quinuclidines has been researched along with pirenzepine in 37 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 19 (51.35) | 18.7374 |
1990's | 14 (37.84) | 18.2507 |
2000's | 2 (5.41) | 29.6817 |
2010's | 2 (5.41) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bartolini, A; Fantetti, L; Ghelardini, C; Giotti, A; Malcangio, M; Malmberg-Aiello, P | 1 |
Fisher, A; Segal, M | 1 |
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK | 1 |
McLeskey, SW; Wojcik, WJ | 1 |
Dwyer, TM; Farley, JM; Ho, IK; Mohan, PM; Yang, CM | 1 |
Matsumoto, M; Morii, K; Saito, H; Togashi, H; Yoshioka, M | 1 |
Fisher, A; Kawanishi, G; Kobayashi, H; Mizobe, F; Mochida, S | 1 |
Kato, T; Mizobe, F; Xu, M; Yamamoto, T | 1 |
Berstein, G; Haga, T; Ichiyama, A | 1 |
Acosta, CG; Ashe, JH; Yarosh, CA | 1 |
Hsu, CT; Hyman, PE; Kao, HW; Ringer, MJ; Snape, WJ; Tomomasa, T | 1 |
Kawanishi, G; Mizobe, F; Ohgane, N; Ono, S; Saito, Y | 1 |
Adem, A; Nordberg, A; Sabbagh, M | 1 |
Ferkany, JW; Kinnier, WJ; Kirkien-Rzeszotarski, A; McPherson, DW; Noronha-Blob, L; Rzeszotarski, WJ | 1 |
de Boer, T; de Graaf, JS; Tonnaer, JA; van Vugt, MA | 1 |
Katayama, S; Kito, S; Matsubayashi, H; Miyoshi, R | 1 |
Roeske, WR; Watson, M; Yamamura, HI | 2 |
Burke, RE | 1 |
Bloom, JW; Halonen, M; Lawrence, LJ; Rould, E; Seaver, NA; Yamamura, HI | 1 |
Roeske, WR; Venter, JC | 1 |
Luthin, GR; Wolfe, BB | 2 |
Gehlert, DR; Roeske, WR; Wamsley, JK; Yamamura, HI | 1 |
Johnson, PC; Roeske, WR; Wamsley, JK; Watson, M; Yamamura, HI | 1 |
Gabelt, BT; Kaufman, PL; Poyer, JF | 1 |
Doods, HN; van Zwieten, PA | 1 |
Gabelt, BT; Kaufman, PL | 1 |
Ohno, M; Watanabe, S; Yamamoto, T | 1 |
Fuse, Y; Higashida, H; Kishida, H; Noda, M; Yamamoto, K | 1 |
Gibson, RE; Gitler, M; Reba, RC; Schneidau, TA; Zeeberg, B | 1 |
Saito, Y | 1 |
Ikeda, T | 1 |
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S | 1 |
Dai, J; Li, Z; Meltzer, HY; Roseman, AS; Snigdha, S | 1 |
Fujino, T; Kageyama, A; Nozawa, Y; Yamada, S; Yoshida, A | 1 |
Chess-Williams, R; Moro, C; Uchiyama, J | 1 |
1 review(s) available for quinuclidines and pirenzepine
Article | Year |
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Muscarinic receptors and drugs in cardiovascular medicine.
Topics: Bradycardia; Cardiovascular Diseases; Cholinergic Agents; Endothelium, Vascular; Humans; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth, Vascular; Nitric Oxide; Parasympatholytics; Pirenzepine; Quinuclidines; Receptors, Muscarinic; Regression Analysis; Structure-Activity Relationship | 1995 |
36 other study(ies) available for quinuclidines and pirenzepine
Article | Year |
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Role of muscarinic receptor subtypes in central antinociception.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesia; Animals; Male; Mice; Pain Measurement; Pirenzepine; Quinuclidines; Receptors, Muscarinic; Thiophenes | 1992 |
AF102B, a muscarinic M1 receptor agonist, mimics some effects of acetylcholine on neurons of rat hippocampus slices.
Topics: Acetylcholine; Animals; Atropine; Electrophysiology; Hippocampus; In Vitro Techniques; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Receptors, Muscarinic; Thiophenes | 1992 |
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine | 1991 |
Identification of muscarinic receptor subtypes present in cerebellar granule cells: prevention of [3H]propylbenzilyl choline mustard binding with specific antagonists.
Topics: Adenylyl Cyclase Inhibitors; Animals; Atropine; Cell Membrane; Cells, Cultured; Cerebellum; Diamines; Electrophoresis, Polyacrylamide Gel; Parasympatholytics; Pirenzepine; Propylbenzilylcholine Mustard; Quinuclidines; Receptors, Muscarinic; Xanthenes | 1990 |
Down-regulation of muscarinic receptors in the striatum of organophosphate-treated swine.
Topics: Acetylcholinesterase; Animals; Binding Sites; Binding, Competitive; Carbachol; Corpus Striatum; Down-Regulation; Guanylyl Imidodiphosphate; Isoflurophate; Magnesium; Male; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Regression Analysis; Swine | 1990 |
Sympathoexcitatory action of a novel muscarinic receptor agonist, AF102B, and its blockade by pirenzepine.
