Page last updated: 2024-08-17

quinoxalines and cyclothiazide

quinoxalines has been researched along with cyclothiazide in 51 studies

Research

Studies (51)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's24 (47.06)18.2507
2000's20 (39.22)29.6817
2010's7 (13.73)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balázs, R; Hack, N1
Berger, T1
Lodge, D; Palmer, AJ1
Mennerick, S; Zorumski, CF1
Trussell, LO; Zhang, S1
Tang, CM; Yamada, KA1
Gallo, V; Holtzclaw, LA; Russell, JT1
Turetsky, DM; Yamada, KA1
Fedele, E; Raiteri, M1
Mendelowitz, D; Mihalevich, M; Neff, RA; Willis, A1
Cebers, G; Hou, YN; Liljequist, S; Terenius, L1
Bristow, DR; Savidge, JR1
Bonfanti, A; Pittaluga, A; Raiteri, M1
Fontana, G; Gemignani, A; Marchese, S; Raiteri, M1
Conti, A; Fedele, E; Raiteri, M1
Ohno, K; Okada, M; Sakamoto, S; Tsutsumi, R; Yamaguchi, T1
Daggett, LP; Deal, C; Hess, SD; Jachec, C; Johnson, EC; Lin, F; Rao, SP; Varney, MA; Veliçelebi, G1
Yamada, KA1
Holmberg, L; Souverbie, F; Sundström, E1
Covey, DF; Hill, MW; Hu, Y; Yamada, KA1
Higashiyama, A; Ishida, N; Kato, N; Yasuda, S1
Badre, SE; Morsette, DJ; Sidorowicz, HE; Sladek, CD1
Arvigo, D; Bonfanti, A; Pittaluga, A; Raiteri, M1
Dzubay, JA; Jahr, CE1
Isaac, JT; Kidd, FL1
Kohda, K; Wang, Y; Yuzaki, M1
Dietrich, D; Dybek, A; Schumacher, TB; Seifert, G; Steinhäuser, C; Weiser, T; Wienrich, M; Wilhelm, D; Zhou, M1
Durkin, JP; Gendron, TF; MacLean, S; Mealing, G; Morley, P; Small, DL; Tremblay, R1
Higashiyama, A; Ishida, N; Kato, N; Morinobu, S; Yasuda, S1
Closier, M; Iop, F; Lestage, P; Lockhart, B1
Kondo, M; Okabe, S; Okado, H; Sumino, R1
Croucher, MJ; Patel, DR; Young, AM1
Linden, DJ1
Allgaier, C; Fischer, W; Franke, H; Illes, P; Scheibler, P1
Chiappalone, M; Davide, F; Marcoli, M; Martinoia, S; Tedesco, MB; Vato, A1
Bruno, V; Caciagli, F; Caricasole, A; Caruso, A; Castiglione, M; Di Giorgi Gerevini, V; Marinelli, F; Melchiorri, D; Moretti, A; Nicoletti, F; Pozzilli, C; Tomassini, V1
Ambrósio, AF; Araújo, IM; Carvalho, CM; Verdasca, MJ1
Li, W; Massey, SC; Trexler, EB1
Cadetti, L; Thoreson, WB; Tranchina, D1
Barygin, OI; Dorofeeva, NA; Magazanik, LG; Salnikov, YI; Tikhonov, DB; Tikhonova, TB1
Bräuner-Osborne, H; Jensen, AA; Strange, M1
Fuda, H; Hanyu, O; Kohjitani, A; Strott, CA1
Bonnot, A; Chub, N; O'Donovan, MJ; Pujala, A1
Eguchi, K; Kanda, T; Takahashi, T; Yamashita, T1
Glowatzki, E; Grant, L; Yi, E1
Chavis, P; Farrugia, F; Garenne, A; Le Masson, G; Manzoni, OJ; Marsicano, G; Piet, R1
Fukui, K; Ishiwata, S; Nishikawa, T; Umino, A; Umino, M; Yorita, K1
Baranovic, J; Kasai, N; Madden, DR; Midgett, CR; Ramanujan, CS; Ryan, JF; Torimitsu, K1
Blachowicz, L; Ghisi, V; Lau, AY; Plested, AJ; Roux, B; Salazar, H1
Asaoka, N; Kaneko, S; Nagayasu, K; Nakagawa, T; Nishitani, N; Shirakawa, H; Yamashiro, M1
Benke, TA; Kirk, ME; Meredith, FL; Rennie, KJ1

