetron

1990
BRL 24924: a potent agonist at a non-classical 5-HT receptor positively coupled with adenylate cyclase in colliculi neurons.
    European journal of pharmacology, 1989, Mar-21, Volume: 162, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cyclic AMP; Embryo, Mammalian; Female; Indoles; Metoclopramide; Mice; Neurons; Pregnancy; Serotonin Antagonists; Tropisetron

1989
[Effect of 5-HT3 receptor antagonists on gastrointestinal motility].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:6

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; In Vitro Techniques; Indazoles; Indoles; Motilin; Ondansetron; Rabbits; Serotonin Antagonists; Tropisetron

1989
Gastrointestinal motility stimulating drugs and 5-HT receptors on myenteric neurons.
    European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Electrophysiology; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Indoles; Male; Metoclopramide; Myenteric Plexus; Neurons; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Stimulation, Chemical; Tropisetron

1989
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1995
Effects of 5-HT1A and 5-HT4 receptor agonists on slow synaptic potentials in enteric neurons.
    European journal of pharmacology, 1995, May-04, Volume: 278, Issue:1

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dose-Response Relationship, Drug; Electrophysiology; Guinea Pigs; Ileum; Indoles; Male; Membrane Potentials; Myenteric Plexus; Neurons; Piperazines; Piperidines; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1995
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron

1994
Ketanserin and granisetron reduce cholera toxin-induced hypersecretion in pig jejunum.
    Scandinavian journal of gastroenterology, 1994, Volume: 29, Issue:10

    Topics: Animals; Animals, Newborn; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholera Toxin; Diarrhea; Dose-Response Relationship, Drug; Drug Therapy, Combination; Granisetron; Indoles; Intestinal Secretions; Jejunum; Ketanserin; Methysergide; Serotonin Antagonists; Swine; Tropisetron

1994
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
    The Journal of surgical research, 1994, Volume: 56, Issue:3

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance

1994
SC-53606, a potent and selective antagonist of 5-hydroxytryptamine4 receptors in isolated rat esophageal tunica muscularis mucosae.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Esophagus; Imidazoles; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Pyrroles; Rats; Receptors, Cell Surface; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Tryptamines

1993