quinpirole has been researched along with clozapine in 51 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 4 (7.84) | 18.7374 |
1990's | 20 (39.22) | 18.2507 |
2000's | 23 (45.10) | 29.6817 |
2010's | 4 (7.84) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Andrieux, M; Besançon, R; Giros, B; Martres, MP; Pilon, C; Schwartz, JC; Sokoloff, P | 1 |
Bouthenet, ML; Giros, B; Martres, MP; Schwartz, JC; Sokoloff, P | 1 |
Gmeiner, P; Hübner, H; Kraxner, J | 1 |
Gmeiner, P; Hübner, H; Löber, S; Utz, W | 1 |
Einsiedel, J; Gmeiner, P; Hübner, H | 2 |
Aboul-Fadl, T; Gmeiner, P; Hübner, H; Löber, S | 1 |
Bergauer, M; Gmeiner, P; Hübner, H | 1 |
Benwell, K; Bickerdike, M; Kennett, G; Knight, AR; Misra, A; Quirk, K; Revell, D | 1 |
Allouchi, H; Argiolas, A; El Hakmaoui, A; Enguehard-Gueiffier, C; Gmeiner, P; Gueiffier, A; Hübner, H; Melis, MR | 1 |
Cohen, AI; Harmon, S; O'Malley, KL; Todd, RD | 1 |
Artz, MT; Cools, AR; Ellenbroek, BA | 1 |
Bakhtiar, R; Bull, DR; Sheehan, MJ | 1 |
Altar, CA; Jiang, LH; Kasser, RJ; Wang, RY | 1 |
Breese, GA; Criswell, HE; Mueller, RA | 1 |
Adamovage, LA; Kreamer, LD; Salama, AI; Saller, CF | 1 |
Ashby, CR; Hitzemann, R; Rubinstein, JE; Wang, RY | 1 |
Hu, XT; Wang, RY | 1 |
Bengtsson, A; Jackson, DM; Malmberg, A; Mohell, N | 1 |
Chio, CL; Drong, RF; Gill, GS; Huff, RM; Riley, DT; Slightom, JL | 1 |
Artigas, F; Ferré, S | 1 |
Bernard, A; Cavegn, C; Chabert, C; Mills, A | 1 |
Ahlenius, S; Karlsson, T; Salmi, P | 1 |
Nowak, JZ; Zawilska, JB | 1 |
Ellerbrock, BR; Sethy, VH; Wu, H | 1 |
Brotchie, J; Fox, S | 1 |
Obuchowicz, E | 1 |
Griffon, N; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P | 1 |
Derbiszewska, T; Nowak, JZ; Zawilska, JB | 1 |
Catalano, M; Civelli, O; Hartman, DS; Henningsen, R; Nobile, M; Smeraldi, E; Zenner, MT | 1 |
Ahlenius, S; Oerther, S | 1 |
Adachi, K; Cools, AR; Hasegawa, M; Hirose, N; Ikeda, H; Koshikawa, N; Sato, M | 1 |
Kulkarni, SK; Ninan, I | 1 |
Jaliffa, CO; Lacoste, FF; Llomovatte, DW; Rosenstein, RE; Sarmiento, MI | 1 |
Alper, RH; Gilliland, SL; Levant, B | 1 |
Armogida, M; Chiacchio, S; Colzi, A; Corsini, GU; DeMontis, MG; Maggio, R; Scarselli, M | 1 |
Hillefors, M; von Euler, G | 1 |
Kaur, G; Kulkarni, SK | 1 |
Arca, A; Casu, MA; Devoto, P; Flore, G; Gessa, GL; Pani, L; Pira, L; Vacca, G | 1 |
Jaliffa, CO; Keller Sarmiento, MI; Minces, L; Rosenstein, RE; Sacca, GB; Sáenz, DA | 1 |
Dong, XY; Duan, LP; Lin, SR; Yang, XL; Zhou, J | 1 |
Aceves, J; Gutiérrez, R; Romo-Parra, H | 1 |
Katsuragi, T; Kita, S; Morishita, H; Sakata, N; Shibata, K | 1 |
Alimohamad, H; Mouyal, J; Rajakumar, N; Rushlow, WJ; Sutton, L | 1 |
Cole, JC; Field, M; Goudie, AJ; Sumnall, HR | 1 |
Amato, D; Borsini, F; Nencini, P; Stasi, MA | 1 |
Li, M; Zhao, C | 2 |
Borsini, F; De Carolis, L; Nencini, P; Serlupi-Crescenzi, O; Stasi, MA | 1 |
Bekker, A; Chen, X; Fan, Q; Fu, R; Li, J; Mei, Q; Shiwalkar, N; Ye, JH; Zuo, W | 1 |
Cao, T; Chen, J; Jiang, Y; Waddington, JL; Wang, C; Wang, P; Zhen, X | 1 |
51 other study(ies) available for quinpirole and clozapine
Article | Year |
---|---|
Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor.
