Page last updated: 2024-08-16

quipazine and piperidines

quipazine has been researched along with piperidines in 42 studies

Research

Studies (42)

TimeframeStudies, this research(%)All Research%
pre-199030 (71.43)18.7374
1990's9 (21.43)18.2507
2000's2 (4.76)29.6817
2010's1 (2.38)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Anzini, M; Cagnotto, A; Campiani, G; Cappelli, A; Skorupska, M; Vomero, S1
Brammer, NT; Charlett, A; Doré, CJ; Fletcher, A; Hudson, S; Minchin, MC; Wann, KT; Wardley-Smith, B1
Eglen, RM; Loury, DN; Michel, AD; Sharif, NA; Stefanich, E; Whiting, RL; Wong, EH1
Bouysset, F; Laubie, M; Schmitt, H; Vayssettes-Courchay, C; Verbeuren, TJ1
Geyer, MA; Tapson, GS; Wing, LL1
Jackson, DA; White, SR1
Bloomquist, WL; Cohen, ML; Fuller, RW; Snoddy, HD1
Amoroso, S; Annunziato, L; Basile, V; Canzoniero, L; Di Renzo, G; Fatatis, A; Taglialatela, M1
Anzini, M; Cagnotto, A; Cappelli, A; Garofalo, A; Vomero, S1
Hurt, SD; Peroutka, SJ; Schmidt, AW1
Raible, LH1
Hewson, G; Hill, RG; Hughes, J; Leighton, GE1
Barrett, JE; Brady, LS1
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL1
Gorzalka, BB; Mendelson, SD3
Godfrey, PP; McClue, SJ; Minchin, MC; Schächter, M; Young, MM1
Hole, DR; Hunter, AJ; Wilson, CA1
Appel, JB; Callahan, PM; Cunningham, KA2
Berendsen, HH; Broekkamp, CL1
Mokler, DJ; Rech, RH; Stoudt, KW1
Dawbarn, D; Long, SK; Pycock, CJ1
Pawłowski, L1
Dandiya, PC; Gurbani, NK; Keshavan, JH1
Shelekhov, SL; Val'dman, AV2
Fuller, RW; Snoddy, HD1
Grahame-Smith, DG; Green, AR; Hammond, M; O'Shaughnessy, K; Schächter, M1
Glennon, RA; Rosecrans, JA; Young, R1
Barbieri, C; Bevilacqua, M; Bigatti, G; Diena, A; Guffanti, A; Norbiato, G; Rauhe, WG; Sala, M; Scorza, D1
Bendotti, C; Borroni, E; Borsini, F; Caccia, S; Invernizzi, R; Mennini, T; Pataccini, R; Samanin, R1
Colpaert, FC; Janssen, PA; Niemegeers, CJ1
Kostowski, W; Puciłowski, O; Płaźnik, A1
Garattini, S; Mennini, T; Samanin, R1
Barrett, RJ; Sanders-Bush, E; Smith, RL1
Angel, I; Garreau, M; Langer, SZ; Prouteau, M; Schoemaker, H1
Fuller, RW; Hemrick-Luecke, SK1
Evans, DC; Hemrick-Luecke, SK1
Kaur, G; Kulkarni, SK1
Lummis, SC; Thompson, AJ1

Other Studies

42 other study(ies) available for quipazine and piperidines

ArticleYear
Synthesis and 5-HT receptors binding studies of some 3-substituted-2-(4-methyl-1-piperazinyl)-4-phenylquinolines.
    Farmaco (Societa chimica italiana : 1989), 1991, Volume: 46, Issue:12

    Topics: Animals; Binding, Competitive; In Vitro Techniques; Ligands; Male; Paroxetine; Piperazines; Piperidines; Quinolones; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists

1991
Exposure to high pressure may produce the 5-HT behavioral syndrome in rats.
    Undersea biomedical research, 1990, Volume: 17, Issue:4

