quinoxalines has been researched along with diazepam in 33 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 18 (54.55) | 18.2507 |
2000's | 8 (24.24) | 29.6817 |
2010's | 6 (18.18) | 24.3611 |
2020's | 1 (3.03) | 2.80 |
Authors | Studies |
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Bas, D; Bruneau, P; Chipot, C; Dorison-Duval, D; Moreau, S | 1 |
Johnston, MV; McDonald, JW; Trescher, WH | 1 |
Castrén, E; Lindholm, D; Thoenen, H; Zafra, F | 1 |
Franklin, SR; Himes, CS; Ho, PM; Tang, AH | 1 |
Oien, TT; Sethy, VH | 1 |
Lees, GJ; Leong, W | 2 |
Karcz-Kubicha, M; Liljequist, S | 1 |
Honoré, T; Jacobsen, P; Swedberg, MD | 1 |
Cook, JM; Koehler, KF; Zhang, P; Zhang, W | 1 |
Hönack, D; Löscher, W | 1 |
Block, F; Schwarz, M | 1 |
al-Zubaidy, ZA; Chapman, AG; Meldrum, BS; Smith, SE | 1 |
Steppuhn, KG; Turski, L | 1 |
Balster, RL; Cristello, AF; Wiley, JL | 1 |
Ashby, CR; Katsumori, H; Minabe, Y; Osawa, M | 1 |
Bowen, CA; Gatto, GJ; Grant, KA | 1 |
Balster, RL; Compton, AD; Holcomb, JD; McCallum, SE; Porter, JH; Varvel, SA; Wiley, JL | 1 |
Ator, NA; Griffiths, RR | 1 |
Chopin, P; Colpaert, FC; Marien, M | 1 |
Kang-Park, MH; Moore, SD; Wilson, WA | 1 |
Balster, RL; Wiley, JL | 1 |
Cock, HR; Nilsen, KE; Walker, MC | 1 |
Accorsi-Mendonça, D; Aguiar, JF; Leão, RM; Machado, BH; Varanda, WA | 1 |
Barkóczy, J; Bilkei-Gorzó, A; Gacsályi, I; Hársing, LG; Hegedus, E; Kapus, GL; Kompagne, H; Lévay, G; Leveleki, C; Vegh, M | 1 |
Bortolatto, CF; Jesse, CR; Nogueira, CW; Savegnago, L; Wilhelm, EA | 1 |
Magara, F; Stoop, R; Terrettaz, T; Viviani, D | 1 |
Fukuhara, A; Goto, Y; Inoue, K; Inui, T; Kume, S; Lee, YH; Miyamoto, Y; Nakajima, H; Nishimura, S; Noda, M; Ohkubo, T; Shimamoto, S; Takeuchi, T; Uchiyama, S | 1 |
Hashimoto, K; Kano, M; Kitamura, K; Miyazaki, T; Nakayama, H; Obata, K; Sakimura, K; Watanabe, M; Yanagawa, Y | 1 |
Carlen, PL; El-Hayek, YH; Wang, J; Wu, C; Ye, H; Zhang, L | 1 |
Bhatt, S; Devadoss, T; Jindal, A; Mahesh, R | 1 |
Jang, HJ; Joo, K; Kim, MJ; Lee, C; Rhie, DJ | 1 |
Divaeva, LN; Ianalieva, LR; Klimenko, AI; Klochkov, VG; Maltsev, DV; Miroshnikov, MV; Morkovnik, AS; Perfiliev, MA; Skripka, MO; Spasov, AA; Vassiliev, PM; Zubenko, AA | 1 |
33 other study(ies) available for quinoxalines and diazepam
Article | Year |
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Rational determination of transfer free energies of small drugs across the water-oil interface.
Topics: Alkanes; Antipyrine; Caffeine; Computer Simulation; Ganciclovir; Glucose; Pharmaceutical Preparations; Solubility; Water | 2002 |
Susceptibility of brain to AMPA induced excitotoxicity transiently peaks during early postnatal development.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analysis of Variance; Animals; Brain; Brain Injuries; Diazepam; Dizocilpine Maleate; Female; Ibotenic Acid; Male; N-Methylaspartate; Neurotoxins; Organ Specificity; Phenytoin; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Seizures | 1992 |
Interplay between glutamate and gamma-aminobutyric acid transmitter systems in the physiological regulation of brain-derived neurotrophic factor and nerve growth factor synthesis in hippocampal neurons.
Topics: Animals; Brain-Derived Neurotrophic Factor; Diazepam; Dizocilpine Maleate; Embryo, Mammalian; Enzyme-Linked Immunosorbent Assay; Female; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Kinetics; Male; Nerve Growth Factors; Nerve Tissue Proteins; Polymerase Chain Reaction; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Glutamate; Receptors, Neurotransmitter; Reference Values; RNA, Messenger; Tetrodotoxin | 1991 |
Behavioral effects of U-78875, a quinoxalinone anxiolytic with potent benzodiazepine antagonist activity.
Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Behavior, Animal; Diazepam; Electroencephalography; Flumazenil; Injections, Intraperitoneal; Male; Motor Activity; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred F344 | 1991 |
Role of cGMP in the mechanism of anxiolytic activity of U-78875.
Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain Chemistry; Carbolines; Cerebellum; Convulsants; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flunitrazepam; Male; Mice; Muscimol; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred Strains; Stress, Psychological | 1991 |
Differential effects of NBQX on the distal and local toxicity of glutamate agonists administered intra-hippocampally.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cell Death; Diazepam; Hippocampus; Injections; Kainic Acid; Limbic System; N-Methylaspartate; Neurons; Quinoxalines; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Glutamate | 1993 |
Synergy between diazepam and NBQX in preventing neuronal death caused by non-NMDA agonists.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cell Death; Diazepam; Drug Synergism; Kainic Acid; Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA | 1994 |
Evidence for an anxiogenic action of AMPA receptor antagonists in the plus-maze test.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Motor Activity; Quinoxalines; Receptors, AMPA | 1995 |
Anticonvulsant, anxiolytic and discriminative effects of the AMPA antagonist 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(f)quinoxaline (NBQX).
Topics: Acoustic Stimulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Excitatory Amino Acid Antagonists; Female; Male; Mice; Mice, Inbred DBA; Morphine; Phencyclidine; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Seizures | 1995 |
Development of a comprehensive pharmacophore model for the benzodiazepine receptor.
Topics: Benzodiazepines; Carbolines; Computer Simulation; Diazepam; Ethanol; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hydrogen Bonding; Ligands; Models, Chemical; Molecular Conformation; Quinoxalines; Receptors, GABA-A; Structure-Activity Relationship | 1995 |
Effects of the non-NMDA antagonists NBQX and the 2,3-benzodiazepine GYKI 52466 on different seizure types in mice: comparison with diazepam and interactions with flumazenil.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Excitatory Amino Acid Antagonists; Flumazenil; Male; Mice; Muscle Relaxants, Central; Pentylenetetrazole; Quinoxalines; Receptors, AMPA; Reflex; Seizures; Synaptic Transmission | 1994 |
The depressant effect of GYKI 52466 on spinal reflex transmission in rats is mediated via non-NMDA and benzodiazepine receptors.
Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; H-Reflex; Injections, Spinal; Male; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex; Synaptic Transmission | 1994 |
Excitatory amino acid antagonists, lamotrigine and BW 1003C87 as anticonvulsants in the genetically epilepsy-prone rat.
Topics: 2-Amino-5-phosphonovalerate; Acoustic Stimulation; Amino Acids; Amino Acids, Cyclic; Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Epilepsy; Female; Lamotrigine; Male; Motor Activity; Phenytoin; Pyrimidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Time Factors; Triazines | 1993 |
Diazepam dependence prevented by glutamate antagonists.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Tolerance; Electroencephalography; Electromyography; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred Strains; Motor Activity; Muscle Tonus; Piperazines; Quinoxalines; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors | 1993 |
Effects of site-selective NMDA receptor antagonists in an elevated plus-maze model of anxiety in mice.
Topics: Amino Acids; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phencyclidine; Punishment; Quinoxalines; Rats; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate | 1995 |
Acute effects of various GABA receptor agonists and glutamate antagonists on focal hippocampal seizures in freely moving rats elicited by low-frequency stimulation.
Topics: Animals; Anticonvulsants; Ataxia; Carbamazepine; Diazepam; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Agonists; Hippocampus; Kynurenic Acid; Male; Muscimol; Pipecolic Acids; Quinoxalines; Rats; Rats, Wistar; Seizures | 1998 |
Assessment of the multiple discriminative stimulus effects of ethanol using an ethanol-pentobarbital-water discrimination in rats.
Topics: Animals; Central Nervous System Depressants; Diazepam; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ethanol; GABA Modulators; Hypnotics and Sedatives; Indoles; Male; Midazolam; Morphine; N-Methylaspartate; Narcotics; Pentobarbital; Phencyclidine; Pregnanolone; Quinoxalines; Rats; Rats, Long-Evans; Serotonin Receptor Agonists; Water | 1997 |
Effects of modulation of NMDA neurotransmission on response rate and duration in a conflict procedure in rats.
Topics: 2-Amino-5-phosphonovalerate; Acetamides; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reward; Synaptic Transmission | 1998 |
Drug discrimination analysis of partial agonists at the benzodiazepine site. I. Differential effects of U-78875 across training conditions in baboons and rats.
Topics: Acoustic Stimulation; Administration, Oral; Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Injections, Intraperitoneal; Lorazepam; Male; Oxadiazoles; Papio; Pentobarbital; Photic Stimulation; Quinoxalines; Rats; Rats, Long-Evans | 1999 |
Effects of acute and subchronic administration of dexefaroxan, an alpha(2)-adrenoceptor antagonist, on memory performance in young adult and aged rodents.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Anti-Anxiety Agents; Avoidance Learning; Basal Nucleus of Meynert; Benzopyrans; Brimonidine Tartrate; Cholinesterase Inhibitors; Cognition; Diazepam; Excitatory Amino Acid Agonists; Ibotenic Acid; Imidazoles; Male; Maze Learning; Memory; Mice; Muscarinic Antagonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Scopolamine; Tacrine | 2002 |
Differential actions of diazepam and zolpidem in basolateral and central amygdala nuclei.
