Page last updated: 2024-08-16

quipazine and ketanserin

quipazine has been researched along with ketanserin in 57 studies

Research

Studies (57)

TimeframeStudies, this research(%)All Research%
pre-199023 (40.35)18.7374
1990's22 (38.60)18.2507
2000's10 (17.54)29.6817
2010's1 (1.75)24.3611
2020's1 (1.75)2.80

Authors

AuthorsStudies
Glennon, RA2
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB1
Conklin, DS; Fitzgerald, LW; Hartig, PR; Iyer, G; Kostich, WA; Krause, CM; Largent, BL; Marshall, AP; Patterson, JP; Tran, DP1
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Jacobs, M; McRee, C; Meyer, DC1
Jeffrey, JJ; Rydelek-Fitzgerald, L; Wilcox, BD1
Alhaider, AA; Mustafa, AA1
Bhattacharya, SK; Datla, KP; Mitra, SK1
Hollingsworth, PJ; Smith, CB; Walker, EA; Woods, JH; Yamamoto, T1
Eison, AS; Margraf, RR; Wright, RN; Yocca, FD1
Geyer, MA; Tapson, GS; Wing, LL1
Jackson, DA; White, SR1
Barrett, RJ; Sanders-Bush, E; Smith, RL2
Lorden, JF; Michela, VL; Stratton, SE1
Bloomquist, WL; Cohen, ML; Fuller, RW; Snoddy, HD1
Nanry, KP; Tilson, HA1
Eison, AS; Eison, MS; Gianutsos, G; Yocca, FD1
Hewson, G; Hill, RG; Hughes, J; Leighton, GE1
Barrett, JE; Brady, LS1
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL1
Gorzalka, BB; Mendelson, SD3
Godfrey, PP; McClue, SJ; Minchin, MC; Schächter, M; Young, MM1
Eberle, KM; Lucki, I; Minugh-Purvis, N1
Barrett, JE; Brady, LS; Witkin, JM1
Hole, DR; Hunter, AJ; Wilson, CA1
Appel, JB; Callahan, PM; Cunningham, KA1
Johnson, JH; Kitts, CS1
Männistö, PT; Tuominen, RK1
Adrien, J; Gorea, E1
Brammer, GL; McGuire, MT; Raleigh, MJ1
Johnson, JH; Lenahan, SE; Seibel, HR1
Fuller, RW; Snoddy, HD1
Glennon, RA; Rosecrans, JA; Young, R1
Barbieri, C; Bevilacqua, M; Bigatti, G; Diena, A; Guffanti, A; Norbiato, G; Rauhe, WG; Sala, M; Scorza, D1
Carrillo, AJ; Liu, B; Signs, SA; Wolford, J1
Ageel, AM; Alhaider, AA; Ginawi, OT1
Jeffrey, JJ; Rydelek-Fitzgerald, L; Teitler, M; Wilcox, BD1
Bobadilla, RA; Castillo, C; Castillo, EF; Hong, E; Ibarra, M1
Fiorella, D; Helsley, S; Rabin, RA; Winter, JC1
Carey, JE; Chen, C; Elliott, JM; Flanigan, TP; Kumar, C; McDonald, B; Newberry, NR; Newton, RA; Phipps, SL1
Byrd, LD; Howell, LL; Schama, KF1
Blakeley, JE; Gurguis, GN; Phan, SP1
Buyse, J; Decuypere, E; Herichová, I; Lamosová, D; Zeman, M1
Pulido, M; Wilson, C1
Hashim, A; Lajtha, A; Sershen, H1
Barrett, RJ; Gresch, PJ; Sanders-Bush, E; Smith, RL1
Burke, T; Hensler, JG; Javors, M; Siafaka-Kapadai, A; Sullivan, NR1
Asgari, K; Body, S; Bradshaw, CM; Fone, KC; Rickard, JF; Szabadi, E; Zhang, Z2
Cavalcante-Lima, HR; Cedraz-Mercez, PL; Côrtes, WS; Medeiros, MA; Olivares, EL; Polo, PA; Reis, LC; Reis, RO1
Gerasimenko, IuP; Kozlovskaia, IB; Moshonkina, TR; Pavlova, NV; Tomilovskaia, ES1
de la Fuente Revenga, M; Dukat, M; González-Maeso, J; Hemanth, P; Jaster, AM; Nassehi, N; Shah, UH; Sierra, S1

