Page last updated: 2024-08-17

quinoxalines and flunitrazepam

quinoxalines has been researched along with flunitrazepam in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (88.89)18.2507
2000's1 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blakeman, DP; Carter, DB; Hamilton, BJ; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Pregenzer, JF1
Harris, LS; Nader, MA; Patrick, GA; Powell, LJ; Winger, G; Woods, JH; Woolverton, WL1
Oien, TT; Sethy, VH1
Catarzi, D; Cecchi, L; Colotta, V; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C; Melani, F2
Catarzi, D; Cecchi, L; Colotta, V; Conti, G; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C1
Belonga, KL; Carter, DB; Im, HK; Im, WB; Jacobsen, EJ; Petke, JD; Sethy, VH; Stelzer, LS; Tang, AH; TenBrink, RE; VonVoigtlander, PF1
Im, HK; Im, WB; Jacobsen, EJ; Pregenzer, JF; Stratman, NC; VonVoigtlander, PF1
Farb, DH; Gibbs, TT; Land, MB; Lyons, HR1

Other Studies

9 other study(ies) available for quinoxalines and flunitrazepam

ArticleYear
Characterization of functional interactions of imidazoquinoxaline derivatives with benzodiazepine-gamma-aminobutyric acidA receptors.
    Molecular pharmacology, 1992, Volume: 42, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chloride Channels; Chlorides; Chlorine; Cloning, Molecular; Drug Interactions; Electrophysiology; Flunitrazepam; GABA-A Receptor Antagonists; Kinetics; Male; Membrane Proteins; Models, Chemical; Molecular Conformation; Oxadiazoles; Quinoxalines; Radioisotopes; Rats; Rats, Inbred Strains; Receptors, GABA-A; Structure-Activity Relationship; Synaptosomes; Tritium

1992
Progress report from the Testing Program for Stimulant and Depressant Drugs (1991).
    NIDA research monograph, 1992, Volume: 119

    Topics: Animals; Anti-Anxiety Agents; Central Nervous System Depressants; Central Nervous System Stimulants; Discrimination, Psychological; Female; Flunitrazepam; Humans; Macaca mulatta; Male; Mice; Nitrazepam; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Self Administration; Substance-Related Disorders

1992
Role of cGMP in the mechanism of anxiolytic activity of U-78875.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain Chemistry; Carbolines; Cerebellum; Convulsants; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flunitrazepam; Male; Mice; Muscimol; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred Strains; Stress, Psychological

1991
Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor.
    Journal of medicinal chemistry, 1994, Sep-02, Volume: 37, Issue:18

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Flunitrazepam; Imidazoles; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Structure-Activity Relationship; Triazoles

1994
Tricyclic heteroaromatic systems pyrazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Pyrazoles; Quinoxalines; Receptors, GABA-A

1993
Tricyclic heteroaromatic systems 1,2,4-triazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
    Farmaco (Societa chimica italiana : 1989), 1993, Volume: 48, Issue:8

    Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Triazoles

1993
High-affinity partial agonist imidazo[1,5-a]quinoxaline amides, carbamates, and ureas at the gamma-aminobutyric acid A/benzodiazepine receptor complex.
    Journal of medicinal chemistry, 1996, Jan-05, Volume: 39, Issue:1

    Topics: Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chlorides; Flunitrazepam; GABA Agonists; GABA Antagonists; Molecular Conformation; Molecular Structure; Oxadiazoles; Pentylenetetrazole; Quinoxalines; Rats; Receptors, GABA-A

1996
Two imidazoquinoxaline ligands for the benzodiazepine site sharing a second low affinity site on rat GABA(A) receptors but with the opposite functionality.
    British journal of pharmacology, 1998, Volume: 123, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Brain; Bridged Bicyclo Compounds, Heterocyclic; Chloride Channels; Cloning, Molecular; Electric Stimulation; Electrophysiology; Flunitrazepam; GABA-A Receptor Agonists; Imidazoles; In Vitro Techniques; Ligands; Membrane Potentials; Patch-Clamp Techniques; Quinolines; Quinoxalines; Rats; Receptors, GABA-A

1998
Distinct signal transduction pathways for GABA-induced GABA(A) receptor down-regulation and uncoupling in neuronal culture: a role for voltage-gated calcium channels.
    Journal of neurochemistry, 2001, Volume: 78, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; Animals; Anti-Anxiety Agents; Brain; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Chick Embryo; Down-Regulation; Excitatory Amino Acid Antagonists; Flunitrazepam; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Nifedipine; Potassium; Quinoxalines; Receptors, GABA-A; Signal Transduction; Tetrodotoxin; Tritium

2001