Page last updated: 2024-08-17

quinoxalines and prazosin

quinoxalines has been researched along with prazosin in 129 studies

Research

Studies (129)

TimeframeStudies, this research(%)All Research%
pre-199034 (26.36)18.7374
1990's65 (50.39)18.2507
2000's21 (16.28)29.6817
2010's8 (6.20)24.3611
2020's1 (0.78)2.80

Authors

AuthorsStudies
Hansson, E; Nilsson, M; Rönnbäck, L1
Pinnock, RD1
Berridge, TL; Doxey, JC; Roach, AG; Smith, CF1
Jansen van't Land, C; van der Laan, JW1
Lefebvre, RA; Smits, GJ1
Deschênes, M; Pinault, D1
Bourreau, JP; Daniel, EE; Kwan, CY; Shimamoto, H1
Minneman, KP; Wilson, KM1
Dunn, WR; McGrath, JC; Wilson, VG2
Bültmann, R; Starke, K; von Kügelgen, I1
Lepor, H1
Flavahan, NA; Komori, K; Miller, VM; Vanhoutte, PM1
Berlan, M; Galitzky, J; Lafontan, M; Montastruc, JL; Senard, JM; Stillings, M1
Alari, L; Axelsson, KL; Persson, ML; Post, C; Uhlén, S; Wikberg, JE1
Guimaraes, S; Nunes, JP1
Altemeyer, KH; Dirks, B; Ensinger, H; Grünert, A1
Rand, MJ; Xiao, XH1
Doxey, JC; John, GW; Reid, JL; Walter, DS1
Guimarães, S; Moura, D; Vaz-da-Silva, MJ1
Brandon, S; Cragoe, EJ; Guyer, CA; Horstman, DA; Limbird, LE; Wilson, AL1
Calvete, J; Hayes, R; Sever, PS; Thom, S1
Lacroix, JS; Lundberg, JM1
Hughes, AD; Martin, GN; Mulvany, MJ; Nielsen, H; Sever, PS; Thom, SM1
Bylund, DB; Ray-Prenger, C1
Albuquerque, AA; Goncalves, J; Paiva, MQ; Proenca, J1
Cattaneo, AG; Doxey, JC; Efendic, S; Ostenson, CG1
Hashimoto, K; Tsujimoto, G1
Edwards, RM; Trizna, W1
Harker, CT; Vanhoutte, PM1
Downing, OA; Stein, W; Wilson, KA; Wilson, VG1
Calvete, J; Hayes, R; Martin, G; Sever, P; Thom, S1
Guimarães, S; Paiva, MQ; Polónia, JJ1
Hesse, IF; Johns, EJ1
Hyman, AL; Kadowitz, PJ2
Dickinson, KE; McKernan, RM; Miles, CM; Sever, PS1
Bassenge, E; Elsner, D; Holtz, J; Sommer, O; Stewart, DJ1
Dettmar, PW; Lord, JA1
Itoh, H; Kohli, JD; Rajfer, SI1
Broadley, KJ; Williamson, KL1
Guimarães, S; Moura, D; Paiva, MQ1
Graham, RM; Powell, WJ; Supple, EW1
Nyman, L; Saano, V; Savola, JM; Virtanen, R1
Uhlén, S; Wikberg, JE1
Gonçalves, J; Guimarães, S; Nunes, JP; Paiva, MQ1
Daly, CJ; McGrath, JC; Wilson, VG1
Messick, K; Ruffolo, RR1
Hyman, AL; Kadowitz, PJ; Lippton, HL1
Pipili, E1
Flavahan, NA; Gisclard, V; Vanhoutte, PM1
Beckeringh, JJ; De Jonge, A; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B1
Hicks, PE1
McWilliam, JR; Meldrum, BS1
Davidoff, RA; Hackman, JC; Holohean, AM; Shope, SB1
Advenier, C; Biyah, K1
Hussain, JF; Kendall, DA; Pinthong, D; Wilson, VG1
Dyamenahalli, U; Haworth, SG; Stuart-Smith, K; Tulloh, RM1
Ge, YZ; Morrison, SF1
Cable, HC; el-Mansoury, A; Morgan, NG1
Gazzola, C; Hunter, RA; Lisle, AT; Magner, T1
Qü, M; Schleicher, A; Zilles, K1
Driessen, B; Starke, K; von Kügelgen, I1
Robinson, NE; Wang, Z; Yu, M1
Kachroo, A; Malhotra, V; Sapru, HN1
Faber, JE; Ikeoka, K1
Crepel, F; Hirsch, JC; Law-Tho, D1
Vanhoutte, PM; Wood, MB; Ye, Z1
Giardinà, D; Gulini, U; Massi, M; Melchiorre, C; Piloni, MG; Pompei, P; Rafaiani, G1
Angel, I; Grosset, A; Langer, SZ; Perrault, G; Schoemaker, H1
Cheetham, SC; Heal, DJ1
Bohmann, C; Riera-Knorrenschild, G; Rump, LC; Schollmeyer, P; Schwertfeger, E; Spillner, G1
Crucianelli, M; Giardinà, D; Melchiorre, C; Taddei, C; Testa, R1
Brown, DR; Malone, ED; Trent, AM; Turner, TA1
Bryant, CE; Clarke, KW1
Bohmann, C; Rist, W; Rump, LC; Schollmeyer, P1
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM1
Intengan, HD; Smyth, DD2
Oriowo, MA; Williams, KI; Yousif, M1
Feltz, P; Hayar, A; Piguet, P1
Nörenberg, W; Schöffel, E; Starke, K; Szabo, B1
Elliott, J1
Guimarães, S; Paiva, MQ; Pereira, O1
Bayliss, DA; Guyenet, PG; Li, YW1
Akaike, N; Arima, J; Ishibashi, H; Kubo, C1
Gallant, CM; Goldstein, I; Gupta, S; Moreland, RB; Traish, A; Yang, S1
Kwan, CY; Mo, FM1
Abysique, A; Bouvier, M; Orsoni, P1
Bredt, DS; Morton, DB1
Hipólide, DC; Nobrega, JN; Raymond, R; Tufik, S1
Soares-da-Silva, P; Vieira-Coelho, MA1
Daniel, EE; Kwan, CY; Loke, JC; Low, AM; Lu-Chao, H1
Borges, AC; Feres, T; Paiva, AC; Paiva, TB; Silva, EG1
Endo, T; Hirafuji, M; Kato, K; Minami, M; Ogawa, T; Satoh, Y; Suzuguchi, T1
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1
Daly, CJ; Mackenzie, JF; McGrath, JC; Naghadeh, MA; Pediani, JD1
Nott, MW; Rand, MJ; Thaina, P1
Fujiki, H; Imaizumi, T; Kambayashi, J; Kimura, Y; Kishi, M; Mori, T; Orito, K; Shimizu, H; Tanaka, M; Teramoto, S; Tominaga, M; Yoshida, K1
Eglen, RM; MacLennan, SJ; Martin, GR; Martin, RS; Reynen, PH1
Eglen, RM; MacLennan, SJ; Martin, GR; Reynen, PH1
Iida, S; Ishihama, K; Kogo, M; Koizumi, H; Matsuya, T; Mori, A; Tanaka, S1
Hillier, C; Jarajapu, YP; MacDonald, A1
Angeli, P; Giardinà, D; Gulini, U; Leonardi, A; Marucci, G; Melchiorre, C; Poggesi, E; Polimanti, O; Sagratini, G1
Adell, A; Amargós-Bosch, M; Artigas, F; Bortolozzi, A; Díaz-Mataix, L; Pons, S; Serrats, J1
Duman, RS; Russell, DS; Tolbert, LM1
Dang, VC; Williams, JT1
Brockhaus, J; Deitmer, JW; Hecker, C; Herold, S1
Gutkowska, J; Menaouar, A; Mukaddam-Daher, S1
Ananthalakshmi, KV; Edafiogho, IO; Kombian, SB1
Kolaj, M; Renaud, LP1
Angeli, P; Buccioni, M; Giardinà, D; Gulini, U; Leonardi, A; Marucci, G; Melchiorre, C; Poggesi, E; Sagratini, G1
Centurión, D; Görnemann, T; Jähnichen, S; Kleuser, B; Pertz, HH; Villalón, CM; von Wenckstern, H1
Koob, GF; Lekic, DM; Mandyam, CD; Wee, S1
Bexis, S; Docherty, JR1
Didier, A; Jourdan, F; Marien, M; Nguyen, V; Veyrac, A1
Bustamante, S; García-Sacristán, A; Hernández, M; Martínez, MP; Navarro-Dorado, J; Orensanz, LM; Prieto, D; Recio, P1
Enokizono, J; Kusuhara, H; Ose, A; Schinkel, AH; Sugiyama, Y1
Imanishi, A; Latifpour, J; Ueda, S; Yamamoto, Y; Yono, M; Yoshida, M1
Cheevers, CV; Donello, JE; Gil, DW; Kedzie, KM; Manlapaz, CA; Rao, S; Tang, E1
Jackson, WF; Moore, AW; Segal, SS1
Man, RY; Ng, KF; Vanhoutte, PM; Wong, ES1
Centurión, D; Hofmann, RA; Jantschak, F; Pertz, HH; Popp, AM; Villalón, CM1
Aston-Jones, G; Smith, RJ1
Aono, Y; Cools, AR; Koshikawa, N; Saigusa, T; Takada, K; Uchida, T; Verheij, MM1
Bult, H; De Meyer, GR; Fransen, P; Martinet, W; Schrijvers, DM; Van Hove, CE; van Langen, JT1
Acheson, AG; Dashwood, MR; Eames, T; Gruss, H; Henry, Y; Rayment, SJ; Scholefield, JH; Simpson, JA; Wilson, VG1
Abdelkarim, H; Albee, LJ; Gao, X; Gaponenko, V; Majetschak, M; Volkman, BF1
Alsufyani, HA; Docherty, JR; McCormick, PA1

