Page last updated: 2024-09-03

renzapride and ondansetron

renzapride has been researched along with ondansetron in 5 studies

Compound Research Comparison

Studies
(renzapride)
Trials
(renzapride)
Recent Studies (post-2010)
(renzapride)
Studies
(ondansetron)
Trials
(ondansetron)
Recent Studies (post-2010) (ondansetron)
701223,3801,216994

Protein Interaction Comparison

ProteinTaxonomyrenzapride (IC50)ondansetron (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)10
Solute carrier family 22 member 2Homo sapiens (human)1.295
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)10
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.0136
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.717
5-hydroxytryptamine receptor 3AHomo sapiens (human)0.0001
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)10
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)10
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.7303
Multidrug and toxin extrusion protein 2Homo sapiens (human)2.4533
GABA theta subunitRattus norvegicus (Norway rat)10
Multidrug and toxin extrusion protein 1Homo sapiens (human)0.0875
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)10
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.0181

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19901 (20.00)18.7374
1990's4 (80.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Candura, SM; Coccini, T; Manzo, L; Onori, L; Rizzi, CA; Tonini, M1
Coleman, J; Lattimer, N; Rhodes, KF1
Itoh, Z; Iwanaga, Y; Mizumoto, A; Yoshida, N1
Ito, A; Ito, T; Iwanaga, H; Karasawa, T; Mizumoto, A; Yoshida, N1
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M1

Other Studies

5 other study(ies) available for renzapride and ondansetron

ArticleYear
The influence of neuronal 5-hydroxytryptamine receptor antagonists on non-cholinergic ganglionic transmission in the guinea-pig enteric excitatory reflex.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Female; Guinea Pigs; Indoles; Intestine, Small; Male; Methiothepin; Muscle Contraction; Ondansetron; Serotonin Antagonists; Synaptic Transmission; Tropisetron

1992
A component of 5-HT-evoked depolarization of the rat isolated vagus nerve is mediated by a putative 5-HT4 receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 346, Issue:5

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; In Vitro Techniques; Male; Neuromuscular Depolarizing Agents; Ondansetron; Potentiometry; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vagus Nerve

1992
Effects of 5-hydroxytryptamine 3 receptor antagonists on gastrointestinal motor activity in conscious dogs.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Digestion; Dogs; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Imidazoles; Indazoles; Indoles; Infusions, Intravenous; Injections, Intravenous; Male; Motilin; Motor Activity; Muscle Contraction; Muscle, Smooth; Ondansetron; Serotonin Antagonists; Time Factors; Tropisetron

1991
[Effect of 5-HT3 receptor antagonists on gastrointestinal motility].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:6

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Dogs; Gastrointestinal Motility; Granisetron; Imidazoles; In Vitro Techniques; Indazoles; Indoles; Motilin; Ondansetron; Rabbits; Serotonin Antagonists; Tropisetron

1989
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
    European journal of pharmacology, 1996, Sep-05, Volume: 311, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists

1996