Topics: Anesthesia; Animals; Blood Pressure; Heart; Heart Rate; In Vitro Techniques; Male; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Sympathomimetics; Thiophenes | 1990 |
Dual synaptic effects of activating M1-muscarinic receptors, in superior cervical ganglia of rabbits.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Animals; Drug Synergism; Electric Stimulation; Evoked Potentials; Ganglia, Sympathetic; In Vitro Techniques; Male; Pirenzepine; Quinuclidines; Rabbits; Receptors, Muscarinic; Synapses; Tubocurarine; Yohimbine | 1988 |
Differential effects of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism in freely moving rats.
Topics: Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes | 1989 |
Effect of the lipid environment on the differential affinity of purified cerebral and atrial muscarinic acetylcholine receptors for pirenzepine.
Topics: Alkylation; Animals; Atrial Function; Brain; Cholesterol Esters; In Vitro Techniques; Membrane Lipids; Phosphatidylcholines; Phosphatidylinositols; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Swine | 1989 |
Modification of nicotinic ganglionic transmission by muscarinic slow postsynaptic potentials in the in vitro rabbit superior cervical ganglion.
Topics: Action Potentials; Animals; Electric Stimulation; Gallamine Triethiodide; Ganglia, Sympathetic; In Vitro Techniques; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Receptors, Nicotinic; Synaptic Transmission | 1988 |
[3H]QNB binding and contraction of rabbit colonic smooth muscle cells.
Topics: Animals; Atropine; Bethanechol; Bethanechol Compounds; Binding, Competitive; Cell Count; Colon; Kinetics; Male; Microbial Collagenase; Muscle Contraction; Muscle, Smooth; Phenethylamines; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Cholinergic | 1987 |
Heterogeneity of muscarinic autoreceptors and heteroreceptors in the rat brain: effects of a novel M1 agonist, AF102B.
Topics: Acetylcholine; Animals; Brain Chemistry; Corpus Striatum; Dopamine; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pirenzepine; Potassium; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes; Thiophenes | 1988 |
Characterization of agonist and antagonist binding to muscarinic cholinergic receptors solubilized from rat cerebral cortex.
Topics: Animals; Atropine; Carbachol; Cerebral Cortex; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1988 |
Affinity and selectivity of the optical isomers of 3-quinuclidinyl benzilate and related muscarinic antagonists.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cattle; Chemical Phenomena; Chemistry; Corpus Striatum; Inositol Phosphates; Male; Muscarine; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship | 1988 |
Differential interactions of muscarinic drugs with binding sites of [3H]pirenzepine and [3H]quinuclidinyl benzilate in rat brain tissue.
Topics: Animals; Binding Sites; Binding, Competitive; Brain Chemistry; Cell Membrane; Male; Parasympatholytics; Parasympathomimetics; Pirenzepine; Protein Binding; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1987 |
Effects of calcium antagonists on muscarinic receptor subtypes in the rat brain.
Topics: Animals; Calcium Channel Blockers; Cerebral Cortex; In Vitro Techniques; Kinetics; Male; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Subcellular Fractions | 1987 |
[3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. I. Characterization and regulation of agonist binding to putative muscarinic subtypes.
Topics: Acetylcholine; Animals; Benzodiazepinones; Buffers; Carbachol; Cerebral Cortex; Guanylyl Imidodiphosphate; In Vitro Techniques; Male; Myocardium; Parasympathomimetics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1986 |
[3H]pirenzepine and (-)-[3H]quinuclidinyl benzilate binding to rat cerebral cortical and cardiac muscarinic cholinergic sites. II. Characterization and regulation of antagonist binding to putative muscarinic subtypes.
Topics: Animals; Benzodiazepinones; Buffers; Cerebral Cortex; Ethylmaleimide; Guanylyl Imidodiphosphate; In Vitro Techniques; Kinetics; Male; Myocardium; Parasympatholytics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1986 |
Gallamine binding to muscarinic M1 and M2 receptors, studied by inhibition of [3H]pirenzepine and [3H]quinuclidinylbenzilate binding to rat brain membranes.
Topics: Alkylation; Animals; Benzodiazepinones; Binding Sites; Binding, Competitive; Brain; Cell Membrane; Cerebral Cortex; Corpus Striatum; Gallamine Triethiodide; Hippocampus; Kinetics; Male; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1986 |
Characterization of high affinity [3H]pirenzepine and (-)-[3H] quinuclidinyl benzilate binding to muscarinic cholinergic receptors in rabbit peripheral lung.
Topics: Animals; Binding, Competitive; Carbachol; Female; Guanylyl Imidodiphosphate; Kinetics; Lung; Male; Myocardium; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Stereoisomerism | 1987 |
The differential loss of [3H]pirenzepine vs [3H] (-) quinuclidinylbenzilate binding to soluble rat brain muscarinic receptors indicates that pirenzepine binds to an allosteric state of the muscarinic receptor.