Reviews

1 review(s) available for quinoxalines and prazosin

ArticleYear
Role of alpha-adrenergic blockers in the treatment of benign prostatic hyperplasia.
    The Prostate. Supplement, 1990, Volume: 3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Carbachol; Humans; Male; Muscle Contraction; Phenylephrine; Prazosin; Prostatic Hyperplasia; Quinoxalines

1990

Trials

1 trial(s) available for quinoxalines and prazosin

ArticleYear
Human vascular smooth muscle responses mediated by alpha 2 mechanisms in vivo and in vitro.
    Clinical science (London, England : 1979), 1985, Volume: 68 Suppl 10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Arteries; Brimonidine Tartrate; Dioxanes; Doxazosin; Forearm; Humans; Idazoxan; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha

1985

Other Studies

127 other study(ies) available for quinoxalines and prazosin

ArticleYear
Receptor-coupled uptake of valproate in rat astroglial primary cultures.
    Neuroscience letters, 1992, Feb-17, Volume: 136, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Astrocytes; Biological Transport; Cells, Cultured; Cerebral Cortex; Clonidine; Drug Interactions; Glutamates; Glutamic Acid; Isoproterenol; Kainic Acid; Ketanserin; Phenylephrine; Prazosin; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter; Serotonin; Valproic Acid; Yohimbine

1992
Activation of kappa-opioid receptors depresses electrically evoked excitatory postsynaptic potentials on 5-HT-sensitive neurones in the rat dorsal raphé nucleus in vitro.
    Brain research, 1992, Jun-26, Volume: 583, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Afferent Pathways; Animals; Benzofurans; Bicuculline; Bombesin; Cholecystokinin; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Evoked Potentials; Glutamates; Glutamic Acid; In Vitro Techniques; Kynurenic Acid; N-Methylaspartate; Naloxone; Naltrexone; Neurons; Picrotoxin; Prazosin; Pyrrolidines; Quinoxalines; Raphe Nuclei; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Synapses; Tetrodotoxin

1992
Selectivity profile of the alpha 2-adrenoceptor antagonist efaroxan in relation to plasma glucose and insulin levels in the rat.
    European journal of pharmacology, 1992, Mar-24, Volume: 213, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Benzofurans; Blood Glucose; Brimonidine Tartrate; Clonidine; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Epinephrine; Idazoxan; Imidazoles; Insulin; Male; Muscles; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Vas Deferens

1992
Chronic infusion of clonidine does not alleviate spontaneous morphine withdrawal symptoms in rats.
    Psychopharmacology, 1992, Volume: 108, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Doxazosin; Drug Implants; Eating; Food; Male; Morphine; Morphine Dependence; Motor Activity; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome

1992
Modulation of non-adrenergic non-cholinergic inhibitory neurotransmission in rat gastric fundus by the alpha 2-adrenoceptor agonist, UK-14,304.
    British journal of pharmacology, 1992, Volume: 107, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Autonomic Nervous System; Brimonidine Tartrate; Electric Stimulation; Gastric Fundus; In Vitro Techniques; Male; Muscle Relaxation; Nitric Oxide; Prazosin; Quinoxalines; Rats; Rats, Wistar; Synaptic Transmission; Vasoactive Intestinal Peptide; Yohimbine

1992
Control of 40-Hz firing of reticular thalamic cells by neurotransmitters.
    Neuroscience, 1992, Volume: 51, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Bicuculline; Electric Conductivity; Female; gamma-Aminobutyric Acid; Ketanserin; Kynurenic Acid; Male; Neurons; Neurotransmitter Agents; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Reticular Formation; Scopolamine; Thalamic Nuclei

1992
Amplification of alpha adrenergic vasoconstriction in canine isolated mesenteric artery and vein.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:3

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Dogs; Dose-Response Relationship, Drug; Endothelins; Female; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Potassium Chloride; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction

1992
Synergistic interactions between alpha 1- and alpha 2-adrenergic receptors in activating 3H-inositol phosphate formation in primary glial cell cultures.
    Journal of neurochemistry, 1991, Volume: 56, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Brain; Brimonidine Tartrate; Cells, Cultured; Dose-Response Relationship, Drug; Inositol Phosphates; Neuroglia; Norepinephrine; Osmolar Concentration; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Time Factors; Tritium; Yohimbine

1991
Postjunctional alpha-adrenoceptors in the rabbit isolated distal saphenous artery: indirect sensitivity to prazosin of responses to noradrenaline mediated via postjunctional alpha 2-adrenoceptors.
    British journal of pharmacology, 1991, Volume: 103, Issue:2

    Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Brimonidine Tartrate; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Yohimbine

1991
Contraction-mediating alpha 2-adrenoceptors in the mouse vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:6

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dioxanes; Drug Interactions; Idazoxan; Male; Mice; Muscle Contraction; Neuropeptide Y; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Suramin; Vas Deferens; Yohimbine

1991
Electrophysiological analysis of adrenergic neurotransmission and its modulation by chronic denervation in canine saphenous veins.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Dogs; Electric Stimulation; Electrophysiology; Female; Membrane Potentials; Muscle Denervation; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Prazosin; Quinoxalines; Saphenous Vein; Synaptic Transmission

