Page last updated: 2024-08-18

quinuclidines and oxotremorine

quinuclidines has been researched along with oxotremorine in 36 studies

Research

Studies (36)

TimeframeStudies, this research(%)All Research%
pre-199027 (75.00)18.7374
1990's7 (19.44)18.2507
2000's2 (5.56)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bürki, HR; Sayers, AC1
Lamble, AP; Lamble, JW1
Gray, DB; Lane, MA; Sastre, A1
Birdsall, NJ; Burgen, AS; Strange, PG1
Kuhar, MJ; Rommelspacher, H1
Maayani, S; Sokolovsky, M; Treister, G1
Cohen, JJ; Gordon, MA; Wilson, IB1
Dulis, BH; Gordon, MA; Wilson, IB1
Roeske, WR; Rosenberger, LB; Yamamura, HI1
Ehlert, FJ; Kokka, N1
Maayani, S; Rehavi, M; Sokolovsky, M1
Cohen, S; Fisher, A; Gitter, S; Weinstock, M1
Cohen, S; Fisher, A; Gitter, S; Grunfeld, Y; Weinstock, M1
Bhattacharya, SK; Das Gupta, G; Sen, AP; Seth, K; Seth, PK1
Fujise, N; Kawanishi, G; Mizobe, F; Nakahara, N1
Iga, Y; Kawanishi, G; Mizobe, F; Ogane, N; Takada, Y1
Iga, Y; Kawanishi, G; Mizobe, F; Nakahara, N; Saito, Y1
Kato, T; Mizobe, F; Xu, M; Yamamoto, T1
Kawanishi, G; Mizobe, F; Ohgane, N; Ono, S; Saito, Y1
Iga, Y; Kawanishi, G; Mizobe, F; Nakahara, N1
Adem, A; Nordberg, A; Sabbagh, M1
Baker, SP; Marchand, S; Meyer, EM; Morgan, E; Otero, DH1
Bering, B; Müller, WE1
Snyder, SH; Yamamura, HI1
Ehler, FJ; Jenden, DJ; Ringdahl, B1
Binder, HJ; Zimmerman, TW1
Jedrych, Z1
Huger, FP; Smith, CP1
Johnson, LR; Seidel, ER1
Abraham, S; Akerman, E; Akselrod, S; Cohen, S; Fisher, A; Lachman, C; Lass, Y1
Gabelt, BT; Kaufman, PL; Poyer, JF1
Freedman, SB; Patel, S1
Arisawa, H; Iga, Y; Ise, M; Takeshita, Y; Yasuda, H1
Brown, AM; Hunter, AJ; Middlemiss, DN; Watson, JM1
Fujii, T; Kawashima, K1
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S1

Other Studies

36 other study(ies) available for quinuclidines and oxotremorine

ArticleYear
Antiacetylcholine activities of psychoactive drugs: a comparison of the [3H]quinuclidinyl benzilate binding assay with conventional methods.
    The Journal of pharmacy and pharmacology, 1976, Volume: 28, Issue:3

    Topics: Acetylcholine; Animals; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; In Vitro Techniques; Methods; Mice; Oxotremorine; Psychotropic Drugs; Pupil; Quinuclidines; Rats

1976
The effect of miotics on the intraocular pressure of conscious owl monkeys.
    Investigative ophthalmology, 1976, Volume: 15, Issue:10

    Topics: Anesthesia, Local; Animals; Aotus trivirgatus; Carbachol; Dose-Response Relationship, Drug; Haplorhini; Intraocular Pressure; Male; Miotics; Oxotremorine; Parasympathomimetics; Pilocarpine; Quinuclidines; Spiro Compounds; Succinimides; Tonometry, Ocular

1976
Muscarinic cholinergic binding sites in the developing avian heart.
    Developmental biology, 1977, Volume: 55, Issue:1

    Topics: Acetylcholine; Animals; Atropine; Benzyl Compounds; Carbachol; Chick Embryo; Heart; Methacholine Compounds; Microsomes; Myocardium; Nicotine; Oxotremorine; Physostigmine; Quaternary Ammonium Compounds; Quinuclidines; Receptors, Cholinergic; Scopolamine; Snake Venoms; Tubocurarine

1977
Occupancy of muscarinic acetylcholine receptors stimulates a guanylate cyclase in neuroblastoma cells.
    Biochemical Society transactions, 1977, Volume: 5, Issue:1