Topics: Animals; Chlorides; CHO Cells; Cricetinae; Dopamine; Dopamine Agents; Dopamine Antagonists; Guanylyl Imidodiphosphate; Humans; Lithium; Lithium Chloride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sodium Chloride; Sulpiride; Transfection | 1992 |
Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics.
Topics: Amino Acid Sequence; Animals; Antipsychotic Agents; Base Sequence; Brain Chemistry; Cell Line; Cloning, Molecular; Cricetinae; DNA; DNA Restriction Enzymes; Dopamine; Guanylyl Imidodiphosphate; Molecular Sequence Data; Nucleic Acid Hybridization; Polymerase Chain Reaction; Rats; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D3; RNA, Messenger; Sequence Homology, Nucleic Acid; Tissue Distribution | 1990 |
Cyanoindole derivatives as highly selective dopamine D(4) receptor partial agonists: solid-phase synthesis, binding assays, and functional experiments.
Topics: Animals; Cell Line; Central Nervous System Agents; Corpus Striatum; Cricetinae; Dopamine Agonists; Humans; In Vitro Techniques; Indoles; Ligands; Mitogens; Piperazines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Structure-Activity Relationship; Thymidine | 2000 |
Rationally based efficacy tuning of selective dopamine d4 receptor ligands leading to the complete antagonist 2-[4-(4-chlorophenyl)piperazin-1-ylmethyl]pyrazolo[1,5-a]pyridine (FAUC 213).
Topics: Animals; Binding, Competitive; Cattle; CHO Cells; Corpus Striatum; Cricetinae; Dopamine Antagonists; Humans; In Vitro Techniques; Ligands; Mitogens; Models, Molecular; Piperazines; Pyrazoles; Pyridines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D4; Stereoisomerism; Structure-Activity Relationship | 2001 |
Benzamide bioisosteres incorporating dihydroheteroazole substructures: EPC synthesis and SAR leading to a selective dopamine D4 receptor partial agonist (FAUC 179).
Topics: Animals; Biochemistry; Cattle; CHO Cells; Clozapine; Cricetinae; Cysteine; Dopamine Antagonists; Drug Design; Humans; In Vitro Techniques; Indoles; Magnetic Resonance Spectroscopy; Molecular Structure; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Serine; Spiperone; Stereoisomerism; Structure-Activity Relationship; Threonine | 2001 |
Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacy.
Topics: Dopamine Agonists; Humans; Ligands; Protein Binding; Pyrazoles; Pyridines; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Structure-Activity Relationship | 2002 |
2,4-Disubstituted pyrroles: synthesis, traceless linking and pharmacological investigations leading to the dopamine D4 receptor partial agonist FAUC 356.
Topics: Animals; Binding Sites; Cattle; CHO Cells; Cloning, Molecular; Cricetinae; Humans; Piperazines; Protein Binding; Pyrroles; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Serotonin; Structure-Activity Relationship; Substrate Specificity; Swine | 2002 |
Cyclic amidines as benzamide bioisosteres: EPC synthesis and SAR studies leading to the selective dopamine D4 receptor agonist FAUC 312.
Topics: Amidines; Animals; Benzamides; Cattle; CHO Cells; Clozapine; Cricetinae; Cyclization; Humans; Kinetics; Ligands; Mitogens; Mitosis; Piperazines; Pyrimidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Stereoisomerism; Structure-Activity Relationship | 2003 |
Pharmacological characterisation of the agonist radioligand binding site of 5-HT(2A), 5-HT(2B) and 5-HT(2C) receptors.