Other Studies

51 other study(ies) available for quinoxalines and cyclothiazide

ArticleYear
Properties of AMPA receptors expressed in rat cerebellar granule cell cultures: Ca2+ influx studies.
    Journal of neurochemistry, 1995, Volume: 65, Issue:3

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Calcium Radioisotopes; Cell Survival; Cells, Cultured; Cerebellum; Cobalt; Concanavalin A; Excitatory Amino Acids; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Wheat Germ Agglutinins

1995
AMPA-type glutamate receptors in glial precursor cells of the rat corpus callosum: ionic and pharmacological properties.
    Glia, 1995, Volume: 14, Issue:2

    Topics: Animals; Benzothiadiazines; Calcium; Chlorides; Concanavalin A; Corpus Callosum; Diuretics; Evans Blue; Kainic Acid; Neuroglia; Patch-Clamp Techniques; Quinoxalines; Rats; Receptors, AMPA; Receptors, Kainic Acid; Sodium Chloride Symporter Inhibitors; Zinc Compounds

1995
Cyclothiazide reverses AMPA receptor antagonism of the 2,3-benzodiazepine, GYKI 53655.
    European journal of pharmacology, 1993, Jan-15, Volume: 244, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Cerebral Cortex; Diuretics; Excitatory Amino Acid Antagonists; Ibotenic Acid; In Vitro Techniques; Kainic Acid; N-Methylaspartate; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1993
Presynaptic influence on the time course of fast excitatory synaptic currents in cultured hippocampal cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Animals, Newborn; Anti-Anxiety Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Evoked Potentials; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kinetics; Magnesium; Neurons; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synapses; Time Factors

1995
Voltage clamp analysis of excitatory synaptic transmission in the avian nucleus magnocellularis.
    The Journal of physiology, 1994, Oct-01, Volume: 480 ( Pt 1)

    Topics: 2-Amino-5-phosphonovalerate; Animals; Basal Ganglia; Benzothiadiazines; Brain Stem; Chick Embryo; Diuretics; Electric Stimulation; Electrophysiology; Evoked Potentials; In Vitro Techniques; Patch-Clamp Techniques; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors; Synapses; Synaptic Transmission; Temperature; Vestibulocochlear Nerve

1994
Benzothiadiazides inhibit rapid glutamate receptor desensitization and enhance glutamatergic synaptic currents.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:9

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzothiadiazines; Cell Line; Cells, Cultured; Diazoxide; Diuretics; Electric Stimulation; Evoked Potentials; Hippocampus; Humans; Kainic Acid; Membrane Potentials; Molecular Structure; N-Methylaspartate; Neurons; Quinoxalines; Quisqualic Acid; Rats; Receptors, Glutamate; Structure-Activity Relationship; Synapses; Time Factors

1993
AMPA receptors shape Ca2+ responses in cortical oligodendrocyte progenitors and CG-4 cells.
    Journal of neuroscience research, 1995, Sep-01, Volume: 42, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cell Line; Cells, Cultured; Dose-Response Relationship, Drug; Glutamic Acid; Kainic Acid; Oligodendroglia; Quinoxalines; Receptors, AMPA; Time Factors

1995
Allosteric interactions between cyclothiazide and AMPA/kainate receptor antagonists.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Allosteric Regulation; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Drug Interactions; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid

1996
Desensitization of AMPA receptors and AMPA-NMDA receptor interaction: an in vivo cyclic GMP microdialysis study in rat cerebellum.
    British journal of pharmacology, 1996, Volume: 117, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cerebellum; Cyclic GMP; Dizocilpine Maleate; Male; Microdialysis; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

1996
Three types of postsynaptic glutamatergic receptors are activated in DMNX neurons upon stimulation of NTS.
    The American journal of physiology, 1996, Volume: 271, Issue:6 Pt 2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzothiadiazines; Brain; Concanavalin A; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Neurons; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Solitary Nucleus; Synapses; Vagus Nerve

