Page last updated: 2024-08-17

quinoxalines and diazepam

quinoxalines has been researched along with diazepam in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's18 (54.55)18.2507
2000's8 (24.24)29.6817
2010's6 (18.18)24.3611
2020's1 (3.03)2.80

Authors

AuthorsStudies
Bas, D; Bruneau, P; Chipot, C; Dorison-Duval, D; Moreau, S1
Johnston, MV; McDonald, JW; Trescher, WH1
Castrén, E; Lindholm, D; Thoenen, H; Zafra, F1
Franklin, SR; Himes, CS; Ho, PM; Tang, AH1
Oien, TT; Sethy, VH1
Lees, GJ; Leong, W2
Karcz-Kubicha, M; Liljequist, S1
Honoré, T; Jacobsen, P; Swedberg, MD1
Cook, JM; Koehler, KF; Zhang, P; Zhang, W1
Hönack, D; Löscher, W1
Block, F; Schwarz, M1
al-Zubaidy, ZA; Chapman, AG; Meldrum, BS; Smith, SE1
Steppuhn, KG; Turski, L1
Balster, RL; Cristello, AF; Wiley, JL1
Ashby, CR; Katsumori, H; Minabe, Y; Osawa, M1
Bowen, CA; Gatto, GJ; Grant, KA1
Balster, RL; Compton, AD; Holcomb, JD; McCallum, SE; Porter, JH; Varvel, SA; Wiley, JL1
Ator, NA; Griffiths, RR1
Chopin, P; Colpaert, FC; Marien, M1
Kang-Park, MH; Moore, SD; Wilson, WA1
Balster, RL; Wiley, JL1
Cock, HR; Nilsen, KE; Walker, MC1
Accorsi-Mendonça, D; Aguiar, JF; Leão, RM; Machado, BH; Varanda, WA1
Barkóczy, J; Bilkei-Gorzó, A; Gacsályi, I; Hársing, LG; Hegedus, E; Kapus, GL; Kompagne, H; Lévay, G; Leveleki, C; Vegh, M1
Bortolatto, CF; Jesse, CR; Nogueira, CW; Savegnago, L; Wilhelm, EA1
Magara, F; Stoop, R; Terrettaz, T; Viviani, D1
Fukuhara, A; Goto, Y; Inoue, K; Inui, T; Kume, S; Lee, YH; Miyamoto, Y; Nakajima, H; Nishimura, S; Noda, M; Ohkubo, T; Shimamoto, S; Takeuchi, T; Uchiyama, S1
Hashimoto, K; Kano, M; Kitamura, K; Miyazaki, T; Nakayama, H; Obata, K; Sakimura, K; Watanabe, M; Yanagawa, Y1
Carlen, PL; El-Hayek, YH; Wang, J; Wu, C; Ye, H; Zhang, L1
Bhatt, S; Devadoss, T; Jindal, A; Mahesh, R1
Jang, HJ; Joo, K; Kim, MJ; Lee, C; Rhie, DJ1
Divaeva, LN; Ianalieva, LR; Klimenko, AI; Klochkov, VG; Maltsev, DV; Miroshnikov, MV; Morkovnik, AS; Perfiliev, MA; Skripka, MO; Spasov, AA; Vassiliev, PM; Zubenko, AA1

Other Studies

33 other study(ies) available for quinoxalines and diazepam

ArticleYear
Rational determination of transfer free energies of small drugs across the water-oil interface.
    Journal of medicinal chemistry, 2002, Jan-03, Volume: 45, Issue:1

    Topics: Alkanes; Antipyrine; Caffeine; Computer Simulation; Ganciclovir; Glucose; Pharmaceutical Preparations; Solubility; Water

2002
Susceptibility of brain to AMPA induced excitotoxicity transiently peaks during early postnatal development.
    Brain research, 1992, Jun-26, Volume: 583, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Aging; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Analysis of Variance; Animals; Brain; Brain Injuries; Diazepam; Dizocilpine Maleate; Female; Ibotenic Acid; Male; N-Methylaspartate; Neurotoxins; Organ Specificity; Phenytoin; Quinoxalines; Quisqualic Acid; Rats; Rats, Inbred Strains; Seizures

1992
Interplay between glutamate and gamma-aminobutyric acid transmitter systems in the physiological regulation of brain-derived neurotrophic factor and nerve growth factor synthesis in hippocampal neurons.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, Nov-15, Volume: 88, Issue:22