1990
Identification of human platelet alpha 2-adrenoceptors with a new antagonist [3H]-RX821002, a 2-methoxy derivative of idazoxan.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Blood Platelets; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; In Vitro Techniques; Kinetics; Male; Membranes; Oxymetazoline; Prazosin; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1990
Antinociceptive actions of alpha 2-adrenoceptor agonists in the rat spinal cord: evidence for antinociceptive alpha 2-adrenoceptor subtypes and dissociation of antinociceptive alpha 2-adrenoceptors from cyclic AMP.
    Journal of neurochemistry, 1990, Volume: 55, Issue:6

    Topics: Adrenergic alpha-Agonists; Animals; Benzylamines; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guanfacine; Male; Neurotoxins; Nociceptors; Pain Measurement; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Spinal Cord; Yohimbine

1990
The effectiveness of alpha 2-adrenoceptor activation increases from the distal to the proximal part of the veins of canine limbs.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Brimonidine Tartrate; Dogs; Extremities; Female; In Vitro Techniques; Male; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Saphenous Vein; Veins; Yohimbine

1990
The role of alpha 1-adrenoceptors in adrenaline-induced hyperkalaemia.
    British journal of anaesthesia, 1990, Volume: 65, Issue:6

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Epinephrine; Hyperkalemia; Pericardium; Phentolamine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Swine

1990
Effects of the alpha 2-adrenoceptor agonist UK14304 on pressor responses in pithed rats.
    Clinical and experimental pharmacology & physiology, 1990, Volume: 17, Issue:10

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Decerebrate State; Dose-Response Relationship, Drug; Drug Synergism; Norepinephrine; Phenylephrine; Prazosin; Pressoreceptors; Quinoxalines; Rats; Vasopressins; Yohimbine

1990
Selective alpha 2-adrenoceptor blockade does not enhance glucose-evoked insulin release.
    European journal of pharmacology, 1990, Oct-23, Volume: 187, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Glucose; Brimonidine Tartrate; Dioxanes; Drug Interactions; Glucose; Idazoxan; Insulin; Male; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains

1990
Alpha-adrenoceptor reserve in the canine cephalic vein.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: Animals; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Female; Forelimb; Male; Phenoxybenzamine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction; Veins; Yohimbine

1990
An aspartate conserved among G-protein receptors confers allosteric regulation of alpha 2-adrenergic receptors by sodium.
    The Journal of biological chemistry, 1990, Dec-15, Volume: 265, Issue:35

    Topics: Affinity Labels; Allosteric Regulation; Amino Acid Sequence; Animals; Aspartic Acid; Brimonidine Tartrate; Dioxanes; DNA Mutational Analysis; Epinephrine; Idazoxan; In Vitro Techniques; Molecular Sequence Data; Oxymetazoline; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Sodium; Structure-Activity Relationship; Swine; Transfection; Yohimbine

1990
In vivo and in vitro studies of alpha 2-adrenoceptor responses in human vascular smooth muscle.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: Adult; Animals; Arm; Brimonidine Tartrate; Dioxanes; Dioxins; Doxazosin; Epinephrine; Humans; Idazoxan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Regional Blood Flow; Vasomotor System

1985
Sympathetic vascular control of the pig nasal mucosa: adrenoceptor mechanisms in blood flow and volume control.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Animals; Antihypertensive Agents; Brimonidine Tartrate; Desipramine; Dioxanes; Electric Stimulation; Female; Idazoxan; Male; Nasal Mucosa; Norepinephrine; Oxymetazoline; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic; Regional Blood Flow; Rheology; Swine; Sympathetic Nervous System

1989
Postjunctional alpha 2-adrenoceptors mediate vasoconstriction in human subcutaneous resistance vessels.
    British journal of pharmacology, 1989, Volume: 97, Issue:3

    Topics: Adult; Aged; Aged, 80 and over; Antihypertensive Agents; Arteries; Azepines; Brimonidine Tartrate; Doxazosin; Female; Humans; In Vitro Techniques; Male; Middle Aged; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Regional Blood Flow; Skin; Vascular Resistance; Vasoconstriction; Veins; Yohimbine

1989
Alpha-2A and alpha-2B adrenergic receptor subtypes: attenuation of cyclic AMP production in cell lines containing only one receptor subtype.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:2

    Topics: Animals; Brimonidine Tartrate; Cyclic AMP; Humans; Isoquinolines; Piperazines; Prazosin; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Tumor Cells, Cultured; Yohimbine

1989
Expression of functional postjunctional alpha 2-adrenoceptors in rabbit isolated distal saphenous artery--a permissive role for angiotensin II?
    British journal of pharmacology, 1989, Volume: 96, Issue:2

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Animals; Arteries; Brimonidine Tartrate; Drug Interactions; In Vitro Techniques; Male; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1989
Hypothermia induces supersensitivity of mouse vas deferens to adrenergic agonists: evidence for postjunctional alpha 2-adrenoceptors.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:1

    Topics: Animals; Antihypertensive Agents; Brimonidine Tartrate; Hypothermia; In Vitro Techniques; Male; Methoxamine; Mice; Muscle, Smooth; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Sympathomimetics; Temperature; Vas Deferens

1989
Alpha-adrenoceptors and insulin release from pancreatic islets of normal and diabetic rats.
    The American journal of physiology, 1989, Volume: 257, Issue:3 Pt 1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Diabetes Mellitus, Experimental; Dioxanes; Female; Glucose; Idazoxan; Insulin; Islets of Langerhans; Male; Phentolamine; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Streptozocin; Yohimbine

1989
Effects of triiodo-L-thyronine (T3)-induced hyperthyroidism on the cardiovascular alpha-adrenoceptor system in young and older rats.
    Japanese journal of pharmacology, 1987, Volume: 44, Issue:4

    Topics: Aging; Animals; Antihypertensive Agents; Blood Pressure; Brimonidine Tartrate; Cardiovascular System; Decerebrate State; Hyperthyroidism; Male; Myocardium; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Triiodothyronine

1987
Characterization of alpha-adrenoceptors on isolated rabbit renal arterioles.
    The American journal of physiology, 1988, Volume: 254, Issue:2 Pt 2

    Topics: Animals; Arterioles; Brimonidine Tartrate; Dose-Response Relationship, Drug; Imidazoles; Kidney Cortex; Male; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction

1988
Cooling the central ear artery of the rabbit: myogenic and adrenergic responses.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Adenosine Triphosphate; Animals; Arteries; Brimonidine Tartrate; Calcium; Cold Temperature; Ear; Electric Stimulation; Indomethacin; Male; Norepinephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Tetrodotoxin; Vasoconstriction; Yohimbine

1988
A comparison of the actions of noradrenaline and UK-14,304 in the longitudinal smooth muscle of the rat isolated portal vein--no evidence for a population of post-junctional alpha 2-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:3

    Topics: Animals; Brimonidine Tartrate; Dioxanes; Idazoxan; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Portal Vein; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha

1988
Pharmacological characterization of postsynaptic alpha-adrenoceptor subtypes in five different dog arteries in-vitro.
    The Journal of pharmacy and pharmacology, 1985, Volume: 37, Issue:3

    Topics: Animals; Antihypertensive Agents; Arteries; Brimonidine Tartrate; Cocaine; Dogs; In Vitro Techniques; Muscle, Smooth, Vascular; Phenylephrine; Prazosin; Propiophenones; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Yohimbine

1985
The role of alpha-adrenoceptors in the regulation of renal tubular sodium reabsorption and renin secretion in the rabbit.
    British journal of pharmacology, 1985, Volume: 84, Issue:3

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Brimonidine Tartrate; Dioxanes; Guanabenz; Hemodynamics; Idazoxan; Kidney; Kidney Tubules; Male; Methoxamine; Natriuresis; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Renin; Sodium