Reviews

2 review(s) available for quipazine and ketanserin

ArticleYear
Central serotonin receptors as targets for drug research.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:1

    Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin

1987
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
    Journal of medicinal chemistry, 2003, Jul-03, Volume: 46, Issue:14

    Topics: Animals; Humans; Ligands; Receptors, Serotonin; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2003

Other Studies

55 other study(ies) available for quipazine and ketanserin

ArticleYear
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature

1993
High-affinity agonist binding correlates with efficacy (intrinsic activity) at the human serotonin 5-HT2A and 5-HT2C receptors: evidence favoring the ternary complex and two-state models of agonist action.
    Journal of neurochemistry, 1999, Volume: 72, Issue:5

    Topics: Amphetamines; Binding, Competitive; Cell Line; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hydrolysis; Isomerism; Ligands; Models, Biological; Phosphatidylinositols; Receptors, Serotonin; Recombinant Proteins; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone

1999
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 2004, Volume: 370, Issue:2

    Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Role of 5-hydroxytryptamine receptors on luteinizing-hormone-releasing hormone release in the ovariectomized, estradiol-treated rat.
    Brain research bulletin, 1992, Volume: 28, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Estradiol; Female; Gonadotropin-Releasing Hormone; Hypothalamus, Middle; Ketanserin; Ovariectomy; Pindolol; Preoptic Area; Quipazine; Radioimmunoassay; Rats; Receptors, Serotonin; Serotonin Antagonists; Suprachiasmatic Nucleus; Tetrahydronaphthalenes

1992
Regulation of collagenase gene expression by serotonin and progesterone in rat uterine smooth muscle cells.
    The Journal of biological chemistry, 1992, Oct-15, Volume: 267, Issue:29

    Topics: Amphetamines; Animals; Cell Nucleus; Cells, Cultured; Collagenases; DNA Probes; Female; Gene Expression Regulation, Enzymologic; Ketanserin; Kinetics; Muscle, Smooth; Myometrium; Progesterone; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Spiperone; Tetradecanoylphorbol Acetate; Transcription, Genetic; Uterus

1992
Enhancement of imipramine-induced rat brain beta-adrenoreceptor desensitization by subacute co-administration of trazodone, zimelidine, quipazine or 5-hydroxytryptophan.
    Psychopharmacology, 1991, Volume: 103, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Brain Chemistry; Drinking Behavior; Female; Fenclonine; Imipramine; Isoproterenol; Ketanserin; Methysergide; Propranolol; Quipazine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Serotonin Antagonists; Trazodone; Zimeldine

1991
Serotonergic modulation of footshock induced aggression in paired rats.
    Indian journal of experimental biology, 1991, Volume: 29, Issue:7

    Topics: 5-Hydroxytryptophan; Aggression; Agonistic Behavior; Animals; Apomorphine; Citalopram; Clorgyline; Drug Interactions; Electroshock; Female; Fenclonine; Fluoxetine; Foot; Ketanserin; Male; Metergoline; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1991
Discriminative-stimulus effects of quipazine and l-5-hydroxytryptophan in relation to serotonin binding sites in the pigeon.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Binding Sites; Binding, Competitive; Brain; Columbidae; Discrimination Learning; Dose-Response Relationship, Drug; Indoles; Ketanserin; Kinetics; Male; Pyrimidines; Quipazine; Rats; Rats, Inbred Strains; Serotonin; Tritium

1991
8-OH-DPAT and buspirone analogs inhibit the ketanserin-sensitive quipazine-induced head shake response in rats.
    Pharmacology, biochemistry, and behavior, 1990, Volume: 35, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Head; Ketanserin; Male; Naphthalenes; Pindolol; Pyrimidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Stereotyped Behavior; Tetrahydronaphthalenes