    Topics: Animals; Brain-Derived Neurotrophic Factor; Diazepam; Dizocilpine Maleate; Embryo, Mammalian; Enzyme-Linked Immunosorbent Assay; Female; gamma-Aminobutyric Acid; Glutamates; Hippocampus; Kinetics; Male; Nerve Growth Factors; Nerve Tissue Proteins; Polymerase Chain Reaction; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, GABA-A; Receptors, Glutamate; Receptors, Neurotransmitter; Reference Values; RNA, Messenger; Tetrodotoxin

1991
Behavioral effects of U-78875, a quinoxalinone anxiolytic with potent benzodiazepine antagonist activity.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Avoidance Learning; Behavior, Animal; Diazepam; Electroencephalography; Flumazenil; Injections, Intraperitoneal; Male; Motor Activity; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred F344

1991
Role of cGMP in the mechanism of anxiolytic activity of U-78875.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Binding, Competitive; Brain Chemistry; Carbolines; Cerebellum; Convulsants; Cyclic GMP; Diazepam; Dose-Response Relationship, Drug; Electroshock; Flunitrazepam; Male; Mice; Muscimol; Oxadiazoles; Quinoxalines; Rats; Rats, Inbred Strains; Stress, Psychological

1991
Differential effects of NBQX on the distal and local toxicity of glutamate agonists administered intra-hippocampally.
    Brain research, 1993, Nov-19, Volume: 628, Issue:1-2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cell Death; Diazepam; Hippocampus; Injections; Kainic Acid; Limbic System; N-Methylaspartate; Neurons; Quinoxalines; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Glutamate

1993
Synergy between diazepam and NBQX in preventing neuronal death caused by non-NMDA agonists.
    Neuroreport, 1994, Oct-27, Volume: 5, Issue:16

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Cell Death; Diazepam; Drug Synergism; Kainic Acid; Neurons; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA

1994
Evidence for an anxiogenic action of AMPA receptor antagonists in the plus-maze test.
    European journal of pharmacology, 1995, Jun-12, Volume: 279, Issue:2-3

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Maze Learning; Mice; Mice, Inbred C57BL; Motor Activity; Quinoxalines; Receptors, AMPA

1995
Anticonvulsant, anxiolytic and discriminative effects of the AMPA antagonist 2,3-dihydroxy-6-nitro-7-sulfamoyl-benzo(f)quinoxaline (NBQX).
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:3

    Topics: Acoustic Stimulation; Animals; Anti-Anxiety Agents; Anticonvulsants; Diazepam; Excitatory Amino Acid Antagonists; Female; Male; Mice; Mice, Inbred DBA; Morphine; Phencyclidine; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Seizures

1995
Development of a comprehensive pharmacophore model for the benzodiazepine receptor.
    Drug design and discovery, 1995, Volume: 12, Issue:3

    Topics: Benzodiazepines; Carbolines; Computer Simulation; Diazepam; Ethanol; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; Hydrogen Bonding; Ligands; Models, Chemical; Molecular Conformation; Quinoxalines; Receptors, GABA-A; Structure-Activity Relationship

1995
Effects of the non-NMDA antagonists NBQX and the 2,3-benzodiazepine GYKI 52466 on different seizure types in mice: comparison with diazepam and interactions with flumazenil.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electroshock; Excitatory Amino Acid Antagonists; Flumazenil; Male; Mice; Muscle Relaxants, Central; Pentylenetetrazole; Quinoxalines; Receptors, AMPA; Reflex; Seizures; Synaptic Transmission

1994
The depressant effect of GYKI 52466 on spinal reflex transmission in rats is mediated via non-NMDA and benzodiazepine receptors.
    European journal of pharmacology, 1994, Apr-21, Volume: 256, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Depression, Chemical; Diazepam; Dose-Response Relationship, Drug; Electric Stimulation; H-Reflex; Injections, Spinal; Male; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, GABA-A; Receptors, N-Methyl-D-Aspartate; Reflex; Synaptic Transmission

1994
Excitatory amino acid antagonists, lamotrigine and BW 1003C87 as anticonvulsants in the genetically epilepsy-prone rat.
    Epilepsy research, 1993, Volume: 15, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; Acoustic Stimulation; Amino Acids; Amino Acids, Cyclic; Analysis of Variance; Animals; Anticonvulsants; Behavior, Animal; Diazepam; Disease Models, Animal; Dizocilpine Maleate; Epilepsy; Female; Lamotrigine; Male; Motor Activity; Phenytoin; Pyrimidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Time Factors; Triazines

1993
Diazepam dependence prevented by glutamate antagonists.
    Proceedings of the National Academy of Sciences of the United States of America, 1993, Jul-15, Volume: 90, Issue:14

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Diazepam; Drug Tolerance; Electroencephalography; Electromyography; Excitatory Amino Acid Antagonists; Male; Mice; Mice, Inbred Strains; Motor Activity; Muscle Tonus; Piperazines; Quinoxalines; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