1985
Evidence for existence of postjunctional alpha 1- and alpha 2-adrenoceptors in cat pulmonary vascular bed.
    The American journal of physiology, 1985, Volume: 249, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Cats; Female; Male; Methoxamine; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Pulmonary Artery; Pulmonary Veins; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1985
Enhancement of alpha- and beta-adrenoceptor responses by elevations in vascular tone in pulmonary circulation.
    The American journal of physiology, 1986, Volume: 250, Issue:6 Pt 2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Cats; Female; Male; Muscle Tonus; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Propanolamines; Pulmonary Circulation; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1986
Heterogeneity between soluble human and rabbit splenic alpha 2-adrenoceptors.
    Biochemical pharmacology, 1986, Oct-15, Volume: 35, Issue:20

    Topics: Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; Lectins; Oxymetazoline; Phentolamine; Prazosin; Quinolizines; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Solubility; Spleen; Sulfhydryl Reagents; Yohimbine

1986
Postsynaptic alpha 1- and alpha 2-adrenergic receptors in adrenergic control of capacitance vessel tone in vivo.
    Hypertension (Dallas, Tex. : 1979), 1986, Volume: 8, Issue:11

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Blood Volume; Brimonidine Tartrate; Compliance; Dogs; Female; Male; Methoxamine; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Splanchnic Circulation; Splenectomy; Tyramine; Vasoconstriction; Yohimbine

1986
The effect of alpha 2-adrenoceptor agonists on the acid secretory responses of rat isolated gastric mucosa to electrical field stimulation.
    British journal of pharmacology, 1986, Volume: 89, Issue:2

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Dioxanes; Electric Stimulation; Gastric Acid; Gastric Mucosa; Histamine; Idazoxan; In Vitro Techniques; Male; Pentagastrin; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains

1986
Pharmacological characterization of the postsynaptic alpha-adrenoceptors in isolated canine mesenteric arteries and veins.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Dogs; Dopamine; Female; In Vitro Techniques; Male; Mesenteric Arteries; Mesenteric Veins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Synapses; Yohimbine

1987
Characterization of the alpha-adrenoceptors mediating positive inotropy of rat left atria by use of selective agonists and antagonists.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 285, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Brimonidine Tartrate; Dioxanes; Idazoxan; Imidazoles; In Vitro Techniques; Isoproterenol; Male; Methoxamine; Muscle Contraction; Myocardial Contraction; Phenylephrine; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Stimulation, Chemical

1987
Alpha 2-adrenoceptor-mediated responses to so-called selective alpha 1-adrenoceptor agonists after partial blockade of alpha 1-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dogs; Drug Interactions; In Vitro Techniques; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Phenoxybenzamine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Verapamil; Yohimbine

1987
Direct effects of alpha 2-adrenergic receptor stimulation on intravascular systemic capacity in the dog.
    Hypertension (Dallas, Tex. : 1979), 1988, Volume: 11, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Volume; Brimonidine Tartrate; Cardiopulmonary Bypass; Central Venous Pressure; Dogs; Hepatic Veins; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Tachyphylaxis; Vascular Resistance; Yohimbine

1988
Characterization of the selectivity, specificity and potency of medetomidine as an alpha 2-adrenoceptor agonist.
    European journal of pharmacology, 1988, May-20, Volume: 150, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brain; Brimonidine Tartrate; Clonidine; Female; Imidazoles; In Vitro Techniques; Male; Medetomidine; Muscle, Smooth; Mydriatics; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Vas Deferens

1988
Inhibition of cyclic AMP production by alpha 2-adrenoceptor stimulation in the guinea-pig spinal cord slices.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Prazosin; Quinoxalines; Spinal Cord; Yohimbine

1988
Loss of selectivity of so-called selective alpha 1-adrenoceptor agonists after phenoxybenzamine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1988, Volume: 338, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Female; Imidazoles; Male; Phenoxybenzamine; Phenylephrine; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1988
Evidence that the population of postjunctional-adrenoceptors mediating contraction of smooth muscle in the rabbit isolated ear vein is predominantly alpha 2.
    British journal of pharmacology, 1988, Volume: 94, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Veins; Yohimbine

1988
Evaluation of the alpha-1 and alpha-2 adrenoceptor-mediated effects of a series of dimethoxy-substituted tolazoline derivatives in the cardiovascular system of the pithed rat.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:1

    Topics: Animals; Blood Pressure; Brimonidine Tartrate; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Heart Rate; Male; Prazosin; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Spinal Cord; Tolazoline; Yohimbine

1985
Nature of alpha 1 and postjunctional alpha 2 adrenoceptors in the pulmonary vascular bed.
    Federation proceedings, 1986, Volume: 45, Issue:9

    Topics: Animals; Azepines; Blood Pressure; Brimonidine Tartrate; Cats; Hydroxydopamines; Methoxamine; Norepinephrine; Oxidopamine; Phenylephrine; Prazosin; Propranolol; Pulmonary Artery; Quinoxalines; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine

1986
A study on the postjunctional excitatory alpha-adrenoreceptor subtypes in the mesenteric arterial bed of the rat.
    Journal of autonomic pharmacology, 1986, Volume: 6, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brimonidine Tartrate; In Vitro Techniques; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Time Factors; Yohimbine

1986
Alpha adrenergic responses of blood vessels of rabbits after ovariectomy and administration of 17 beta-estradiol.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 240, Issue:2

    Topics: Animals; Blood Vessels; Brimonidine Tartrate; Estradiol; Female; Muscle, Smooth, Vascular; Norepinephrine; Ovariectomy; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Vasoconstriction; Vasomotor System; Yohimbine

1987
The contractions induced in rat and guinea-pig aortic strips by the alpha 2-adrenoceptor selective agonists B-HT 920 and UK 14,304 are mediated by alpha 1-adrenoceptors.
    European journal of pharmacology, 1984, Sep-17, Volume: 104, Issue:3-4

    Topics: Adrenergic alpha-Agonists; Animals; Aorta; Azepines; Brimonidine Tartrate; Dose-Response Relationship, Drug; Gallopamil; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Yohimbine

1984
alpha-adrenoreceptor-mediated phasic and tonic activity in rat portal vein in vitro.
    Journal of autonomic pharmacology, 1983, Volume: 3, Issue:2

    Topics: Animals; Brimonidine Tartrate; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Portal Vein; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha

1983
Noradrenergic regulation of growth hormone secretion in the baboon.
    Endocrinology, 1983, Volume: 112, Issue:1

    Topics: Albuterol; Animals; Brimonidine Tartrate; Dose-Response Relationship, Drug; Female; Growth Hormone; Male; Papio; Practolol; Prazosin; Propanolamines; Propranolol; Quinoxalines; Receptors, Adrenergic

1983
Activation of alpha-adrenoceptors indirectly facilitates sodium pumping in frog motoneurons.
    Brain research, 1993, Dec-10, Volume: 630, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Clonidine; Motor Neurons; N-Methylaspartate; Norepinephrine; Prazosin; Propranolol; Quinoxalines; Rana pipiens; Sodium-Potassium-Exchanging ATPase; Spinal Cord; Tetrodotoxin

1993
Effects of three alpha 2-adrenoceptor agonists, rilmenidine, UK 14304 and clonidine on bradykinin- and substance P-induced airway microvascular leakage in guinea-pigs.
    Neuropeptides, 1995, Volume: 28, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Bradykinin; Brimonidine Tartrate; Capillaries; Capillary Permeability; Clonidine; Dioxanes; Extravascular Lung Water; Guinea Pigs; Idazoxan; Oxazoles; Prazosin; Quinoxalines; Rilmenidine; Substance P; Trachea