    Topics: Acetylcholine; Atropine; Carbachol; Cell Line; Cell Membrane; Enzyme Activation; Guanylate Cyclase; Kinetics; Neuroblastoma; Oxotremorine; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1977
Effects of drugs and axotomy on acetylcholine levels in central cholinergic neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 291, Issue:1

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Axons; Benzilates; Hippocampus; Oxotremorine; Parasympathetic Nervous System; Parasympathomimetics; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Septal Nuclei; Septum Pellucidum; Synaptic Transmission

1975
Drugs affecting the cholinergic system in the intact mammalian eye. I. Evaluation of the miotic activity of acetylcholine-like drugs in the mouse eye.
    Investigative ophthalmology, 1975, Volume: 14, Issue:3

    Topics: Acetylcholine; Animals; Arecoline; Carbachol; Guinea Pigs; Hydrogen-Ion Concentration; Miotics; Oxotremorine; Phencyclidine; Pupil; Quinuclidines

1975
Muscarinic cholinergic receptors in murine lymphocytes: demonstration by direct binding.
    Proceedings of the National Academy of Sciences of the United States of America, 1978, Volume: 75, Issue:6

    Topics: Animals; Atropine; Binding, Competitive; Ligands; Lymphocytes; Male; Mice; Oxotremorine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1978
Identification of muscarinic binding sites in human neutrophils by direct binding.
    Molecular pharmacology, 1979, Volume: 15, Issue:1

    Topics: Atropine; Benzilates; Binding, Competitive; Humans; In Vitro Techniques; Kinetics; Neutrophils; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic

1979
The regulation of muscarinic cholinergic receptors by guanine nucleotides in cardiac tissue.
    European journal of pharmacology, 1979, Volume: 56, Issue:1-2

    Topics: Animals; Atropine; Benzilates; Guanine Nucleotides; Guanosine Triphosphate; Guanylyl Imidodiphosphate; Male; Myocardium; Oxotremorine; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic

1979
Decrease in (3H)-quinuclidinyl bezilate binding to the muscarinic cholinergic receptor in the longitudinal muscle of the rat ileum following chronic administration of diisopropylfuorophosphate.
    Proceedings of the Western Pharmacology Society, 1977, Volume: 20

    Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cholinesterases; Depression, Chemical; Ileum; In Vitro Techniques; Isoflurophate; Male; Muscle, Smooth; Myocardium; Oxotremorine; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Time Factors

1977
Enzymatic resolution and cholinergic properties of (+/-)3-quinuclidinol derivatives.
    Life sciences, 1977, Nov-01, Volume: 21, Issue:9

    Topics: Animals; Brain; Butyrylcholinesterase; Cholinesterases; Dose-Response Relationship, Drug; Guinea Pigs; Horses; Ileum; Kinetics; Male; Oxotremorine; Quinuclidines; Radioligand Assay; Rats; Receptors, Muscarinic; Reflex, Abnormal; Stereoisomerism; Structure-Activity Relationship

1977
A new probe for heterogeneity in muscarinic receptors: 2-methyl-spiro-(1, 3-dioxolane-4, 3')-quinuclidine.
    European journal of pharmacology, 1976, Volume: 37, Issue:2

    Topics: Animals; Blood Pressure; Cricetinae; Depression, Chemical; Ganglia, Spinal; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Mydriatics; Oxotremorine; Parasympathomimetics; Physostigmine; Quinuclidines; Receptors, Cholinergic; Salivation; Spiro Compounds; Tremor

1976
A study of muscarinic receptor heterogeneity with weak antagonists.
    European journal of pharmacology, 1976, Volume: 38, Issue:1

    Topics: Animals; Cats; Cholinesterase Inhibitors; Ganglia, Spinal; Ganglionic Stimulants; Guinea Pigs; Ileum; In Vitro Techniques; Mice; Oxotremorine; Parasympatholytics; Parasympathomimetics; Quinuclidines; Receptors, Cholinergic; Structure-Activity Relationship

1976
Central muscarinic receptor subtypes and carrageenin-induced paw oedema in rats.
    Research in experimental medicine. Zeitschrift fur die gesamte experimentelle Medizin einschliesslich experimenteller Chirurgie, 1991, Volume: 191, Issue:1

    Topics: Animals; Arecoline; Carbachol; Carrageenan; Cerebellum; Corpus Striatum; Edema; Female; Foot; Gallamine Triethiodide; Inflammation; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine

1991
Central muscarinic activities of an M1-selective agonist: preferential effect on reversal of amnesia.
    Brain research, 1990, Jan-15, Volume: 507, Issue:1

    Topics: Animals; Avoidance Learning; Hypothermia; Male; Memory; Mice; Oxotremorine; Quinuclidines; Receptors, Muscarinic; Thiophenes

1990
Effects of a M1 muscarinic receptor agonist on the central cholinergic system, evaluated by brain microdialysis.
    Neuroscience letters, 1990, Jun-22, Volume: 114, Issue:1

    Topics: Acetylcholine; Animals; Brain; Cerebral Cortex; Corpus Striatum; Dialysis; Hippocampus; Kinetics; Male; Oxotremorine; Parasympathomimetics; Quinuclidines; Rats; Rats, Inbred Strains; Scopolamine; Thiophenes; Time Factors

1990
Beneficial effects of FKS-508 (AF102B), a selective M1 agonist, on the impaired working memory in AF64A-treated rats.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:4

    Topics: Animals; Aziridines; Cerebral Cortex; Choline; Choline O-Acetyltransferase; Hippocampus; Learning; Male; Memory; Neuromuscular Blocking Agents; Oxotremorine; Parasympathomimetics; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes

1989
Differential effects of M1- and M2-muscarinic drugs on striatal dopamine release and metabolism in freely moving rats.
    Brain research, 1989, Aug-28, Volume: 495, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Male; Oxotremorine; Pirenzepine; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Thiophenes

1989
Heterogeneity of muscarinic autoreceptors and heteroreceptors in the rat brain: effects of a novel M1 agonist, AF102B.
    European journal of pharmacology, 1988, Oct-11, Volume: 155, Issue:1-2

    Topics: Acetylcholine; Animals; Brain Chemistry; Corpus Striatum; Dopamine; Hippocampus; In Vitro Techniques; Male; Oxotremorine; Parasympathomimetics; Pirenzepine; Potassium; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Synaptosomes; Thiophenes

1988
Amelioration of experimental amnesia (passive avoidance failure) in rodents by the selective M1 agonist AF102B.
    Japanese journal of pharmacology, 1988, Volume: 48, Issue:4

    Topics: Amnesia; Animals; Arecoline; Aziridines; Choline; Male; Memory; Mice; Mice, Inbred Strains; Oxotremorine; Parasympathomimetics; Quinuclidines; Retention, Psychology; Scopolamine; Thiophenes

1988
Characterization of agonist and antagonist binding to muscarinic cholinergic receptors solubilized from rat cerebral cortex.
    Journal of neural transmission, 1988, Volume: 72, Issue:1

    Topics: Animals; Atropine; Carbachol; Cerebral Cortex; In Vitro Techniques; Male; Oxotremorine; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic

1988
Effects of acetylethylcholine mustard on [3H]quinuclidinyl benzilate binding and acetylcholine release in rat brain synaptosomes.
    Journal of neurochemistry, 1987, Volume: 48, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Brain; Dose-Response Relationship, Drug; Hemicholinium 3; Kinetics; Male; Oxotremorine; Potassium; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Synaptosomes

1987
Stereospecific 3H-QNB binding to human erythrocyte membranes associated with muscarinic cholinergic receptors.
    Journal of neural transmission, 1987, Volume: 68, Issue:1-2

    Topics: Adult; Aging; Animals; Atropine; Brain; Carbachol; Erythrocyte Membrane; Female; Guanylyl Imidodiphosphate; Humans; In Vitro Techniques; Male; Middle Aged; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Stereoisomerism

1987
Muscarinic cholinergic binding in rat brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1974, Volume: 71, Issue:5

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Benzilates; Binding Sites; Binding, Competitive; Brain; Brompheniramine; Carbachol; Chlorpheniramine; Hydrogen-Ion Concentration; In Vitro Techniques; Kinetics; Male; Methacholine Compounds; Microsomes; Mitochondria; Oxotremorine; Pilocarpine; Quaternary Ammonium Compounds; Quinuclidines; Rats; Receptors, Cholinergic; Scopolamine; Temperature; Time Factors; Tritium

1974
Muscarinic activity and receptor binding of the enantiomers of aceclidine and its methiodide.
    Molecular pharmacology, 1982, Volume: 21, Issue:3

