Page last updated: 2024-09-04

r115777 and lonafarnib

r115777 has been researched along with lonafarnib in 3 studies

Compound Research Comparison

Studies
(r115777)
Trials
(r115777)
Recent Studies (post-2010)
(r115777)
Studies
(lonafarnib)
Trials
(lonafarnib)
Recent Studies (post-2010) (lonafarnib)
8042243490
804603

Protein Interaction Comparison

ProteinTaxonomyr115777 (IC50)lonafarnib (IC50)
Chain A, Protein farnesyltransferase alpha subunitRattus norvegicus (Norway rat)0.0019
Chain B, Protein farnesyltransferase beta subunitRattus norvegicus (Norway rat)0.0019
GTPase HRasHomo sapiens (human)0.07
ATP-dependent translocase ABCB1Homo sapiens (human)2.7
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaBos taurus (cattle)0.0083
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaHomo sapiens (human)0.1498
Protein farnesyltransferase subunit betaBos taurus (cattle)0.0083
Protein farnesyltransferase subunit betaHomo sapiens (human)0.1498
Protein farnesyltransferase subunit betaRattus norvegicus (Norway rat)0.0019
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaRattus norvegicus (Norway rat)0.0019
Geranylgeranyl transferase type-1 subunit betaBos taurus (cattle)0.0083

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Claiborne, A; Cohen, J; Frost, D; Gu, WZ; Hutchins, C; Li, Q; Lin, NH; Rosenberg, SH; Sham, HL; Stoll, VS; Wang, W; Woods, KW1
Bauer, KD; Bendale, P; Buckner, FS; Chakrabarti, D; Floyd, D; Gelb, MH; Hamilton, A; Hornéy, CP; Lombardo, LJ; Nallan, L; Pendyala, PR; Rivas, K; Sebti, S; Van Voorhis, WC; Weber, PC; Williams, DK; Windsor, WT; Yokoyama, K1
Cohen, J; Frost, D; Galicia, T; Gu, WZ; Hutchins, C; Li, Q; Li, T; Rosenberg, SH; Sham, HL; Stoll, VS; Woods, KW1

Other Studies

3 other study(ies) available for r115777 and lonafarnib

ArticleYear
Design, synthesis, and activity of achiral analogs of 2-quinolones and indoles as non-thiol farnesyltransferase inhibitors.
    Bioorganic & medicinal chemistry letters, 2005, Apr-15, Volume: 15, Issue:8

    Topics: Alkyl and Aryl Transferases; Animals; Cattle; Drug Design; Enzyme Inhibitors; Farnesyltranstransferase; Hydroxyquinolines; Indoles; Mice; NIH 3T3 Cells; Quinolones; Stereoisomerism

2005
Protein farnesyltransferase inhibitors exhibit potent antimalarial activity.
    Journal of medicinal chemistry, 2005, Jun-02, Volume: 48, Issue:11

    Topics: Alkyl and Aryl Transferases; Animals; Antimalarials; Cells, Cultured; Electrophoresis, Polyacrylamide Gel; Erythrocytes; Farnesyltranstransferase; Female; Humans; Malaria; Mice; Mice, Inbred BALB C; Microscopy, Fluorescence; Plasmodium berghei; Plasmodium falciparum; Protein Prenylation; Quinolones; Rats; Structure-Activity Relationship

2005
Benzimidazolones and indoles as non-thiol farnesyltransferase inhibitors based on tipifarnib scaffold: synthesis and activity.
    Bioorganic & medicinal chemistry letters, 2005, Jun-02, Volume: 15, Issue:11

    Topics: Alkyl and Aryl Transferases; Animals; Benzimidazoles; Enzyme Inhibitors; Farnesyltranstransferase; Indoles; Mice; NIH 3T3 Cells; Quinolones

2005
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