quinpirole and bp 897
quinpirole has been researched along with bp 897 in 8 studies
Research
Studies (8)
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 8 (100.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
Authors
| Authors | Studies |
|---|---|
| Bettinetti, L; Gmeiner, P; Hübner, H; Schlotter, K | 1 |
| Aiello, F; Butini, S; Cagnotto, A; Campiani, G; Carnovali, F; Catalanotti, B; Cervo, L; Fattorusso, C; Fumagalli, E; Gemma, S; Mennini, T; Nacci, V; Novellino, E; Stark, JA; Trotta, F | 1 |
| Berardi, F; Colabufo, NA; Contino, M; Lacivita, E; Leopoldo, M; Perrone, R | 1 |
| Boeckler, F; Gmeiner, P; Hübner, H; Schlotter, K | 1 |
| Berardi, F; Contino, M; De Giorgio, P; Lacivita, E; Leopoldo, M; Perrone, R | 1 |
| Avenell, KY; Boyfield, I; Jewitt, FR; Nash, DJ; Riley, GJ; Wood, MD | 1 |
| Garcia-Ladona, J; Wicke, K | 1 |
| Beardsley, PM; Cook, CD; Newman, JL; Winfree, JC | 1 |
Other Studies
8 other study(ies) available for quinpirole and bp 897
| Article | Year |
|---|---|
Interactive SAR studies: rational discovery of super-potent and highly selective dopamine D3 receptor antagonists and partial agonists.
Topics: Animals; CHO Cells; Cricetinae; Dopamine Agonists; Dopamine Antagonists; Humans; Ligands; Mitosis; Piperazines; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Swine; Thiophenes | 2002 |
Synthesis and pharmacological evaluation of potent and highly selective D3 receptor ligands: inhibition of cocaine-seeking behavior and the role of dopamine D3/D2 receptors.
Topics: Animals; Behavior, Addictive; Brain; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Extinction, Psychological; In Vitro Techniques; Ligands; Male; Models, Molecular; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Administration; Structure-Activity Relationship | 2003 |
First structure-activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure.
Topics: Amides; Animals; CHO Cells; Cricetinae; Cricetulus; Humans; Piperazines; Radioligand Assay; Receptors, Dopamine D3; Stereoisomerism; Structure-Activity Relationship | 2005 |
Fancy bioisosteres: novel paracyclophane derivatives as super-affinity dopamine D3 receptor antagonists.
Topics: Amides; Animals; Benzene Derivatives; Benzofurans; Binding Sites; Bridged-Ring Compounds; Central Nervous System Agents; CHO Cells; Corpus Striatum; Cricetinae; Cricetulus; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Mutation; Radioligand Assay; Receptors, Dopamine D3; Stereoisomerism; Structure-Activity Relationship; Swine; Thymidine | 2006 |
Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands with optimal lipophilicity for brain imaging of the dopamine D3 receptor. Part II.
Topics: Amides; Drug Design; Humans; Ligands; Piperazines; Positron-Emission Tomography; Protein Binding; Radiopharmaceuticals; Receptors, Dopamine D3 | 2009 |
Evidence for antagonist activity of the dopamine D3 receptor partial agonist, BP 897, at human dopamine D3 receptor.
Topics: Animals; Azepines; CHO Cells; Cricetinae; Dopamine Agonists; Humans; Piperazines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3 | 2000 |
The dopamine D3 receptor partial agonist, BP 897, is an antagonist at human dopamine D3 receptors and at rat somatodendritic dopamine D3 receptors.
Topics: Animals; Benzopyrans; Binding, Competitive; CHO Cells; Cricetinae; Dendrites; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Electrophysiology; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Neurons; Oxazines; Piperazines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Substantia Nigra; Sulfur Radioisotopes; Tetrahydronaphthalenes | 2001 |
Modulation of the locomotor activating effects of the noncompetitive NMDA receptor antagonist MK801 by dopamine D2/3 receptor agonists in mice.
Topics: Animals; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Naphthalenes; Piperazines; Pyrrolidines; Quinolines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, N-Methyl-D-Aspartate; Salicylamides; Stereotyped Behavior | 2004 |