1996
Characterization of NMDA- and AMPA-induced enhancement of AP-1 DNA binding activity in rat cerebellar granule cells.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Cerebellum; Dizocilpine Maleate; DNA-Binding Proteins; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Kinetics; N-Methylaspartate; Neurons; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Transcription Factor AP-1

1997
Distribution of Ca(2+)-permeable AMPA receptors among cultured rat cerebellar granule cells.
    Neuroreport, 1997, May-27, Volume: 8, Issue:8

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cells, Cultured; Cerebellum; Culture Media; Culture Media, Serum-Free; Diuretics; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fluorescent Dyes; Fura-2; Manganese; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1997
Differential desensitization of ionotropic non-NMDA receptors having distinct neuronal location and function.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:1

    Topics: Acetylcholine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cerebral Cortex; Choline; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; In Vitro Techniques; Kainic Acid; Male; Norepinephrine; Potassium; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Serotonin; Synaptosomes

1997
Neuropeptide Y release from cultured hippocampal neurons: stimulation by glutamate acting at N-methyl-D-aspartate and AMPA receptors.
    Neuroscience, 1997, Volume: 81, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antibody Specificity; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Chromatography, High Pressure Liquid; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Kainic Acid; Magnesium; Neurons; Neuropeptide Y; Quinoxalines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tetrodotoxin

1997
The glutamate receptor/NO/cyclic GMP pathway in the hippocampus of freely moving rats: modulation by cyclothiazide, interaction with GABA and the behavioural consequences.
    Neuropharmacology, 1997, Volume: 36, Issue:10

    Topics: Animals; Behavior, Animal; Benzothiadiazines; Cyclic GMP; Diuretics; Drug Interactions; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Nitric Oxide; Nitric Oxide Synthase; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors

1997
The AMPA-receptor antagonist YM90K reduces AMPA receptor-mediated excitotoxicity in rat hippocampal cultures.
    Japanese journal of pharmacology, 1998, Volume: 76, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Cells, Cultured; Diuretics; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Kainic Acid; Neurons; Neuroprotective Agents; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1998
Pharmacological characterization of the human ionotropic glutamate receptor subtype GluR3 stably expressed in mammalian cells.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 285, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Binding, Competitive; Brain; Cells, Cultured; Diuretics; Electrophysiology; Excitatory Amino Acid Antagonists; Hippocampus; Humans; Kidney; Quinoxalines; Rats; Receptors, AMPA; Sodium Chloride Symporter Inhibitors

1998
AMPA receptor activation potentiated by the AMPA modulator 1-BCP is toxic to cultured rat hippocampal neurons.
    Neuroscience letters, 1998, Jun-19, Volume: 249, Issue:2-3

    Topics: Animals; Benzothiadiazines; Cell Survival; Cells, Cultured; Dioxoles; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Neurons; Neurotoxins; Piperidines; Quinoxalines; Rats; Receptors, AMPA

1998
NMDA and AMPA receptors evoke transmitter release from noradrenergic axon terminals in the rat spinal cord.
    Neurochemical research, 1998, Volume: 23, Issue:12

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Concanavalin A; Dizocilpine Maleate; In Vitro Techniques; Kainic Acid; Male; N-Methylaspartate; Norepinephrine; Presynaptic Terminals; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Tetrodotoxin

1998
The diazoxide derivative 7-chloro-3-methyl-3,4-dihydro-2H-1,2,4-benzothiadiazine-S,S-dioxide augments AMPA- and GABA-mediated synaptic responses in cultured hippocampal neurons.
    Neurobiology of disease, 1998, Volume: 5, Issue:3

    Topics: Animals; Animals, Newborn; Antihypertensive Agents; Benzothiadiazines; Cells, Cultured; Dizocilpine Maleate; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glutamic Acid; Hippocampus; Neural Inhibition; Neurons; Neurotoxins; Patch-Clamp Techniques; Quinoxalines; Rats; Receptors, AMPA; Receptors, GABA; Synapses; Synaptic Transmission

1998
[Running fit and generalized tonic-clonic seizure are differently controlled by different subtype receptors in the brainstem].
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 1998, Volume: 18, Issue:4

    Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anticonvulsants; Benzothiadiazines; Brain Stem; Dizocilpine Maleate; Epilepsy, Tonic-Clonic; Excitatory Amino Acid Agonists; Inferior Colliculi; N-Methylaspartate; Neuroprotective Agents; Propylthiouracil; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Seizures

