r 84760 has been researched along with naloxone in 1 studies
Studies (r 84760) | Trials (r 84760) | Recent Studies (post-2010) (r 84760) | Studies (naloxone) | Trials (naloxone) | Recent Studies (post-2010) (naloxone) |
---|---|---|---|---|---|
7 | 0 | 0 | 20,134 | 1,257 | 3,321 |
Protein | Taxonomy | r 84760 (IC50) | naloxone (IC50) |
---|---|---|---|
Cytochrome P450 2D6 | Homo sapiens (human) | 2 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 0.043 | |
Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0219 | |
Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0019 | |
Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0019 | |
Mu-type opioid receptor | Homo sapiens (human) | 0.0397 | |
Delta-type opioid receptor | Homo sapiens (human) | 0.1896 | |
Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.05 | |
Kappa-type opioid receptor | Homo sapiens (human) | 0.0795 | |
Mu-type opioid receptor | Mus musculus (house mouse) | 0.0154 | |
Mu-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0089 | |
Beta-2 adrenergic receptor | Cavia porcellus (domestic guinea pig) | 0.0055 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Fujibayashi, K; Iizuka, Y; Sakamoto, K; Watanabe, M | 1 |
1 other study(ies) available for r 84760 and naloxone
Article | Year |
---|---|
Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist.
Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Benzoquinones; Binding, Competitive; Diuretics; Drug Tolerance; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Molecular Sequence Data; Naloxone; Pain; Postural Balance; Pyrrolidines; Rabbits; Receptors, Opioid, kappa; Substance-Related Disorders; Thiazines; Vas Deferens | 1994 |