1995
Comparison of the interaction of agmatine and crude methanolic extracts of bovine lung and brain with alpha 2-adrenoceptor binding sites.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Binding, Competitive; Brimonidine Tartrate; Cattle; Cerebral Cortex; Clonidine; Dioxanes; Idazoxan; Imidazoles; Lung; Methanol; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Yohimbine

1995
Adrenoceptor-stimulated endothelium-dependent relaxation in porcine intrapulmonary arteries.
    Pulmonary pharmacology, 1994, Volume: 7, Issue:5

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Arginine; Brimonidine Tartrate; Dose-Response Relationship, Drug; Endothelium, Vascular; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; Prazosin; Pulmonary Artery; Quinoxalines; Swine; Yohimbine

1994
Adrenergic modulation of a spinal sympathetic reflex in the rat.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:1

    Topics: Animals; Brimonidine Tartrate; Clonidine; Male; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reflex; Spinal Cord; Sympathetic Nervous System

1995
Activation of alpha-2-adrenoceptors results in an increase in F-actin formation in HIT-T15 pancreatic B-cells.
    The Biochemical journal, 1995, Apr-01, Volume: 307 ( Pt 1)

    Topics: Actins; Adenoma, Islet Cell; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Biopolymers; Brimonidine Tartrate; Cytochalasins; Dioxanes; Drug Interactions; Exocytosis; Fluorescent Dyes; Gene Expression Regulation; Idazoxan; Insulin; Insulin Secretion; Islets of Langerhans; Neoplasm Proteins; Norepinephrine; Pertussis Toxin; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Tumor Cells, Cultured; Virulence Factors, Bordetella

1995
Effects of alpha-adrenoceptor agonists and antagonists on metabolic rate in cattle.
    Comparative biochemistry and physiology. Part A, Physiology, 1995, Volume: 111, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Basal Metabolism; Body Temperature; Brimonidine Tartrate; Cattle; Clonidine; Dioxanes; Female; Guanfacine; Heart Rate; Idazoxan; Male; Prazosin; Quinoxalines

1995
Regional distribution and heterogeneity of alpha-adrenoceptors in the rat and human central nervous system.
    Journal fur Hirnforschung, 1993, Volume: 34, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Autoradiography; Brain; Brain Chemistry; Brimonidine Tartrate; Humans; Organ Specificity; Prazosin; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Species Specificity; Tritium; Yohimbine

1993
Neural ATP release and its alpha 2-adrenoceptor-mediated modulation in guinea-pig vas deferens.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:4

    Topics: Adenosine Triphosphate; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurons; Norepinephrine; Prazosin; Purinergic P2 Receptor Antagonists; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Purinergic P2; Suramin; Vas Deferens; Yohimbine

1993
Prejunctional alpha 2-adrenoceptors inhibit acetylcholine release from cholinergic nerves in equine airways.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 1

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Horses; Idazoxan; In Vitro Techniques; Isometric Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Sympathetic Nervous System; Trachea; Yohimbine

1993
Role of alpha 1-adrenergic receptors in the intermediolateral column in mediating the pressor responses elicited by the stimulation of ventrolateral medullary pressor area.
    Brain research, 1993, Oct-29, Volume: 626, Issue:1-2

    Topics: Adrenal Glands; Adrenergic alpha-Agonists; Amino Acids; Animals; Blood Pressure; Epinephrine; Male; Mesenteric Arteries; Microinjections; Neurons; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spinal Cord; Sympathetic Nervous System

1993
ANG II reverses selective inhibition of alpha 2-adrenoceptor sensitivity after in vitro isolation of arterioles.
    The American journal of physiology, 1993, Volume: 265, Issue:6 Pt 2

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Animals; Arterioles; Brimonidine Tartrate; Histological Techniques; In Vitro Techniques; Phenylephrine; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Yohimbine

1993
Noradrenaline decreases transmission of NMDA- and non-NMDA-receptor mediated monosynaptic EPSPs in rat prefrontal neurons in vitro.
    The European journal of neuroscience, 1993, Nov-01, Volume: 5, Issue:11

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adrenergic Antagonists; Afferent Pathways; Animals; Clonidine; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; In Vitro Techniques; Isoproterenol; Membrane Potentials; Methoxamine; Neurons; Norepinephrine; Phentolamine; Phenylephrine; Prazosin; Prefrontal Cortex; Propranolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

1993
Alpha-adrenergic receptor responsiveness in vascular smooth muscle of canine bone.
    Clinical orthopaedics and related research, 1993, Issue:287

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Female; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Regional Blood Flow; Tibia; Yohimbine

1993
Structure-activity relationships in prazosin-related compounds. 2. Role of the piperazine ring on alpha-blocking activity.
    Journal of medicinal chemistry, 1993, Mar-19, Volume: 36, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Hemodynamics; Male; Piperazines; Prazosin; Quinazolines; Quinoxalines; Rats; Rats, Inbred SHR; Stereoisomerism; Structure-Activity Relationship

1993
In vivo pharmacological profile of SL 84.0418, a new selective, peripherally active alpha 2-adrenoceptor antagonist.
    European journal of pharmacology, 1993, Apr-06, Volume: 234, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Glucose; Blood Pressure; Brimonidine Tartrate; Clonidine; Decerebrate State; Dioxanes; Epinephrine; Heart Rate; Hyperglycemia; Idazoxan; Indoles; Male; Mice; Motor Activity; Norepinephrine; Peripheral Nerves; Prazosin; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Vasoconstriction

1993
Evidence that RU 24969-induced locomotor activity in C57/B1/6 mice is specifically mediated by the 5-HT1B receptor.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Biogenic Monoamines; Brain Chemistry; Indoles; Male; Methoxydimethyltryptamines; Mice; Mice, Inbred C57BL; Motor Activity; Prazosin; Quinoxalines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Dopaminergic and alpha-adrenergic control of neurotransmission in human right atrium.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Benzazepines; Brimonidine Tartrate; Domperidone; Dopamine Agonists; Dopamine Antagonists; Electric Stimulation; Ergolines; Female; Fenoldopam; Heart Atria; Humans; In Vitro Techniques; Male; Methoxamine; Middle Aged; Norepinephrine; Prazosin; Quinoxalines; Quinpirole; Receptors, Adrenergic, alpha; Receptors, Dopamine; Sulpiride; Synaptic Transmission; Yohimbine

1995
Receptor binding profile of cyclazosin, a new alpha 1B-adrenoceptor antagonist.
    European journal of pharmacology, 1995, Dec-04, Volume: 287, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Male; Prazosin; Quinazolines; Quinoxalines; Rats; Receptors, Adrenergic, alpha-1

1995
Influence of adrenergic and cholinergic mediators on the equine jejunum in vitro.
    American journal of veterinary research, 1996, Volume: 57, Issue:6

    Topics: Acetylcholine; Adrenergic Agonists; Adrenergic Antagonists; Animals; Atropine; Brimonidine Tartrate; Calcium Channel Blockers; Cholinergic Agonists; Cholinergic Antagonists; Dose-Response Relationship, Drug; Horses; Isoproterenol; Jejunum; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxymetazoline; Parasympathetic Nervous System; Phentolamine; Phenylephrine; Prazosin; Quinoxalines; Sympathetic Nervous System; Tetrodotoxin; Verapamil; Yohimbine

1996
The actions of medetomidine may not be mediated exclusively by alpha 2-adrenoceptors in the equine saphenous vein.
    Journal of veterinary pharmacology and therapeutics, 1996, Volume: 19, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Dose-Response Relationship, Drug; Electric Stimulation; Endothelium, Vascular; Female; Horses; Imidazoles; Male; Medetomidine; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Saphenous Vein; Structure-Activity Relationship