1998
Role of non-NMDA receptors in osmotic and glutamate stimulation of vasopressin release: effect of rapid receptor desensitization.
    Journal of neuroendocrinology, 1998, Volume: 10, Issue:12

    Topics: Animals; Benzothiadiazines; Concanavalin A; Down-Regulation; Excitatory Amino Acid Antagonists; Glutamic Acid; Hypothalamo-Hypophyseal System; In Vitro Techniques; Magnesium; Male; Osmolar Concentration; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Sodium Chloride; Vasopressins

1998
Aniracetam, 1-BCP and cyclothiazide differentially modulate the function of NMDA and AMPA receptors mediating enhancement of noradrenaline release in rat hippocampal slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Dioxoles; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Heterocyclic Compounds; Hippocampus; In Vitro Techniques; Kynurenic Acid; Male; N-Methylaspartate; Nootropic Agents; Norepinephrine; Piperidines; Pyrrolidinones; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Tritium

1999
The concentration of synaptically released glutamate outside of the climbing fiber-Purkinje cell synaptic cleft.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-01, Volume: 19, Issue:13

    Topics: Amino Acid Transport System X-AG; Animals; ATP-Binding Cassette Transporters; Benzothiadiazines; Cell Membrane; Dose-Response Relationship, Drug; Glutamic Acid; In Vitro Techniques; Kinetics; Models, Biological; Neuroglia; Patch-Clamp Techniques; Probability; Purkinje Cells; Quinoxalines; Rats; Receptors, AMPA; Synapses; Temperature

1999
Glutamate transport blockade has a differential effect on AMPA and NMDA receptor-mediated synaptic transmission in the developing barrel cortex.
    Neuropharmacology, 2000, Mar-03, Volume: 39, Issue:5

    Topics: Amino Acid Transport System X-AG; Animals; Aspartic Acid; ATP-Binding Cassette Transporters; Benzothiadiazines; Biological Transport; Dicarboxylic Acids; Diuretics; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glutamic Acid; In Vitro Techniques; Kainic Acid; Neurotransmitter Uptake Inhibitors; Picrotoxin; Pyrrolidines; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Sodium Chloride Symporter Inhibitors; Somatosensory Cortex; Synaptic Transmission; Thalamus

2000
Mutation of a glutamate receptor motif reveals its role in gating and delta2 receptor channel properties.
    Nature neuroscience, 2000, Volume: 3, Issue:4

    Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Cell Line; Conserved Sequence; Dizocilpine Maleate; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Humans; Ion Channel Gating; Kainic Acid; Kidney; Mice; Mice, Neurologic Mutants; Molecular Sequence Data; Mutagenesis; Neuromuscular Depolarizing Agents; Patch-Clamp Techniques; Purkinje Cells; Quinoxalines; Receptors, Glutamate; Transfection

2000
Developmental regulation of AMPA-receptor properties in CA1 pyramidal neurons of rat hippocampus.
    Neuropharmacology, 2000, Apr-03, Volume: 39, Issue:6

    Topics: Alternative Splicing; Animals; Animals, Newborn; Benzodiazepines; Benzothiadiazines; Excitatory Amino Acid Antagonists; Female; Hippocampus; In Vitro Techniques; Kinetics; Patch-Clamp Techniques; Pyramidal Cells; Quinoxalines; Rats; Receptors, AMPA; Receptors, Kainic Acid

2000
Pharmacological and molecular characterization of glutamate receptors in the MIN6 pancreatic beta-cell line.
    Neurological research, 2000, Volume: 22, Issue:4

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Biological Transport; Calcium; Cell Survival; DNA Primers; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glutamic Acid; Islets of Langerhans; Kainic Acid; Protein Kinase C; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Spider Venoms; Tumor Cells, Cultured

2000
Characterization of audiogenic-like seizures in naive rats evoked by activation of AMPA and NMDA receptors in the inferior colliculus.
    Experimental neurology, 2000, Volume: 164, Issue:2