1990
5HT-2 mediation of acute behavioral effects of hallucinogens in rats.
    Psychopharmacology, 1990, Volume: 100, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; DOM 2,5-Dimethoxy-4-Methylamphetamine; Dose-Response Relationship, Drug; Hallucinogens; Ketanserin; Male; Mescaline; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Ritanserin; Serotonin; Tetrahydronaphthalenes

1990
Receptor subtypes mediating facilitation by serotonin of excitability of spinal motoneurons.
    Neuropharmacology, 1990, Volume: 29, Issue:9

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; In Vitro Techniques; Injections, Intravenous; Iontophoresis; Ketanserin; Male; Methysergide; Microelectrodes; Motor Neurons; Piperidines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Spinal Cord; Tetrahydronaphthalenes

1990
Adaptation of brain 5HT2 receptors after mianserin treatment: receptor sensitivity, not receptor binding, more accurately correlates with behavior.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2

    Topics: Animals; Brain; Dose-Response Relationship, Drug; Injections, Subcutaneous; Ketanserin; Male; Mianserin; Phosphatidylinositols; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin

1990
Enhanced sensitivity to quipazine in the genetically dystonic rat (dt).
    Pharmacology, biochemistry, and behavior, 1990, Volume: 37, Issue:1

    Topics: Aging; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Dystonia; Ketanserin; Phenotype; Quipazine; Rats; Rats, Mutant Strains; Receptors, Serotonin; Tremor

1990
Lack of a difference between ketanserin and ritanserin in central vs. peripheral serotonin receptor antagonism.
    Life sciences, 1989, Volume: 45, Issue:13

    Topics: Animals; Blood Pressure; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists

1989
The role of 5HT1A receptors in the modulation of the acoustic startle reflex in rats.
    Psychopharmacology, 1989, Volume: 97, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Dose-Response Relationship, Drug; Ketanserin; Male; Metergoline; Methoxydimethyltryptamines; Quipazine; Rats; Rats, Inbred F344; Receptors, Serotonin; Reflex, Startle; Serotonin Antagonists; Tetrahydronaphthalenes

1989
Effects of imipramine and serotonin-2 agonists and antagonists on serotonin-2 and beta-adrenergic receptors following noradrenergic or serotonergic denervation.
    Life sciences, 1989, Volume: 44, Issue:19

    Topics: 5,7-Dihydroxytryptamine; Animals; Cerebral Cortex; Cerebral Ventricles; Fluoxetine; Imipramine; Ketanserin; Kinetics; Male; Neurons; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reference Values; Serotonin; Stereotyped Behavior

1989
Quipazine reduces food intake in the rat by activation of 5-HT2-receptors.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Animals; Diet; Dose-Response Relationship, Drug; Eating; Histamine H2 Antagonists; Imidazoles; Ketanserin; Methysergide; Ondansetron; Pindolol; Piperidines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Ritanserin; Serotonin Antagonists

1988
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri

1985
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:3

    Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium

1985
Serotonin type 2 antagonists inhibit lordosis behavior in the female rat: reversal with quipazine.
    Life sciences, 1986, Jan-06, Volume: 38, Issue:1

    Topics: Analysis of Variance; Animals; Butyrophenones; Cyproheptadine; Estradiol; Female; Ketanserin; Methiothepin; Piperidines; Pizotyline; Posture; Progesterone; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists; Sexual Behavior, Animal

1986
Serotonergic agonists stimulate inositol lipid metabolism in rabbit platelets.
    Life sciences, 1985, Oct-28, Volume: 37, Issue:17

    Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Inositol Phosphates; Ketanserin; Lysergic Acid Diethylamide; Phosphatidylinositols; Piperidines; Quipazine; Rabbits; Receptors, Serotonin; Serotonin

1985
The role of the aural head shake reflex in serotonin-mediated head shaking behavior.
    Psychopharmacology, 1987, Volume: 92, Issue:2

    Topics: Animals; Behavior, Animal; Habituation, Psychophysiologic; Injections, Subcutaneous; Ketanserin; Male; Phenelzine; Quipazine; Rats; Rats, Inbred Strains; Reflex; Serotonin

