Page last updated: 2024-08-17

quinoxalines and medetomidine

quinoxalines has been researched along with medetomidine in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19901 (6.67)18.7374
1990's11 (73.33)18.2507
2000's3 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andersson, RG; Grundström, N; Jacobsson, L1
Crosson, CE; Heath, AR; Ogidigben, MJ; Potter, DE1
Nyman, L; Saano, V; Savola, JM; Virtanen, R1
Dalley, JW; Stanford, SC1
Ohisalo, JJ; Raasmaja, A; Savola, JM; Vikman, HL1
Hein, L; Limbird, LE; MacMillan, LB; Piascik, MT; Smith, MS1
Bryant, CE; Clarke, KW1
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM1
Calcutt, NA; Chaplan, SR1
Audinot, V; Chaput, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Nicolas, JP; Richard, N; Touzard, M; Verrièle, L1
Buerkle, H; Yaksh, TL1
Haapalinna, A; Jolkkonen, J; Kauppinen, R; Koistinaho, J; Nieminen, L; Puurunen, K; Sivenius, J1
Colpaert, FC; Pauwels, PJ1
Hein, L; Klebroff, W; Meyer, A; Philipp, M; Starke, K; Trendelenburg, AU1
Chen, W; Marvizón, JC; Song, B1

Other Studies

15 other study(ies) available for quinoxalines and medetomidine

ArticleYear
Influence of some alpha 2-receptor agonists and antagonists on the excitatory non-adrenergic, non-cholinergic neurotransmission in the airways of guinea-pigs in vivo.
    Acta physiologica Scandinavica, 1991, Volume: 142, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Electric Stimulation; Guinea Pigs; Imidazoles; Male; Medetomidine; Quinoxalines; Respiratory Muscles; Respiratory System; Synaptic Transmission; Vagus Nerve

1991
Functional evidence for heterogeneity of ocular alpha 2-adrenoceptors.
    Proceedings of the Western Pharmacology Society, 1990, Volume: 33

    Topics: Anesthesia; Animals; Brimonidine Tartrate; Cats; Ciliary Body; Cyclic AMP; Dose-Response Relationship, Drug; Eye; Imidazoles; In Vitro Techniques; Iris; Isoproterenol; Medetomidine; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide

1990
Characterization of the selectivity, specificity and potency of medetomidine as an alpha 2-adrenoceptor agonist.
    European journal of pharmacology, 1988, May-20, Volume: 150, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brain; Brimonidine Tartrate; Clonidine; Female; Imidazoles; In Vitro Techniques; Male; Medetomidine; Muscle, Smooth; Mydriatics; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Vas Deferens

1988
Contrasting effects of the imidazol(in)e alpha 2-adrenoceptor agonists, medetomidine, clonidine and UK 14,304 on extraneuronal levels of noradrenaline in the rat frontal cortex: evaluation using in vivo microdialysis and synaptosomal uptake studies.
    British journal of pharmacology, 1995, Volume: 114, Issue:8

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Frontal Lobe; Imidazoles; Male; Medetomidine; Microdialysis; Norepinephrine; Quinoxalines; Rats; Rats, Sprague-Dawley; Synaptosomes; Time Factors

1995
Alpha 2A-adrenergic regulation of cyclic AMP accumulation and lipolysis in human omental and subcutaneous adipocytes.
    International journal of obesity and related metabolic disorders : journal of the International Association for the Study of Obesity, 1996, Volume: 20, Issue:2

    Topics: Abdomen; Adipocytes; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Brimonidine Tartrate; Cyclic AMP; Epinephrine; Female; Glycerol; Humans; Imidazoles; Isoproterenol; Lipolysis; Male; Medetomidine; Middle Aged; Omentum; Quinoxalines; Receptors, Adrenergic, alpha

1996
Central hypotensive effects of the alpha2a-adrenergic receptor subtype.
    Science (New York, N.Y.), 1996, Aug-09, Volume: 273, Issue:5276

