Page last updated: 2024-08-17

quinoxalines and colforsin

quinoxalines has been researched along with colforsin in 102 studies

Research

Studies (102)

TimeframeStudies, this research(%)All Research%
pre-199011 (10.78)18.7374
1990's52 (50.98)18.2507
2000's28 (27.45)29.6817
2010's11 (10.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gnegy, ME; Mangels, LA1
Bourne, HR; Conklin, BR; Wong, YH1
Atkinson, BN; Minneman, KP1
Dieudonne, MN; Giudicelli, Y; Pecquery, R1
Coupry, I; Downing, S; Duzic, E; Lanier, SM1
Duzic, E; Lanier, SM1
Newman, ME1
Ball, SG; Ong, ML; Vaughan, PF1
McKenzie, FR; Milligan, G1
Osborne, NN1
Areso, P; García-Sevilla, JA; Giralt, MT; Guimón, J; Padró, D1
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D1
Alari, L; Axelsson, KL; Persson, ML; Post, C; Uhlén, S; Wikberg, JE1
Giudicelli, Y; Leneveu, MC; Pecquery, R1
Pratt, BL; Takahashi, JS1
Galzin, AM; Langer, SZ; Ramdine, R1
Uhlén, S; Wikberg, JE2
García-Sáinz, JA; Martínez, OM1
Areso, P; García-Sevilla, JA; Giralt, MT; Ulibarri, I1
Bylund, DB; Ray-Prenger, C; Turner, JT1
Bylund, DB; Jones, SB; Toews, ML; Turner, JT1
Duman, RS; Enna, SJ; Nomura, S1
Duman, RS; Enna, SJ1
Agneter, E; Boehm, S; Drobny, H; Huck, S; Koth, G; Singer, EA1
Bouloumie, A; Galitzky, J; Lafontan, M; Langin, D; Remaury, A; Tavernier, G; Valet, P1
Hara, M; Inoue, M; Irie, T; Mikami, T; Mikami, Y; Minato, A; Omori, K; Uyama, M; Yasukura, T; Zeng, XT1
Berlan, M; Bousquet-Mélou, A; Galitzky, J; Lafontan, M1
Regunathan, S; Reis, DJ1
Chetkovich, DM; Sweatt, JD1
Gean, PW; Huang, CC; Tsai, JJ1
Kurose, H; Lefkowitz, RJ1
Milligan, G1
Malik, KU; Schwartz, DD1
Soares-da-Silva, P1
Kellermann, O; Launay, JM; Loric, S; Maroteaux, L1
Abel, PW; Bockman, CS; Gonzalez-Cabrera, I1
Arner, P; Hellström, L; Langin, D; Reynisdottir, S; Rössner, S1
Ogihara, M1
Glitsch, M; Llano, I; Marty, A1
Itoh, Y; Kimura, K; Oka, M; Shimidzu, T; Ukai, Y; Yoshikuni, Y1
Goldstein, I; Huang, YH; Moreland, RB; Traish, AM1
Després, JP; Marcotte, M; Mauriège, P; Prud'Homme, D; Tremblay, A; Yoshioka, M1
Correze, C; Dib, K; el Jamali, A; Lambert, B; Wrisez, F1
Durham, PL; Russo, AF; Sharma, RV1
Huang, L; Huynh, LP; Mangrum, AJ; Momose-Hotokezaka, A; Okusa, MD1
Lu, L; Ordway, GA1
Katusic, ZS; Onoue, H1
Kendall, DA; Roberts, RE; Tomlinson, AE; Wilson, VG1
Minneman, KP; Williams, NG; Zhong, H1
Soares-da-Silva, P; Vieira-Coelho, MA1
Milligan, G; Sautel, M1
Polte, T; Schröder, H1
Albert, PR; Ghahremani, MH; Lembo, PM1
Borea, PA; Caiazza, A; Gessi, S; Portaluppi, F; Rastelli, G; Varani, K1
Durham, PL; Russo, AF1
Kendall, DA; Roberts, RE; Wilson, VG2
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1
Carlson, EJ; Drewett, JG; Kreklau, EL1
Eikenburg, DC; Shivachar, AC1
Gong, GX; Scholz, PM; Straznicka, M; Tse, J; Weiss, HR; Yan, L1
Gupte, SA; Phillibert, D; Rupawalla, T; Wolin, MS1
Kitazawa, T; Maezono, Y; Taneike, T1
Dick, JM; Lefebvre, RA1
Després, JP; Imbeault, P; Mauriège, P; Prud'Homme, D; Tremblay, A1
Berggren, PO; Cooney, RV; Sjöholm, A1
Eguchi, D; Katusic, ZS1
García-Barrado, MJ; Iglesias-Osma, MC; Moratinos, J; Sancho, C1
Blaylock, NA; Chan, SL; Dunn, WR; Minyan, W; Wilson, VG1
Flammer, J; Haefliger, IO; Liu, R1
Gupte, SA; Okada, T1
Argibay, J; Hoebeke, J; Nascimento, JH; Peineau, N; Sallé, L1
Jacobson, KL; Ott, SM; Singh, JC; Watson, EL1
Bessard, G; Bréant, D; Caron, F; Corompt, E; Devillier, P1
Bers, DM; Katoh, H; Ziolo, MT1
Flammer, J; Haefliger, IO; Liu, R; Wu, R1
Chen, YH; LaPolt, PS; Ngo, A; Tafoya, M1
Diamond, J; Sandirasegarane, L1
Barahona, MV; Benedito, S; García-Sacristán, A; Hernández, M; Martínez, AC; Orensanz, LM; Prieto, D; Recio, P; Rivera, L1
Eglen, RM; Kendall, DA; Maclennan, SJ; Pinthong, D; Wilson, VG1
Barnes, NY; Parent, AT; Sisodia, SS; Taniguchi, Y; Thinakaran, G1
MacNaughton, WK; Skinn, AC1
Elmedal Laursen, B; Mulvany, MJ; Simonsen, U1
Antunes, E; Baracat, JS; Claudino, MA; De Nucci, G; Priviero, FB; Teixeira, CE; Webb, RC1
Ivenshitz, M; Segal, M1
Haefliger, I; Wu, R; Yao, K; Yin, J1
Fraga, S; Jose, PA; Simão, S; Soares-da-Silva, P1
Genade, S; Genis, A; Huisamen, B; Lochner, A; Ytrehus, K1
Behr, J; Breustedt, J; Fidzinski, P; Maier, N; Schmitz, D; Wozny, C1
Baki, A; Bekes, Z; Boros, A; Bugovics, G; Gere, A; Ignácz-Szendrei, G; Kolok, S; Kurko, D; Nagy, J; Szombathelyi, Z1
Bylund, DB; Montgomery, MD1
Goy, D; Gummersbach, C; Hemmrich, K; Kröncke, KD; Pallua, N; Paul, NE; Suschek, CV1
Arnoletti, E; Baragli, A; Ghè, C; Ghigo, E; Granata, R; Muccioli, G1
Bernier, BE; Morikawa, H; Whitaker, LR1
Moonen, RM; Villamor, E1
Blouquit-Laye, S; Braun, C; Chinet, T; Dannhoffer, L; Dinh-Xuan, AT; Sage, E1
Agazatian, D; Froehlich, O; Kim, YH; Pech, V; Thumova, M; Verlander, JW; Wall, SM; Wang, X1
Colbert, CM; Eskin, A; Pita-Almenar, JD; Zou, S1
Bae, H; Bang, H; Kim, JH; Kim, K; Kim, T; Ko, JH; Lee, HJ; Lim, I1
Alexander, SP; Garle, MJ; Randall, MD; Roberts, RE; Wong, PS1
Fernández-Fernández, D; Kroker, KS; Rosenbrock, H1