    Topics: Acoustic Stimulation; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Animals, Suckling; Benzothiadiazines; Dizocilpine Maleate; Drug Administration Routes; Excitatory Amino Acid Antagonists; Female; Hypothyroidism; Inferior Colliculi; Injections, Intraventricular; Male; Maternal Exposure; N-Methylaspartate; Propylthiouracil; Proto-Oncogene Proteins c-fos; Quinoxalines; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Seizures

2000
(S)-2,3-dihydro-[3,4]cyclopentano-1,2,4-benzothiadiazine-1,1-dioxide: (S18986-1) a positive modulator of AMPA receptors enhances (S)-AMPA-mediated [3H]noradrenaline release from rat hippocampal and frontal cortex slices.
    European journal of pharmacology, 2000, Aug-04, Volume: 401, Issue:2

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Frontal Lobe; Hippocampus; In Vitro Techniques; Male; Norepinephrine; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Stereoisomerism; Tetrodotoxin; Tritium

2000
A high GluR1 : GluR2 expression ratio is correlated with expression of Ca2+-binding proteins in rat forebrain neurons.
    The European journal of neuroscience, 2000, Volume: 12, Issue:8

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Antihypertensive Agents; Benzothiadiazines; Biological Transport; Calbindin 1; Calbindins; Calcium; Calcium Channel Blockers; Cells, Cultured; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Gene Expression; In Situ Hybridization; Neurons; Parvalbumins; Prosencephalon; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; RNA, Messenger; S100 Calcium Binding Protein G

2000
Presynaptic alpha-amino-3-hydroxy-5-methyl-4-isoxazole propionate receptor-mediated stimulation of glutamate and GABA release in the rat striatum in vivo: a dual-label microdialysis study.
    Neuroscience, 2001, Volume: 102, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Anti-Anxiety Agents; Antihypertensive Agents; Benzodiazepines; Benzothiadiazines; Calcium; Carbon Radioisotopes; Corpus Striatum; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Kynurenic Acid; Male; Microdialysis; Nootropic Agents; Potassium; Presynaptic Terminals; Pyrrolidinones; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Tritium

2001
The expression of cerebellar LTD in culture is not associated with changes in AMPA-receptor kinetics, agonist affinity, or unitary conductance.
    Proceedings of the National Academy of Sciences of the United States of America, 2001, Nov-20, Volume: 98, Issue:24

    Topics: 2-Amino-5-phosphonovalerate; Animals; Benzothiadiazines; Cells, Cultured; Cerebellum; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Long-Term Potentiation; Mice; Phorbol Esters; Quinoxalines; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2001
AMPA-induced Ca(2+) influx in cultured rat cortical nonpyramidal neurones: pharmacological characterization using fura-2 microfluorimetry.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzodiazepines; Benzothiadiazines; Calcium; Cells, Cultured; Cerebral Cortex; Cobalt; Diazoxide; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Fluorescence; Fluorometry; Fura-2; gamma-Aminobutyric Acid; Immunohistochemistry; N-Methylaspartate; Neurons; Piperazines; Quinoxalines; Rats; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate

2002
Networks of neurons coupled to microelectrode arrays: a neuronal sensory system for pharmacological applications.
    Biosensors & bioelectronics, 2003, Volume: 18, Issue:5-6

    Topics: Algorithms; Animals; Benzothiadiazines; Biosensing Techniques; Cells, Cultured; Cells, Immobilized; Chick Embryo; Chickens; Dizocilpine Maleate; Microelectrodes; Nerve Net; Quinoxalines; Signal Processing, Computer-Assisted

2003
Testosterone amplifies excitotoxic damage of cultured oligodendrocytes.
    Journal of neurochemistry, 2004, Volume: 88, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Calcium; Cells, Cultured; Drug Synergism; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression; Kainic Acid; L-Lactate Dehydrogenase; Neurotoxins; Oligodendroglia; Quinoxalines; Rats; Receptors, AMPA; Receptors, Androgen; Receptors, Kainic Acid; Testosterone; Time Factors

2004
Nitric oxide inhibits complex I following AMPA receptor activation via peroxynitrite.
    Neuroreport, 2004, Sep-15, Volume: 15, Issue:13

