Page last updated: 2024-08-17

quinoxalines and cgs 12066b

quinoxalines has been researched along with cgs 12066b in 71 studies

Research

Studies (71)

TimeframeStudies, this research(%)All Research%
pre-19903 (4.23)18.7374
1990's46 (64.79)18.2507
2000's16 (22.54)29.6817
2010's6 (8.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Higgins, GA; Jones, BJ; Oakley, NR1
Reid, A; Sawynok, J2
Clement, HW; Gemsa, D; Wesemann, W1
Newman, ME1
Levine, JD; Taiwo, YO1
Martin, P; Puech, AJ1
Donát, P; Rodgers, RJ; Shepherd, JK1
Frances, H; Monier, C2
Cloëz, I; Fillion, G; Harel-Dupas, C1
Benjamin, D; Lal, H; Meyerson, LR1
Bervoets, K; Colpaert, FC; Millan, MJ1
Baudrie, V; Chaouloff, F; Laude, D; Martin, GR1
Cooper, SJ; Neill, JC1
Fallon, SL; Sinton, CM1
Boyar, WC; Fallon, SL; Glaeser, BS; Martin, LL; Neale, RF; Sinton, CM; Stone, GA; Wasley, JW; Williams, M1
Heckman, CJ; Miller, JF; Paul, KD; Rymer, WZ1
Bell, R; Donaldson, C; Gracey, D1
Gradin, K; Persson, B1
Hashim, A; Lajtha, A; Sershen, H3
Goldstein, DS; Kopin, IJ; Pacak, K; Yadid, G1
Hiraga, Y; Ikeda, Y; Izumi, J; Miura, N; Washizuka, M1
Bolaños-Jiménez, F; Fillion, G; Manhães de Castro, R1
Bolaños-Jiménez, F; de Castro, RM; Fillion, G1
Cheetham, SC; Heal, DJ1
Muck-Seler, D; Pericić, D1
Ellinwood, EH; Joyner, CM; King, GR1
Heckman, CJ; Lee, RH; Miller, JF; Paul, KD; Rymer, WZ1
Bagdy, E; Harsing, LG1
Abraini, JH; Kriem, B; Rostain, JC1
Kellermann, O; Launay, JM; Loric, S; Maroteaux, L1
Koob, GF; Parsons, LH; Weiss, F1
Pickard, GE; Rea, MA; Riberdy, AF; Scott, PA; Weber, ET1
Mamede Rosa, ML; Prado, WA1
Joppa, MA; Meisel, RL; Rowe, RK1
Cologer-Clifford, A; Lu, SF; Simon, NG; Smoluk, SA1
Katz, LC; Roerig, B1
Colombo, G; Gatto, GJ; Grant, KA1
Durham, PL; Russo, AF; Sharma, RV1
Durham, PL; Russo, AF2
Gean, PW; Lu, KT1
Empson, RM; Gloveli, T; Heinemann, U; Schmitz, D1
Bowen, CA; Gatto, GJ; Grant, KA1
Rainnie, DG1
Delville, Y; Ferris, CF; Stolberg, T1
Khan, NA; Poisson, JP1
O'Neill, MF; Tomkins, DM1
Russo, AF; Wood, JL1
Gao, X; Wu, G; Yang, Z; Zhang, Y1
Garraway, SM; Hochman, S1
Garcia, MM; Minor, LD; Paul, D; Yao, D; Zhu, P1
Blier, P; Diksic, M; Fikre Merid, M; Tohyama, Y; Yamane, F1
Amstislavskaya, TG; Popova, NK1
Adaikan, PG; Hayes, ES1
Grant, KA; Porcu, P1
Jang, MJ; Jeong, HS; Park, JS1
Brumley, MR; Robinson, SR1
Ando, RD; Bagdy, G; Benko, A; Ferrington, L; Kelly, PA; Kirilly, E1
Calama, E; Martín, ML; Morán, A; Ortíz de Urbina, AV; San Román, L1
Odagaki, Y; Toyoshima, R1
Coppinger, D; Maciag, D; Paul, IA1
Aoyama, T; Hattori, T; Kato, S; Kurosawa, S; Nahata, M; Ohno, S; Ro, S; Sakurada, T; Takabayashi, H; Tamai, M; Yakabi, K; Yuzurihara, M1
Jiang, Z; Shang, J; Wang, W; Zhang, H; Zhang, L1
Bakhtiari, A; Salari, AA; Solati, J1
Khatri, N; Lin, RC; Paul, IA; Simpson, KL1
García, M; García-Pedraza, JÁ; Martín, ML; Morán, A1
Avdonin, PP; Avdonin, PV; Goncharov, NV; Mironova, GY; Nadeev, AD; Zharkikh, IL1

