quipazine has been researched along with 1-(3-trifluoromethylphenyl)piperazine in 32 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 14 (43.75) | 18.7374 |
1990's | 14 (43.75) | 18.2507 |
2000's | 4 (12.50) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Glennon, RA | 1 |
Glennon, RA; Lyon, RA; McKenney, JD; Slusher, RM; Titeler, M | 1 |
Audia, JE; Baez, M; Cohen, ML; Kursar, JD; Lucaites, VL; Nelson, DL; Nissen, JS; Schenck, KW; Wainscott, DB | 1 |
Abdel-Rahman, AA; Dukat, M; Glennon, RA; Gyermek, L; Ingher, S; Ismaiel, AM; Teitler, M | 1 |
Dupre, A; Egan, C; Grinde, E; Hake, M; Herrick-Davis, K; Roth, BL; Teitler, M | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Cloëz-Tayarani, I; Fillion, G; Harel-Dupas, C | 1 |
Bloomquist, W; Cohen, ML; Robertson, DW; Wong, DT | 1 |
Cloëz, I; Fillion, G; Harel-Dupas, C | 1 |
McKearney, JW | 2 |
Breeding, M; Sanders-Bush, E | 1 |
Cooper, SJ; Neill, JC | 1 |
Barrett, JE; Brady, LS | 1 |
Clineschmidt, BV; Pettibone, DJ; Reiss, DR; Robinson, JL | 1 |
Balestre, MN; Bockaert, J; Cory, RN; Guillon, G; Rouot, B; Sladeczek, F | 1 |
Amedro, J; Brown, L; Smith, D; Williams, G | 1 |
Dinwiddie, WG; Fuller, RW; Lin, TM; Warrick, MW | 1 |
Clemens, JA; Fuller, RW; Hemrick-Luecke, SK; Mason, NR; Snoddy, HD | 1 |
Boddeke, HW; Kalkman, HO; Timmermans, PB; Van Zwieten, PA | 1 |
Cohen, ML; Fuller, RW | 1 |
Clemens, JA; Roush, ME | 1 |
Fuller, RW; Stamm, NB; Yen, TT | 1 |
Audinot, V; Brocco, M; Gobert, A; Millan, MJ; Schreiber, R; Veiga, S | 1 |
Fuller, RW; Hemrick-Luecke, SK | 1 |
Ageel, AM; Alhaider, AA; Ginawi, OT | 1 |
Fiorella, D; Helsley, S; Rabin, RA; Winter, JC | 1 |
Schechter, MD | 1 |
Berg, KA; Clarke, WP; Goldfarb, J; Leff, P; Maayani, S; Scaramellini, C | 1 |
Caldarola-Pastuszka, M; Jackson, A; Price, T; Trevino, A; Uphouse, L; Wolf, A | 1 |
Berg, KA; Clarke, WP; Cropper, JD; Emeson, RB; Niswender, CM; Sanders-Bush, E | 1 |
Adaikan, PG; Hayes, ES | 1 |
1 review(s) available for quipazine and 1-(3-trifluoromethylphenyl)piperazine
Article | Year |
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Central serotonin receptors as targets for drug research.
Topics: Animals; Humans; Receptors, Serotonin; Research Design; Serotonin | 1987 |
31 other study(ies) available for quipazine and 1-(3-trifluoromethylphenyl)piperazine
Article | Year |
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5-HT1 and 5-HT2 binding characteristics of some quipazine analogues.
Topics: Animals; DOM 2,5-Dimethoxy-4-Methylamphetamine; Generalization, Stimulus; In Vitro Techniques; Male; Piperazines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Structure-Activity Relationship | 1986 |
Pharmacological characteristics of the newly cloned rat 5-hydroxytryptamine2F receptor.
Topics: Animals; Binding Sites; Cell Line; Cloning, Molecular; Gastric Fundus; Inositol 1,4,5-Trisphosphate; Male; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Temperature | 1993 |
Structure-activity relationships for the binding of arylpiperazines and arylbiguanides at 5-HT3 serotonin receptors.
Topics: Animals; Biguanides; Heart Rate; Male; Molecular Structure; Muscle Contraction; Piperazines; Rabbits; Rats; Receptors, Serotonin; Reflex; Serotonin Antagonists; Serotonin Receptor Agonists; Structure-Activity Relationship; Urinary Bladder | 1996 |
Agonist high and low affinity state ratios predict drug intrinsic activity and a revised ternary complex mechanism at serotonin 5-HT(2A) and 5-HT(2C) receptors.