Trials

2 trial(s) available for quinoxalines and colforsin

ArticleYear
Platelet alpha2-adrenoceptor alterations in patients with essential hypertension.
    British journal of clinical pharmacology, 1999, Volume: 47, Issue:2

    Topics: Adrenergic alpha-Antagonists; Blood Platelets; Brimonidine Tartrate; Colforsin; Cyclic AMP; Epinephrine; Female; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypertension; Male; Middle Aged; Protein Binding; Quinoxalines; Receptors, Adrenergic, alpha-2; Thermodynamics

1999
Adipose tissue metabolism in young and middle-aged men after control for total body fatness.
    The Journal of clinical endocrinology and metabolism, 2000, Volume: 85, Issue:7

    Topics: Adipose Tissue; Adrenergic Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic beta-Agonists; Adult; Aging; Body Composition; Brimonidine Tartrate; Bucladesine; Cell Separation; Colforsin; Epinephrine; Glycerol; Humans; Isoproterenol; Lipolysis; Lipoprotein Lipase; Male; Middle Aged; Quinoxalines; Theophylline

2000

Other Studies

100 other study(ies) available for quinoxalines and colforsin

ArticleYear
Cyclic AMP accumulation alters calmodulin localization in SK-N-SH human neuroblastoma cells.
    Brain research. Molecular brain research, 1992, Volume: 12, Issue:1-3

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Alprostadil; Analgesics; Brimonidine Tartrate; Bucladesine; Calcium; Calmodulin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Cytosol; Edetic Acid; Egtazic Acid; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Humans; Kinetics; Neuroblastoma; Quinoxalines; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1992
Gz-mediated hormonal inhibition of cyclic AMP accumulation.
    Science (New York, N.Y.), 1992, Jan-17, Volume: 255, Issue:5042

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Dinoprostone; Dopamine; Gene Expression Regulation; GTP-Binding Proteins; Hormones; In Vitro Techniques; Lysophospholipids; Pertussis Toxin; Quinoxalines; Rats; Signal Transduction; Transfection; Virulence Factors, Bordetella

1992
Preferential desensitization of beta- versus alpha 2-adrenergic receptors accelerates loss of response to norepinephrine in primary glial cultures.
    Molecular pharmacology, 1992, Volume: 41, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Female; Isoproterenol; Neuroglia; Norepinephrine; Pregnancy; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1992
Characteristics of the alpha 2/beta-adrenoceptor-coupled adenylate cyclase system and their relationship with adrenergic responsiveness in hamster fat cells from different anatomical sites.
    European journal of biochemistry, 1992, Apr-15, Volume: 205, Issue:2

    Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Colforsin; Cricetinae; Dioxanes; Epididymis; Epinephrine; GTP-Binding Proteins; Idazoxan; Isoproterenol; Kinetics; Lipolysis; Macromolecular Substances; Male; Mesocricetus; Organ Specificity; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Skin; Theophylline

1992
Factors determining the specificity of signal transduction by guanine nucleotide-binding protein-coupled receptors. I. Coupling of alpha 2-adrenergic receptor subtypes to distinct G-proteins.
    The Journal of biological chemistry, 1992, May-15, Volume: 267, Issue:14

    Topics: 3T3 Cells; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cell Membrane; Colforsin; Cyclic AMP; Epinephrine; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Kinetics; Mice; Pertussis Toxin; Quinoxalines; Receptors, Adrenergic, alpha; RNA, Messenger; Signal Transduction; Transfection; Virulence Factors, Bordetella; Yohimbine

1992
Factors determining the specificity of signal transduction by guanine nucleotide-binding protein-coupled receptors. III. Coupling of alpha 2-adrenergic receptor subtypes in a cell type-specific manner.
    The Journal of biological chemistry, 1992, Nov-25, Volume: 267, Issue:33

    Topics: 3T3 Cells; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Cell Line; Colforsin; Cyclic AMP; Edetic Acid; Egtazic Acid; Epinephrine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Kinetics; Manganese; Mice; Muscle, Smooth; PC12 Cells; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, beta; Signal Transduction; Transfection; Virulence Factors, Bordetella

1992
Serotonin inhibits adenylate cyclase in human platelet membranes.
    European journal of pharmacology, 1992, Aug-03, Volume: 226, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Binding Sites; Blood Platelets; Colforsin; Dose-Response Relationship, Drug; Humans; Methysergide; Quinoxalines; Receptors, Serotonin; Serotonin; Spiperone; Yohimbine

1992
Regulation of noradrenaline release from rat occipital cortex tissue chops by alpha 2-adrenergic agonists.
    Journal of neurochemistry, 1991, Volume: 56, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Brimonidine Tartrate; Bucladesine; Clonidine; Colforsin; Cyclic AMP; Histological Techniques; Male; Norepinephrine; Occipital Lobe; Quinoxalines; Rats; Rats, Inbred Strains

1991
Cholera toxin impairment of opioid-mediated inhibition of adenylate cyclase in neuroblastoma x glioma hybrid cells is due to a toxin-induced decrease in opioid receptor levels.
    The Biochemical journal, 1991, Apr-01, Volume: 275 ( Pt 1)

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Brimonidine Tartrate; Cholera Toxin; Colforsin; Enkephalin, Leucine-2-Alanine; Glioma; GTP Phosphohydrolases; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hybrid Cells; Immunoblotting; Neuroblastoma; Pertussis Toxin; Quinoxalines; Receptors, Opioid; Receptors, Opioid, delta; Signal Transduction; Tumor Cells, Cultured; Virulence Factors, Bordetella

1991
Inhibition of cAMP production by alpha 2-adrenoceptor stimulation in rabbit retina.
    Brain research, 1991, Jul-05, Volume: 553, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; GTP-Binding Proteins; In Vitro Techniques; Pertussis Toxin; Phosphoric Diester Hydrolases; Quinoxalines; Rabbits; Retina; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella

1991
Alpha 2-adrenoceptor-mediated inhibition of platelet adenylate cyclase and induction of aggregation in major depression. Effect of long-term cyclic antidepressant drug treatment.
    Archives of general psychiatry, 1990, Volume: 47, Issue:2

    Topics: Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Adult; Aged; Antidepressive Agents, Tricyclic; Blood Platelets; Brimonidine Tartrate; Colforsin; Depressive Disorder; Epinephrine; Female; Humans; Male; Middle Aged; Platelet Aggregation; Quinoxalines; Receptors, Adrenergic, alpha

1990
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
    Biochemical pharmacology, 1990, Aug-01, Volume: 40, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1990
Antinociceptive actions of alpha 2-adrenoceptor agonists in the rat spinal cord: evidence for antinociceptive alpha 2-adrenoceptor subtypes and dissociation of antinociceptive alpha 2-adrenoceptors from cyclic AMP.
    Journal of neurochemistry, 1990, Volume: 55, Issue:6