1996
Low concentrations of angiotensin II unmask vasoconstrictory alpha 2-adrenoceptors in isolated perfused kidneys of spontaneously hypertensive rats.
    Cardiovascular research, 1995, Volume: 30, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Angiotensin II; Animals; Blood Pressure; Brimonidine Tartrate; Dioxanes; Dose-Response Relationship, Drug; Hypertension; Idazoxan; Imidazoles; Kidney; Methoxamine; Perfusion; Prazosin; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction

1995
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine

1996
Clonidine-induced increase in osmolar clearance and free water clearance via activation of two distinct alpha 2-adrenoceptor sites.
    British journal of pharmacology, 1996, Volume: 119, Issue:4

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Male; Naltrexone; Osmolar Concentration; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Water

1996
Characterization of alpha-adrenoceptor subtype(s) mediating vasoconstriction in the perfused rabbit ovarian vascular bed.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Dose-Response Relationship, Drug; Electric Stimulation; Female; Ovary; Oxidopamine; Perfusion; Prazosin; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction

1996
Adrenergic responses in silent and putative inhibitory pacemaker-like neurons of the rat rostral ventrolateral medulla in vitro.
    Neuroscience, 1997, Volume: 77, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Bicuculline; Biological Clocks; Brimonidine Tartrate; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; GABA Antagonists; Glycine Agents; Interneurons; Ion Channel Gating; Isoproterenol; Medulla Oblongata; Norepinephrine; Prazosin; Quinoxalines; Rats; Rats, Wistar; Strychnine; Synaptic Transmission; Tetrodotoxin; Yohimbine

1997
Alpha-2a/d adrenoceptor subtype stimulation by guanfacine increases osmolar clearance.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Body Water; Brimonidine Tartrate; Guanfacine; Idazoxan; Kidney; Male; Naltrexone; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2

1997
Subtype determination of soma-dendritic alpha2-autoreceptors in slices of rat locus coeruleus.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Brimonidine Tartrate; Dendrites; In Vitro Techniques; Locus Coeruleus; Maprotiline; Neurons; Norepinephrine; Phentolamine; Prazosin; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Yohimbine

1997
Alpha-adrenoceptors in equine digital veins: evidence for the presence of both alpha1 and alpha2-receptors mediating vasoconstriction.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Dopamine; Horses; Idazoxan; In Vitro Techniques; Isometric Contraction; Methoxamine; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction; Veins; Yohimbine

1997
Alpha-adrenoceptor-mediated prejunctional effects of chloroethylclonidine in the canine saphenous vein.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 282, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Autoreceptors; Brimonidine Tartrate; Clonidine; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Saphenous Vein; Yohimbine

1997
Voltage-dependent calcium currents in bulbospinal neurons of neonatal rat rostral ventrolateral medulla: modulation by alpha2-adrenergic receptors.
    Journal of neurophysiology, 1998, Volume: 79, Issue:2

    Topics: Action Potentials; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Animals, Newborn; Brimonidine Tartrate; Calcium; Calcium Channels; Calcium Channels, L-Type; Dihydropyridines; Fluorescent Dyes; Ion Channel Gating; Medulla Oblongata; omega-Agatoxin IVA; omega-Conotoxin GVIA; Patch-Clamp Techniques; Peptides; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Spider Venoms; Tyrosine 3-Monooxygenase

1998
alpha2-Adrenoceptor-mediated potassium currents in acutely dissociated rat locus coeruleus neurones.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: 4-Aminopyridine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cell Membrane Permeability; Cells, Cultured; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Isoquinolines; Kinetics; Locus Coeruleus; Membrane Potentials; Neurons; Nystatin; Patch-Clamp Techniques; Piperazines; Potassium; Potassium Channel Blockers; Potassium Channels; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Thionucleotides; Yohimbine

1998
The expression of functional postsynaptic alpha2-adrenoceptors in the corpus cavernosum smooth muscle.
    British journal of pharmacology, 1998, Volume: 123, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Cyclic AMP; Male; Muscle Contraction; Muscle, Smooth; Oxymetazoline; Penis; Phenylephrine; Prazosin; Quinoxalines; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha-2; Second Messenger Systems; Synapses; Tritium; Yohimbine

1998
Alpha-adrenoceptor subtypes of dog saphenous vein: another unusual property.
    Life sciences, 1998, Volume: 62, Issue:17-18

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Dogs; Female; Fluorescence; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Potassium Chloride; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Saphenous Vein; Signal Transduction; Yohimbine

1998
Evidence for supraspinal nervous control of external anal sphincter motility in the cat.
    Brain research, 1998, Jun-08, Volume: 795, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Anal Canal; Animals; Blood Pressure; Brimonidine Tartrate; Cats; Clonidine; Efferent Pathways; Electric Stimulation; Electromyography; Enkephalin, Leucine; Female; Injections, Intravenous; Injections, Intraventricular; Injections, Spinal; Locus Coeruleus; Male; Morphine; Narcotics; Nicergoline; Norepinephrine; Peripheral Nerves; Phenylephrine; Prazosin; Quinoxalines; Reflex; Spinal Cord

1998
Norepinephrine increases cyclic GMP levels in cerebellar cells from neuronal nitric oxide synthase knockout mice.
    Journal of neurochemistry, 1998, Volume: 71, Issue:1

    Topics: Animals; Astrocytes; Cerebellum; Cyclic GMP; Enzyme Inhibitors; Guanylate Cyclase; Mice; Mice, Knockout; Nerve Tissue Proteins; Neuronal Plasticity; Neurons; Nitric Oxide Synthase; Nitric Oxide Synthase Type I; Nitroarginine; Norepinephrine; Oxadiazoles; Prazosin; Quinoxalines; Sympatholytics; Sympathomimetics

1998
Heterogeneous effects of rapid eye movement sleep deprivation on binding to alpha- and beta-adrenergic receptor subtypes in rat brain.
    Neuroscience, 1998, Volume: 86, Issue:3

    Topics: Animals; Autoradiography; Brain; Brimonidine Tartrate; Iodine Radioisotopes; Kinetics; Male; Organ Specificity; Pindolol; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sleep Deprivation; Sleep, REM; Tritium

1998
Alpha2-adrenoceptors mediate the effect of dopamine on adult rat jejunal electrolyte transport.
    European journal of pharmacology, 1998, Aug-28, Volume: 356, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amiloride; Animals; Brimonidine Tartrate; Bucladesine; Cardiotonic Agents; Colforsin; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electric Impedance; Electrolytes; Furosemide; Ion Transport; Jejunum; Male; Ouabain; Phentolamine; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2

1998
Insights into the unusual alpha adrenoceptor subtype in dog saphenous vein using phenoxybenzamine.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Alkylating Agents; Alkylation; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Phenoxybenzamine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, alpha-2; Saphenous Vein; Yohimbine

1999
Impaired function of alpha-2 adrenoceptors in smooth muscle of mesenteric arteries from spontaneously hypertensive rats.
    British journal of pharmacology, 1998, Volume: 125, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apamin; Biological Factors; Brimonidine Tartrate; Endothelium, Vascular; Enzyme Inhibitors; Female; Hypertension; In Vitro Techniques; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nitric Oxide; Nitroarginine; Prazosin; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha-2

1998
[Signal transduction of serotonin release from enterochromaffin cells in mouse ileal crypts].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1998, Volume: 112 Suppl 1

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Clonidine; Enterochromaffin Cells; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Norepinephrine; Phosphodiesterase Inhibitors; Prazosin; Pyrrolidinones; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Rolipram; Serotonin; Signal Transduction; Yohimbine