    Topics: Analysis of Variance; Animals; Antihypertensive Agents; Benzothiadiazines; Cells, Cultured; Cyclic GMP; Drug Interactions; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Hippocampus; Immunohistochemistry; Kainic Acid; Microtubule-Associated Proteins; Neurons; NG-Nitroarginine Methyl Ester; Nitric Oxide; Peroxynitrous Acid; Proton Pumps; Quinoxalines; Rats; Receptors, AMPA; Tyrosine

2004
Simultaneous contribution of two rod pathways to AII amacrine and cone bipolar cell light responses.
    Journal of neurophysiology, 2005, Volume: 93, Issue:3

    Topics: Amacrine Cells; Animals; Benzodiazepines; Benzothiadiazines; Diagnostic Imaging; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; Fluorescein; GABA Antagonists; Glycine Agents; In Vitro Techniques; Light; Male; Membrane Potentials; Models, Biological; Neurons; Patch-Clamp Techniques; Picrotoxin; Quinoxalines; Rabbits; Retina; Retinal Rod Photoreceptor Cells; Strychnine; Synapses; Synaptic Transmission; Visual Pathways

2005
A comparison of release kinetics and glutamate receptor properties in shaping rod-cone differences in EPSC kinetics in the salamander retina.
    The Journal of physiology, 2005, Dec-15, Volume: 569, Issue:Pt 3

    Topics: Animals; Benzodiazepines; Benzothiadiazines; Calcium; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Kinetics; Models, Biological; Neurotransmitter Agents; Quinoxalines; Receptors, AMPA; Receptors, Glutamate; Retinal Bipolar Cells; Retinal Cone Photoreceptor Cells; Retinal Horizontal Cells; Retinal Rod Photoreceptor Cells; Synaptic Transmission; Synaptic Vesicles; Urodela

2005
Action of extracellular divalent cations on native alpha-amino-3-hydroxy-5-methylisoxazole-4-propionate (AMPA) receptors.
    Journal of neurochemistry, 2005, Volume: 95, Issue:6

    Topics: Algorithms; Animals; Benzothiadiazines; Binding, Competitive; Cations, Divalent; Excitatory Amino Acid Agonists; Extracellular Space; Hippocampus; Kainic Acid; Pyramidal Cells; Quinoxalines; Rats; Receptors, AMPA

2005
Functional characterisation of homomeric ionotropic glutamate receptors GluR1-GluR6 in a fluorescence-based high throughput screening assay.
    Combinatorial chemistry & high throughput screening, 2006, Volume: 9, Issue:2

    Topics: Aniline Compounds; Benzothiadiazines; Calcium; Cell Line; Combinatorial Chemistry Techniques; Concanavalin A; Drug Evaluation, Preclinical; Electrophysiology; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Fluorescence; Glutamic Acid; Humans; Kainic Acid; Quinoxalines; Receptors, AMPA; Receptors, Glutamate; Signal Transduction; Xanthenes

2006
Regulation of SULT2B1a (pregnenolone sulfotransferase) expression in rat C6 glioma cells: relevance of AMPA receptor-mediated NO signaling.
    Neuroscience letters, 2008, Jan-03, Volume: 430, Issue:1

    Topics: Animals; Benzothiadiazines; Cell Line, Tumor; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glioma; Glutamic Acid; Isoenzymes; Neuroglia; Nitric Oxide; Pregnenolone; Quinoxalines; Rats; Receptors, AMPA; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfotransferases

2008
Excitatory actions of ventral root stimulation during network activity generated by the disinhibited neonatal mouse spinal cord.
    Journal of neurophysiology, 2009, Volume: 101, Issue:6

    Topics: Action Potentials; Animals; Animals, Newborn; Benzothiadiazines; Bicuculline; Biophysics; Carbodiimides; Chromones; Electric Stimulation; Electroporation; Excitatory Amino Acid Antagonists; Functional Laterality; GABA Antagonists; Glycine Agents; In Vitro Techniques; Mice; Motor Neurons; Neural Inhibition; Neural Pathways; Organic Chemicals; Quinoxalines; Reaction Time; Spectrum Analysis; Spinal Cord; Spinal Nerve Roots; Strychnine; Time Factors

2009
Vesicular glutamate filling and AMPA receptor occupancy at the calyx of Held synapse of immature rats.
    The Journal of physiology, 2009, May-15, Volume: 587, Issue:Pt 10