    Topics: Adrenergic alpha-Agonists; Animals; Benzylamines; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guanfacine; Male; Neurotoxins; Nociceptors; Pain Measurement; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Spinal Cord; Yohimbine

1990
Influence of androgenic status on the alpha 2/beta-adrenergic control of lipolysis in white fat cells: predominant alpha 2-antilipolytic response in testosterone-treated-castrated hamsters.
    Endocrinology, 1988, Volume: 122, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; Isoproterenol; Lipolysis; Male; Mesocricetus; Niacin; Orchiectomy; Phentolamine; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Testosterone

1988
Vasoactive intestinal polypeptide and alpha 2-adrenoceptor agonists regulate adenosine 3',5'-monophosphate accumulation and melatonin release in chick pineal cell cultures.
    Endocrinology, 1989, Volume: 125, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Brimonidine Tartrate; Cells, Cultured; Chickens; Colforsin; Cyclic AMP; Kinetics; Melatonin; Molecular Sequence Data; Pineal Gland; Quinoxalines; Radioimmunoassay; Sequence Homology, Nucleic Acid; Structure-Activity Relationship; Vasoactive Intestinal Peptide

1989
Involvement of adenylate cyclase and protein kinase C in the alpha 2-adrenoceptor-mediated inhibition of noradrenaline and 5-hydroxytryptamine release in rat hypothalamic slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Antihypertensive Agents; Brimonidine Tartrate; Colforsin; Dioxanes; Electric Stimulation; Hypothalamus; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin

1989
Alpha 2-adrenoceptors mediate inhibition of cyclic AMP production in the spinal cord after stimulation of cyclic AMP with forskolin but not after stimulation with capsaicin or vasoactive intestinal peptide.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Adenine; Animals; Brimonidine Tartrate; Capsaicin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Guinea Pigs; Male; Quinoxalines; Receptors, Adrenergic, alpha; Spinal Cord; Tissue Distribution; Vasoactive Intestinal Peptide

1989
Functional alpha 2-adrenoceptors in rat adipocytes: inhibition of cyclic AMP accumulation.
    Biochemistry international, 1989, Volume: 19, Issue:4

    Topics: Adenylate Cyclase Toxin; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Male; Pertussis Toxin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella

1989
Uncoupling of the platelet alpha 2-adrenoceptor adenylate cyclase system by N-ethylmaleimide and the resulting effect on receptor density and sensitivity.
    European journal of pharmacology, 1988, Jan-05, Volume: 145, Issue:1

    Topics: Adenylyl Cyclases; Adult; Antihypertensive Agents; Blood Platelets; Brimonidine Tartrate; Colforsin; Ethylmaleimide; Humans; In Vitro Techniques; Kinetics; Male; Quinoxalines; Receptors, Adrenergic, alpha; Sulfhydryl Reagents

1988
Alpha 2-adrenergic receptors in the human cell line, HT29. Characterization with the full agonist radioligand [3H]UK-14,304 and inhibition of adenylate cyclase.
    Molecular pharmacology, 1985, Volume: 28, Issue:5

    Topics: Adenocarcinoma; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Brimonidine Tartrate; Cell Line; Clonidine; Colforsin; Colonic Neoplasms; Dose-Response Relationship, Drug; Guanosine Triphosphate; Humans; Kinetics; Magnesium; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine

1985
Alpha 2-adrenergic receptor-mediated sensitization of forskolin-stimulated cyclic AMP production.
    Proceedings of the National Academy of Sciences of the United States of America, 1987, Volume: 84, Issue:5

    Topics: Adenine; Adenocarcinoma; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Cell Line; Colforsin; Colonic Neoplasms; Cyclic AMP; Humans; Kinetics; Norepinephrine; Quinoxalines; Receptors, Adrenergic, alpha

1987
In vivo or in vitro exposure to imipramine reduces alpha 2-adrenoceptor-mediated inhibition of cyclic AMP production in rat brain cerebral cortical slices.
    Brain research, 1987, Apr-28, Volume: 410, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Interactions; Imipramine; Male; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta

1987
Inhibition of cyclic AMP production by alpha 2-adrenoceptor stimulation in the guinea-pig spinal cord slices.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Prazosin; Quinoxalines; Spinal Cord; Yohimbine

1988
A procedure for measuring alpha 2-adrenergic receptor-mediated inhibition of cyclic AMP accumulation in rat brain slices.
    Brain research, 1986, Oct-08, Volume: 384, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Animals; Brain; Brimonidine Tartrate; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Mianserin; Norepinephrine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide

1986
Alpha 2-adrenoceptor-mediated inhibition of electrically evoked [3H]noradrenaline release from chick sympathetic neurons: role of cyclic AMP.
    Journal of neurochemistry, 1994, Volume: 63, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Adrenergic Fibers; Animals; Brimonidine Tartrate; Calcium Channels; Cells, Cultured; Chick Embryo; Cholera Toxin; Colforsin; Cyclic AMP; Electric Stimulation; Neurons; Norepinephrine; Quinoxalines; Receptors, Adrenergic, alpha-2; Tritium

1994
Molecular mechanisms underlying regional variations of catecholamine-induced lipolysis in rat adipocytes.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Base Sequence; Brimonidine Tartrate; Bucladesine; Catecholamines; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dioxanes; DNA Primers; Epididymis; Gene Expression; Idazoxan; Isoproterenol; Lipase; Lipolysis; Male; Molecular Sequence Data; Organ Specificity; Polymerase Chain Reaction; Propanolamines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger; Skin

1995
Adrenergic receptor-mediated Cl- transport in rabbit corneal endothelial cells.
    Japanese journal of pharmacology, 1995, Volume: 67, Issue:4

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetates; Acetazolamide; Adrenergic Agonists; Adrenergic Antagonists; Affinity Labels; Animals; Brimonidine Tartrate; Cells, Cultured; Chlorides; Colforsin; Dose-Response Relationship, Drug; Endothelium, Corneal; Fluorescent Dyes; Ion Transport; Isoproterenol; Microscopy, Fluorescence; Norepinephrine; Phentolamine; Phenylephrine; Photometry; Quinolines; Quinoxalines; Rabbits; Receptors, Adrenergic; Yohimbine

1995
Control of lipolysis in intra-abdominal fat cells of nonhuman primates: comparison with humans.
    Journal of lipid research, 1995, Volume: 36, Issue:3

    Topics: Abdomen; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenocorticotropic Hormone; Aged; Animals; Brimonidine Tartrate; Bucladesine; Callithrix; Colforsin; Female; Humans; In Vitro Techniques; Lipolysis; Macaca fascicularis; Male; Middle Aged; Papio; Peptide YY; Peptides; Primates; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Species Specificity

1995
Effects of moxonidine, an imidazoline antihypertensive agent, on second messenger systems in rat brain.
    European journal of pharmacology, 1994, Oct-14, Volume: 269, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Antihypertensive Agents; Brain Chemistry; Brain Stem; Brimonidine Tartrate; Cerebral Cortex; Colforsin; Cyclic AMP; Cyclic GMP; Imidazoles; In Vitro Techniques; Norepinephrine; Phosphatidylinositols; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Second Messenger Systems; Yohimbine

