Page last updated: 2024-08-17

quinoxalines and thiourea

quinoxalines has been researched along with thiourea in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.14)18.2507
2000's13 (92.86)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hathway, GJ; Humphrey, PP; Kendrick, KM1
Costa, G; García-Pascual, A; Jiménez, E; Labadía, A; Triguero, D1
Bergamini, A; Bolacchi, F; Caccia, S; Campiani, G; Coletta, M; Fabbrini, M; Faggioli, E; Fracasso, C; Greco, G; Maga, G; Marini, S; Morelli, E; Nacci, V; Novellino, E; Spadari, S; Uccella, I1
Breder, J; Opitz, T; Reymann, KG; Sabelhaus, CF; Schröder, UH1
Aiello, F; Armaroli, S; Bergamini, A; Bolacchi, F; Bongiovanni, B; Caccia, S; Campiani, G; Capozzi, M; Coletta, M; Fabbrini, M; Garofalo, A; Greco, G; Guiso, G; Maga, G; Marini, S; Morelli, E; Nacci, V; Novellino, E; Ramunno, A; Spadari, S; Ventura, L1
Deng, A; Thomson, SC1
Kahlert, S; Martínez-Sánchez, M; Reiser, G; Reymann, KG; Schröder, UH; Striggow, F1
Kiedrowski, L1
Jung, SY; Kim, YT; Park, YJ; Seo, WS; Suh, CK1
Kim, YT; Kwak, J; Namkung, YL; Suh, CK1
Bannon, AW; Deng, H; Gavva, NR; Gore, A; Han, B; Hovland, DN; Juan, T; Klionsky, L; Kuang, R; Le, A; Lehto, SG; Louis, JC; Magal, E; Norman, MH; Surapaneni, S; Tamir, R; Treanor, JJ; Wang, J; Youngblood, B; Zhu, D1
Bahekar, RH; Goel, A; Gupta, AA; Jadav, PA; Jain, MR; Patel, DN; Patel, PR; Prajapati, VM1
Abou-Zied, AH; El-Shaieb, KM; Hassan, AA; Mourad, AF1
Majewski, H; Zhao, J1

Other Studies

14 other study(ies) available for quinoxalines and thiourea

ArticleYear
Evidence that somatostatin sst2 receptors mediate striatal dopamine release.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Aminopyridines; Animals; Corpus Striatum; Dopamine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Neurotransmitter Agents; Oligopeptides; Peptides, Cyclic; Quinoxalines; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin; Thiourea

1999
Spontaneous photo-relaxation of urethral smooth muscle from sheep, pig and rat and its relationship with nitrergic neurotransmission.
    The Journal of physiology, 2000, Feb-01, Volume: 522 Pt 3

    Topics: Adenine; Animals; Citrulline; Cold Temperature; Culture Techniques; Electric Stimulation; Enzyme Inhibitors; Female; Light; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Oxadiazoles; Oxyhemoglobins; Phosphodiesterase Inhibitors; Photic Stimulation; Potassium; Purinones; Quinoxalines; Rats; Rats, Wistar; Sheep; Superoxides; Swine; Synaptic Transmission; Tetrodotoxin; Thiourea; Time Factors; Urethra

2000
Non-nucleoside HIV-1 reverse transcriptase inhibitors: synthesis and biological evaluation of novel quinoxalinylethylpyridylthioureas as potent antiviral agents.
    Antiviral chemistry & chemotherapy, 2000, Volume: 11, Issue:2

    Topics: Amino Acid Substitution; Animals; HIV Reverse Transcriptase; HIV-1; Humans; Male; Mice; Mice, Inbred Strains; Mutation; Nucleosides; Quinoxalines; Reverse Transcriptase Inhibitors; Thiourea

2000
Inhibition of different pathways influencing Na(+) homeostasis protects organotypic hippocampal slice cultures from hypoxic/hypoglycemic injury.
    Neuropharmacology, 2000, Jul-24, Volume: 39, Issue:10

    Topics: Animals; Brain Ischemia; Cell Death; Culture Techniques; Dizocilpine Maleate; Electrophysiology; Hippocampus; Homeostasis; Hypoglycemia; Hypoxia; Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sodium; Sodium Channel Blockers; Sodium Channels; Sodium-Calcium Exchanger; Tetrodotoxin; Thiourea

2000
Quinoxalinylethylpyridylthioureas (QXPTs) as potent non-nucleoside HIV-1 reverse transcriptase (RT) inhibitors. Further SAR studies and identification of a novel orally bioavailable hydrazine-based antiviral agent.
    Journal of medicinal chemistry, 2001, Feb-01, Volume: 44, Issue:3

    Topics: Animals; Anti-HIV Agents; Biological Availability; Cell Line; Didanosine; Drug Synergism; HIV Reverse Transcriptase; HIV-1; Humans; Mice; Models, Molecular; Pyridines; Quinoxalines; Reverse Transcriptase Inhibitors; Stereoisomerism; Structure-Activity Relationship; Thiourea; Zidovudine

2001
Cyclic GMP mediates influence of macula densa nitric oxide over tubuloglomerular feedback.
    Kidney & blood pressure research, 2003, Volume: 26, Issue:1