Topics: Binding Sites; Binding, Competitive; Cell Line; Humans; Radioligand Assay; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2B; Receptor, Serotonin, 5-HT2C; Recombinant Proteins; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT2 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2004 |
2-[(4-phenylpiperazin-1-yl)methyl]imidazo(di)azines as selective D4-ligands. Induction of penile erection by 2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine (PIP3EA), a potent and selective D4 partial agonist.
Topics: Animals; Cattle; CHO Cells; Cricetinae; Cricetulus; Erectile Dysfunction; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Imidazoles; Ligands; Male; Mitosis; Penile Erection; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Rats; Receptors, Dopamine D4; Structure-Activity Relationship | 2006 |
Photoreceptors of mouse retinas possess D4 receptors coupled to adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Benzamides; Clozapine; Cyclic AMP; Ergolines; Gene Expression; In Situ Hybridization; Mice; Mice, Inbred C57BL; Mice, Mutant Strains; Molecular Sequence Data; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Quinpirole; Receptors, Dopamine; Retina; RNA, Messenger; Spiperone | 1992 |
The involvement of dopamine D1 and D2 receptors in the effects of the classical neuroleptic haloperidol and the atypical neuroleptic clozapine.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Clozapine; Dopamine Agents; Dopamine Antagonists; Drug Interactions; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1991 |
Characterization of dopamine autoreceptors in the amygdala: a fast cyclic voltammetric study in vitro.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Amygdala; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Dopamine; Electric Stimulation; Ergolines; Male; Metoclopramide; Neurotransmitter Uptake Inhibitors; Nialamide; Piperazines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Secretory Rate; Sulpiride | 1991 |
One year of continuous treatment with haloperidol or clozapine fails to induce a hypersensitive response of caudate putamen neurons to dopamine D1 and D2 receptor agonists.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Administration, Oral; Animals; Clozapine; Dibenzazepines; Dopamine Agents; Drug Interactions; Ergolines; Haloperidol; Male; Neurons; Putamen; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine | 1990 |
Clozapine antagonism of D-1 and D-2 dopamine receptor-mediated behaviors.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Appetite Depressants; Behavior, Animal; Benzazepines; Clozapine; Dibenzazepines; Ergolines; Female; Hydroxydopamines; Motor Activity; Oxidopamine; Pregnancy; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Cholinergic; Receptors, Dopamine; Receptors, Serotonin | 1989 |
Dopamine receptor occupancy in vivo: measurement using N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ).
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clozapine; Corpus Striatum; Ergolines; Haloperidol; Male; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1989 |
One year treatment with haloperidol or clozapine fails to alter neostriatal D1- and D2-dopamine receptor sensitivity in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Colforsin; Corpus Striatum; Cyclic AMP; Dibenzazepines; Drug Synergism; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1989 |
Haloperidol and clozapine: differential effects on the sensitivity of caudate-putamen neurons to dopamine agonists and cholecystokinin following one month continuous treatment.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Animals; Benzazepines; Cholecystokinin; Clozapine; Corpus Striatum; Dibenzazepines; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Sincalide | 1989 |
Why does clozapine stimulate the motor activity of reserpine-pretreated rats when combined with a dopamine D1 receptor agonist?
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; alpha-Methyltyrosine; Animals; Antipsychotic Agents; Clozapine; Dopamine Antagonists; Drug Therapy, Combination; Enzyme Inhibitors; Ergolines; Male; Methyltyrosines; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Reserpine; Stimulation, Chemical; Tyrosine 3-Monooxygenase | 1995 |
D4 dopamine receptor-mediated signaling events determined in transfected Chinese hamster ovary cells.
Topics: Amiloride; Animals; Arachidonic Acid; Base Sequence; Butaclamol; CHO Cells; Cloning, Molecular; Clozapine; Cricetinae; Cyclic AMP; DNA; Dopamine; Dopamine Antagonists; Ergolines; Genes, Synthetic; Haloperidol; Humans; Kinetics; Molecular Sequence Data; Pertussis Toxin; Protein Kinase C; Quinpirole; Raclopride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Signal Transduction; Sodium-Hydrogen Exchangers; Transfection; Virulence Factors, Bordetella | 1994 |
Clozapine decreases serotonin extracellular levels in the nucleus accumbens by a dopamine receptor-independent mechanism.
Topics: Animals; Clozapine; Dopamine; Dopamine Agonists; Ergolines; Haloperidol; Microdialysis; Nucleus Accumbens; Quinpirole; Raclopride; Rats; Receptors, Dopamine; Salicylamides; Serotonin; Time Factors | 1995 |
Characterization of the functional activity of dopamine ligands at human recombinant dopamine D4 receptors.