1994
nMDA receptor activation increases cyclic AMP in area CA1 of the hippocampus via calcium/calmodulin stimulation of adenylyl cyclase.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenylyl Cyclases; Animals; Ascorbic Acid; Calcium; Calmodulin; Cell Membrane; Colforsin; Cyclic AMP; Deoxyadenosines; Dopamine; Enzyme Activation; Evoked Potentials; Glycine; Hippocampus; In Vitro Techniques; Isoproterenol; Kinetics; Models, Neurological; N-Methylaspartate; Pyramidal Tracts; Quinoxalines; Rats; Receptors, N-Methyl-D-Aspartate; Sulfonamides; Theophylline; Trifluoperazine

1993
Enhancement of NMDA receptor-mediated synaptic potential by isoproterenol is blocked by Rp-adenosine 3',5'-cyclic monophosphothioate.
    Neuroscience letters, 1993, Oct-29, Volume: 161, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Evoked Potentials; In Vitro Techniques; Isoproterenol; Neurons; Picrotoxin; Quinoxalines; Rats; Receptors, N-Methyl-D-Aspartate; Synapses; Thionucleotides

1993
Differential desensitization and phosphorylation of three cloned and transfected alpha 2-adrenergic receptor subtypes.
    The Journal of biological chemistry, 1994, Apr-01, Volume: 269, Issue:13

    Topics: Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Base Sequence; Blotting, Western; Brimonidine Tartrate; Cell Line; CHO Cells; Cloning, Molecular; Colforsin; Cricetinae; Kinetics; Molecular Sequence Data; Molecular Weight; Norepinephrine; Phosphates; Phosphorylation; Quinoxalines; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Transfection

1994
Specificity and functional applications of antipeptide antisera which identify G-protein alpha subunits.
    Methods in enzymology, 1994, Volume: 237

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Antibody Specificity; Blotting, Western; Brimonidine Tartrate; Cell Line; Cell Membrane; Colforsin; Electrophoresis, Polyacrylamide Gel; Enzyme-Linked Immunosorbent Assay; Erythrocyte Membrane; GTP Phosphohydrolases; GTP-Binding Proteins; Immune Sera; Immunoassay; Indicators and Reagents; Kinetics; Macromolecular Substances; Molecular Sequence Data; Peptides; Quinoxalines; Recombinant Proteins; Turkeys

1994
Cyclic AMP modulates but does not mediate the inhibition of [3H]norepinephrine release by activation of alpha-2 adrenergic receptors in cultured rat ganglion cells.
    Neuroscience, 1993, Volume: 52, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Animals, Newborn; Brimonidine Tartrate; Cells, Cultured; Chromatography, Paper; Colforsin; Cyclic AMP; Electric Stimulation; Ganglia, Sympathetic; In Vitro Techniques; Norepinephrine; Quinoxalines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Thionucleotides

1993
Renal tubular dopamine outward transfer during Na(+)-H+ exchange activation by alpha 1- and alpha 2-adrenoceptor agonists.
    British journal of pharmacology, 1993, Volume: 109, Issue:2

    Topics: Adrenergic alpha-Agonists; Amiloride; Animals; Bucladesine; Colforsin; Dopamine; Hydrogen; In Vitro Techniques; Kidney Tubules; Levodopa; Phenylephrine; Phorbol 12,13-Dibutyrate; Quinoxalines; Rats; Sodium; Sphingosine

1993
Sequential onset of three 5-HT receptors during the 5-hydroxytryptaminergic differentiation of the murine 1C11 cell line.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Antiparkinson Agents; Cells, Cultured; Colforsin; Cyclic AMP; Ergolines; Gene Expression; Quinoxalines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Time Factors

1996
Alpha-2 adrenoceptor subtype causing nitric oxide-mediated vascular relaxation in rats.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Colforsin; Cyclic AMP; Endothelium, Vascular; In Vitro Techniques; Kinetics; Mesenteric Arteries; Nitric Oxide; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Swine; Vasodilation

1996
Regulation of lipolysis in fat cells of obese women during long-term hypocaloric diet.
    International journal of obesity and related metabolic disorders : journal of the International Association for the Study of Obesity, 1996, Volume: 20, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipocytes; Adrenergic beta-Agonists; Adult; Brimonidine Tartrate; Bucladesine; Catecholamines; Colforsin; Dobutamine; Energy Intake; Female; Food Deprivation; Glucose; Humans; Insulin; Insulin Resistance; Isoproterenol; Lipolysis; Middle Aged; Obesity; Propanolamines; Quinoxalines; Terbutaline; Time Factors

1996
Cell-density-dependent expression of the alpha(2)-adrenergic response by epidermal growth factor (EGF) in primary cultures of adult rat hepatocytes.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Cell Count; Cells, Cultured; Colforsin; Cyclic AMP; Cycloheximide; Cytochalasin B; Epidermal Growth Factor; Genistein; Isoflavones; Liver; Male; Oxymetazoline; Pertussis Toxin; Protein Biosynthesis; Proteins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella; Yohimbine

1996
Glutamate as a candidate retrograde messenger at interneurone-Purkinje cell synapses of rat cerebellum.
    The Journal of physiology, 1996, Dec-01, Volume: 497 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; Alanine; Animals; Benzoates; Colforsin; Cyclopropanes; Electrophysiology; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Interneurons; Kinetics; Presynaptic Terminals; Purkinje Cells; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Tetrodotoxin

1996
Involvement of metabotropic glutamate receptors in Gi- and Gs-dependent modulation of adenylate cyclase activity induced by a novel cognition enhancer NS-105 in rat brain.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Alanine; Animals; Baclofen; Brimonidine Tartrate; Cell Membrane; Cerebral Cortex; Cholera Toxin; Cognition; Colforsin; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoproterenol; Kinetics; Male; Manganese; Pertussis Toxin; Piperidines; Proline; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurotransmitter; Virulence Factors, Bordetella; Yohimbine

1997
Expression of functional alpha2-adrenergic receptor subtypes in human corpus cavernosum and in cultured trabecular smooth muscle cells.
    Receptors & signal transduction, 1997, Volume: 7, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Humans; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Penis; Quinoxalines; Radioisotopes; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA, Messenger; Yohimbine

1997
Regional differences in adipose tissue metabolism between sedentary and endurance-trained women.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: Abdomen; Adipocytes; Adipose Tissue; Adrenergic alpha-Agonists; Adult; Analysis of Variance; Brimonidine Tartrate; Bucladesine; Cells, Cultured; Colforsin; Epinephrine; Exercise Test; Female; Humans; Life Style; Lipolysis; Lipoprotein Lipase; Oxygen Consumption; Physical Endurance; Physical Fitness; Quinoxalines; Regression Analysis; Respiration; Skin; Thigh

1997
Sodium saccharin inhibits adenylyl cyclase activity in non-taste cells.
    Cellular signalling, 1997, Volume: 9, Issue:6

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adipocytes; Adrenergic alpha-Agonists; Animals; Astrocytes; Brimonidine Tartrate; Carcinogens; Cell Fractionation; Cell Membrane; Cerebral Cortex; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; GTP-Binding Proteins; Idazoxan; Male; Pertussis Toxin; Phenylisopropyladenosine; Quinoxalines; Rats; Rats, Wistar; Saccharin; Signal Transduction; Swine; Taste; Thyroid Gland; Virulence Factors, Bordetella