    Topics: Analgesics; Animals; Body Temperature; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Mice; Muscle Contraction; Muscle, Smooth; Oxotremorine; Parasympathomimetics; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic; Stereoisomerism

1982
Muscarinic receptors on rat isolated colonic epithelial cells. A correlation between inhibition of [3H]quinuclidinyl benzilate binding and alteration in ion transport.
    Gastroenterology, 1982, Volume: 83, Issue:6

    Topics: Animals; Bethanechol; Bethanechol Compounds; Binding, Competitive; Colon; Dimethylphenylpiperazinium Iodide; Electrolytes; Electrophysiology; Epithelium; In Vitro Techniques; Oxotremorine; Parasympatholytics; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Muscarinic

1982
Cholinolytic activity of 3-hydroxyquinuclidyl-1-phenyl-1-cyclohexyl-1-carboxylate hydrochloride (ANC-821).
    Polish journal of pharmacology and pharmacy, 1983, Volume: 35, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Bronchi; Electrocardiography; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Rats; Rats, Inbred Strains

1983
Effect of zinc on [3H]-QNB displacement by cholinergic agonists and antagonists.
    Biochemical pharmacology, 1983, Jan-15, Volume: 32, Issue:2

    Topics: Acetylcholine; Animals; Arecoline; Atropine; Binding, Competitive; Male; Oxotremorine; Parasympatholytics; Parasympathomimetics; Physostigmine; Pilocarpine; Quinuclidines; Quinuclidinyl Benzilate; Rats; Zinc

1983
Contraction and [3H]QNB binding in collagenase isolated fundic smooth muscle cells.
    The American journal of physiology, 1983, Volume: 245, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Guinea Pigs; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Ouabain; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Stomach

1983
Does rigidity in structure of muscarinic agonists and antagonists reflect drug specificity?
    Monographs in neural sciences, 1980, Volume: 7

    Topics: Acetylcholine; Animals; Behavior, Animal; Biological Assay; Dogs; Guinea Pigs; Male; Mice; Molecular Conformation; Oxotremorine; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic; Structure-Activity Relationship

1980
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
    Experimental eye research, 1994, Volume: 59, Issue:6

    Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines

1994
The muscarinic receptor agonist L-658,903 modulates the in vivo accumulation of inositol monophosphates in mouse brain.
    European journal of pharmacology, 1994, May-17, Volume: 267, Issue:3

    Topics: Animals; Binding Sites; Brain; Dose-Response Relationship, Drug; In Vitro Techniques; Inositol Phosphates; Lithium Chloride; Male; Mice; N-Methylscopolamine; Oxadiazoles; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Receptors, Muscarinic; Scopolamine; Scopolamine Derivatives

1994
Modulation of rhythmical slow activity, long-term potentiation and memory by muscarinic receptor agonists.
    European journal of pharmacology, 1996, Jul-11, Volume: 308, Issue:1

    Topics: Administration, Oral; Animals; Avoidance Learning; Dose-Response Relationship, Drug; Electric Stimulation; Electroencephalography; Hippocampus; Long-Term Potentiation; Male; Memory; Mice; Mice, Inbred Strains; Muscarinic Agonists; Oxotremorine; Quinuclidines; Rats; Rats, Wistar; Scopolamine; Synaptic Transmission; Theta Rhythm; Thiophenes

1996
In vitro characterisation of the muscarinic receptor partial agonist, sabcomeline, in rat cortical and heart membranes.
    European journal of pharmacology, 1999, Apr-01, Volume: 370, Issue:1

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cell Membrane; Cells, Cultured; Cerebral Cortex; Drug Interactions; Heart; Imines; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth, Vascular; Myocardium; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Radioligand Assay; Rats; Rats, Sprague-Dawley

1999
YM905, a novel M3 antagonist, inhibits Ca2+ signaling and c-fos gene expression mediated via muscarinic receptors in human T cells.
    General pharmacology, 2000, Volume: 35, Issue:2

    Topics: Calcium Signaling; Cells, Cultured; Genes, fos; Humans; Isoquinolines; Muscarinic Antagonists; Oxotremorine; Quinuclidines; Receptor, Muscarinic M3; Receptors, Muscarinic; RNA, Messenger; Solifenacin Succinate; T-Lymphocytes; Tetrahydroisoquinolines

2000
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:3

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection

2007