renzapride has been researched along with tropisetron in 20 studies
Studies (renzapride) | Trials (renzapride) | Recent Studies (post-2010) (renzapride) | Studies (tropisetron) | Trials (tropisetron) | Recent Studies (post-2010) (tropisetron) |
---|---|---|---|---|---|
70 | 12 | 2 | 944 | 218 | 150 |
Protein | Taxonomy | renzapride (IC50) | tropisetron (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 4 | Cavia porcellus (domestic guinea pig) | 3.1623 | |
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 3.1623 | |
Muscarinic acetylcholine receptor M5 | Homo sapiens (human) | 3.45 | |
Neuronal acetylcholine receptor subunit beta-4 | Homo sapiens (human) | 1.8 | |
Sodium-dependent serotonin transporter | Homo sapiens (human) | 0.488 | |
Neuronal acetylcholine receptor subunit alpha-3 | Homo sapiens (human) | 1.8 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (15.00) | 18.7374 |
1990's | 17 (85.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ansanay, H; Dumuis, A; Giraldo, E; Gozlan, H; Ladinsky, H; Monferini, E; Rizzi, CA; Schiantarelli, P; Sebben, M; Turconi, M | 1 |
Candura, SM; Coccini, T; Manzo, L; Onori, L; Rizzi, CA; Tonini, M | 1 |
Clarke, DE; Craig, DA | 1 |
Brown, AM; Brown, MJ; Kaumann, AJ; Murray, KJ; Sanders, L | 1 |
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N | 1 |
Gullikson, GW; Loeffler, RF; Viriña, MA | 1 |
Kaumann, AJ | 1 |
den Boer, MO; Heiligers, JP; Saxena, PR; Villalón, CM | 1 |
Andrade, R; Araneda, RC; Chaput, Y | 1 |
Boddeke, HW; Kalkman, HO | 1 |
Bockaert, J; Dumuis, A; Sebben, M | 2 |
Ito, A; Ito, T; Iwanaga, H; Karasawa, T; Mizumoto, A; Yoshida, N | 1 |
Gullikson, GW; Nemeth, PR | 1 |
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ | 1 |
Galligan, JJ; Pan, H | 1 |
Buchheit, KH; Buhl, T | 1 |
Hansen, MB; Skadhauge, E | 1 |
Hansen, MB; Jaffe, BM | 1 |
Flynn, DL; Goldstin, B; Gullikson, GW; Moormann, AE; Yang, DC | 1 |
20 other study(ies) available for renzapride and tropisetron
Article | Year |
---|---|
Characterization of a novel 5-HT4 receptor antagonist of the azabicycloalkyl benzimidazolone class: DAU 6285.
Topics: Animals; Benzamides; Benzimidazoles; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Cyclic AMP; Embryo, Mammalian; Heart Rate; Indoles; Kinetics; Mesencephalon; Mice; Rats; Receptors, Serotonin; Reflex; Serotonin; Serotonin Antagonists; Stimulation, Chemical; Tropisetron | 1992 |
The influence of neuronal 5-hydroxytryptamine receptor antagonists on non-cholinergic ganglionic transmission in the guinea-pig enteric excitatory reflex.
Topics: Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Female; Guinea Pigs; Indoles; Intestine, Small; Male; Methiothepin; Muscle Contraction; Ondansetron; Serotonin Antagonists; Synaptic Transmission; Tropisetron | 1992 |
Peristalsis evoked by 5-HT and renzapride: evidence for putative 5-HT4 receptor activation.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Guinea Pigs; In Vitro Techniques; Indoles; Male; Peristalsis; Receptors, Serotonin; Serotonin; Tropisetron | 1991 |
A 5-HT4-like receptor in human right atrium.