    Topics: 2-Amino-5-phosphonovalerate; Action Potentials; Animals; Aspartic Acid; Benzothiadiazines; Brain Stem; Excitatory Postsynaptic Potentials; Glutamic Acid; Kynurenic Acid; Patch-Clamp Techniques; Presynaptic Terminals; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Vesicles; Temperature; Tetrodotoxin

2009
Two modes of release shape the postsynaptic response at the inner hair cell ribbon synapse.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Mar-24, Volume: 30, Issue:12

    Topics: Animals; Animals, Newborn; Benzothiadiazines; Biophysics; Cochlea; Cochlear Nerve; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Hair Cells, Auditory, Inner; Hearing; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Sprague-Dawley; Synapses

2010
State-dependent, bidirectional modulation of neural network activity by endocannabinoids.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Nov-16, Volume: 31, Issue:46

    Topics: 4-Aminopyridine; Action Potentials; Animals; Animals, Newborn; Benzothiadiazines; Brain; Cannabinoid Receptor Modulators; Cells, Cultured; Electric Stimulation; Endocannabinoids; Excitatory Amino Acid Antagonists; GABA Antagonists; In Vitro Techniques; Mice; Mice, Transgenic; Nerve Net; Neural Inhibition; Neurons; Organophosphorus Compounds; Picrotoxin; Piperidines; Potassium Channel Blockers; Pyrazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Sodium Channel Blockers; Tetrodotoxin; Valine

2011
Modulation of extracellular d-serine content by calcium permeable AMPA receptors in rat medial prefrontal cortex as revealed by in vivo microdialysis.
    The international journal of neuropsychopharmacology, 2013, Volume: 16, Issue:6

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Area Under Curve; Benzothiadiazines; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Excitatory Amino Acid Agents; Extracellular Fluid; Fluorometry; Gas Chromatography-Mass Spectrometry; Male; Microdialysis; Prefrontal Cortex; Quinoxalines; Rats; Rats, Wistar; Receptors, AMPA; Serine; Spermine; Time Factors

2013
Reconstitution of homomeric GluA2(flop) receptors in supported lipid membranes: functional and structural properties.
    The Journal of biological chemistry, 2013, Mar-22, Volume: 288, Issue:12

    Topics: Animals; Benzothiadiazines; Glutamic Acid; Ion Channel Gating; Lipid Bilayers; Lipids; Liposomes; Membrane Potentials; Microscopy, Atomic Force; Protein Conformation; Quinoxalines; Rats; Receptors, AMPA

2013
A conformational intermediate in glutamate receptor activation.
    Neuron, 2013, Aug-07, Volume: 79, Issue:3

    Topics: Benzothiadiazines; Biophysical Phenomena; Cell Line, Transformed; Crystallography, X-Ray; Cysteine; Dithionitrobenzoic Acid; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Glutamic Acid; Humans; In Vitro Techniques; Membrane Potentials; Models, Molecular; Molecular Conformation; Mutation; Patch-Clamp Techniques; Phenanthrolines; Protein Structure, Tertiary; Quinoxalines; Receptors, Glutamate; Uncoupling Agents

2013
Raphe AMPA receptors and nicotinic acetylcholine receptors mediate ketamine-induced serotonin release in the rat prefrontal cortex.
    The international journal of neuropsychopharmacology, 2014, Volume: 17, Issue:8

    Topics: Animals; Antidepressive Agents; Benzothiadiazines; Dihydro-beta-Erythroidine; Dorsal Raphe Nucleus; Dose-Response Relationship, Drug; Injections, Subcutaneous; Ketamine; Male; Microdialysis; Microinjections; Nicotinic Antagonists; Prefrontal Cortex; Quinoxalines; Rats; Receptors, AMPA; Receptors, Nicotinic; Serotonin; Spermine

2014
AMPA receptor-mediated rapid EPSCs in vestibular calyx afferents.
    Journal of neurophysiology, 2017, 06-01, Volume: 117, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Benzothiadiazines; Calcium Channel Blockers; Calcium Channels, L-Type; Cells, Cultured; Dipeptides; Excitatory Postsynaptic Potentials; Female; Gerbillinae; Hair Cells, Vestibular; Male; Nifedipine; Quinoxalines; Receptors, AMPA; Strontium; Synapses

2017