Topics: Animals; Cell Line; Clozapine; DNA; Dopamine; Dopamine Agents; Ergolines; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Humans; Ligands; Moths; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone; Sulfur Radioisotopes; Tritium | 1994 |
Antagonism by SCH 23390 of clozapine-induced hypothermia in the rat.
Topics: Amphetamines; Animals; Benzazepines; Body Temperature; Body Temperature Regulation; Chromans; Clonidine; Clozapine; Dopamine Agents; Dopamine D2 Receptor Antagonists; Ergolines; Hypothermia; Injections, Subcutaneous; Male; Oxotremorine; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Salicylamides; Serotonin Antagonists | 1994 |
Dopamine receptor regulating serotonin N-acetyltransferase activity in chick retina represents a D4-like subtype: pharmacological characterization.
Topics: Animals; Arylamine N-Acetyltransferase; Benzamides; Benzazepines; Chickens; Circadian Rhythm; Clozapine; Dopamine; Dopamine Antagonists; Ergolines; Ketanserin; Male; Quinpirole; Receptors, Dopamine; Retina; Spiperone; Sulpiride | 1994 |
Comparative dopaminergic and muscarinic antagonist activity of clozapine and haloperidol.
Topics: Acetylcholine; Animals; Cerebellum; Clozapine; Corpus Striatum; Cyclic GMP; Dopamine Antagonists; Ergolines; Haloperidol; Male; Mice; Muscarinic Antagonists; Oxotremorine; Quinpirole; Rats; Rats, Sprague-Dawley | 1996 |
Normethylclozapine potentiates the action of quinpirole in the 6-hydroxydopamine lesioned rat.
Topics: Animals; Behavior, Animal; Clozapine; Dopamine Agonists; Drug Synergism; Functional Laterality; Male; Oxidopamine; Quinpirole; Rats; Rats, Sprague-Dawley; Rotation; Serotonin Antagonists; Stereotyped Behavior; Sympathectomy, Chemical | 1996 |
Long-term treatment with chlorpromazine and haloperidol but not with sulpiride and clozapine markedly elevates neuropeptide Y-like immunoreactivity in the rat hypothalamus.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Antipsychotic Agents; Benzazepines; Chlorpromazine; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Gene Expression Regulation; Haloperidol; Hypothalamus; Male; Neuropeptide Y; Prazosin; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Sulpiride | 1996 |
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1996 |
Pharmacological modifications in dopaminergic neurotransmission affect the quinpirole-evoked suppression of serotonin N-acetyltransferase activity in chick retina: an impact on dopamine D4-like receptors.
Topics: Animals; Antipsychotic Agents; Arylamine N-Acetyltransferase; Chickens; Circadian Rhythm; Clozapine; Dopamine Agents; Enzyme Inhibitors; Levodopa; Male; Quinpirole; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Retina; Salicylamides; Sulpiride; Synaptic Transmission | 1996 |
Expression and characterization of a dopamine D4R variant associated with delusional disorder.
Topics: Animals; Antipsychotic Agents; CHO Cells; Clozapine; Cricetinae; Dopamine; Dopamine Agonists; Dopamine Antagonists; Epinephrine; Genetic Variation; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kinetics; Norepinephrine; Polymorphism, Genetic; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Schizophrenia, Paranoid; Transfection | 1998 |
Atypical antipsychotics and dopamine D(1) receptor agonism: an in vivo experimental study using core temperature measurements in the rat.
