r 59022 and r 59949

r 59022 has been researched along with r 59949 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (10.00)18.2507
2000's5 (50.00)29.6817
2010's4 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Baldanzi, G; Bertoni, A; Capello, D; Fresu, LG; Gesu, A; Graziani, A; Massarotti, A; Ruffo, E; Snow, AL; Talmon, M; Tron, GC; Varma, KSS; Velnati, S1
de Chaffoy de Courcelles, D1
Alfranca, A; Aragonés, J; Jones, DR; Landázuri, MO; Martin, S; Mérida, I; San Juan, MA; Vara, A; Vidal, F1
Eppinger, E; Meinhardt, G; Schmidmaier, R1
de Boschero, MG; Giusto, NM; Zulian, SE1
Kawada-Matsuo, M; Li, D; Saito, N; Shibata, Y; Shirai, Y; Yamashita, Y1
Abounader, R; Dominguez, CL; Floyd, DH; Harris, TE; Kefas, BA; Lee, JK; Mullins, GR; Purow, BW; Wilson, GM; Xiao, A; Xin, W; Yacur, MN1
Kunii, N; Liu, K; Mizuno, H; Saga, H; Sakai, H; Sakane, F; Sasaki, S; Sato, M1

Reviews

1 review(s) available for r 59022 and r 59949

ArticleYear
The use of diacylglycerol kinase inhibitors for elucidating the roles of protein kinase C.
    Advances in second messenger and phosphoprotein research, 1990, Volume: 24

    Topics: Animals; Blood Platelets; Diacylglycerol Kinase; Diglycerides; Enzyme Activation; Humans; Neutrophils; Phosphotransferases; Piperidines; Protein Kinase C; Pyrimidinones; Quinazolines; Quinazolinones; Rabbits; Receptors, Cell Surface; Second Messenger Systems; Thiazoles

1990

Other Studies

9 other study(ies) available for r 59022 and r 59949

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Identification of a novel DGKα inhibitor for XLP-1 therapy by virtual screening.
    European journal of medicinal chemistry, 2019, Feb-15, Volume: 164

    Topics: Cell Death; Computer Simulation; Diacylglycerol Kinase; Drug Evaluation, Preclinical; Humans; Lymphoproliferative Disorders; Piperidines; Protein Kinase Inhibitors; Pyrimidinones; Quinazolinones; Ritanserin; Thiazoles

2019
Evidence for the involvement of diacylglycerol kinase in the activation of hypoxia-inducible transcription factor 1 by low oxygen tension.
    The Journal of biological chemistry, 2001, Mar-30, Volume: 276, Issue:13

    Topics: Cell Nucleus; Diacylglycerol Kinase; Diglycerides; DNA; DNA-Binding Proteins; Dose-Response Relationship, Drug; Enzyme Inhibitors; HeLa Cells; Humans; Hypoxia; Hypoxia-Inducible Factor 1; Hypoxia-Inducible Factor 1, alpha Subunit; Immunoblotting; Luciferases; Nuclear Proteins; Oxygen; Phosphatidic Acids; Phospholipids; Piperidines; Plasmids; Pyrimidinones; Quinazolines; Quinazolinones; Recombinant Proteins; Signal Transduction; Thiazoles; Transcription Factors; Transcription, Genetic; Transcriptional Activation; Transfection

2001
Effect of novel modulators of protein kinase C activity upon chemotherapy-induced differentiation and apoptosis in myeloid leukemic cells.
    Anti-cancer drugs, 2002, Volume: 13, Issue:7

    Topics: Antineoplastic Agents; Apoptosis; CD11c Antigen; CD4 Antigens; Cell Cycle; Cell Differentiation; Diacylglycerol Kinase; Enzyme Activators; Enzyme Inhibitors; Farnesol; Flow Cytometry; Genes, fos; Genes, jun; Humans; Immunoblotting; Isoenzymes; Leukemia, Myeloid; Naphthalenes; Oncogene Protein p21(ras); Piperidines; Protein Kinase C; Pyrimidinones; Quinazolines; Quinazolinones; Sulfonamides; Thiazoles; Triazoles; Tumor Cells, Cultured

2002
Insulin action on polyunsaturated phosphatidic acid formation in rat brain: an "in vitro" model with synaptic endings from cerebral cortex and hippocampus.
    Neurochemical research, 2009, Volume: 34, Issue:7

    Topics: Animals; Cerebral Cortex; Chromones; Cyclosporine; Diacylglycerol Kinase; Diglycerides; Genistein; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Insulin; Insulin Antagonists; Morpholines; Okadaic Acid; Phosphatidic Acids; Phosphoprotein Phosphatases; Piperidines; Pyrimidinones; Quinazolinones; Rats; Rats, Wistar; Sodium Fluoride; Synaptosomes; Thiazoles; Vanadates

2009
Streptococcus mutans diacylglycerol kinase homologue: a potential target for anti-caries chemotherapy.
    Journal of medical microbiology, 2011, Volume: 60, Issue:Pt 5

    Topics: Cariostatic Agents; Dental Caries; Diacylglycerol Kinase; Enzyme Inhibitors; Genes, Bacterial; Humans; Hydrogen-Ion Concentration; Mutation; Piperidines; Pyrimidinones; Quinazolinones; Streptococcus mutans; Thiazoles

2011
Diacylglycerol kinase α is a critical signaling node and novel therapeutic target in glioblastoma and other cancers.
    Cancer discovery, 2013, Volume: 3, Issue:7

    Topics: Apoptosis; Brain Neoplasms; Cell Line, Tumor; Diacylglycerol Kinase; Gene Expression Regulation, Neoplastic; Glioblastoma; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Molecular Targeted Therapy; Piperidines; Pyrimidinones; Quinazolinones; RNA, Small Interfering; Thiazoles

2013
Evaluations of the selectivities of the diacylglycerol kinase inhibitors R59022 and R59949 among diacylglycerol kinase isozymes using a new non-radioactive assay method.
    Pharmacology, 2013, Volume: 92, Issue:1-2

    Topics: Animals; Chlorocebus aethiops; COS Cells; Diacylglycerol Kinase; Enzyme Inhibitors; High-Throughput Screening Assays; Isoenzymes; Piperidines; Pyrimidinones; Quinazolinones; Thiazoles

2013