Page last updated: 2024-09-04

r 84760 and naloxone

r 84760 has been researched along with naloxone in 1 studies

Compound Research Comparison

Studies
(r 84760)
Trials
(r 84760)
Recent Studies (post-2010)
(r 84760)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
70020,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomyr 84760 (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujibayashi, K; Iizuka, Y; Sakamoto, K; Watanabe, M1

Other Studies

1 other study(ies) available for r 84760 and naloxone

ArticleYear
Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist.
    European journal of pharmacology, 1994, Aug-11, Volume: 261, Issue:1-2

    Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Benzoquinones; Binding, Competitive; Diuretics; Drug Tolerance; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Molecular Sequence Data; Naloxone; Pain; Postural Balance; Pyrrolidines; Rabbits; Receptors, Opioid, kappa; Substance-Related Disorders; Thiazines; Vas Deferens

1994