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Base Sequence; Blood Pressure; Brain Stem; Brimonidine Tartrate; Gene Targeting; Heart Rate; Imidazoles; Medetomidine; Mice; Mice, Inbred C57BL; Molecular Sequence Data; Point Mutation; Quinoxalines; Receptors, Adrenergic, alpha-2

1996
The actions of medetomidine may not be mediated exclusively by alpha 2-adrenoceptors in the equine saphenous vein.
    Journal of veterinary pharmacology and therapeutics, 1996, Volume: 19, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Brimonidine Tartrate; Dose-Response Relationship, Drug; Electric Stimulation; Endothelium, Vascular; Female; Horses; Imidazoles; Male; Medetomidine; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Saphenous Vein; Structure-Activity Relationship

1996
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine

1996
Spinal pharmacology of tactile allodynia in diabetic rats.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: 2-Amino-5-phosphonovalerate; Analgesics, Non-Narcotic; Analgesics, Opioid; Animals; Anti-Bacterial Agents; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Female; Imidazoles; Injections, Spinal; Medetomidine; Morphine; Pain; Quinoxalines; Rats; Rats, Sprague-Dawley; Spinal Cord; Streptozocin

1997
Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole, and the agonist, dexmedetomidine, are highly selective for alpha2A adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brimonidine Tartrate; CHO Cells; Cricetinae; Guanfacine; Humans; Idazoxan; Imidazoles; Ligands; Medetomidine; Quinoxalines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Yohimbine

1998
Pharmacological evidence for different alpha 2-adrenergic receptor sites mediating analgesia and sedation in the rat.
    British journal of anaesthesia, 1998, Volume: 81, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesia; Analgesics, Non-Narcotic; Animals; Brimonidine Tartrate; Clonidine; Conscious Sedation; Hypnotics and Sedatives; Imidazoles; Injections, Intraventricular; Injections, Spinal; Male; Medetomidine; Pain Threshold; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Yohimbine

1998
Neuroprotection by the alpha2-adrenoceptor agonist, dexmedetomidine, in rat focal cerebral ischemia.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Arterial Occlusive Diseases; Body Weight; Cerebral Arteries; Cerebral Cortex; Cerebral Infarction; Corpus Striatum; Excitatory Amino Acid Antagonists; Imidazoles; Ischemic Attack, Transient; Male; Medetomidine; Neuroprotective Agents; Pipecolic Acids; Quinoxalines; Rats; Rats, Wistar

1999
Partial to complete antagonism by putative antagonists at the wild-type alpha(2C)-adrenoceptor based on kinetic analyses of agonist:antagonist interactions.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Azepines; Brimonidine Tartrate; Calcium; CHO Cells; Clonidine; Cricetinae; DNA, Recombinant; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; Idazoxan; Kinetics; Medetomidine; Mice; Oxymetazoline; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Transfection

2000
All three alpha2-adrenoceptor types serve as autoreceptors in postganglionic sympathetic neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoreceptors; Brimonidine Tartrate; Cattle; Cells, Cultured; Drug Interactions; Female; Ganglia, Sympathetic; Gene Expression; Heart Atria; Hippocampus; Male; Medetomidine; Mice; Mice, Inbred C57BL; Mice, Knockout; Occipital Lobe; Parietal Lobe; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Sympathetic Fibers, Postganglionic; Vas Deferens

2003
Inhibition of opioid release in the rat spinal cord by alpha2C adrenergic receptors.
    Neuropharmacology, 2008, Volume: 54, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics, Opioid; Animals; Brimonidine Tartrate; Clonidine; Data Interpretation, Statistical; Electric Stimulation; Enkephalins; Guanfacine; Immunohistochemistry; Male; Medetomidine; Microscopy, Confocal; Oligopeptides; Protease Inhibitors; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Opioid, mu; Spinal Cord; Veratridine

2008