qx-314 and benzocaine

qx-314 has been researched along with benzocaine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19903 (27.27)18.7374
1990's4 (36.36)18.2507
2000's3 (27.27)29.6817
2010's1 (9.09)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ikemoto, Y; Oda, M; Yoshida, A1
Keynes, RD1
Danilo, P; Rosen, MR; Spinelli, W1
Gintant, GA; Hoffman, BF; Naylor, RE1
Quan, C; Wang, GK; Wang, S1
Quan, C; Wang, GK; Wang, SY1
Arledge, JA; Durieux, ME; Hönemann, CW; Sullivan, LM1
Byford, AM; Durieux, ME; Fischer, LG; Hollmann, MW1
de Klaver, M; Durieux, ME; Henle, P; Hollmann, MW; Kamatchi, GL; Ritter, CH1
Ahern, CA; Dougherty, DA; Eastwood, AL; Horn, R1
Ahern, CA; Goodchild, SJ; Lee, S1

Other Studies

11 other study(ies) available for qx-314 and benzocaine

ArticleYear
Blockade by local anaesthetics of the single Ca(2+)-activated K+ channel in rat hippocampal neurones.
    British journal of pharmacology, 1992, Volume: 105, Issue:1

    Topics: Anesthetics, Local; Animals; Benzocaine; Calcium; Female; Hippocampus; In Vitro Techniques; Lidocaine; Male; Neurons; Potassium Channels; Rats; Rats, Inbred Strains

1992
Properties of the sodium gating current in the squid giant axon.
    Annals of the New York Academy of Sciences, 1986, Volume: 479

    Topics: Anesthetics, Local; Animals; Axons; Benzocaine; Ion Channels; Lidocaine; Membrane Potentials; Neural Conduction; Sodium; Tetrodotoxin

1986
Reduction of Vmax by QX-314 and benzocaine in neonatal and adult canine cardiac Purkinje fibers.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Action Potentials; Animals; Animals, Newborn; Benzocaine; Dogs; Heart Conduction System; Kinetics; Lidocaine; Membrane Potentials; Purkinje Fibers

1988
The influence of molecular form of local anesthetic-type antiarrhythmic agents on reduction of the maximum upstroke velocity of canine cardiac Purkinje fibers.
    Circulation research, 1983, Volume: 52, Issue:6

    Topics: Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Benzocaine; Dogs; Heart Conduction System; Ion Channels; Lidocaine; Membrane Potentials; Molecular Conformation; Purkinje Fibers; Sodium; Tocainide

1983
A common local anesthetic receptor for benzocaine and etidocaine in voltage-gated mu1 Na+ channels.
    Pflugers Archiv : European journal of physiology, 1998, Volume: 435, Issue:2

    Topics: Amino Acid Sequence; Anesthetics, Local; Benzocaine; Cell Line; Electric Conductivity; Embryo, Mammalian; Etidocaine; Humans; Kidney; Lidocaine; Molecular Sequence Data; Mutagenesis, Site-Directed; Receptors, Drug; Sodium Channels

1998
Local anesthetic block of batrachotoxin-resistant muscle Na+ channels.
    Molecular pharmacology, 1998, Volume: 54, Issue:2

    Topics: Anesthetics, Local; Batrachotoxins; Benzocaine; Cells, Cultured; Drug Resistance; Etidocaine; Humans; Lidocaine; Muscles; Sodium Channels

1998
Synergistic inhibition of lysophosphatidic acid signaling by charged and uncharged local anesthetics.
    Anesthesia and analgesia, 1999, Volume: 88, Issue:5

    Topics: Anesthetics, Local; Animals; Benzocaine; Chloride Channels; Dose-Response Relationship, Drug; Female; Guanosine 5'-O-(3-Thiotriphosphate); Lidocaine; Lysophospholipids; Protein Kinase C; Signal Transduction; Xenopus

1999
Local anesthetic inhibition of m1 muscarinic acetylcholine signaling.
    Anesthesiology, 2000, Volume: 93, Issue:2

    Topics: Acetylcholine; Anesthetics, Local; Animals; Benzocaine; Binding Sites; Cells, Cultured; CHO Cells; Choline; Cricetinae; Electrophysiology; GTP-Binding Proteins; Lidocaine; Patch-Clamp Techniques; Quinuclidinyl Benzilate; Receptors, Muscarinic; Signal Transduction; Xenopus

2000
Inhibition of m3 muscarinic acetylcholine receptors by local anaesthetics.
    British journal of pharmacology, 2001, Volume: 133, Issue:1

    Topics: Anesthetics, Local; Animals; Benzocaine; CHO Cells; Cricetinae; Female; Heterotrimeric GTP-Binding Proteins; Inhibitory Concentration 50; Lidocaine; Models, Biological; Muscarinic Antagonists; Oocytes; Rats; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Xenopus laevis

2001
Electrostatic contributions of aromatic residues in the local anesthetic receptor of voltage-gated sodium channels.
    Circulation research, 2008, Jan-04, Volume: 102, Issue:1

    Topics: Amino Acids, Aromatic; Anesthetics, Local; Animals; Benzocaine; Binding Sites; Humans; Lidocaine; Muscle Proteins; NAV1.4 Voltage-Gated Sodium Channel; Oocytes; Sodium Channel Blockers; Sodium Channels; Static Electricity; Transfection; Xenopus

2008
Local anesthetic inhibition of a bacterial sodium channel.
    The Journal of general physiology, 2012, Volume: 139, Issue:6

    Topics: Acetanilides; Anesthetics, Local; Bacillus; Benzocaine; Binding Sites; Cell Line, Transformed; Cytoplasm; Eukaryota; HEK293 Cells; Humans; Hydrophobic and Hydrophilic Interactions; Ion Channel Gating; Kinetics; Lidocaine; Piperazines; Ranolazine; Sodium; Sodium Channels

2012