1997
Repression of the calcitonin gene-related peptide promoter by 5-HT1 receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-15, Volume: 17, Issue:24

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enhancer Elements, Genetic; Gene Expression Regulation; Genes, Reporter; Neurons; Promoter Regions, Genetic; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin Receptor Agonists; Sumatriptan; Thyroid Neoplasms; Time Factors; Transcription, Genetic; Trigeminal Ganglion; Tumor Cells, Cultured

1997
Regulation of adenylyl cyclase in polarized renal epithelial cells by G protein-coupled receptors.
    The American journal of physiology, 1997, Volume: 273, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Cell Line; Cell Membrane; Cell Polarity; Colforsin; Cyclic AMP; Epithelial Cells; Gene Expression Regulation; GTP-Binding Proteins; Kidney; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Purinergic P1; Recombinant Proteins; Transfection

1997
Alpha2C-adrenoceptors mediate inhibition of forskolin-stimulated cAMP production in rat striatum.
    Brain research. Molecular brain research, 1997, Dec-15, Volume: 52, Issue:2

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Colforsin; Corpus Striatum; Cyclic AMP; Functional Laterality; In Vitro Techniques; Kinetics; Male; Oligonucleotides, Antisense; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; RNA, Messenger; Transcription, Genetic

1997
The effect of 1H-[1,2,4]oxadiazolo[4,3-a]quinoxalin-1-one (ODQ) and charybdotoxin (CTX) on relaxations of isolated cerebral arteries to nitric oxide.
    Brain research, 1998, Feb-23, Volume: 785, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Bradykinin; Cerebral Arteries; Charybdotoxin; Colforsin; Cyclic GMP; Dogs; Endothelium, Vascular; Enzyme Inhibitors; Guanylate Cyclase; Hydrazines; In Vitro Techniques; Isometric Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitrogen Oxides; Oxadiazoles; Quinoxalines; Uridine Triphosphate

1998
Alpha2-adrenoceptor-mediated contractions of the porcine isolated ear artery: evidence for a cyclic AMP-dependent and a cyclic AMP-independent mechanism.
    British journal of pharmacology, 1998, Volume: 124, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Angiotensin II; Animals; Arteries; Brimonidine Tartrate; Colforsin; Cyclic AMP; Ear; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Nitroprusside; Quinoxalines; Receptors, Adrenergic, alpha-2; Swine

1998
Differential coupling of alpha1-, alpha2-, and beta-adrenergic receptors to mitogen-activated protein kinase pathways and differentiation in transfected PC12 cells.
    The Journal of biological chemistry, 1998, Sep-18, Volume: 273, Issue:38

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium-Calmodulin-Dependent Protein Kinases; Cell Differentiation; Colforsin; Enzyme Activation; Inositol Phosphates; Isopropyl Thiogalactoside; JNK Mitogen-Activated Protein Kinases; Kinetics; Mitogen-Activated Protein Kinases; Nerve Growth Factors; Norepinephrine; p38 Mitogen-Activated Protein Kinases; PC12 Cells; Quinoxalines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Recombinant Proteins; Signal Transduction; Transfection

1998
Alpha2-adrenoceptors mediate the effect of dopamine on adult rat jejunal electrolyte transport.
    European journal of pharmacology, 1998, Aug-28, Volume: 356, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amiloride; Animals; Brimonidine Tartrate; Bucladesine; Cardiotonic Agents; Colforsin; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electric Impedance; Electrolytes; Furosemide; Ion Transport; Jejunum; Male; Ouabain; Phentolamine; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2

1998
Loss of activation of Gs but not Gi following expression of an alpha2A-adrenoceptor-Gi1alpha fusion protein.
    FEBS letters, 1998, Sep-25, Volume: 436, Issue:1

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Binding Sites; Brimonidine Tartrate; Cholera Toxin; Colforsin; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Oxymetazoline; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Virulence Factors, Bordetella

1998
Cyclic AMP mediates endothelial protection by nitric oxide.
    Biochemical and biophysical research communications, 1998, Oct-20, Volume: 251, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclase Inhibitors; Alkaloids; Animals; Carbazoles; Cattle; Cell Line; Cell Survival; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic N-Oxides; Dideoxyadenosine; Endothelium, Vascular; Enzyme Inhibitors; Free Radical Scavengers; Imidazoles; Indoles; Kinetics; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Penicillamine; Pulmonary Artery; Pyrroles; Quinoxalines; S-Nitroso-N-Acetylpenicillamine; Tumor Necrosis Factor-alpha

1998
Receptor selectivity of the cloned opossum G protein-coupled receptor kinase 2 (GRK2) in intact opossum kidney cells: role in desensitization of endogenous alpha2C-adrenergic but not serotonin 1B receptors.
    Molecular endocrinology (Baltimore, Md.), 1999, Volume: 13, Issue:1

    Topics: Adrenergic alpha-Agonists; Amino Acid Sequence; Animals; Base Sequence; beta-Adrenergic Receptor Kinases; Blotting, Northern; Brimonidine Tartrate; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP-Dependent Protein Kinases; G-Protein-Coupled Receptor Kinase 2; Kidney; Molecular Sequence Data; Mutation; Opossums; Quinoxalines; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Recombinant Proteins; Sequence Homology, Amino Acid

1999
Regulation of calcitonin gene-related peptide secretion by a serotonergic antimigraine drug.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, May-01, Volume: 19, Issue:9

    Topics: Animals; Animals, Newborn; Calcitonin Gene-Related Peptide; Cells, Cultured; Colforsin; Cyclic AMP; HeLa Cells; Humans; Inflammation; Kinetics; Models, Neurological; Neurons; Okadaic Acid; Oxadiazoles; Potassium Chloride; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Serotonin Receptor Agonists; Sumatriptan; Transfection; Trigeminal Ganglion; Tryptamines

1999
A study of NPY-mediated contractions of the porcine isolated ear artery.
    British journal of pharmacology, 1999, Volume: 127, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Angiotensin II; Animals; Brimonidine Tartrate; Colforsin; Cyclic AMP; Ear, External; In Vitro Techniques; Isometric Contraction; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Neuropeptide Y; Nitroprusside; Quinoxalines; Receptors, Adrenergic, alpha-2; Receptors, Neuropeptide Y; Regional Blood Flow; Swine; Vasoconstrictor Agents; Vasodilator Agents

1999
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999
Nitric oxide inhibits human aldosteronogenesis without guanylyl cyclase stimulation.
    Molecular and cellular endocrinology, 1999, Jul-20, Volume: 153, Issue:1-2

    Topics: Adrenal Cortex; Aldosterone; Angiotensin II; Animals; Cell Line; Colforsin; Cyclic GMP; Enzyme Inhibitors; Guanylate Cyclase; Humans; Hydroxycholesterols; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Nitroso Compounds; Oxadiazoles; PC12 Cells; Quinoxalines; Rats

1999
Differential effects of epinephrine and norepinephrine on cAMP response and g(i3)alpha protein expression in cultured sympathetic neurons.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:1

    Topics: Adrenergic Agonists; Animals; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; Isoproterenol; Neurons; Norepinephrine; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Superior Cervical Ganglion

1999
Cyclic GMP and cyclic AMP induced changes in control and hypertrophic cardiac myocyte function interact through cyclic GMP affected cyclic-AMP phosphodiesterases.
    Canadian journal of physiology and pharmacology, 1999, Volume: 77, Issue:6