    Topics: Animals; Citrulline; Cyclic GMP; Enzyme Inhibitors; Feedback, Physiological; Glomerular Filtration Rate; Guanylate Cyclase; Juxtaglomerular Apparatus; Male; Nephrons; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Thiourea

2003
Na(+) and Ca(2+) homeostasis pathways, cell death and protection after oxygen-glucose-deprivation in organotypic hippocampal slice cultures.
    Neuroscience, 2004, Volume: 128, Issue:4

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Boron Compounds; Calcium; Calcium Channel Blockers; Cell Death; Clonazepam; Dantrolene; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Fura-2; Glucose; Hippocampus; Hypoxia; In Situ Nick-End Labeling; Indoles; Intracellular Space; Ion Exchange; Lidocaine; Mibefradil; Nimodipine; Organ Culture Techniques; Quinoxalines; Rats; Rats, Wistar; Sodium; Sodium Channel Blockers; Thiazepines; Thiourea; Time Factors

2004
High activity of K+-dependent plasmalemmal Na+/Ca2+ exchangers in hippocampal CA1 neurons.
    Neuroreport, 2004, Sep-15, Volume: 15, Issue:13

    Topics: Animals; Calcium; Cells, Cultured; Cesium; Embryo, Mammalian; Excitatory Amino Acid Antagonists; Female; Gluconates; Gramicidin; Hippocampus; Ion Transport; Lithium; Male; Meglumine; Neurons; Potassium; Pregnancy; Quinoxalines; Rats; Sodium; Sodium-Calcium Exchanger; Thiourea

2004
Effects of Na+-Ca2+ exchanger activity on the alpha-amino-3-hydroxy-5-methyl-4-isoxazolone-propionate-induced Ca2+ influx in cerebellar Purkinje neurons.
    Neuroscience, 2005, Volume: 131, Issue:3

    Topics: Agatoxins; Animals; Animals, Newborn; Bepridil; Calbindins; Calcium; Calcium Channel Blockers; Cells, Cultured; Cerebellum; Diagnostic Imaging; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fluorescent Antibody Technique; Glutamic Acid; Isoxazoles; Microscopy, Confocal; Oligonucleotides, Antisense; Polyamines; Propionates; Purkinje Cells; Quinoxalines; Rats; S100 Calcium Binding Protein G; Sodium; Sodium Channel Blockers; Sodium-Calcium Exchanger; Thiourea

2005
Involvement of Na+-Ca2+ exchanger on metabotropic glutamate receptor 1-mediated [Ca2+]i transients in rat cerebellar Purkinje neurons.
    Neuroscience, 2007, Apr-25, Volume: 146, Issue:1

    Topics: Animals; Animals, Newborn; Bepridil; Calcium; Calcium Channel Blockers; Cells, Cultured; Cerebellum; Drug Interactions; Enzyme Activation; Excitatory Amino Acid Antagonists; Methoxyhydroxyphenylglycol; Oligodeoxyribonucleotides, Antisense; Purkinje Cells; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Sodium-Calcium Exchanger; Thiourea

2007
The vanilloid receptor TRPV1 is tonically activated in vivo and involved in body temperature regulation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2007, Mar-28, Volume: 27, Issue:13

    Topics: Acrylamides; Animals; Benzothiazoles; Blood-Brain Barrier; Body Temperature Regulation; Bridged Bicyclo Compounds, Heterocyclic; Capsaicin; Cells, Cultured; CHO Cells; Conserved Sequence; Cricetinae; Cricetulus; Dogs; Female; Fever; Humans; Hypothermia; Macaca fascicularis; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Species Specificity; Sulfonamides; Thiourea; TRPV Cation Channels

2007
Synthesis and antidiabetic activity of 3,6,7-trisubstituted-2-(1H-imidazol-2-ylsulfanyl)quinoxalines and quinoxalin-2-yl isothioureas.
    Archiv der Pharmazie, 2007, Volume: 340, Issue:7

    Topics: Animals; Cell Line, Tumor; Dose-Response Relationship, Drug; Hypoglycemic Agents; Imidazoles; Insulin; Insulin Secretion; Insulin-Secreting Cells; Quinoxalines; Rats; Stereoisomerism; Structure-Activity Relationship; Sulfones; Thiourea

2007
Synthesis of 1,3,4-thiadiazole, 1,3,4-thiadiazine, 1,3,6-thiadiazepane and quinoxaline derivatives from symmetrical dithiobiureas and thioureidoethylthiourea derivatives.
    Molecules (Basel, Switzerland), 2005, Aug-31, Volume: 10, Issue:7

    Topics: Disulfides; Heterocyclic Compounds; Models, Molecular; Molecular Conformation; Quinoxalines; Sulfhydryl Compounds; Thiadiazines; Thiadiazoles; Thiazoles; Thioacetamide; Thiourea; Toluene

2005
Endothelial nitric oxide attenuates Na+/Ca2+ exchanger-mediated vasoconstriction in rat aorta.
    British journal of pharmacology, 2008, Volume: 154, Issue:5

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Aorta, Thoracic; Dinoprost; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; In Vitro Techniques; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroprusside; Oxadiazoles; Potassium; Prostaglandin-Endoperoxide Synthases; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium; Sodium-Calcium Exchanger; Thiourea; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents

2008