1987
Antagonism by ketanserin of the behavioral effects of quipazine but not l-5-hydroxytryptophan in squirrel monkeys.
    Psychopharmacology, 1988, Volume: 94, Issue:3

    Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Ketanserin; Male; Methysergide; Quinolines; Quipazine; Saimiri

1988
Studies into the dual effects of serotonergic pharmacological agents on female sexual behaviour in the rat: preliminary evidence that endogenous 5HT is stimulatory.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:1

    Topics: 5-Hydroxytryptophan; Adrenalectomy; Alanine; Animals; Castration; Cinanserin; Female; Ketanserin; Metergoline; Methysergide; Mianserin; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Sexual Behavior, Animal; Zimeldine

1985
Differentiation between the stimulus effects of l-5-hydroxytryptophan and LSD.
    European journal of pharmacology, 1985, Jan-22, Volume: 108, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Benserazide; Cues; Discrimination, Psychological; Ketanserin; Lysergic Acid Diethylamide; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains

1985
Serotonin antagonist pirenperone inhibits sexual behavior in the male rat: attenuation by quipazine.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:4

    Topics: Animals; Dose-Response Relationship, Drug; Fenclonine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Serotonin Antagonists; Sexual Behavior, Animal; Tranquilizing Agents

1985
A facilitatory role for serotonin in the sexual behavior of the female rat.
    Pharmacology, biochemistry, and behavior, 1985, Volume: 22, Issue:6

    Topics: Animals; Castration; Estradiol; Female; Ketanserin; Methysergide; Piperidines; Progesterone; Quipazine; Rats; Rats, Inbred Strains; Receptors, Dopamine; Serotonin; Sexual Behavior, Animal; Spiperone

1985
Serotonergic mediation of a negative feedback effect of estrogen on luteinizing hormone release in ovariectomized rats.
    Endocrinology, 1988, Volume: 123, Issue:5

    Topics: Animals; Estradiol; Estrogens; Feedback; Female; Ketanserin; Luteinizing Hormone; Metergoline; Methysergide; Ovariectomy; Quipazine; Rats; Receptors, Serotonin; Serotonin; Software

1988
Further studies of serotonergic activity in the regulation of the cold stimulated thyrotropin secretion in male rats.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:2

    Topics: Animals; Cold Temperature; Injections, Intraventricular; Ketanserin; Male; Metergoline; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Thyrotropin

1988
Serotonergic regulation of noradrenergic coerulean neurons: electrophysiological evidence for the involvement of 5-HT2 receptors.
    European journal of pharmacology, 1988, Sep-23, Volume: 154, Issue:3

    Topics: Action Potentials; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electrophysiology; Ketanserin; Locus Coeruleus; Male; Neurons; Norepinephrine; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Synapses

1988
Similarity of 5-HT2 receptor sites in dominant and subordinate vervet monkeys.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 27, Issue:4

    Topics: Animals; Binding Sites; Brain; Chlorocebus aethiops; Dominance-Subordination; Ketanserin; Male; Quipazine; Receptors, Serotonin; Social Dominance; Tissue Distribution

1987
Opiate-serotonin synergism stimulating luteinizing hormone release in estrogen-progesterone-primed ovariectomized rats: mediation by serotonin2 receptors.
    Endocrinology, 1987, Volume: 120, Issue:4

    Topics: Animals; Estradiol; Female; Ketanserin; Luteinizing Hormone; Methysergide; Morphine; Ovariectomy; Progesterone; Quinolines; Quipazine; Rats; Receptors, Serotonin; Serotonin

1987
Central serotonin antagonist activity of ketanserin.
    Research communications in chemical pathology and pharmacology, 1984, Volume: 46, Issue:1

    Topics: Animals; Brain; Corticosterone; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists

1984
Antagonism of the effects of the hallucinogen DOM and the purported 5-HT agonist quipazine by 5-HT2 antagonists.
    European journal of pharmacology, 1983, Jul-22, Volume: 91, Issue:2-3

