Page last updated: 2024-08-16

quipazine and tropisetron

quipazine has been researched along with tropisetron in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19901 (9.09)18.7374
1990's9 (81.82)18.2507
2000's1 (9.09)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bryce, D; Chalabi, PM; Furman, J; Guarino, KJ; Ives, JL; McLean, S; Nagel, AA; Rosen, T; Roth, RW; Seeger, TF1
Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT1
Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC1
Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG1
Borrelli, G; Budriesi, R; Butini, S; Caccia, S; Cagnotto, A; Campiani, G; Catalanotti, B; Chiarini, A; Coccone, SS; Colovic, M; Fattorusso, C; Fiorini, I; Fracasso, C; Gemma, S; Hamon, M; Ioan, P; Mennini, T; Morelli, E; Nacci, V; Novellino, E; Persico, M; Ros, S1
Cloëz-Tayarani, I; Fillion, G; Harel-Dupas, C1
Smith, DJ; Smith, DL; Williams, GM1
Bouysset, F; Laubie, M; Schmitt, H; Vayssettes-Courchay, C; Verbeuren, TJ1
Perry, DC1
Peroutka, SJ1
Abraham, C; Giesen-Crouse, E; Lacoste, JM; Laubie, M; Malen, C; Morain, P1

Other Studies

11 other study(ies) available for quipazine and tropisetron

ArticleYear
Synthesis, in vitro binding profile, and central nervous system penetrability of the highly potent 5-HT3 receptor antagonist [3H]-4-(2-methoxyphenyl)-2-[4(5)-methyl-5(4)-imidazolylmethyl]thiazole.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:11

    Topics: Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry; Glioma; Imidazoles; Mice; Molecular Structure; Neuroblastoma; Serotonin Antagonists; Thiazoles; Tumor Cells, Cultured

1990
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:12

    Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes

1990
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:6

    Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1990
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
    Journal of medicinal chemistry, 1998, Jan-29, Volume: 41, Issue:3

    Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists

1998
Specific targeting of peripheral serotonin 5-HT(3) receptors. Synthesis, biological investigation, and structure-activity relationships.
    Journal of medicinal chemistry, 2009, Jun-11, Volume: 52, Issue:11

    Topics: Animals; Baroreflex; Chemical Phenomena; Female; Guinea Pigs; Heart; Heart Atria; Male; Mice; Models, Molecular; Myocardium; Pyrroles; Quinoxalines; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin 5-HT3 Receptor Agonists; Structure-Activity Relationship

2009
Inhibition of [3H] gamma-aminobutyric acid release from guinea-pig hippocampal synaptosomes by serotonergic agents.
    Fundamental & clinical pharmacology, 1992, Volume: 6, Issue:8-9

    Topics: Animals; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Methiothepin; Piperazines; Quipazine; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptosomes; Tropisetron

1992
5-HT3 receptors are not involved in the modulation of the K(+)-evoked release of [3H]5-HT from spinal cord synaptosomes of rat.
    Neuropharmacology, 1992, Volume: 31, Issue:8

    Topics: Animals; Biguanides; Bufotenin; Hydroxyindoleacetic Acid; In Vitro Techniques; Indoles; Male; Potassium; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Spinal Cord; Synaptosomes; Tropisetron

1992
The cardiovascular effects of quipazine are mediated by peripheral 5-HT2 and 5-HT3 receptors in anaesthetized rats.
    European journal of pharmacology, 1990, Aug-02, Volume: 184, Issue:1

    Topics: Amidines; Anesthesia; Animals; Blood Pressure; Carotid Body; Denervation; Heart Rate; Hemodynamics; Hexamethonium Compounds; In Vitro Techniques; Indoles; Lung; Male; Myocardium; Piperidines; Prazosin; Pressoreceptors; Propanolamines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Renin-Angiotensin System; Ritanserin; Sympathetic Nervous System; Thiophenes; Tropisetron; Vagotomy

1990
Autoradiography of [3H]quipazine in rodent brain.
    European journal of pharmacology, 1990, Oct-02, Volume: 187, Issue:1

    Topics: Animals; Autoradiography; Brain; Cricetinae; Gerbillinae; Guinea Pigs; In Vitro Techniques; Indoles; Male; Membranes; Mesocricetus; Mice; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Species Specificity; Tropisetron

1990
Species variations in 5-HT3 recognition sites labeled by 3H-quipazine in the central nervous system.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:5

    Topics: Animals; Cattle; Cerebral Cortex; Chickens; Cocaine; Dogs; Guinea Pigs; Humans; Indoles; Mice; Quinolines; Quipazine; Rabbits; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin; Species Specificity; Swine; Tropanes; Tropisetron; Turtles

1988
The antagonist properties of S 11978 on 5HT3 receptors in N1E-115 neuroblastoma cells.
    Fundamental & clinical pharmacology, 1993, Volume: 7, Issue:5

    Topics: Animals; Binding, Competitive; Electrophysiology; Indoles; Kinetics; Mice; Neuroblastoma; Ondansetron; Quipazine; Serotonin Antagonists; Thiophenes; Tritium; Tropisetron; Tumor Cells, Cultured

1993