1998
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999
Importance of agonists in alpha-adrenoceptor classification and localisation of alpha1-adrenoceptors in human prostate.
    European urology, 1999, Volume: 36 Suppl 1

    Topics: Adrenergic alpha-Agonists; Animals; Binding, Competitive; Brimonidine Tartrate; Calcium; Carotid Artery, Common; Cells, Cultured; Fibroblasts; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phenylephrine; Prazosin; Prostate; Quinoxalines; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Saphenous Vein

1999
Effects of some imidazolidine alpha2-adrenoceptor agonists in rat isolated atria.
    Journal of autonomic pharmacology, 1999, Volume: 19, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Clonidine; Drug Interactions; Electric Stimulation; Female; Heart Atria; Heart Rate; Idazoxan; Imidazoles; In Vitro Techniques; Muscle Contraction; Norepinephrine; Pargyline; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Time Factors

1999
Mechanisms of action of OPC-28326, a selective hindlimb vasodilator.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Adrenergic Antagonists; Anesthesia; Aniline Compounds; Animals; Blood Pressure; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Female; Femoral Artery; Hemodynamics; Hindlimb; In Vitro Techniques; Male; Perfusion; Phenylephrine; Piperidines; Prazosin; Quinoxalines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Vasodilator Agents; Yohimbine

1999
Characterization of human recombinant alpha(2A)-adrenoceptors expressed in Chinese hamster lung cells using extracellular acidification rate changes.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Cell Line; Cricetinae; Dexmedetomidine; Dose-Response Relationship, Drug; Doxazosin; Gene Expression; Humans; Hydrogen-Ion Concentration; Imidazoles; Norepinephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Tetrahydronaphthalenes; Yohimbine

2000
Characterization of human recombinant alpha(2A)-adrenoceptors expressed in Chinese hamster lung cells using intracellular Ca(2+) changes: evidence for cross-talk between recombinant alpha(2A)- and native alpha(1)-adrenoceptors.
    British journal of pharmacology, 2000, Volume: 129, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aniline Compounds; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Calcium; Cell Line; Cricetinae; Dexmedetomidine; Dose-Response Relationship, Drug; Doxazosin; Estrenes; Fluorescence; Gene Expression; Humans; Imidazoles; Norepinephrine; Prazosin; Pyrrolidinones; Quinoxalines; Radioligand Assay; Receptor Cross-Talk; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Signal Transduction; Tetrahydronaphthalenes; Thapsigargin; Xanthenes; Yohimbine

2000
Effect of norepinephrine receptors on trigeminal rhythm generation in newborn rats.
    Brain research bulletin, 2000, Sep-15, Volume: 53, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Bicuculline; Brimonidine Tartrate; Idazoxan; Mastication; Motor Neurons; N-Methylaspartate; Neural Pathways; Norepinephrine; Organ Culture Techniques; Phenylephrine; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Trigeminal Nuclei

2000
The alpha(1A)-adrenoceptor subtype mediates contraction in rat femoral resistance arteries.
    European journal of pharmacology, 2001, Jun-22, Volume: 422, Issue:1-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Femoral Artery; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Naphthyridines; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Tetrahydronaphthalenes; Vascular Resistance; Vasoconstriction

2001
Searching for cyclazosin analogues as alpha(1B)-adrenoceptor antagonists.
    Farmaco (Societa chimica italiana : 1989), 2003, Volume: 58, Issue:7

    Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Binding Sites; CHO Cells; Clone Cells; Cricetinae; Guinea Pigs; Humans; Male; Prazosin; Quinazolines; Quinoxalines; Rats; Receptors, Adrenergic, alpha-1; Spleen; Vas Deferens

2003
In vivo modulation of 5-hydroxytryptamine release in mouse prefrontal cortex by local 5-HT(2A) receptors: effect of antipsychotic drugs.
    The European journal of neuroscience, 2003, Volume: 18, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Aminopyridines; Anesthetics, Local; Animals; Antipsychotic Agents; Benzopyrans; Blotting, Western; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Antagonists; Fluorobenzenes; Immunohistochemistry; In Situ Hybridization; Indoles; Indophenol; Male; Mice; Mice, Inbred C57BL; Microdialysis; Piperidines; Prazosin; Prefrontal Cortex; Quinoxalines; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Thiazoles; Time Factors

2003
Norepinephrine activates extracellular-regulated kinase in cortical neurons.
    Biological psychiatry, 2003, Nov-15, Volume: 54, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Blotting, Western; Brimonidine Tartrate; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Interactions; Embryo, Mammalian; Enzyme Inhibitors; Extracellular Space; Female; Isoproterenol; Male; Mitogen-Activated Protein Kinases; Neurons; Norepinephrine; Pertussis Toxin; Phosphorylation; Prazosin; Pregnancy; Propranolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Time Factors; Yohimbine

2003
Chronic morphine treatment reduces recovery from opioid desensitization.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Sep-01, Volume: 24, Issue:35

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cocaine; Drug Tolerance; Enkephalin, Methionine; Leucine; Locus Coeruleus; Male; Monensin; Morphine; Morphine Dependence; Morphine Derivatives; Norepinephrine; Phosphorylation; Prazosin; Protein Kinase C; Protein Processing, Post-Translational; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Opioid, mu; Staurosporine; Thiorphan; Yohimbine

2004
alpha1-Adrenergic modulation of synaptic input to Purkinje neurons in rat cerebellar brain slices.
    Journal of neuroscience research, 2005, Nov-15, Volume: 82, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Adenosine Triphosphate; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Animals, Newborn; Cerebellum; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Isoproterenol; Membrane Potentials; Norepinephrine; Patch-Clamp Techniques; Phentolamine; Phenylephrine; Picrotoxin; Prazosin; Purkinje Cells; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Synapses; Tetrodotoxin; Time Factors

2005
Receptors involved in moxonidine-stimulated atrial natriuretic peptide release from isolated normotensive rat hearts.
    European journal of pharmacology, 2006, Jul-10, Volume: 541, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Atrial Natriuretic Factor; Bridged Bicyclo Compounds; Brimonidine Tartrate; Clonidine; Coronary Circulation; Drug Synergism; Female; Heart; Heart Rate; Heptanes; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Myocardium; Perfusion; Phenoxybenzamine; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Yohimbine

2006
Enaminones and norepinephrine employ convergent mechanisms to depress excitatory synaptic transmission in the rat nucleus accumbens in vitro.
    The European journal of neuroscience, 2006, Volume: 24, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cyclohexanes; Dopamine; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Antagonists; In Vitro Techniques; Male; Neural Inhibition; Norepinephrine; Nucleus Accumbens; Phosphinic Acids; Prazosin; Propanolamines; Quinoxalines; Rats; Rats, Sprague-Dawley; Synaptic Transmission

2006
Presynaptic alpha-adrenoceptors in median preoptic nucleus modulate inhibitory neurotransmission from subfornical organ and organum vasculosum lamina terminalis.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2007, Volume: 292, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cells, Cultured; Hypothalamus; Idazoxan; Imidazoles; Isoproterenol; Norepinephrine; Prazosin; Preoptic Area; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Signal Transduction; Subfornical Organ

2007
Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.
    Bioorganic & medicinal chemistry, 2007, Mar-15, Volume: 15, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Binding, Competitive; Furans; Male; Molecular Structure; Prazosin; Quinazolines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Stereoisomerism; Structure-Activity Relationship; Vas Deferens

