Page last updated: 2024-09-04

r 84760 and naltrexone

r 84760 has been researched along with naltrexone in 1 studies

Compound Research Comparison

Studies
(r 84760)
Trials
(r 84760)
Recent Studies (post-2010)
(r 84760)
Studies
(naltrexone)
Trials
(naltrexone)
Recent Studies (post-2010) (naltrexone)
7008,7451,2282,642

Protein Interaction Comparison

ProteinTaxonomyr 84760 (IC50)naltrexone (IC50)
Cytochrome P450 2D6Homo sapiens (human)1
Delta-type opioid receptorMus musculus (house mouse)0.0051
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0063
Kappa-type opioid receptorMus musculus (house mouse)0.006
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0005
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0005
Mu-type opioid receptorHomo sapiens (human)0.006
Delta-type opioid receptorHomo sapiens (human)0.0319
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0093
Kappa-type opioid receptorHomo sapiens (human)0.0377
Mu-type opioid receptorMus musculus (house mouse)0.0076
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0004

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Butelman, ER; Ho, A; Kreek, MJ; Schlussman, SD; Zhang, Y1

Other Studies

1 other study(ies) available for r 84760 and naltrexone

ArticleYear
Effect of the kappa opioid agonist R-84760 on cocaine-induced increases in striatal dopamine levels and cocaine-induced place preference in C57BL/6J mice.
    Psychopharmacology, 2004, Volume: 173, Issue:1-2

    Topics: Analysis of Variance; Animals; Behavior, Animal; Chromatography, High Pressure Liquid; Cocaine; Conditioning, Operant; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Food; Male; Mice; Mice, Inbred C57BL; Microdialysis; Motor Activity; Naltrexone; Narcotic Antagonists; Neostriatum; Pyrrolidines; Receptors, Opioid, kappa; Thiazines

2004