Page last updated: 2024-09-03

renzapride and sdz 205-557

renzapride has been researched along with sdz 205-557 in 5 studies

Compound Research Comparison

Studies
(renzapride)
Trials
(renzapride)
Recent Studies (post-2010)
(renzapride)
Studies
(sdz 205-557)
Trials
(sdz 205-557)
Recent Studies (post-2010) (sdz 205-557)
701225609

Protein Interaction Comparison

ProteinTaxonomyrenzapride (IC50)sdz 205-557 (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.2512
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.2512

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ1
Buchheit, KH; Buhl, T1
Flynn, DL; Goldstin, B; Gullikson, GW; Moormann, AE; Yang, DC1
Ito, H; Kamato, T; Miyata, K; Nagakura, Y; Nishida, A; Yamano, M1
Hillsley, K; Mawe, GM1

Other Studies

5 other study(ies) available for renzapride and sdz 205-557

ArticleYear
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1995
Stimulant effects of 5-hydroxytryptamine on guinea pig stomach preparations in vitro.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: 4-Aminobenzoic Acid; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Atropine; Benzamides; Binding Sites; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Electric Stimulation; Female; Guinea Pigs; In Vitro Techniques; Indoles; Ligands; Male; Metoclopramide; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stomach; Tetrodotoxin; Tropanes; Tropisetron

1994
SC-53606, a potent and selective antagonist of 5-hydroxytryptamine4 receptors in isolated rat esophageal tunica muscularis mucosae.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Carbachol; Esophagus; Imidazoles; In Vitro Techniques; Indoles; Male; Mucous Membrane; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Pyrroles; Rats; Receptors, Cell Surface; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron; Tryptamines

1993
Characterization of 5-hydroxytryptamine (5-HT) receptor subtypes influencing colonic motility in conscious dogs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Benzimidazoles; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dogs; Dose-Response Relationship, Drug; Gastrointestinal Motility; Hexamethonium; Injections, Intravenous; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Transducers

1996
5-HT is present in nerves of guinea pig sphincter of Oddi and depolarizes sphincter of Oddi neurons.
    The American journal of physiology, 1998, Volume: 275, Issue:5

    Topics: 4-Aminobenzoic Acid; 5,7-Dihydroxytryptamine; Animals; Atropine; Benzamides; Bridged Bicyclo Compounds, Heterocyclic; Evoked Potentials; Ganglia, Autonomic; Guinea Pigs; Immunohistochemistry; Indazoles; Membrane Potentials; Myenteric Plexus; Nerve Fibers; Neurons; Organ Culture Techniques; para-Aminobenzoates; Serotonin; Serotonin Antagonists; Sphincter of Oddi; Tetrodotoxin; Tropanes

1998