2007
Characterization of the postjunctional alpha 2C-adrenoceptor mediating vasoconstriction to UK14304 in porcine pulmonary veins.
    British journal of pharmacology, 2007, Volume: 151, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Gene Expression; Imidazoles; In Vitro Techniques; Indoles; Isoindoles; Isoquinolines; Neuromuscular Junction; Norepinephrine; Piperazines; Prazosin; Pulmonary Veins; Quinolizines; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Swine; Vasoconstriction; Yohimbine

2007
Alpha 1-noradrenergic system role in increased motivation for cocaine intake in rats with prolonged access.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2008, Volume: 18, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Betaxolol; Brain Chemistry; Brimonidine Tartrate; Cocaine-Related Disorders; Conditioning, Operant; Data Interpretation, Statistical; Dose-Response Relationship, Drug; Immunohistochemistry; Male; Motivation; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Self Administration; Septal Nuclei

2008
Role of alpha1-adrenoceptor subtypes in the effects of methylenedioxy methamphetamine (MDMA) on body temperature in the mouse.
    British journal of pharmacology, 2008, Volume: 153, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Animals; Body Temperature; Fever; Male; Mice; N-Methyl-3,4-methylenedioxyamphetamine; Piperazines; Prazosin; Quinazolines; Quinoxalines; Receptors, Adrenergic, alpha-1; Thymine

2008
Noradrenergic control of odor recognition in a nonassociative olfactory learning task in the mouse.
    Learning & memory (Cold Spring Harbor, N.Y.), 2007, Volume: 14, Issue:12

    Topics: Adrenergic Agents; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Association Learning; Benzopyrans; Benzylamines; Brimonidine Tartrate; Imidazoles; Male; Mental Recall; Mice; Mice, Inbred C57BL; Norepinephrine; Odorants; Prazosin; Propranolol; Quinoxalines; Recognition, Psychology; Smell

2007
Noradrenergic vasoconstriction of pig prostatic small arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 2008, Volume: 376, Issue:6

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Arteries; Brimonidine Tartrate; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Signaling; Dose-Response Relationship, Drug; Electric Stimulation; Guanethidine; In Vitro Techniques; Indoles; Male; Norepinephrine; Piperazines; Prazosin; Prostate; Quinoxalines; Swine; Thymine; Vasoconstriction; Yohimbine

2008
Quantitative investigation of the role of breast cancer resistance protein (Bcrp/Abcg2) in limiting brain and testis penetration of xenobiotic compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Brain; Cell Line; Dantrolene; Dogs; Imidazoles; LLC-PK1 Cells; Male; Mice; Mice, Knockout; Prazosin; Quinoxalines; Swine; Testis; Triamterene; Xenobiotics

2008
Differential effects of prazosin and naftopidil on pelvic blood flow and nitric oxide synthase levels in spontaneously hypertensive rats.
    Journal of receptor and signal transduction research, 2008, Volume: 28, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Hypertension; Male; Naphthalenes; Nitric Oxide Synthase; Pelvis; Penis; Piperazines; Prazosin; Prostate; Quinazolines; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Adrenergic, alpha; Regional Blood Flow; Urinary Bladder

2008
Alpha-1-adrenergic receptor agonist activity of clinical alpha-adrenergic receptor agonists interferes with alpha-2-mediated analgesia.
    Anesthesiology, 2009, Volume: 110, Issue:2

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics; Animals; Brimonidine Tartrate; Calcium; Clonidine; Dinoprostone; Drug Interactions; Excitatory Amino Acid Agonists; Exploratory Behavior; Hyperalgesia; Injections, Spinal; Mice; Mice, Inbred C57BL; Mice, Knockout; N-Methylaspartate; Pain Measurement; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2

2009
Regional heterogeneity of α-adrenoreceptor subtypes in arteriolar networks of mouse skeletal muscle.
    The Journal of physiology, 2010, Nov-01, Volume: 588, Issue:Pt 21

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic beta-Antagonists; Animals; Arterioles; Brimonidine Tartrate; Isoproterenol; Male; Mice; Mice, Inbred C57BL; Models, Animal; Muscle, Skeletal; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2

2010
Dexmedetomidine induces both relaxations and contractions, via different {alpha}2-adrenoceptor subtypes, in the isolated mesenteric artery and aorta of the rat.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Aorta; Brimonidine Tartrate; Clonidine; Dexmedetomidine; Endothelium, Vascular; In Vitro Techniques; Indomethacin; Male; Mesenteric Arteries; Models, Biological; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Naphthalenes; NG-Nitroarginine Methyl Ester; Pertussis Toxin; Prazosin; Propionates; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Thromboxane

2010
Postjunctional α2C-adrenoceptors mediate vasoconstriction in rat tail artery: influence of precontraction and temperature on vasoreactivity.
    Naunyn-Schmiedeberg's archives of pharmacology, 2010, Volume: 382, Issue:5-6

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Brimonidine Tartrate; Dioxanes; Imidazoles; In Vitro Techniques; Isoindoles; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Piperazines; Prazosin; Quinolizines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Serotonin; Tail; Temperature; Vasoconstriction; Yohimbine

2010
α(2) Adrenergic and imidazoline receptor agonists prevent cue-induced cocaine seeking.
    Biological psychiatry, 2011, Oct-15, Volume: 70, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Cocaine; Cues; Dose-Response Relationship, Drug; Drug Interactions; Drug-Seeking Behavior; Extinction, Psychological; Guanfacine; Imidazoles; Imidazoline Receptors; Isoquinolines; Male; Motor Activity; Naphthyridines; Prazosin; Propranolol; Pyrimidines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration

2011
The α₁-, but not α₂-, adrenoceptor in the nucleus accumbens plays an inhibitory role upon the accumbal noradrenaline and dopamine efflux of freely moving rats.
    European journal of pharmacology, 2012, Aug-05, Volume: 688, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Brimonidine Tartrate; Clonidine; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; Idazoxan; Male; Methoxamine; Movement; Neurons; Norepinephrine; Nucleus Accumbens; Prazosin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2

2012
Contribution of α-adrenoceptor stimulation by phenylephrine to basal nitric oxide production in the isolated mouse aorta.
    Journal of cardiovascular pharmacology, 2013, Volume: 61, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Aorta, Thoracic; Brimonidine Tartrate; Dose-Response Relationship, Drug; Imidazoles; Isoindoles; Male; Mice; Mice, Inbred C57BL; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Vasoconstrictor Agents; Yohimbine

2013
Dual effects of α2 -adrenoceptors in modulating myogenic tone in sheep isolated internal anal sphincter.
    Neurogastroenterology and motility, 2014, Volume: 26, Issue:8

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Anal Canal; Animals; Brimonidine Tartrate; Clonidine; Dexmedetomidine; Muscle Contraction; Prazosin; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Sheep; Tissue Culture Techniques

2014
Partial agonist activity of α1-adrenergic receptor antagonists for chemokine (C-X-C motif) receptor 4 and atypical chemokine receptor 3.
    PloS one, 2018, Volume: 13, Issue:9

    Topics: Adrenergic alpha-1 Receptor Antagonists; beta-Arrestins; Binding Sites; Cells, Cultured; Chemokine CXCL12; Chemotaxis; Drug Evaluation, Preclinical; Drug Repositioning; HEK293 Cells; Humans; MAP Kinase Signaling System; Myocytes, Smooth Muscle; Nuclear Magnetic Resonance, Biomolecular; Prazosin; Quinazolines; Quinoxalines; Receptors, CXCR; Receptors, CXCR4

2018
Both α
    Pharmacological reports : PR, 2021, Volume: 73, Issue:1

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Male; Muscle Contraction; Norepinephrine; Phenylephrine; Piperazines; Prazosin; Quinazolines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Spleen; Thymine; Yohimbine

2021