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quinoxalines and guanosine 5'-o-(3-thiotriphosphate)

quinoxalines has been researched along with guanosine 5'-o-(3-thiotriphosphate) in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (47.62)18.2507
2000's9 (42.86)29.6817
2010's2 (9.52)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Duzic, E; Lanier, SM1
Illes, P; Regenold, JT1
Dingus, J; Hildebrandt, JD; Kataoka, R; Lanier, SM; Sato, M; Wilcox, M1
Barnes, JM; Henley, JM; Kirkham, D; Murphy, PA1
Itoh, Y; Kimura, K; Oka, M; Shimidzu, T; Ukai, Y; Yoshikuni, Y1
Akaike, N; Arima, J; Ishibashi, H; Kubo, C1
Bahia, DS; Fanelli, F; Lee, M; Milligan, G; Rees, S; Wise, A1
Bell, MI; Lee, K; Richardson, PJ1
Borea, PA; Caiazza, A; Gessi, S; Portaluppi, F; Rastelli, G; Varani, K1
Borea, PA; Campi, F; Gessi, S; Varani, K1
Bylund, DB; Happe, HK; Murrin, LC1
García-Sevilla, JA; González-Maeso, J; Guimón, J; Meana, JJ1
Barat, A; Burgos, JS; Ramírez, G1
Birdsall, NJ; Leppik, RA1
Pauwels, PJ; Rauly, I; Wurch, T1
Hoffrén, AM; Johnson, MS; Kanerva, L; Marjamäki, A; Nyrönen, T; Peltonen, JM; Pihlavisto, M; Savola, JM; Scheinin, M; Wurster, S; Xhaard, H1
Odagaki, Y; Toyoshima, R1
Pulges, O; Rinken, A1
Callado, LF; Erdozain, AM; Meana, JJ; Ortega, JE; Rodriguez, F; Rozas, I1
Aldana, I; Ancizu, S; Caignard, DH; Castrillo, N; Delagrange, P; Galiano, S; Monge, A; Pérez-Silanes, S1
Beck, SG; Calizo, LH; Campbell, K; Piel, D; Rood, BD; Spangler, ZP1

Trials

1 trial(s) available for quinoxalines and guanosine 5'-o-(3-thiotriphosphate)

ArticleYear
Platelet alpha2-adrenoceptor alterations in patients with essential hypertension.
    British journal of clinical pharmacology, 1999, Volume: 47, Issue:2

    Topics: Adrenergic alpha-Antagonists; Blood Platelets; Brimonidine Tartrate; Colforsin; Cyclic AMP; Epinephrine; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypertension; Male; Middle Aged; Protein Binding; Quinoxalines; Receptors, Adrenergic, alpha-2; Thermodynamics

1999

Other Studies

20 other study(ies) available for quinoxalines and guanosine 5'-o-(3-thiotriphosphate)

ArticleYear
Factors determining the specificity of signal transduction by guanine nucleotide-binding protein-coupled receptors. III. Coupling of alpha 2-adrenergic receptor subtypes in a cell type-specific manner.
    The Journal of biological chemistry, 1992, Nov-25, Volume: 267, Issue:33

    Topics: 3T3 Cells; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Cell Line; Colforsin; Cyclic AMP; Edetic Acid; Egtazic Acid; Epinephrine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Manganese; Mice; Muscle, Smooth; PC12 Cells; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, beta; Signal Transduction; Transfection; Virulence Factors, Bordetella

1992
Interaction between neuropeptide Y and noradrenaline on central catecholamine neurons.
    Nature, 1990, Mar-01, Volume: 344, Issue:6261

    Topics: Action Potentials; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Enkephalins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; In Vitro Techniques; Locus Coeruleus; Neuropeptide Y; Norepinephrine; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu; Thionucleotides; Yohimbine

1990
Factors determining specificity of signal transduction by G-protein-coupled receptors. Regulation of signal transfer from receptor to G-protein.
    The Journal of biological chemistry, 1995, Jun-23, Volume: 270, Issue:25