Topics: Animals; Cell Line; Computer Simulation; GTP-Binding Proteins; Inositol Phosphates; Kinetics; Phosphatidylinositols; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Recombinant Proteins; Serotonin Receptor Agonists; Signal Transduction; Transfection; Tritium | 2000 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
Inhibition of [3H] gamma-aminobutyric acid release from guinea-pig hippocampal synaptosomes by serotonergic agents.
Topics: Animals; gamma-Aminobutyric Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Indoles; Male; Methiothepin; Piperazines; Quipazine; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptosomes; Tropisetron | 1992 |
mCPP but not TFMPP is an antagonist at cardiac 5HT3 receptors.
Topics: Animals; Cerebral Cortex; Heart; Heart Rate; In Vitro Techniques; Male; Piperazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1992 |
The inhibitory effect of trifluoromethylphenylpiperazine on [3H]acetylcholine release in guinea pig hippocampal synaptosomes is mediated by a 5-hydroxytryptamine1 receptor distinct from 1A, 1B, and 1C subtypes.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Guinea Pigs; Hippocampus; Male; Piperazines; Potassium; Quinoxalines; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Synaptosomes; Tetrahydronaphthalenes | 1991 |
Effects of serotonin agonists on operant behavior in the squirrel monkey: quipazine, MK-212, trifluoromethylphenylpiperazine, and chlorophenylpiperazine.
Topics: Animals; Conditioning, Operant; Male; Piperazines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri; Serotonin Antagonists | 1990 |
Serotonin1c receptor reserve in choroid plexus masks receptor subsensitivity.
Topics: Animals; Binding Sites; Choroid Plexus; Lysergic Acid Diethylamide; Male; Mianserin; Phenoxybenzamine; Piperazines; Quinolines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1990 |
Selective reduction by serotonergic agents of hypertonic saline consumption in rats: evidence for possible 5-HT1C receptor mediation.
Topics: Animals; Dose-Response Relationship, Drug; Drinking Behavior; Fenfluramine; Fluoxetine; Hypertonic Solutions; Indoles; Male; Piperazines; Pyrazines; Quinoxalines; Quipazine; Rats; Receptors, Serotonin; Serotonin | 1989 |
Serotonin-antagonist effects of 1-(1-naphthyl)piperazine on operant behavior of squirrel monkeys.
Topics: Animals; Conditioning, Operant; DOM 2,5-Dimethoxy-4-Methylamphetamine; Electroshock; Female; Food; Male; Piperazines; Quipazine; Reinforcement Schedule; Saimiri; Serotonin Antagonists | 1989 |
Effects of serotonin receptor agonists and antagonists on schedule-controlled behavior of squirrel monkeys.
Topics: 5-Hydroxytryptophan; Animals; Cinanserin; Conditioning, Operant; Cyproheptadine; Electroshock; Female; Ketanserin; Male; Metergoline; Methysergide; Piperazines; Piperidines; Pyrazines; Quipazine; Receptors, Serotonin; Saimiri | 1985 |
Characterization of 5-hydroxytryptamine receptors in rat stomach fundus.
Topics: Animals; Binding, Competitive; Brain Chemistry; Gastric Fundus; In Vitro Techniques; Ketanserin; Male; Muscle Contraction; Piperazines; Piperidines; Propranolol; Pyrazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Tritium | 1985 |
The 5-hydroxytryptamine (5-HT2) receptor stimulates inositol phosphate formation in intact and broken WRK1 cells: determination of occupancy-response relationships for 5-HT agonists.
Topics: 5-Methoxytryptamine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Bufotenin; Cell Line; Dibenzylchlorethamine; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine Triphosphate; Indoles; Inositol Phosphates; Kinetics; Mammary Neoplasms, Experimental; Mathematics; N,N-Dimethyltryptamine; Piperazines; Quipazine; Rats; Receptors, Serotonin; Sugar Phosphates; Tetrahydronaphthalenes; Tryptamines | 1987 |
A pharmacological analysis of the rat spinal cord serotonin (5-HT) autoreceptor.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Ergolines; Male; Piperazines; Potassium; Quipazine; Rats; Receptors, Serotonin; Serotonin; Spinal Cord; Spiperone; Tetrahydronaphthalenes; Tritium | 1988 |
Antidiarrhoeal effects of quipazine and l-(m-trifluoromethylphenyl)piperazine in mice.
Topics: 5-Hydroxytryptophan; Animals; Antidiarrheals; Diarrhea; Mice; Piperazines; Quinolines; Quipazine | 1981 |
Substituted piperazines as central serotonin agonists: comparative specificity of the postsynaptic actions of quipazine and m-trifluoromethylphenylpiperazine.