    Topics: 5-Hydroxytryptophan; Animals; Atmospheric Pressure; Behavior, Animal; Brain; Carbidopa; Central Nervous System Diseases; Fenclonine; High Pressure Neurological Syndrome; Hydroxyindoleacetic Acid; Male; Niacinamide; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1990
Characteristics of 5-HT3 binding sites in NG108-15, NCB-20 neuroblastoma cells and rat cerebral cortex using [3H]-quipazine and [3H]-GR65630 binding.
    British journal of pharmacology, 1991, Volume: 102, Issue:4

    Topics: Animals; Binding, Competitive; Cell Line; Cerebral Cortex; Imidazoles; Indoles; Kinetics; Ligands; Mice; Nervous System Neoplasms; Neuroblastoma; Paroxetine; Piperidines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Tumor Cells, Cultured

1991
The cardiovascular effects of quipazine are mediated by peripheral 5-HT2 and 5-HT3 receptors in anaesthetized rats.
    European journal of pharmacology, 1990, Aug-02, Volume: 184, Issue:1

    Topics: Amidines; Anesthesia; Animals; Blood Pressure; Carotid Body; Denervation; Heart Rate; Hemodynamics; Hexamethonium Compounds; In Vitro Techniques; Indoles; Lung; Male; Myocardium; Piperidines; Prazosin; Pressoreceptors; Propanolamines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Renin-Angiotensin System; Ritanserin; Sympathetic Nervous System; Thiophenes; Tropisetron; Vagotomy

1990
5HT-2 mediation of acute behavioral effects of hallucinogens in rats.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Tetrahydronaphthalenes

1990
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes

1990
Lack of a difference between ketanserin and ritanserin in central vs. peripheral serotonin receptor antagonism.
    Life sciences, 1989, Volume: 45, Issue:13

    Topics: Animals; Blood Pressure; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1989
Pharmacological characterization of serotonin receptors involved in the control of prolactin secretion.
    European journal of pharmacology, 1989, Mar-21, Volume: 162, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Fenfluramine; Indoles; Male; Piperidines; Prolactin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Tetrahydronaphthalenes

1989
Synthesis and 5HT-receptors affinity of some 4-phenylquinoline derivatives.
    Farmaco (Societa chimica italiana : 1989), 1989, Volume: 44, Issue:6

    Topics: Animals; Brain; Chemical Phenomena; Chemistry; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Paroxetine; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Synapses

1989
'[3H]quipazine' degradation products label 5-HT uptake sites.
    European journal of pharmacology, 1989, Nov-14, Volume: 171, Issue:1

    Topics: Animals; Chromatography, High Pressure Liquid; In Vitro Techniques; Paroxetine; Piperidines; Quinolines; Quipazine; Radioligand Assay; Rats; Receptors, Serotonin

1989
Inhibitory action of alpha-melanocyte stimulating hormone on lordosis in rats: possible involvement of serotonin.
    Pharmacology, biochemistry, and behavior, 1988, Volume: 30, Issue:1

    Topics: alpha-MSH; Animals; Female; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal

1988
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1988
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri

1985
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1985
Serotonin type 2 antagonists inhibit lordosis behavior in the female rat: reversal with quipazine.
    Life sciences, 1986, Jan-06, Volume: 38, Issue:1

    Topics: Analysis of Variance; Animals; Butyrophenones; Cyproheptadine; Estradiol; Female; Ketanserin; Methiothepin; Piperidines; Pizotyline; Posture; Progesterone; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sexual Behavior, Animal

1986
Serotonergic agonists stimulate inositol lipid metabolism in rabbit platelets.
    Life sciences, 1985, Oct-28, Volume: 37, Issue:17

    Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Piperidines; Quipazine; Rabbits; Receptors, Serotonin; Serotonin

1985
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine

1985
Differentiation between the stimulus effects of l-5-hydroxytryptophan and LSD.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Benserazide; Cues; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains

1985
Serotonin antagonist pirenperone inhibits sexual behavior in the male rat: attenuation by quipazine.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Fenclonine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Serotonin Antagonists; Sexual Behavior, Animal; Tranquilizing Agents

