Page last updated: 2024-09-03

renzapride and methysergide

renzapride has been researched along with methysergide in 5 studies

Compound Research Comparison

Studies
(renzapride)
Trials
(renzapride)
Recent Studies (post-2010)
(renzapride)
Studies
(methysergide)
Trials
(methysergide)
Recent Studies (post-2010) (methysergide)
701222,9358180

Protein Interaction Comparison

ProteinTaxonomyrenzapride (IC50)methysergide (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.0021
Alpha-2A adrenergic receptorHomo sapiens (human)1.631
D(2) dopamine receptorHomo sapiens (human)0.807
Alpha-2B adrenergic receptorHomo sapiens (human)4.763
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.054
D(1A) dopamine receptorHomo sapiens (human)0.943
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.013
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0021
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.054
D(3) dopamine receptorHomo sapiens (human)0.172
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0006
5-hydroxytryptamine receptor 6Homo sapiens (human)0.162

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Delarue, C; Idres, S; Lefebvre, H; Vaudry, H1
Hansen, MB; Skadhauge, E1
Beubler, E; Hansen, MB; Skadhauge, E; Thørboll, JE1
Hansen, MB; Jaffe, BM1
Ito, H; Kamato, T; Miyata, K; Nagakura, Y; Nishida, A; Yamano, M1

Other Studies

5 other study(ies) available for renzapride and methysergide

ArticleYear
Benzamide derivatives provide evidence for the involvement of a 5-HT4 receptor type in the mechanism of action of serotonin in frog adrenocortical cells.
    Brain research. Molecular brain research, 1991, Volume: 10, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenal Cortex; Adrenal Cortex Hormones; Aldosterone; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Corticosterone; In Vitro Techniques; Kinetics; Methysergide; Piperidines; Rana ridibunda; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1991
Ketanserin and granisetron reduce cholera toxin-induced hypersecretion in pig jejunum.
    Scandinavian journal of gastroenterology, 1994, Volume: 29, Issue:10

    Topics: Animals; Animals, Newborn; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cholera Toxin; Diarrhea; Dose-Response Relationship, Drug; Drug Therapy, Combination; Granisetron; Indoles; Intestinal Secretions; Jejunum; Ketanserin; Methysergide; Serotonin Antagonists; Swine; Tropisetron

1994
Effect of indomethacin, renzapride, methysergide, ketanserin, granisetron and citalopram on serotonin-induced fluid accumulation in pig jejunum.
    Physiological research, 1994, Volume: 43, Issue:2

    Topics: Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Citalopram; Dose-Response Relationship, Drug; Granisetron; Indomethacin; Intestinal Absorption; Jejunum; Ketanserin; Methysergide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Swine

1994
5-HT receptor subtypes involved in luminal serotonin-induced secretion in rat intestine in vivo.
    The Journal of surgical research, 1994, Volume: 56, Issue:3

    Topics: 5-Methoxytryptamine; Animals; Benzamides; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Ileum; Indoles; Jejunum; Ketanserin; Male; Methysergide; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Tropisetron; Water-Electrolyte Balance

1994
Characterization of 5-hydroxytryptamine (5-HT) receptor subtypes influencing colonic motility in conscious dogs.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: 4-Aminobenzoic Acid; Animals; Benzamides; Benzimidazoles; Biguanides; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dogs; Dose-Response Relationship, Drug; Gastrointestinal Motility; Hexamethonium; Injections, Intravenous; Ketanserin; Male; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Transducers

1996