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Cardiomegaly; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Heart; Milrinone; Oxadiazoles; Oxygen Consumption; Purinones; Quinoxalines

1999
alpha(2)-adrenoceptor and NPY receptor-mediated contractions of porcine isolated blood vessels: evidence for involvement of the vascular endothelium.
    British journal of pharmacology, 1999, Volume: 128, Issue:8

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic Agonists; Animals; Brimonidine Tartrate; Colforsin; Endothelium, Vascular; Humans; Neuropeptide Y; Quinoxalines; Receptors, Adrenergic, alpha-2; Swine; Vasoconstriction; Vasoconstrictor Agents; Vasodilation

1999
NADPH and heme redox modulate pulmonary artery relaxation and guanylate cyclase activation by NO.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Animals; Cattle; Colforsin; Cyclic GMP; Electron Transport; Enzyme Activation; Enzyme Inhibitors; Ferricyanides; Flavoproteins; Glutathione; Guanylate Cyclase; Heme; In Vitro Techniques; NADH, NADPH Oxidoreductases; NADP; Nitric Oxide; Oxadiazoles; Oxidation-Reduction; Penicillamine; Pentose Phosphate Pathway; Pulmonary Artery; Quinoxalines; Reactive Oxygen Species; Sulfhydryl Compounds

1999
The mechanisms of alpha(2)-adrenoceptor agonist-induced contraction in longitudinal muscle of the porcine uterus.
    European journal of pharmacology, 2000, Feb-25, Volume: 390, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Calcium Channel Blockers; Clonidine; Colforsin; Cyclic AMP; Female; Fluorescent Dyes; Fura-2; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myometrium; Pertussis Toxin; Quinoxalines; Swine; Uterus; Verapamil; Virulence Factors, Bordetella

2000
Interplay between nitric oxide and vasoactive intestinal polypeptide in the pig gastric fundus smooth muscle.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Adenine; Adenylyl Cyclase Inhibitors; Amidines; Animals; Arginine; Benzylamines; Carbazoles; Colforsin; Cyclic AMP; Dexamethasone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gastric Fundus; In Vitro Techniques; Indoles; Isoquinolines; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Nitroarginine; Oxadiazoles; Protein Kinase Inhibitors; Pyrroles; Quinoxalines; Sulfonamides; Swine; Thionucleotides; Vasoactive Intestinal Peptide

2000
gamma-tocopherol partially protects insulin-secreting cells against functional inhibition by nitric oxide.
    Biochemical and biophysical research communications, 2000, Oct-22, Volume: 277, Issue:2

    Topics: Adenylyl Cyclases; Animals; Calcium; Calcium Channels; Carbachol; Cell Division; Cell Line; Cell Survival; Cholinergic Agonists; Colforsin; Cyclic GMP; Enzyme Inhibitors; Insulin; Insulin Secretion; Insulinoma; Interleukin-1; Islets of Langerhans; Models, Chemical; Nitric Oxide; Nitrogen Oxides; Oxadiazoles; Phorbol Esters; Protein Kinase C; Quinoxalines; Rats; Spermine; Type C Phospholipases; Vitamin E

2000
Inhibitory effect of valves on endothelium-dependent relaxations to calcium ionophore in canine saphenous vein.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Calcimycin; Calcium; Colforsin; Cyclic GMP; Cyclooxygenase Inhibitors; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Hydrazines; In Vitro Techniques; Indomethacin; Ionophores; NG-Nitroarginine Methyl Ester; Nitric Oxide Donors; Nitrogen Oxides; Oxadiazoles; Potassium Chloride; Quinoxalines; Saphenous Vein; Vasoconstrictor Agents; Vasodilation

2001
Effects of verapamil and elgodipine on isoprenaline-induced metabolic responses in rabbits.
    European journal of pharmacology, 2001, Mar-09, Volume: 415, Issue:1

    Topics: Adipose Tissue; Animals; Blood Glucose; Brimonidine Tartrate; Calcium Channel Blockers; Colforsin; Consciousness; Dihydropyridines; Dose-Response Relationship, Drug; Epinephrine; Glucose; In Vitro Techniques; Insulin; Islets of Langerhans; Isoproterenol; Male; Metabolism; Potassium; Quinoxalines; Rabbits; Verapamil

2001
Evidence for a non-adrenoceptor, imidazoline-mediated contractile response to oxymetazoline in the porcine isolated rectal artery.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Animals; Arteries; Benzofurans; Brimonidine Tartrate; Colforsin; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Potassium Chloride; Quinoxalines; Receptors, Adrenergic; Rectum; Swine; Vasoconstriction

2001
Brimonidine and inhibition of nitrite production in isolated porcine ciliary processes.
    Klinische Monatsblatter fur Augenheilkunde, 2001, Volume: 218, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Aqueous Humor; Brimonidine Tartrate; Ciliary Body; Colforsin; Intraocular Pressure; Nitric Oxide; Nitrites; Quinoxalines; Swine

2001
Prostaglandins and nitric oxide mediate superoxide-induced myocardial contractile dysfunction in isolated rat hearts.
    Journal of molecular and cellular cardiology, 2001, Volume: 33, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Aspartate Aminotransferases; Colforsin; Enzyme Inhibitors; Heart; Myocardial Contraction; Myocardium; Nitrates; Nitric Acid; Nitroarginine; Nitroglycerin; Nitroprusside; Oxadiazoles; Phosphodiesterase Inhibitors; Platelet Aggregation Inhibitors; Prostaglandins; Quinoxalines; Rats; Superoxides; Thromboxane A2; Vasodilator Agents

2001
cGMP-mediated inhibition of cardiac L-type Ca(2+) current by a monoclonal antibody against the M(2) ACh receptor.
    American journal of physiology. Cell physiology, 2001, Volume: 281, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Antibodies, Monoclonal; Autoantibodies; Calcium Channels, L-Type; Colforsin; Cyclic GMP; Enzyme Inhibitors; Guanosine; Guinea Pigs; Heart Ventricles; In Vitro Techniques; Isoproterenol; Membrane Potentials; Muscle Fibers, Skeletal; Myocardium; Oxadiazoles; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Quinoxalines; Receptor, Muscarinic M2; Receptors, Muscarinic

2001
Nitric oxide inhibition of cAMP synthesis in parotid acini: regulation of type 5/6 adenylyl cyclase.
    Cellular signalling, 2001, Volume: 13, Issue:10

    Topics: Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Isoenzymes; Isoproterenol; Mice; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Parotid Gland; Phosphoric Diester Hydrolases; Quinoxalines; Thapsigargin; Triazoles

2001
Relaxation and modulation of cyclic AMP production in response to atrial natriuretic peptides in guinea pig tracheal smooth muscle.
    European journal of pharmacology, 2001, Nov-02, Volume: 430, Issue:2-3

    Topics: Adenylyl Cyclases; Animals; Apamin; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Natriuretic Peptide, C-Type; Nitroprusside; Oxadiazoles; Peptide Fragments; Peptides; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Quinoxalines; Rolipram; Trachea

2001
Expression of inducible nitric oxide synthase depresses beta-adrenergic-stimulated calcium release from the sarcoplasmic reticulum in intact ventricular myocytes.
    Circulation, 2001, Dec-11, Volume: 104, Issue:24