    Topics: 3T3 Cells; Adrenergic alpha-Agonists; Animals; Brain; Brimonidine Tartrate; Cattle; Cell Line; Cell Membrane; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Kinetics; Mice; PC12 Cells; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Signal Transduction; Transfection; Virulence Factors, Bordetella

1995
Interaction of guanine nucleotides with [3H]kainate and 6-[3H]cyano-7-nitroquinoxaline-2,3-dione binding in goldfish brain.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenine Nucleotides; Animals; Autoradiography; Binding Sites; Brain; Cell Membrane; Goldfish; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Kainic Acid; Kinetics; Magnesium; Quinoxalines; Radioligand Assay; Receptors, Kainic Acid; Sodium; Tritium

1993
Involvement of metabotropic glutamate receptors in Gi- and Gs-dependent modulation of adenylate cyclase activity induced by a novel cognition enhancer NS-105 in rat brain.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Alanine; Animals; Baclofen; Brimonidine Tartrate; Cell Membrane; Cerebral Cortex; Cholera Toxin; Cognition; Colforsin; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoproterenol; Kinetics; Male; Manganese; Pertussis Toxin; Piperidines; Proline; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurotransmitter; Virulence Factors, Bordetella; Yohimbine

1997
alpha2-Adrenoceptor-mediated potassium currents in acutely dissociated rat locus coeruleus neurones.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: 4-Aminopyridine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cell Membrane Permeability; Cells, Cultured; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Triphosphate; Isoquinolines; Kinetics; Locus Coeruleus; Membrane Potentials; Neurons; Nystatin; Patch-Clamp Techniques; Piperazines; Potassium; Potassium Channel Blockers; Potassium Channels; Prazosin; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Thionucleotides; Yohimbine

1998
Hydrophobicity of residue351 of the G protein Gi1 alpha determines the extent of activation by the alpha 2A-adrenoceptor.
    Biochemistry, 1998, Aug-18, Volume: 37, Issue:33

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Brimonidine Tartrate; Cell Line; Cysteine; Glycine; GTP-Binding Protein alpha Subunits, Gi-Go; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kidney; Molecular Sequence Data; Mutagenesis, Site-Directed; Pertussis Toxin; Protein Binding; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Transfection; Virulence Factors, Bordetella

1998
Characterization of the mechanism of action of tachykinins in rat striatal cholinergic interneurons.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Chelating Agents; Corpus Striatum; Diazonium Compounds; Electric Stimulation; Estrenes; Excitatory Amino Acid Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Interneurons; Male; Membrane Potentials; Patch-Clamp Techniques; Phenoxyacetates; Phosphodiesterase Inhibitors; Photochemistry; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin

1998
Alpha2-adrenergic agonist modulation of [35S]GTPgammaS binding to guanine-nucleotide-binding-proteins in human platelet membranes.
    Life sciences, 1999, Volume: 64, Issue:16

    Topics: Adrenergic alpha-Agonists; Blood Platelets; Brimonidine Tartrate; Cell Membrane; Cyclic AMP; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Humans; Kinetics; Quinoxalines; Sodium Chloride; Sulfur Radioisotopes

1999
Alpha(2)-adrenoceptor-stimulated GTP gamma S binding in rat brain: an autoradiographic study.
    European journal of pharmacology, 2000, Jun-30, Volume: 399, Issue:1

    Topics: Animals; Autoradiography; Brain; Brimonidine Tartrate; Dose-Response Relationship, Drug; Epinephrine; Female; Guanosine 5'-O-(3-Thiotriphosphate); Idazoxan; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Serotonin

2000
mu-opioid receptor and alpha2-adrenoceptor agonist stimulation of [35S]GTPgammaS binding to G-proteins in postmortem brains of opioid addicts.
    Molecular psychiatry, 2000, Volume: 5, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adult; Autopsy; Brain; Brimonidine Tartrate; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Opioid-Related Disorders; Postmortem Changes; Quinoxalines; Receptors, Opioid, mu; Reference Values; Sulfur Radioisotopes