1993
Effects of site-selective NMDA receptor antagonists in an elevated plus-maze model of anxiety in mice.
    European journal of pharmacology, 1995, Dec-27, Volume: 294, Issue:1

    Topics: Amino Acids; Animals; Anti-Anxiety Agents; Anxiety; Diazepam; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Modulators; Male; Mice; Mice, Inbred ICR; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phencyclidine; Punishment; Quinoxalines; Rats; Receptors, Glycine; Receptors, N-Methyl-D-Aspartate

1995
Acute effects of various GABA receptor agonists and glutamate antagonists on focal hippocampal seizures in freely moving rats elicited by low-frequency stimulation.
    Synapse (New York, N.Y.), 1998, Volume: 28, Issue:1

    Topics: Animals; Anticonvulsants; Ataxia; Carbamazepine; Diazepam; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Agonists; Hippocampus; Kynurenic Acid; Male; Muscimol; Pipecolic Acids; Quinoxalines; Rats; Rats, Wistar; Seizures

1998
Assessment of the multiple discriminative stimulus effects of ethanol using an ethanol-pentobarbital-water discrimination in rats.
    Behavioural pharmacology, 1997, Volume: 8, Issue:4

    Topics: Animals; Central Nervous System Depressants; Diazepam; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ethanol; GABA Modulators; Hypnotics and Sedatives; Indoles; Male; Midazolam; Morphine; N-Methylaspartate; Narcotics; Pentobarbital; Phencyclidine; Pregnanolone; Quinoxalines; Rats; Rats, Long-Evans; Serotonin Receptor Agonists; Water

1997
Effects of modulation of NMDA neurotransmission on response rate and duration in a conflict procedure in rats.
    Neuropharmacology, 1998, Volume: 37, Issue:12

    Topics: 2-Amino-5-phosphonovalerate; Acetamides; Animals; Anti-Anxiety Agents; Chlordiazepoxide; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Electroshock; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Reward; Synaptic Transmission

1998
Drug discrimination analysis of partial agonists at the benzodiazepine site. I. Differential effects of U-78875 across training conditions in baboons and rats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Acoustic Stimulation; Administration, Oral; Animals; Anti-Anxiety Agents; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; GABA-A Receptor Agonists; Injections, Intraperitoneal; Lorazepam; Male; Oxadiazoles; Papio; Pentobarbital; Photic Stimulation; Quinoxalines; Rats; Rats, Long-Evans

1999
Effects of acute and subchronic administration of dexefaroxan, an alpha(2)-adrenoceptor antagonist, on memory performance in young adult and aged rodents.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 301, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Anti-Anxiety Agents; Avoidance Learning; Basal Nucleus of Meynert; Benzopyrans; Brimonidine Tartrate; Cholinesterase Inhibitors; Cognition; Diazepam; Excitatory Amino Acid Agonists; Ibotenic Acid; Imidazoles; Male; Maze Learning; Memory; Mice; Muscarinic Antagonists; Quinoxalines; Rats; Rats, Sprague-Dawley; Scopolamine; Tacrine

2002
Differential actions of diazepam and zolpidem in basolateral and central amygdala nuclei.
    Neuropharmacology, 2004, Volume: 46, Issue:1

    Topics: Amygdala; Animals; Animals, Newborn; Bicuculline; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; GABA Modulators; In Vitro Techniques; Male; Neural Inhibition; Patch-Clamp Techniques; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Valine; Zolpidem

2004
Effects of modulators of N-methyl-D-aspartate receptor-mediated neurotransmission on diazepam discrimination in rats.
    Life sciences, 2004, May-28, Volume: 75, Issue:2

    Topics: Amino Acids; Animals; Biguanides; Binding Sites; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Agonists; Male; N-Methylaspartate; Pentobarbital; Phencyclidine; Piperazines; Quinolones; Quinoxalines; Rats; Rats, Sprague-Dawley; Riluzole

2004
Characterization of the tetanus toxin model of refractory focal neocortical epilepsy in the rat.
    Epilepsia, 2005, Volume: 46, Issue:2

    Topics: Animals; Anticonvulsants; Behavior, Animal; Brain; Diazepam; Disease Models, Animal; Electroencephalography; Electromyography; Epilepsies, Partial; Exploratory Behavior; Male; Motor Activity; Neocortex; Phenytoin; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Tetanus Toxin

2005
Urethane inhibits the GABAergic neurotransmission in the nucleus of the solitary tract of rat brain stem slices.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2007, Volume: 292, Issue:1

    Topics: Anesthetics, Intravenous; Anesthetics, Local; Animals; Brain Stem; Diazepam; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Synaptic Transmission; Tetrodotoxin; Urethane