Topics: Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Cyclic AMP; Embryo, Mammalian; Female; Heart Atria; Humans; Indoles; Male; Middle Aged; Myocardial Contraction; Piperidines; Protein Kinases; Receptors, Serotonin; Serotonin; Structure-Activity Relationship; Tropisetron | 1991 |
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron | 1991 |
Relationship of serotonin-3 receptor antagonist activity to gastric emptying and motor-stimulating actions of prokinetic drugs in dogs.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Cisplatin; Dogs; Dose-Response Relationship, Drug; Female; Gastric Emptying; Gastrointestinal Motility; Indoles; Injections, Intravenous; Male; Metoclopramide; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Tropisetron | 1991 |
Piglet sinoatrial 5-HT receptors resemble human atrial 5-HT4-like receptors.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cardiotonic Agents; Cisapride; Female; Heart; Heart Atria; Humans; In Vitro Techniques; Indoles; Male; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sinoatrial Node; Swine; Tropisetron | 1990 |
Mediation of 5-hydroxytryptamine-induced tachycardia in the pig by the putative 5-HT4 receptor.
Topics: Anesthesia; Animals; Benzamides; Blood Pressure; Brain; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Heart; Heart Rate; In Vitro Techniques; Indoles; Isoproterenol; Myocardium; Receptors, Serotonin; Serotonin; Swine; Tropisetron | 1990 |
Pharmacological and functional analysis of a novel serotonin receptor in the rat hippocampus.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Hippocampus; In Vitro Techniques; Indoles; Male; Neurons; Pyramidal Tracts; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tropanes; Tropisetron | 1990 |
Zacopride and BRL 24924 induce an increase in EEG-energy in rats.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electroencephalography; Indoles; Injections, Intraventricular; Male; Rats; Rats, Inbred Strains; Scopolamine; Serotonin Antagonists; Tropisetron | 1990 |
Pharmacological characterization of 5-hydroxytryptamine4(5-HT4) receptors positively coupled to adenylate cyclase in adult guinea pig hippocampal membranes: effect of substituted benzamide derivatives.
Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Enzyme Activation; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Receptors, Serotonin; Serotonin; Signal Transduction; Spiperone; Structure-Activity Relationship; Tropisetron | 1990 |
BRL 24924: a potent agonist at a non-classical 5-HT receptor positively coupled with adenylate cyclase in colliculi neurons.
Topics: Adenylyl Cyclases; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Bridged-Ring Compounds; Cyclic AMP; Embryo, Mammalian; Female; Indoles; Metoclopramide; Mice; Neurons; Pregnancy; Serotonin Antagonists; Tropisetron | 1989 |
[Effect of 5-HT3 receptor antagonists on gastrointestinal motility].
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; In Vitro Techniques; Indazoles; Indoles; Motilin; Ondansetron; Rabbits; Serotonin Antagonists; Tropisetron | 1989 |
Gastrointestinal motility stimulating drugs and 5-HT receptors on myenteric neurons.
Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Electrophysiology; Gastrointestinal Motility; Guinea Pigs; In Vitro Techniques; Indoles; Male; Metoclopramide; Myenteric Plexus; Neurons; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Stimulation, Chemical; Tropisetron | 1989 |
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1995 |
Effects of 5-HT1A and 5-HT4 receptor agonists on slow synaptic potentials in enteric neurons.
Topics: 5-Methoxytryptamine; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Dose-Response Relationship, Drug; Electrophysiology; Guinea Pigs; Ileum; Indoles; Male; Membrane Potentials; Myenteric Plexus; Neurons; Piperazines; Piperidines; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1995 |
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron | 1994 |
Ketanserin and granisetron reduce cholera toxin-induced hypersecretion in pig jejunum.
Topics: Animals; Animals, Newborn; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholera Toxin; Diarrhea; Dose-Response Relationship, Drug; Drug Therapy, Combination; Granisetron; Indoles; Intestinal Secretions; Jejunum; Ketanserin; Methysergide; Serotonin Antagonists; Swine; Tropisetron | 1994 |
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance | 1994 |
SC-53606, a potent and selective antagonist of 5-hydroxytryptamine4 receptors in isolated rat esophageal tunica muscularis mucosae.
Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Esophagus; Imidazoles; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Pyrroles; Rats; Receptors, Cell Surface; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Tryptamines | 1993 |