2000
Guanine nucleotides block agonist-driven 45Ca2+ influx in chick embryo retinal explants.
    Neuroreport, 2000, Jul-14, Volume: 11, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Biological Transport; Calcium; Calcium Radioisotopes; Chick Embryo; Excitatory Amino Acid Antagonists; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Guanosine Monophosphate; N-Methylaspartate; Organ Culture Techniques; Quinoxalines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Retina; Thionucleotides

2000
Agonist binding and function at the human alpha(2A)-adrenoceptor: allosteric modulation by amilorides.
    Molecular pharmacology, 2000, Volume: 58, Issue:5

    Topics: Adrenergic alpha-Agonists; Allosteric Regulation; Amiloride; Animals; Brimonidine Tartrate; CHO Cells; Cricetinae; Diuretics; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Quinoxalines; Receptors, Adrenergic, alpha-2; Sulfur Radioisotopes; Transfection

2000
Dissimilar pharmacological responses by a new series of imidazoline derivatives at precoupled and ligand-activated alpha 2A-adrenoceptor states: evidence for effector pathway-dependent differential antagonism.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 305, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Benzopyrans; Binding Sites; Brimonidine Tartrate; CHO Cells; Cricetinae; Cyclic AMP; Epinephrine; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Idazoxan; Imidazoles; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Sulfur Radioisotopes; Tumor Cells, Cultured

2003
Molecular mechanisms of ligand-receptor interactions in transmembrane domain V of the alpha2A-adrenoceptor.
    British journal of pharmacology, 2003, Volume: 140, Issue:2

    Topics: Adrenergic Agonists; Amino Acid Sequence; Amino Acid Substitution; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Catecholamines; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Idazoxan; Ligands; Membrane Proteins; Models, Molecular; Molecular Structure; Mutation; Protein Structure, Tertiary; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Sequence Homology, Amino Acid; Sulfur Radioisotopes; Tritium

2003
5-HT1A receptor-mediated G protein activation assessed by [35S]GTPgammaS binding in rat cerebral cortex.
    European journal of pharmacology, 2005, Oct-03, Volume: 521, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Enzyme Activation; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Hippocampus; Magnesium Chloride; Male; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride; Sulfur Radioisotopes

2005
Alpha 2A-adrenoceptor-specific stimulation of [35S]GTP gamma S binding to membrane preparations of rat frontal cortex.
    Neurochemical research, 2008, Volume: 33, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brimonidine Tartrate; Clonidine; Emotions; Guanfacine; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoquinolines; Kinetics; Membranes; Naphthyridines; Prefrontal Cortex; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Signal Transduction; Stress, Psychological

2008
Guanidine and 2-aminoimidazoline aromatic derivatives as alpha2-adrenoceptor ligands: searching for structure-activity relationships.
    Journal of medicinal chemistry, 2009, Feb-12, Volume: 52, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Brimonidine Tartrate; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Imidazoles; Microdialysis; Neurons; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Structure-Activity Relationship

2009
New quinoxaline derivatives as potential MT₁ and MT₂ receptor ligands.
    Molecules (Basel, Switzerland), 2012, Jun-25, Volume: 17, Issue:7

    Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Indoles; Ligands; Naphthalenes; Quinolines; Quinoxalines; Receptor, Melatonin, MT1; Receptor, Melatonin, MT2; Structure-Activity Relationship

2012
Dorsal raphe serotonin neurons in mice: immature hyperexcitability transitions to adult state during first three postnatal weeks suggesting sensitive period for environmental perturbation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Apr-02, Volume: 34, Issue:14

    Topics: Age Factors; Animals; Animals, Newborn; Bacterial Proteins; Bicuculline; Environment; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Luminescent Proteins; Male; Mice; Mice, Transgenic; Quinoxalines; Raphe Nuclei; Serotonergic Neurons; Serotonin; Serotonin Receptor Agonists; Transcription Factors

2014