1985
A facilitatory role for serotonin in the sexual behavior of the female rat.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone

1985
Drug-induced penile erections in rats: indications of serotonin1B receptor mediation.
    European journal of pharmacology, 1987, Mar-31, Volume: 135, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Apomorphine; Benserazide; Haloperidol; Male; Nialamide; Penile Erection; Piperidines; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tranquilizing Agents

1987
The 5HT2 antagonist pirenperone reverses disruption of FR-40 by hallucinogenic drugs.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:5

    Topics: Animals; Conditioning, Operant; Hallucinogens; Lisuride; Lysergic Acid Diethylamide; Male; Mescaline; N,N-Dimethyltryptamine; Piperidines; Quipazine; Rats; Rats, Inbred Strains

1985
Increased central 5-hydroxytryptamine receptor mechanisms in rats after chronic neuroleptic treatment.
    British journal of pharmacology, 1981, Volume: 73, Issue:1

    Topics: Animals; Anisoles; Antipsychotic Agents; Behavior, Animal; Brain; Female; Fenfluramine; Piperidines; Quipazine; Rats; Receptors, Dopamine; Receptors, Serotonin; Serotonin

1981
Amitriptyline and femoxetine, but not clomipramine or citalopram, antagonize hyperthermia induced by directly acting 5-hydroxytryptamine-like drugs in heat adapted rats.
    The Journal of pharmacy and pharmacology, 1984, Volume: 36, Issue:3

    Topics: Adaptation, Physiological; Amitriptyline; Animals; Body Temperature; Citalopram; Clomipramine; Dose-Response Relationship, Drug; Hot Temperature; Male; Piperazines; Piperidines; Propylamines; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists

1984
Discriminative stimulus properties of lergotrile.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Animals; Apomorphine; Discrimination Learning; Dose-Response Relationship, Drug; Ergolines; Ergonovine; Haloperidol; Lisuride; Lysergic Acid Diethylamide; Male; Piperidines; Pizotyline; Quipazine; Rats; Rats, Inbred Strains; Sulpiride

1984
Quipazine induced wet dog shake behaviour in rats: mechanism of action.
    Pharmacological research communications, 1980, Volume: 12, Issue:8

    Topics: Animals; Brain Chemistry; Hydroxyindoleacetic Acid; Motor Activity; Norepinephrine; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Serotonin

1980
[Effect of serotoninergic substances on escape behavior in acute stress situations].
    Biulleten' eksperimental'noi biologii i meditsiny, 1983, Volume: 96, Issue:8

    Topics: 5-Hydroxytryptophan; Animals; Antidepressive Agents; Brompheniramine; Cyproheptadine; Escape Reaction; Humans; Male; Piperazines; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Stress, Psychological; Tranquilizing Agents; Trazodone; Zimeldine

1983
[Neurochemical analysis of the mechanism of action of serotoninergic substances on avoidance behavior in situations of acute stress].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 97, Issue:4

    Topics: 5-Hydroxytryptophan; Acute Disease; Animals; Avoidance Learning; Cyproheptadine; Humans; Hydrazines; Male; Piperazines; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Stress, Psychological; Tranquilizing Agents; Zimeldine

1984
Central serotonin antagonist activity of ketanserin.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 46, Issue:1

    Topics: Animals; Brain; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1984
Inhibition of 5-hydroxytryptamine-mediated behaviour by the putative 5-HT2 antagonist pirenperone.
    Neuropharmacology, 1983, Volume: 22, Issue:5

    Topics: 5-Hydroxytryptophan; Animals; Carbidopa; Haloperidol; Male; Methamphetamine; Motor Activity; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Tranylcypromine; Tryptophan

1983
Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists

1983
Serotonergic regulation of cortisol secretion in dogs.
    Endocrinology, 1984, Volume: 115, Issue:2

    Topics: Animals; Dogs; Fenfluramine; Hydrocortisone; Ketanserin; Piperidines; Quipazine; Serotonin; Time Factors