Topics: Allosteric Site; Animals; Benzodiazepinones; Brain; Drug Stability; Half-Life; Pirenzepine; Protein Conformation; Quinuclidines; Quinuclidinyl Benzilate; Rats; Receptors, Muscarinic | 1984 |
Comparison of [3H]pirenzepine and [3H]quinuclidinylbenzilate binding to muscarinic cholinergic receptors in rat brain.
Topics: Animals; Benzodiazepinones; Brain; Guanosine Triphosphate; In Vitro Techniques; Kinetics; Male; Parasympatholytics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1984 |
Muscarinic antagonist binding site heterogeneity as evidenced by autoradiography after direct labeling with [3H]-QNB and [3H]-pirenzepine.
Topics: Animals; Autoradiography; Benzodiazepinones; Brain; Male; Organ Specificity; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Tritium | 1984 |
Light microscopic autoradiographic localization of [3H]pirenzepine and [3H](-)quinuclidinyl benzilate binding in human stellate ganglia.
Topics: Autoradiography; Benzodiazepinones; Humans; Parasympatholytics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Muscarinic; Stellate Ganglion; Tritium | 1984 |
[3H]Pirenzepine and [3H]quinuclidinyl benzilate binding to brain muscarinic cholinergic receptors. Differences in measured receptor density are not explained by differences in receptor isomerization.
Topics: Animals; Benzodiazepinones; Cerebral Cortex; Isomerism; Kinetics; Male; Mathematics; Models, Neurological; Parasympatholytics; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic | 1984 |
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines | 1994 |
Inhibition of aceclidine-stimulated outflow facility, accommodation and miosis in rhesus monkeys by muscarinic receptor subtype antagonists.
Topics: Accommodation, Ocular; Animals; Aqueous Humor; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Muscarinic Antagonists; Parasympatholytics; Piperidines; Pirenzepine; Pupil; Quinuclidines | 1994 |
Blockade of hippocampal M1 muscarinic receptors impairs working memory performance of rats.
Topics: Animals; Conditioning, Operant; Diamines; Dose-Response Relationship, Drug; Hippocampus; Injections; Male; Memory, Short-Term; Muscarinic Agonists; Muscarinic Antagonists; Parasympatholytics; Parasympathomimetics; Pirenzepine; Psychomotor Performance; Quinuclidines; Rats; Rats, Wistar; Thiophenes | 1994 |
Activation of inward current associated with M-potassium current inhibition in m1-muscarinic receptor-transformed NG108-15 cells by KST-5452, a novel cognition enhancer.
Topics: Acetylcholine; Animals; Benzylidene Compounds; Cell Line, Transformed; Cognition; Electrophysiology; Membrane Potentials; Pirenzepine; Potassium Channels; Quinuclidines; Rats; Receptors, Muscarinic; Tumor Cells, Cultured | 1994 |
Muscarinic receptor selectivities of 3-Quinuclidinyl 8-xanthenecarboxylate (QNX) in rat brain.
Topics: Animals; Brain; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Xanthenes | 1994 |
[Effect of a muscarinic (M1) receptor agonist on sympathetic nerve activity in rats].
Topics: Adrenal Medulla; Animals; Blood Pressure; Dose-Response Relationship, Drug; Electrophysiology; Heart; Heart Rate; Male; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Wistar; Receptors, Muscarinic; Sympathetic Nervous System; Thiophenes | 1993 |
[Functional role of muscarinic M1 receptor for the ganglionic transmission in the rat superior cervical ganglion].
Topics: Animals; Dimethylphenylpiperazinium Iodide; Ganglionic Stimulants; Hexamethonium; Laser-Doppler Flowmetry; Male; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Parasympathomimetics; Pirenzepine; Quinuclidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Nicotinic; Superior Cervical Ganglion; Synaptic Transmission; Thiophenes; Thyroid Gland | 1997 |
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection | 2007 |
Effect of muscarinic receptor agonists xanomeline and sabcomeline on acetylcholine and dopamine efflux in the rat brain; comparison with effects of 4-[3-(4-butylpiperidin-1-yl)-propyl]-7-fluoro-4H-benzo[1,4]oxazin-3-one (AC260584) and N-desmethylclozapine
Topics: Acetylcholine; Animals; Antipsychotic Agents; Benzoxazines; Brain; Clozapine; Dopamine; Drug Synergism; Imines; Male; Nucleus Accumbens; Pirenzepine; Prefrontal Cortex; Pyridines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Risperidone; Thiadiazoles | 2008 |
Loss of muscarinic and purinergic receptors in urinary bladder of rats with hydrochloric acid-induced cystitis.
Topics: Adenosine Triphosphate; Animals; Benzhydryl Compounds; Benzofurans; Cresols; Cystitis; Disease Models, Animal; Down-Regulation; Female; Hydrochloric Acid; Mandelic Acids; N-Methylscopolamine; Organophosphonates; Phenols; Phenylpropanolamine; Pirenzepine; Polycyclic Compounds; Pyridoxal Phosphate; Pyrrolidines; Quinuclidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Receptors, Purinergic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urination; Urodynamics | 2010 |
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium | 2011 |