    Topics: Amphetamines; Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Ketanserin; Male; Piperidines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Serotonin Antagonists

1983
Serotonergic regulation of cortisol secretion in dogs.
    Endocrinology, 1984, Volume: 115, Issue:2

    Topics: Animals; Dogs; Fenfluramine; Hydrocortisone; Ketanserin; Piperidines; Quipazine; Serotonin; Time Factors

1984
Neurochemical and behavioral evidence that quipazine-ketanserin discrimination is mediated by serotonin2A receptor.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: Animals; Brain Mapping; Discrimination Learning; Dose-Response Relationship, Drug; Fluorobenzenes; Ketanserin; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Serotonergic involvement in the regulation of prolactin and vasoactive intestinal peptide mRNA expression in the rat anterior pituitary.
    Molecular and cellular endocrinology, 1994, Volume: 105, Issue:2

    Topics: 5-Hydroxytryptophan; alpha-Methyltyrosine; Animals; Blotting, Northern; Bromocriptine; Gene Expression Regulation; Haloperidol; Ketanserin; Male; Methiothepin; Methoxydimethyltryptamines; Methyltyrosines; Pituitary Gland, Anterior; Prolactin; Quipazine; Rats; Rats, Sprague-Dawley; RNA, Messenger; Serotonin; Time Factors; Transcription, Genetic; Vasoactive Intestinal Peptide

1994
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
    Neuropharmacology, 1993, Volume: 32, Issue:12

    Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes

1993
Serotonin-mediated 5-HT2 receptor gene regulation in rat myometrial smooth muscle cells.
    Molecular and cellular endocrinology, 1993, Volume: 92, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Biguanides; Cells, Cultured; Cycloheximide; Female; Gene Expression Regulation; Ketanserin; Medroxyprogesterone Acetate; Myometrium; Piperazines; Quipazine; Rats; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Sulpiride; Transcription, Genetic; Up-Regulation

1993
A comparative study of the effects of some 5-HT1A receptor agonists on the blood pressure of pithed rats.
    Archives of medical research, 1995,Autumn, Volume: 26, Issue:3

    Topics: 5-Methoxytryptamine; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Blood Pressure; Buspirone; Decerebrate State; Ketanserin; Male; Methoxamine; Pindolol; Prazosin; Pyrimidines; Quipazine; Rats; Rats, Wistar; Serotonin Receptor Agonists

1995
5-HT2C receptor-mediated phosphoinositide turnover and the stimulus effects of m-chlorophenylpiperazine.
    Psychopharmacology, 1995, Volume: 122, Issue:3

    Topics: Animals; Choroid Plexus; Conditioning, Operant; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Interactions; Ketanserin; Lysergic Acid Diethylamide; Ondansetron; Phosphatidylinositols; Piperazines; Pyrazines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1995
Characterisation of human 5-hydroxytryptamine2A and 5-hydroxytryptamine2C receptors expressed in the human neuroblastoma cell line SH-SY5Y: comparative stimulation by hallucinogenic drugs.
    Journal of neurochemistry, 1996, Volume: 67, Issue:6

    Topics: Adrenergic alpha-Agonists; Amphetamines; Antiparkinson Agents; Calcium; Choroid Plexus; Electrophysiology; Ergolines; Ergotamine; Frontal Lobe; Hallucinogens; Humans; Hydrolysis; Ketanserin; Lysergic Acid Diethylamide; Mescaline; Methoxydimethyltryptamines; Neuroblastoma; Phosphatidylinositols; Piperazines; Quipazine; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium; Tumor Cells, Cultured

1996
Serotonergic modulation of the discriminative-stimulus effects of cocaine in squirrel monkeys.
    Psychopharmacology, 1997, Volume: 132, Issue:1

    Topics: Animals; Cocaine; Discrimination Learning; Drug Interactions; Ketanserin; Male; Narcotics; Quipazine; Saimiri; Serotonin Agents

1997
Characteristics of agonist displacement of [3H]ketanserin binding to platelet 5-HT2A receptors: implications for psychiatric research.
    Psychiatry research, 1998, Sep-21, Volume: 80, Issue:3

