quipazine has been researched along with granisetron in 9 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 8 (88.89) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 1 (11.11) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Bloomquist, W; Cohen, ML; Reid, LR; Robertson, DW; Schenck, K; Wong, DT | 1 |
| Carr, AA; Hibert, MF; Hoffmann, R; Miller, RC | 1 |
| Bourguignon, JJ; Didier, B; Hoffmann, R; Rival, Y; Rybaltchenko, V; Wermuth, CG | 1 |
| Anzini, M; Bruni, G; Cappelli, A; De Benedetti, PG; Doucet, E; Hamon, M; Langer, T; Makovec, F; Mennuni, L; Menziani, MC; Romeo, MR; Vomero, S | 1 |
| Anzini, M; Bruni, G; Canullo, L; Cappelli, A; De Benedetti, PG; Donati, A; Doucet, E; Giorgi, G; Hamon, M; Makovec, F; Mennuni, L; Menziani, MC; Romeo, MR; Vomero, S | 1 |
| Bonhaus, DW; Eglen, RM; Lee, JA; Loury, DN; Wong, EH; Wu, I | 1 |
| Angel, I; Garreau, M; Langer, SZ; Prouteau, M; Schoemaker, H | 1 |
| Barnes, JM; Barnes, NM | 1 |
| Lummis, SC; Thompson, AJ | 1 |
9 other study(ies) available for quipazine and granisetron
| Article | Year |
|---|---|
Synthesis and biochemical evaluation of tritium-labeled 1-methyl-N-(8-methyl-8-azabicyclo[3.2.1]oct-3-yl)-1H-indazole-3-carboxa mide, a useful radioligand for 5HT3 receptors.
Topics: Animals; Cell Membrane; Cerebral Cortex; Guinea Pigs; Heart Rate; Ileum; Indazoles; Male; Methylation; Myocardium; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Structure-Activity Relationship; Tritium; Tropanes | 1990 |
Conformation-activity relationship study of 5-HT3 receptor antagonists and a definition of a model for this receptor site.
Topics: Animals; Binding Sites; Guinea Pigs; Mice; Protein Conformation; Rabbits; Rats; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship | 1990 |
5-HT3 antagonists derived from aminopyridazine-type muscarinic M1 agonists.
Topics: Animals; Brain Stem; Hippocampus; In Vitro Techniques; Models, Molecular; Muscarinic Agonists; Myocardium; Protein Conformation; Pyridazines; Rats; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists | 1998 |
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 1. Mapping the central 5-HT3 receptor binding site by arylpiperazine derivatives.
Topics: Animals; Benzene; Binding Sites; Glioma; Guanidine; Mice; Models, Molecular; Molecular Structure; Neuroblastoma; Phenanthridines; Piperazines; Quinolines; Quipazine; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Tumor Cells, Cultured | 1998 |
Novel potent and selective central 5-HT3 receptor ligands provided with different intrinsic efficacy. 2. Molecular basis of the intrinsic efficacy of arylpiperazine derivatives at the central 5-HT3 receptors.
Topics: Animals; Binding, Competitive; Brain; Cell Line; Granisetron; In Vitro Techniques; Ligands; Male; Mice; Models, Molecular; Piperazines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship | 1999 |
Different densities of 5-HT3 receptors are labeled by [3H]quipazine, [3H]GR 65630 and [3H]granisetron.
Topics: Animals; Binding, Competitive; Cerebral Cortex; Cricetinae; Granisetron; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Neuroblastoma; Quipazine; Rabbits; Rats; Serotonin Antagonists; Tumor Cells, Cultured | 1993 |
Litoxetine: a selective 5-HT uptake inhibitor with concomitant 5-HT3 receptor antagonist and antiemetic properties.
Topics: Animals; Antiemetics; Binding, Competitive; Cerebral Cortex; Cisplatin; Dose-Response Relationship, Drug; Ferrets; Fluoxetine; Granisetron; Indazoles; Male; Piperidines; Quipazine; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Vomiting | 1993 |
Differential binding characteristics of agonists at 5-HT3 receptor recognition sites in NG108-15 neuroblastoma-glioma cells labelled by [3H]-(S)-zacopride and [3H]granisetron.
Topics: Animals; Benzamides; Biguanides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cell Membrane; Glioma; Granisetron; Indazoles; Kinetics; Neuroblastoma; Ondansetron; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 1993 |
A single channel mutation alters agonist efficacy at 5-HT3A and 5-HT3AB receptors.
Topics: Animals; Dopamine; Drug Partial Agonism; Female; Granisetron; HEK293 Cells; Humans; Mutation; Oocytes; Patch-Clamp Techniques; Piperidines; Quinoxalines; Quipazine; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin 5-HT3 Receptor Agonists; Time Factors; Xenopus laevis | 2013 |