Topics: Animals; Antipsychotic Agents; Benzazepines; Benzodiazepines; Clozapine; Dibenzothiazepines; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Fever; Hypothermia; Male; Olanzapine; Pirenzepine; Quetiapine Fumarate; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Risperidone; Time Factors | 2000 |
Effects of chronic haloperidol and clozapine on vacuous chewing and dopamine-mediated jaw movements in rats: evaluation of a revised animal model of tardive dyskinesia.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Behavior, Animal; Clozapine; Disease Models, Animal; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dyskinesia, Drug-Induced; Haloperidol; Jaw; Male; Mastication; Quinpirole; Rats; Rats, Sprague-Dawley; Reproducibility of Results; Serotonin Antagonists | 1999 |
Quinpirole, 8-OH-DPAT and ketanserin modulate catalepsy induced by high doses of atypical antipsychotics.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Benzodiazepines; Catalepsy; Clozapine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Imidazoles; Indoles; Ketanserin; Male; Mice; Mice, Inbred BALB C; Olanzapine; Pirenzepine; Quinpirole; Random Allocation; Rats; Rats, Wistar; Risperidone; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Species Specificity | 1999 |
Dopamine decreases melatonin content in golden hamster retina.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Benzazepines; Chromatography, High Pressure Liquid; Circadian Rhythm; Clozapine; Cricetinae; Cyclic AMP; Depression, Chemical; Dopamine; Dopamine Agonists; Dopamine Antagonists; Kinetics; Male; Melatonin; Mesocricetus; Quinpirole; Receptors, Dopamine; Retina; Spiperone | 2000 |
Pharmacology of quinpirole-stimulated [35S]GTPgammaS binding: discrepancy with receptor binding profile.
Topics: Animals; Benzazepines; Binding, Competitive; Clorgyline; Clozapine; Corpus Striatum; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); Haloperidol; Male; Membranes; Monoamine Oxidase Inhibitors; Quinpirole; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Selegiline; Spiperone; Sulfur Radioisotopes; Thiazoles | 2000 |
Reconstitution of functional dopamine D(2s) receptor by co-expression of amino- and carboxyl-terminal receptor fragments.
Topics: Animals; Apomorphine; Binding, Competitive; Clozapine; Colforsin; COS Cells; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gene Expression; Haloperidol; Membranes; Peptide Fragments; Pergolide; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Transfection; Tritium | 2000 |
Pharmacology of [3H]R(+)-7-OH-DPAT binding in the rat caudate-putamen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Caudate Nucleus; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Guanidines; Guanosine Triphosphate; Haloperidol; Heterotrimeric GTP-Binding Proteins; Indans; Kinetics; Magnesium; Male; Oxazines; Protein Binding; Putamen; Quinpirole; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Remoxipride; Sodium; Specific Pathogen-Free Organisms; Sulfones; Sulpiride; Tetrahydronaphthalenes | 2001 |
Studies on modulation of feeding behavior by atypical antipsychotics in female mice.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adipose Tissue; Animals; Antipsychotic Agents; Body Weight; Clozapine; Eating; Feeding Behavior; Female; Fluoxetine; Hyperphagia; Mice; Mice, Inbred Strains; Organ Size; Quinpirole; Quipazine; Selective Serotonin Reuptake Inhibitors; Weight Gain | 2002 |
Co-release of noradrenaline and dopamine from noradrenergic neurons in the cerebral cortex induced by clozapine, the prototype atypical antipsychotic.
Topics: Adrenergic alpha-Agonists; Animals; Antipsychotic Agents; Cerebral Cortex; Chromatography, High Pressure Liquid; Clonidine; Clozapine; Dopamine; Dopamine Agonists; Extracellular Space; Immunohistochemistry; Male; Microdialysis; Neurons; Norepinephrine; Occipital Lobe; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley | 2003 |
Photic regulation of heme oxygenase activity in the golden hamster retina: involvement of dopamine.
Topics: Animals; Benzazepines; Bilirubin; Bucladesine; Circadian Rhythm; Clozapine; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Activation; Enzyme Inhibitors; Heme Oxygenase (Decyclizing); In Vitro Techniques; Male; Mesocricetus; Photoperiod; Quinpirole; Retina; Spiperone; Thiobarbituric Acid Reactive Substances | 2003 |
[The roles of dopamine 4 receptor in MPTP-induced gastrointestinal mucosal injury in rats].
Topics: Animals; Clozapine; Cytoprotection; Female; Gastric Mucosa; Intestinal Mucosa; MPTP Poisoning; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D4 | 2003 |
Tonic modulation of inhibition by dopamine D4 receptors in the rat hippocampus.
Topics: Animals; Clozapine; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; GABA Antagonists; Hippocampus; Male; Neural Inhibition; Neural Pathways; Organ Culture Techniques; Perforant Pathway; Pyridines; Pyrroles; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D4; Synapses | 2005 |
A new approach to finding specific dopamine D4 receptor agonists.
Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Apomorphine; Blotting, Western; Bromocriptine; Cloning, Molecular; Clozapine; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Synergism; Guinea Pigs; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Phenethylamines; Prazosin; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Alignment; Sequence Homology, Amino Acid; Vas Deferens | 2005 |
The effects of antipsychotics on beta-catenin, glycogen synthase kinase-3 and dishevelled in the ventral midbrain of rats.
Topics: Adaptor Proteins, Signal Transducing; Amphetamine; Animals; Antipsychotic Agents; Benzazepines; beta Catenin; Blotting, Western; Central Nervous System Stimulants; Clozapine; Cytoskeletal Proteins; Dishevelled Proteins; Dopamine Agonists; Female; Glycogen Synthase Kinase 3; Haloperidol; Immunohistochemistry; Intercellular Signaling Peptides and Proteins; Male; Mesencephalon; Phosphoproteins; Quinpirole; Rats; Rats, Sprague-Dawley; Risperidone; Signal Transduction; Trans-Activators; Wnt Proteins; Wnt1 Protein | 2005 |
Potentiation of olanzapine substitution in rats discriminating clozapine by the D2/3 agonist quinpirole.
Topics: Animals; Antipsychotic Agents; Benzodiazepines; Clozapine; Discrimination Learning; Discrimination, Psychological; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Female; Olanzapine; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3 | 2007 |
Haloperidol both prevents and reverses quinpirole-induced nonregulatory water intake, a putative animal model of psychogenic polydipsia.
Topics: Administration, Oral; Animals; Antipsychotic Agents; Benzodiazepines; Clomipramine; Clozapine; Disease Models, Animal; Dose-Response Relationship, Drug; Drinking; Haloperidol; Male; Olanzapine; Piperazines; Pyrroles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Thiazepines | 2008 |
The receptor mechanisms underlying the disruptive effects of haloperidol and clozapine on rat maternal behavior: a double dissociation between dopamine D(2) and 5-HT(2A/2C) receptors.
Topics: Amphetamines; Animals; Antipsychotic Agents; Clozapine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Female; Haloperidol; Maternal Behavior; Nesting Behavior; Postpartum Period; Pregnancy; Quinpirole; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptor, Serotonin, 5-HT2C; Receptors, Dopamine D2; Serotonin Receptor Agonists | 2009 |
c-Fos identification of neuroanatomical sites associated with haloperidol and clozapine disruption of maternal behavior in the rat.
Topics: Amphetamines; Animals; Animals, Newborn; Antipsychotic Agents; Biomarkers; Brain; Clozapine; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Female; Haloperidol; Immunohistochemistry; Male; Maternal Behavior; Neostriatum; Nucleus Accumbens; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D2; Septum of Brain; Serotonin 5-HT2 Receptor Antagonists; Serotonin Receptor Agonists | 2010 |
The effects of clozapine on quinpirole-induced non-regulatory drinking and prepulse inhibition disruption in rats.
Topics: Animals; Antipsychotic Agents; Brain; Brain-Derived Neurotrophic Factor; Clozapine; Disease Models, Animal; Dopamine Agonists; Dose-Response Relationship, Drug; Drinking; Gene Expression Regulation; Haloperidol; Male; Proto-Oncogene Proteins c-fos; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Schizophrenia | 2010 |
Alcohol withdrawal drives depressive behaviors by activating neurons in the rostromedial tegmental nucleus.
Topics: 2-Amino-5-phosphonovalerate; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Clozapine; Dopaminergic Neurons; Ethanol; gamma-Aminobutyric Acid; Male; Microinjections; Neural Inhibition; Neural Pathways; Nucleus Accumbens; Proto-Oncogene Proteins c-fos; Quinoxalines; Quinpirole; Rats; Substance Withdrawal Syndrome; Tegmentum Mesencephali; Ventral Tegmental Area | 2019 |
D2 receptor-mediated miRNA-143 expression is associated with the effects of antipsychotic drugs on phencyclidine-induced schizophrenia-related locomotor hyperactivity and with Neuregulin-1 expression in mice.
Topics: Animals; Benzazepines; Clozapine; Dopamine D2 Receptor Antagonists; Haloperidol; Hippocampus; Male; Mice; Mice, Transgenic; MicroRNAs; Motor Activity; Neuregulin-1; Phencyclidine; Prefrontal Cortex; Primary Cell Culture; Quinpirole; Receptors, Dopamine D2; Salicylamides | 2019 |