2007
Antagonism of AMPA receptors produces anxiolytic-like behavior in rodents: effects of GYKI 52466 and its novel analogues.
    Psychopharmacology, 2008, Volume: 198, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Conflict, Psychological; Data Interpretation, Statistical; Diazepam; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Male; Membrane Potentials; Mice; Motor Activity; Neurons; Patch-Clamp Techniques; Piperazines; Quinoxalines; Radioligand Assay; Rats; Rats, Wistar; Receptors, AMPA; Telencephalon

2008
Anticonvulsant and antioxidant effects of 3-alkynyl selenophene in 21-day-old rats on pilocarpine model of seizures.
    Brain research bulletin, 2009, Jun-30, Volume: 79, Issue:5

    Topics: Animals; Anticonvulsants; Antioxidants; Brain; Diazepam; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Kainic Acid; Male; Organoselenium Compounds; Pentylenetetrazole; Pilocarpine; Quinoxalines; Rats; Rats, Wistar; Seizures; Time Factors; Treatment Outcome

2009
Oxytocin enhances the inhibitory effects of diazepam in the rat central medial amygdala.
    Neuropharmacology, 2010, Volume: 58, Issue:1

    Topics: Amygdala; Animals; Anti-Anxiety Agents; Diazepam; Drug Synergism; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Neural Inhibition; Neurons; Oxytocin; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Sprague-Dawley

2010
Drug delivery system for poorly water-soluble compounds using lipocalin-type prostaglandin D synthase.
    Journal of controlled release : official journal of the Controlled Release Society, 2012, Apr-10, Volume: 159, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain Ischemia; CA1 Region, Hippocampal; Diazepam; Disease Models, Animal; Drug Delivery Systems; Gerbillinae; Glutathione Transferase; Intramolecular Oxidoreductases; Lipocalins; Male; Mice; Pyramidal Cells; Quinoxalines; Recombinant Fusion Proteins; Solubility; Water

2012
GABAergic inhibition regulates developmental synapse elimination in the cerebellum.
    Neuron, 2012, Apr-26, Volume: 74, Issue:2

    Topics: Agatoxins; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Bicuculline; Biophysical Phenomena; Biophysics; Calbindins; Calcium; Calcium Channels; Cerebellum; Chromones; Cytochromes c; Dendrites; Diazepam; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Modulators; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation, Developmental; Glutamate Decarboxylase; Green Fluorescent Proteins; In Vitro Techniques; Membrane Potentials; Mice; Mice, Inbred C57BL; Mice, Transgenic; Microscopy, Confocal; Microscopy, Electron, Transmission; Nerve Tissue Proteins; Neurotoxins; Patch-Clamp Techniques; Phospholipase C beta; Protein Kinase C; Purkinje Cells; Quinoxalines; Receptors, Glutamate; Receptors, Metabotropic Glutamate; S100 Calcium Binding Protein G; Synapses; Vesicular Inhibitory Amino Acid Transport Proteins

2012
Hippocampal excitability is increased in aged mice.
    Experimental neurology, 2013, Volume: 247

    Topics: Action Potentials; Age Factors; Aging; Animals; Biophysics; Brain Waves; Diazepam; Electric Stimulation; Electroencephalography; Excitatory Amino Acid Antagonists; Hippocampus; Hypnotics and Sedatives; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neurons; Patch-Clamp Techniques; Quinoxalines; Wakefulness

2013
Anxiolytic-like effect of N-n-butyl-3-methoxyquinoxaline-2-carboxamide (60) in experimental mouse models of anxiety.
    Indian journal of experimental biology, 2013, Volume: 51, Issue:7

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Behavior, Animal; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Male; Mice; Molecular Structure; Quinoxalines; Receptors, Serotonin, 5-HT3

2013
GluN2B-containing N-methyl-D-aspartate receptors compensate for the inhibitory control of synaptic plasticity during the early critical period in the rat visual cortex.
    Journal of neuroscience research, 2015, Volume: 93, Issue:9

    Topics: 2-Amino-5-phosphonovalerate; Age Factors; Animals; Animals, Newborn; Bicuculline; Diazepam; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Modulators; GABA-A Receptor Antagonists; Gene Expression Regulation, Developmental; Long-Term Potentiation; Male; Neural Inhibition; Piperidines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, N-Methyl-D-Aspartate; Visual Cortex

2015
Design, Synthesis and Pharmacological Evaluation of Novel C
    International journal of molecular sciences, 2022, Nov-19, Volume: 23, Issue:22

    Topics: Anti-Anxiety Agents; Diazepam; Elevated Plus Maze Test; Motor Activity; Quinoxalines

2022