Topics: Amygdala; Animals; Animals, Newborn; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; GABA Modulators; In Vitro Techniques; Male; Neural Inhibition; Patch-Clamp Techniques; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Valine; Zolpidem | 2004 |
Effects of modulators of N-methyl-D-aspartate receptor-mediated neurotransmission on diazepam discrimination in rats.
Topics: Amino Acids; Animals; Biguanides; Binding Sites; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Male; N-Methylaspartate; Pentobarbital; Phencyclidine; Piperazines; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Riluzole | 2004 |
Characterization of the tetanus toxin model of refractory focal neocortical epilepsy in the rat.
Topics: Animals; Anticonvulsants; Behavior, Animal; Brain; Diazepam; Disease Models, Animal; Electroencephalography; Electromyography; Epilepsies, Partial; Exploratory Behavior; Male; Motor Activity; Neocortex; Phenytoin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetanus Toxin | 2005 |
Urethane inhibits the GABAergic neurotransmission in the nucleus of the solitary tract of rat brain stem slices.
Topics: Anesthetics, Intravenous; Anesthetics, Local; Animals; Brain Stem; Diazepam; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Synaptic Transmission; Tetrodotoxin; Urethane | 2007 |
Antagonism of AMPA receptors produces anxiolytic-like behavior in rodents: effects of GYKI 52466 and its novel analogues.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Conflict, Psychological; Data Interpretation, Statistical; Diazepam; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Male; Membrane Potentials; Mice; Motor Activity; Neurons; Patch-Clamp Techniques; Piperazines; Quinoxalines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Telencephalon | 2008 |
Anticonvulsant and antioxidant effects of 3-alkynyl selenophene in 21-day-old rats on pilocarpine model of seizures.
Topics: Animals; Anticonvulsants; Antioxidants; Brain; Diazepam; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Kainic Acid; Male; Organoselenium Compounds; Pentylenetetrazole; Pilocarpine; Quinoxalines; Rats; Rats, Wistar; Seizures; Time Factors; Treatment Outcome | 2009 |
Oxytocin enhances the inhibitory effects of diazepam in the rat central medial amygdala.
Topics: Amygdala; Animals; Anti-Anxiety Agents; Diazepam; Drug Synergism; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Neurons; Oxytocin; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Sprague-Dawley | 2010 |
Drug delivery system for poorly water-soluble compounds using lipocalin-type prostaglandin D synthase.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain Ischemia; CA1 Region, Hippocampal; Diazepam; Disease Models, Animal; Drug Delivery Systems; Gerbillinae; Glutathione Transferase; Intramolecular Oxidoreductases; Lipocalins; Male; Mice; Pyramidal Cells; Quinoxalines; Recombinant Fusion Proteins; Solubility; Water | 2012 |
GABAergic inhibition regulates developmental synapse elimination in the cerebellum.
Topics: Agatoxins; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Bicuculline; Biophysical Phenomena; Biophysics; Calbindins; Calcium; Calcium Channels; Cerebellum; Chromones; Cytochromes c; Dendrites; Diazepam; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Microscopy, Confocal; Microscopy, Electron, Transmission; Nerve Tissue Proteins; Neurotoxins; Patch-Clamp Techniques; Phospholipase C beta; Protein Kinase C; Purkinje Cells; Quinoxalines; Receptors, Glutamate; Receptors, Metabotropic Glutamate; S100 Calcium Binding Protein G; Synapses; Vesicular Inhibitory Amino Acid Transport Proteins | 2012 |
Hippocampal excitability is increased in aged mice.
Topics: Action Potentials; Age Factors; Aging; Animals; Biophysics; Brain Waves; Diazepam; Electric Stimulation; Electroencephalography; Excitatory Amino Acid Antagonists; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Quinoxalines; Wakefulness | 2013 |
Anxiolytic-like effect of N-n-butyl-3-methoxyquinoxaline-2-carboxamide (60) in experimental mouse models of anxiety.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Molecular Structure; Quinoxalines; Receptors, Serotonin, 5-HT3 | 2013 |
GluN2B-containing N-methyl-D-aspartate receptors compensate for the inhibitory control of synaptic plasticity during the early critical period in the rat visual cortex.
Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Modulators; GABA-A Receptor Antagonists; Gene Expression Regulation, Developmental; Long-Term Potentiation; Male; Neural Inhibition; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Visual Cortex | 2015 |
Design, Synthesis and Pharmacological Evaluation of Novel C
Topics: Anti-Anxiety Agents; Diazepam; Elevated Plus Maze Test; Motor Activity; Quinoxalines | 2022 |