    Topics: Animals; Calcium; Colforsin; Cyclic GMP; Enzyme Inhibitors; Guanidines; Guanylate Cyclase; Heart Failure; Heart Ventricles; Humans; Lipopolysaccharides; Male; Middle Aged; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Sarcoplasmic Reticulum

2001
Inhibition by brimonidine of forskolin-induced nitrite production in isolated pig ciliary processes.
    Investigative ophthalmology & visual science, 2002, Volume: 43, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Ciliary Body; Colforsin; Dose-Response Relationship, Drug; GTP-Binding Protein alpha Subunits, Gi-Go; Nitrites; Pertussis Toxin; Quinoxalines; Receptors, Adrenergic, alpha-2; Swine; Virulence Factors, Bordetella

2002
Effects of nitric oxide and cGMP on inhibin A and inhibin subunit mRNA levels from cultured rat granulosa cells.
    Fertility and sterility, 2003, Volume: 79 Suppl 1

    Topics: Animals; Blotting, Northern; Colforsin; Cyclic GMP; Dibutyryl Cyclic GMP; Enzyme Inhibitors; Estradiol; Female; Follicle Stimulating Hormone; Granulosa Cells; Inhibins; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Quinoxalines; Rats; Rats, Sprague-Dawley; RNA, Messenger

2003
Pertussis toxin-sensitive G protein but not NO/cGMP pathway mediates the negative inotropic effect of carbachol in adult rat cardiomyocytes.
    Pharmacology, 2004, Volume: 70, Issue:1

    Topics: Adenylyl Cyclases; Animals; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Electric Stimulation; GTP-Binding Proteins; Injections, Intraperitoneal; Isoproterenol; Male; Myocardial Contraction; Myocytes, Cardiac; Nitric Oxide Synthase; omega-N-Methylarginine; Oxadiazoles; Pertussis Toxin; Quinoxalines; Rats; Time Factors

2004
Heterogeneity of neuronal and smooth muscle receptors involved in the VIP- and PACAP-induced relaxations of the pig intravesical ureter.
    British journal of pharmacology, 2004, Volume: 141, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Apamin; Capsaicin; Charybdotoxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Female; Guanylate Cyclase; Male; Muscle, Smooth; Neurons, Afferent; Neuropeptide Y; Neuropeptides; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; omega-Conotoxin GVIA; Oxadiazoles; Peptide Fragments; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium Channels, Calcium-Activated; Quinoxalines; Receptors, Calcitonin Gene-Related Peptide; Receptors, Peptide; Receptors, Vasoactive Intestinal Peptide; Rolipram; Sensory Receptor Cells; Swine; Tetraethylammonium; Ureter; Vasoactive Intestinal Peptide

2004
No evidence for activation of alpha(2)-adrenoceptors by methanolic extracts of bovine brain and lung containing clonidine-displacing substance.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Animals; Brain Chemistry; Brimonidine Tartrate; Cattle; Clonidine; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Lung; Male; Methanol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Swine; Tissue Extracts; Vas Deferens; Veins

2003
Presenilin attenuates receptor-mediated signaling and synaptic function.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Feb-09, Volume: 25, Issue:6

    Topics: Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Carbamates; Carbazoles; Cell Adhesion Molecules; Cell Line, Tumor; Cell Membrane; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DCC Receptor; Dipeptides; Endopeptidases; Excitatory Postsynaptic Potentials; Genes, DCC; Glutamic Acid; Indoles; Lidocaine; Membrane Proteins; Memory; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurites; Neuroblastoma; Neurons; Piperazines; Presenilin-1; Protein Processing, Post-Translational; Pyrroles; Quinoxalines; Rats; Receptors, Cell Surface; Recombinant Fusion Proteins; Second Messenger Systems; Synaptic Transmission; Transfection; Tumor Suppressor Proteins

2005
Nitric oxide inhibits cAMP-dependent CFTR trafficking in intestinal epithelial cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2005, Volume: 289, Issue:4

    Topics: Cell Line; Cell Membrane; Cell Membrane Permeability; Chlorides; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Inhibitors; Epithelial Cells; Fluorescent Antibody Technique; Guanylate Cyclase; Humans; Intestinal Mucosa; Intestines; Isoquinolines; Nitric Oxide; Nitric Oxide Donors; Nocodazole; Oxadiazoles; Quinoxalines; Sulfonamides

2005
Involvement of guanylyl cyclase, protein kinase A and Na+ K+ ATPase in relaxations of bovine isolated bronchioles induced by GEA 3175, an NO donor.
    Pulmonary pharmacology & therapeutics, 2006, Volume: 19, Issue:3

    Topics: Animals; Bronchi; Calcium; Cattle; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Guanylate Cyclase; In Vitro Techniques; Molsidomine; Muscle Relaxation; Nitric Oxide; Nitric Oxide Donors; Ouabain; Oxadiazoles; Peptides; Potassium; Quinoxalines; S-Nitrosoglutathione; Serotonin; Sodium-Potassium-Exchanging ATPase; Thionucleotides; Triazoles

2006
Stimulation of soluble guanylyl cyclase by BAY 41-2272 relaxes anococcygeus muscle: interaction with nitric oxide.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: Animals; Carbachol; Carbolines; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Drug Synergism; Electric Stimulation; Enzyme Activation; Enzyme Inhibitors; Guanylate Cyclase; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroglycerin; Oxadiazoles; Pyrazoles; Pyridines; Quinoxalines; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Soluble Guanylyl Cyclase; Tadalafil; Tetrodotoxin

2006
Simultaneous NMDA-dependent long-term potentiation of EPSCs and long-term depression of IPSCs in cultured rat hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Evoked Potentials; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Neuronal Plasticity; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin; Thionucleotides; Time Factors

2006
Inhibition by brimonidine of forskolin-induced nitric oxide synthase expression in human ciliary bodies in vitro.
    Molecular vision, 2007, Apr-02, Volume: 13

    Topics: Adrenergic alpha-Agonists; Blotting, Western; Brimonidine Tartrate; Ciliary Body; Colforsin; Cryopreservation; Humans; In Vitro Techniques; Nitric Oxide Synthase; Quinoxalines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tissue and Organ Harvesting

2007
Oxidative stress plays a permissive role in alpha2-adrenoceptor-mediated events in immortalized SHR proximal tubular epithelial cells.
    Molecular and cellular biochemistry, 2008, Volume: 315, Issue:1-2

    Topics: Acetophenones; Actins; Animals; Brimonidine Tartrate; Bucladesine; Cell Line, Transformed; Chloride-Bicarbonate Antiporters; Colforsin; Epithelial Cells; Hydrogen Peroxide; Kidney Tubules, Proximal; Membrane Glycoproteins; NADPH Oxidase 2; NADPH Oxidases; Oxidative Stress; Pertussis Toxin; Quinoxalines; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2

2008
Melatonin receptor-mediated protection against myocardial ischaemia/reperfusion injury: role of its anti-adrenergic actions.
    Journal of pineal research, 2008, Volume: 45, Issue:4

