raubasine has been researched along with clonidine in 6 studies
Studies (raubasine) | Trials (raubasine) | Recent Studies (post-2010) (raubasine) | Studies (clonidine) | Trials (clonidine) | Recent Studies (post-2010) (clonidine) |
---|---|---|---|---|---|
7 | 0 | 3 | 13,692 | 2,044 | 1,394 |
140 | 8 | 22 | 13,692 | 2,044 | 1,394 |
Protein | Taxonomy | raubasine (IC50) | clonidine (IC50) |
---|---|---|---|
Alpha-2A adrenergic receptor | Homo sapiens (human) | 0.101 | |
Alpha-2B adrenergic receptor | Homo sapiens (human) | 0.0353 | |
Alpha-2C adrenergic receptor | Homo sapiens (human) | 0.0115 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 5.365 | |
Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.0173 | |
Alpha-1D adrenergic receptor | Homo sapiens (human) | 1.21 | |
5-hydroxytryptamine receptor 1B | Rattus norvegicus (Norway rat) | 5.365 | |
Alpha-2A adrenergic receptor | Bos taurus (cattle) | 0.002 | |
Nischarin | Rattus norvegicus (Norway rat) | 0.3662 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (83.33) | 18.7374 |
1990's | 1 (16.67) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bondinell, W; Hieble, JP; Ruffolo, RR | 1 |
Guez, D; Sebban, C; Tesolin, B | 1 |
Demichel, P; Roquebert, J | 1 |
Demichel, P; Gomond, P; Roquebert, J | 2 |
Aarhus, LL; Rimele, TJ; Rooke, TW; Vanhoutte, PM | 1 |
1 review(s) available for raubasine and clonidine
Article | Year |
---|---|
Alpha- and beta-adrenoceptors: from the gene to the clinic. 2. Structure-activity relationships and therapeutic applications.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Humans; Molecular Conformation; Molecular Structure; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Structure-Activity Relationship | 1995 |
5 other study(ies) available for raubasine and clonidine
Article | Year |
---|---|
[Quantified electroencephalogram: value in the evaluation of therapy of cerebral aging].
Topics: Almitrine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Central Nervous System Stimulants; Cerebral Cortex; Clonidine; Dementia; Drug Combinations; Drug Evaluation; Electroencephalography; Humans; Piperazines; Rats; Secologanin Tryptamine Alkaloids; Yohimbine | 1987 |
Effects of raubasine stereoisomers on pre- and postsynaptic alpha-adrenoceptors in the rat vas deferens.
Topics: Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Secologanin Tryptamine Alkaloids; Stereoisomerism; Vas Deferens; Yohimbine | 1984 |
Pre- and postsynaptic alpha-adrenoceptor blocking activity of raubasine in the rat vas deferens.
Topics: Adrenergic beta-Antagonists; Animals; Clonidine; Cocaine; Dose-Response Relationship, Drug; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, beta; Secologanin Tryptamine Alkaloids; Synapses; Vas Deferens; Yohimbine | 1981 |
alpha-Adrenoceptor blocking properties of raubasine in pithed rats.
Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Clonidine; Decerebrate State; Electric Stimulation; Heart Rate; Male; Phenylephrine; Rats; Rats, Inbred Strains; Secologanin Tryptamine Alkaloids; Spinal Cord; Yohimbine | 1982 |
Alpha-1 adrenoceptors and calcium in isolated canine coronary arteries.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channel Blockers; Clonidine; Coronary Vessels; Dogs; Female; Imidazoles; Male; Methoxamine; Muscle Contraction; Norepinephrine; Phenylephrine; Prazosin; Secologanin Tryptamine Alkaloids; Yohimbine | 1983 |