Topics: Animals; Brain; Brain Chemistry; Corticosterone; Drinking Behavior; Hydroxyindoleacetic Acid; Male; Monoamine Oxidase Inhibitors; Piperazines; Prolactin; Quinolines; Quipazine; Rats; Serotonin; Synapses | 1981 |
Calcium-dependency of the pressor responses to selective 5-hydroxytryptamine receptor agonists in pithed rats.
Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Calcium; Indoles; Methoxydimethyltryptamines; Piperazines; Prazosin; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spinal Cord; Yohimbine | 1983 |
Antagonism of vascular serotonin receptors by m-chlorophenylpiperazine and m-trifluoromethylphenylpiperazine.
Topics: Animals; Depression, Chemical; Jugular Veins; Male; Muscle Contraction; Muscle, Smooth, Vascular; Piperazines; Quipazine; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Serotonin Antagonists | 1983 |
Inhibition of prolactin release by stimulation of presynaptic serotonin autoreceptors.
Topics: Animals; Brain Stem; Depression, Chemical; Male; Methoxydimethyltryptamines; Piperazines; Prolactin; Quipazine; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin | 1982 |
Lowering of blood pressure by direct- and indirect-acting serotonin agonists in spontaneously hypertensive rats.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Fenfluramine; Hypertension; Male; Metergoline; Piperazines; Quinolines; Quipazine; Rats; Time Factors | 1981 |
(1-(2,5-dimethoxy-4 iodophenyl)-2-aminopropane)-induced head-twitches in the rat are mediated by 5-hydroxytryptamine (5-HT) 2A receptors: modulation by novel 5-HT2A/2C antagonists, D1 antagonists and 5-HT1A agonists.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Behavior, Animal; Benzazepines; Dopamine Antagonists; Male; Piperazines; Quipazine; Rats; Rats, Wistar; Receptors, Adrenergic; Receptors, Dopamine D1; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1995 |
Decreased hypothalamic epinephrine concentration by quipazine and other serotonin agonists in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Down-Regulation; Epinephrine; Hypothalamus; Male; Medulla Oblongata; Piperazines; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists | 1995 |
The quipazine- and TFMPP-increased conditioned avoidance response in rats: role of 5HT1C/5-HT2 receptors.
Topics: Animals; Avoidance Learning; Conditioning, Operant; Ketanserin; Male; Mianserin; Nadolol; Pindolol; Piperazines; Prazosin; Quipazine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Reference Values; Serotonin Antagonists; Serotonin Receptor Agonists; Spiperone; Tropanes | 1993 |
5-HT2C receptor-mediated phosphoinositide turnover and the stimulus effects of m-chlorophenylpiperazine.
Topics: Animals; Choroid Plexus; Conditioning, Operant; DOM 2,5-Dimethoxy-4-Methylamphetamine; Drug Interactions; Ketanserin; Lysergic Acid Diethylamide; Ondansetron; Phosphatidylinositols; Piperazines; Pyrazines; Quipazine; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1995 |
Serotonergic mediation of fenfluramine discriminative stimuli in fawn-hooded rats.
Topics: Animals; Discrimination Learning; Dose-Response Relationship, Drug; Fenfluramine; Fluoxetine; Ibogaine; Male; Methoxydimethyltryptamines; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Agents; Serotonin Receptor Agonists | 1997 |
Effector pathway-dependent relative efficacy at serotonin type 2A and 2C receptors: evidence for agonist-directed trafficking of receptor stimulus.
Topics: Animals; Bufotenin; CHO Cells; Cricetinae; Humans; Lysergic Acid Diethylamide; Models, Chemical; Neuropeptides; Phospholipases A; Phospholipases A2; Piperazines; Pituitary Adenylate Cyclase-Activating Polypeptide; Quipazine; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Signal Transduction; Type C Phospholipases | 1998 |
Attenuation of the lordosis-inhibiting effects of 8-OH-DPAT by TFMPP and quipazine.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Estrus; Female; Piperazines; Posture; Quipazine; Rats; Rats, Inbred F344; Serotonin Receptor Agonists; Sexual Behavior, Animal | 1998 |
RNA-editing of the 5-HT(2C) receptor alters agonist-receptor-effector coupling specificity.
Topics: Amphetamines; Animals; Arachidonic Acid; Binding, Competitive; Bufotenin; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Ergolines; Inositol Phosphates; Lysergic Acid Diethylamide; Piperazines; Protein Isoforms; Quipazine; Radioligand Assay; Receptor, Serotonin, 5-HT2C; Receptors, Serotonin; RNA Editing; Serotonin; Serotonin Receptor Agonists; Tritium | 2001 |
Metachlorophenylpiperazine (m-CPP) induced intracavernous pressure responses in anaesthetized rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Anesthesia; Animals; Male; Penile Erection; Penis; Piperazines; Pressure; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Sexual Behavior, Animal | 2002 |