    Topics: Adrenergic Antagonists; Animals; Colforsin; Cyclic AMP; Guanylate Cyclase; Heart; Indoles; Isoproterenol; Male; Maleimides; Melatonin; Myocardial Infarction; Myocardial Reperfusion Injury; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxadiazoles; p38 Mitogen-Activated Protein Kinases; Propranolol; Protein Kinase C; Quinoxalines; Rats; Rats, Wistar; Receptors, Melatonin; Tryptamines

2008
Differential cAMP signaling at hippocampal output synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Dec-31, Volume: 28, Issue:53

    Topics: Action Potentials; Analysis of Variance; Animals; Calcium; Colforsin; Cyclic AMP; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Isoquinolines; Neurons; Oligopeptides; Patch-Clamp Techniques; Protein Kinase Inhibitors; Pyridazines; Quinoxalines; Rats; Signal Transduction; Sulfonamides; Synapses; Time Factors

2008
Comparative pharmacology of adrenergic alpha(2C) receptors coupled to Ca(2+) signaling through different Galpha proteins.
    Neurochemistry international, 2009, Volume: 55, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Calcium Signaling; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Fluorometry; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Humans; Quinoxalines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Recombinant Proteins; RNA, Messenger; Transfection

2009
Lack of effect of the alpha2C-adrenoceptor Del322-325 polymorphism on inhibition of cyclic AMP production in HEK293 cells.
    British journal of pharmacology, 2010, Volume: 159, Issue:4

    Topics: Adenylyl Cyclases; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Binding, Competitive; Brimonidine Tartrate; Cell Line; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Humans; Linear Models; Norepinephrine; Polymorphism, Genetic; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Signal Transduction; Transfection

2010
Nitric oxide and downstream second messenger cGMP and cAMP enhance adipogenesis in primary human preadipocytes.
    Cytotherapy, 2010, Volume: 12, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adipocytes; Adipogenesis; Adult; Cell Proliferation; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; DDT; Guanylate Cyclase; Humans; Male; Middle Aged; Nitric Oxide; Oxadiazoles; Quinoxalines; Second Messenger Systems; Stem Cells; Subcutaneous Fat; Tissue Engineering

2010
Acylated and unacylated ghrelin attenuate isoproterenol-induced lipolysis in isolated rat visceral adipocytes through activation of phosphoinositide 3-kinase γ and phosphodiesterase 3B.
    Biochimica et biophysica acta, 2011, Volume: 1811, Issue:6

    Topics: Acylation; Adipocytes; Adrenergic beta-Agonists; Animals; Benzimidazoles; Blotting, Western; Cells, Cultured; Class Ib Phosphatidylinositol 3-Kinase; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Drug Interactions; Ghrelin; Glycerol; Intra-Abdominal Fat; Isoproterenol; Lipolysis; Male; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinolones; Quinoxalines; Rats; Rats, Wistar; Thiazolidinediones

2011
Previous ethanol experience enhances synaptic plasticity of NMDA receptors in the ventral tegmental area.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2011, Apr-06, Volume: 31, Issue:14

    Topics: Amphibian Proteins; Analysis of Variance; Animals; Biophysics; Central Nervous System Depressants; Cocaine; Colforsin; Conditioning, Operant; Corticotropin-Releasing Hormone; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Ethanol; Excitatory Amino Acid Antagonists; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Long-Term Potentiation; Male; Methoxyhydroxyphenylglycol; Mice; Mice, Inbred C57BL; Neuronal Plasticity; Neurons; Peptide Hormones; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Salicylamides; Ventral Tegmental Area

2011
Developmental changes in mesenteric artery reactivity in embryonic and newly hatched chicks.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2011, Volume: 181, Issue:8

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Animals, Newborn; Body Weight; Chick Embryo; Chickens; Colforsin; Embryonic Development; Endothelin-1; Enzyme Inhibitors; Mesenteric Arteries; NG-Nitroarginine Methyl Ester; Nitroprusside; Norepinephrine; Oxadiazoles; Potassium Chloride; Quinoxalines; Vasoconstriction; Vasodilation

2011
Effect of nitric oxide on epithelial ion transports in noncystic fibrosis and cystic fibrosis human proximal and distal airways.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Oct-01, Volume: 303, Issue:7

    Topics: Adenosine Triphosphate; Adult; Aged; Amiloride; Bronchi; Chloride Channels; Colforsin; Cyclic GMP; Cyclic N-Oxides; Cystic Fibrosis; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Free Radical Scavengers; Guanylate Cyclase; Humans; Imidazoles; Middle Aged; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Oxadiazoles; Purinones; Quinoxalines; Young Adult

2012
Pendrin protein abundance in the kidney is regulated by nitric oxide and cAMP.
    American journal of physiology. Renal physiology, 2012, Sep-15, Volume: 303, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Anion Transport Proteins; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Inhibitors; Imidazoles; Kidney Tubules, Collecting; Mice; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroso Compounds; Oxadiazoles; Quinoxalines; Sulfate Transporters; Triazines

2012
Relationship between increase in astrocytic GLT-1 glutamate transport and late-LTP.
    Learning & memory (Cold Spring Harbor, N.Y.), 2012, Nov-19, Volume: 19, Issue:12

    Topics: Alanine Transaminase; Analysis of Variance; Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Biophysics; Biotinylation; Cells, Cultured; Colforsin; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Excitatory Postsynaptic Potentials; Flow Cytometry; Glial Fibrillary Acidic Protein; Glutamates; Glutamic Acid; Glycine; Hippocampus; In Vitro Techniques; Indoles; Kainic Acid; Long-Term Potentiation; Male; Neurons; Protein Transport; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin; Valine

2012
The stimulating effects of nitric oxide on intermediate conductance Ca²⁺-activated K⁺ channels in human dermal fibroblasts through PKG pathways but not the PKA pathways.
    The Chinese journal of physiology, 2014, Jun-30, Volume: 57, Issue:3

    Topics: 4-Aminopyridine; Calcium; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dermis; Enzyme Inhibitors; Fibroblasts; Humans; Intermediate-Conductance Calcium-Activated Potassium Channels; Nitric Oxide; Oxadiazoles; Patch-Clamp Techniques; Peptides; Potassium Channel Blockers; Quinoxalines; Signal Transduction; Toxins, Biological; Wound Healing

2014
A role for the sodium pump in H2O2-induced vasorelaxation in porcine isolated coronary arteries.
    Pharmacological research, 2014, Volume: 90

    Topics: Animals; Bradykinin; Carbenoxolone; Catalase; Colforsin; Coronary Vessels; Female; Hydrogen Peroxide; In Vitro Techniques; Indomethacin; Male; NG-Nitroarginine Methyl Ester; Nitroprusside; Ouabain; Oxadiazoles; Peptides; Polyethylene Glycols; Quinoxalines; Sodium-Potassium-Exchanging ATPase; Swine; Vasoconstrictor Agents; Vasodilation; Verapamil

2014
Inhibition of PDE2A, but not PDE9A, modulates presynaptic short-term plasticity measured by paired-pulse facilitation in the CA1 region of the hippocampus.
    Synapse (New York, N.Y.), 2015, Volume: 69, Issue:10

    Topics: Adenosine; Animals; CA1 Region, Hippocampal; Cadmium Chloride; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 2; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Long-Term Potentiation; Male; Morpholines; Neurons; Oxadiazoles; Presynaptic Terminals; Pyrimidines; Quinoxalines; Rats; Rats, Wistar

2015