    Topics: Adult; Binding Sites; Female; Humans; Ketanserin; Male; Middle Aged; Platelet Aggregation Inhibitors; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1998
Role of melatonin in the control of growth and growth hormone secretion in poultry.
    Domestic animal endocrinology, 1999, Volume: 17, Issue:2-3

    Topics: Animals; Coturnix; Growth Hormone; Ketanserin; Male; Melatonin; Photoperiod; Quipazine; Radioimmunoassay; Random Allocation; Serotonin Antagonists; Serotonin Receptor Agonists; Thyrotropin-Releasing Hormone

1999
Effects of serotonergic agents on the transport response in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:3

    Topics: Age Factors; Analysis of Variance; Animals; Cinanserin; Female; Growth; Ketanserin; Metergoline; Motor Activity; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Serotonin-mediated striatal dopamine release involves the dopamine uptake site and the serotonin receptor.
    Brain research bulletin, 2000, Volume: 53, Issue:3

    Topics: Animals; Bicuculline; Cocaine; Corpus Striatum; Dizocilpine Maleate; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; Ketanserin; Male; Methiothepin; Mice; Mice, Inbred C57BL; Oxymetazoline; Piperazines; Quinoxalines; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Stimulus generalization by fenfluramine in a quipazine-ketanserin drug discrimination is not dependent on indirect serotonin release.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 72, Issue:1-2

    Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Fenfluramine; Ketanserin; Male; Quipazine; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin

2002
Effect of valproic acid on serotonin-2A receptor signaling in C6 glioma cells.
    Journal of neurochemistry, 2004, Volume: 90, Issue:5

    Topics: Animals; Anticonvulsants; Binding Sites; Cell Line; Dose-Response Relationship, Drug; Glioma; Ketanserin; Mice; Phosphatidylinositols; Quipazine; Receptor, Serotonin, 5-HT2A; Signal Transduction; Time Factors; Tritium; Valproic Acid

2004
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on the discrimination of durations: evidence for the involvement of 5-HT2A but not 5-HT3 receptors.
    Behavioural pharmacology, 2005, Volume: 16, Issue:1

    Topics: Animals; Biguanides; Discrimination Learning; Discrimination, Psychological; Female; Ketanserin; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Tropanes

2005
Effects of quipazine and m-chlorophenylbiguanide (m-CPBG) on temporal differentiation: evidence for the involvement of 5-HT2A but not 5-HT3 receptors in interval timing behaviour.
    Psychopharmacology, 2005, Volume: 181, Issue:2

    Topics: Animals; Biguanides; Conditioning, Operant; Dose-Response Relationship, Drug; Female; Injections, Intraperitoneal; Injections, Subcutaneous; Ketanserin; Psychometrics; Quipazine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin, 5-HT3; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin 5-HT3 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Task Performance and Analysis; Time Perception; Tropanes

2005
Behavioral and neuropharmacological evidence that serotonin crosses the blood-brain barrier in Coturnix japonica (Galliformes; Aves).
    Brazilian journal of biology = Revista brasleira de biologia, 2007, Volume: 67, Issue:1

    Topics: Animals; Blood-Brain Barrier; Coturnix; Dose-Response Relationship, Drug; Ketanserin; Male; Quipazine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sleep; Yawning

2007
[Serotoninergic system morphofunctional aspects in control of postural and locomotion function].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 2012, Volume: 98, Issue:12

    Topics: Animals; Exercise Test; Gait; Hindlimb; Injections, Intraperitoneal; Ketanserin; Locomotion; Male; Posture; Quipazine; Rats; Rats, Sprague-Dawley; Serotonergic Neurons; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Spinal Cord Injuries; Thoracic Vertebrae

2012
Psychedelic-like Properties of Quipazine and Its Structural Analogues in Mice.
    ACS chemical neuroscience, 2021, 03-03, Volume: 12, Issue:5

    Topics: Animals; Hallucinogens; Ketanserin; Mice; Mice, Knockout; Quipazine; Receptor, Serotonin, 5-HT2A; Serotonin

2021