1984
Further studies on the mechanism of serotonin-dependent anorexia in rats.
    Psychopharmacology, 1980, Volume: 68, Issue:1

    Topics: Animals; Anorexia; Brain; Feeding and Eating Disorders; Feeding Behavior; Female; Fenfluramine; Humans; Piperazines; Piperidines; Quipazine; Rats; Serotonin; Serotonin Antagonists; Synaptosomes; Time Factors

1980
A drug discrimination analysis of lysergic acid diethylamide (LSD): in vivo agonist and antagonist effects of purported 5-hydroxytryptamine antagonists and of pirenperone, a LSD-antagonist.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 221, Issue:1

    Topics: Animals; Discrimination, Psychological; Dose-Response Relationship, Drug; Generalization, Stimulus; Lysergic Acid Diethylamide; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists

1982
Effect of stimulation of brain serotonergic system on mouse-killing behavior in rats.
    Physiology & behavior, 1980, Volume: 25, Issue:2

    Topics: Aggression; Animals; Benzofurans; Brain; Electric Stimulation; Humans; Male; Mesencephalon; Mice; Piperidines; Quipazine; Raphe Nuclei; Rats; Receptors, Serotonin; Serotonin

1980
Evidence that it is possible to cause anorexia by increasing release and/or directly stimulating postsynaptic serotonin receptors in the brain.
    Progress in neuro-psychopharmacology, 1980, Volume: 4, Issue:4-5

    Topics: Animals; Anorexia; Appetite Depressants; Brain; Feeding Behavior; Fenfluramine; Piperazines; Piperidines; Quipazine; Rats; Receptors, Serotonin; Serotonin; Synaptosomes

1980
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Brain Mapping; Discrimination Learning; Dose-Response Relationship, Drug; Fluorobenzenes; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Litoxetine: a selective 5-HT uptake inhibitor with concomitant 5-HT3 receptor antagonist and antiemetic properties.
    European journal of pharmacology, 1993, Mar-02, Volume: 232, Issue:2-3

    Topics: Animals; Antiemetics; Binding, Competitive; Cerebral Cortex; Cisplatin; Dose-Response Relationship, Drug; Ferrets; Fluoxetine; Granisetron; Indazoles; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Vomiting

1993
Involvement of 5-HT2A receptors in the elevation of rat serum corticosterone concentrations by quipazine and MK-212.
    European journal of pharmacology, 1996, Sep-12, Volume: 311, Issue:2-3

    Topics: Animals; Corticosterone; Fluorobenzenes; Indoles; Male; Piperidines; Pyrazines; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Urea

1996
Comparison of the potency of MDL 100,907 and SB 242084 in blocking the serotonin (5-HT)(2) receptor agonist-induced increases in rat serum corticosterone concentrations: evidence for 5-HT(2A) receptor mediation of the HPA axis.
    Neuropharmacology, 2002, Volume: 42, Issue:2

    Topics: Aminopyridines; Amphetamines; Animals; Corticosterone; Dose-Response Relationship, Drug; Ethylamines; Fluorobenzenes; Hypothalamo-Hypophyseal System; Indoles; Male; Piperazines; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Evidence for serotonergic modulation of progesterone-induced hyperphagia, depression and algesia in female mice.
    Brain research, 2002, Jul-12, Volume: 943, Issue:2

    Topics: Analgesics; Animals; Antidepressive Agents, Second-Generation; Brain; Depression; Disease Models, Animal; Drug Interactions; Female; Fluoxetine; Hyperphagia; Menstrual Cycle; Mice; Mice, Inbred Strains; Motor Activity; Pain; Pain Measurement; Piperidines; Progesterone; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists

2002
A single channel mutation alters agonist efficacy at 5-HT3A and 5-HT3AB receptors.
    British journal of pharmacology, 2013, Volume: 170, Issue:2

    Topics: Animals; Dopamine; Drug Partial Agonism; Female; Granisetron; HEK293 Cells; Humans; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Quinoxalines; Quipazine; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Agonists; Time Factors; Xenopus laevis

2013