Other Studies

71 other study(ies) available for quinoxalines and cgs 12066b

ArticleYear
Effect of 5-HT1A receptor agonists in two models of anxiety after dorsal raphe injection.
    Psychopharmacology, 1992, Volume: 106, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anxiety; Conflict, Psychological; Injections; Interpersonal Relations; Male; Microinjections; Piperazines; Pyrimidines; Quinoxalines; Raphe Nuclei; Rats; Receptors, N-Methyl-D-Aspartate; Receptors, Serotonin; Tetrahydronaphthalenes

1992
Noradrenergic mediation of spinal antinociception by 5-hydroxytryptamine: characterization of receptor subtypes.
    European journal of pharmacology, 1992, Nov-13, Volume: 223, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic alpha-Antagonists; Amphetamines; Animals; Desipramine; In Vitro Techniques; Male; Nociceptors; Norepinephrine; Oxidopamine; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Spinal Cord

1992
Serotonin-norepinephrine interactions: a voltammetric study on the effect of serotonin receptor stimulation followed in the N. raphe dorsalis and the Locus coeruleus of the rat.
    Journal of neural transmission. General section, 1992, Volume: 88, Issue:1

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Drug Interactions; Electrophysiology; Hydroxyindoleacetic Acid; Locus Coeruleus; Male; Microelectrodes; Norepinephrine; Quinoxalines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1992
Serotonin inhibits adenylate cyclase in human platelet membranes.
    European journal of pharmacology, 1992, Aug-03, Volume: 226, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Binding Sites; Blood Platelets; Colforsin; Dose-Response Relationship, Drug; Humans; Methysergide; Quinoxalines; Receptors, Serotonin; Serotonin; Spiperone; Yohimbine

1992
Serotonin is a directly-acting hyperalgesic agent in the rat.
    Neuroscience, 1992, Volume: 48, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Hydroxyurea; Hyperalgesia; Indomethacin; Male; Nociceptors; Oxidopamine; Pain; Quinoxalines; Rats; Rats, Inbred Strains; Reflex; Sensory Thresholds; Serotonin; Serotonin Antagonists; Tetrahydronaphthalenes

1992
Is there a relationship between 5-HT1B receptors and the mechanisms of action of antidepressant drugs in the learned helplessness paradigm in rats?
    European journal of pharmacology, 1991, Jan-03, Volume: 192, Issue:1

    Topics: Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Avoidance Learning; Electroshock; Helplessness, Learned; Male; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Synaptic Transmission

1991
Differential effects of novel ligands for 5-HT receptor subtypes on nonopioid defensive analgesia in male mice.
    Neuroscience and biobehavioral reviews, 1991,Winter, Volume: 15, Issue:4

    Topics: Aggression; Analgesia; Animals; Dioxins; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred DBA; Pyrazines; Quinolines; Quinoxalines; Reaction Time; Receptors, Serotonin; Ritanserin; Serotonin Antagonists; Spiro Compounds

1991
Isolation increases a behavioral response to the selective 5-HT 1B agonist CGS 120 66B.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 40, Issue:2

    Topics: Animals; Behavior, Animal; Male; Mice; Piperazines; Quinoxalines; Receptors, Serotonin; Social Isolation

1991
The inhibitory effect of trifluoromethylphenylpiperazine on [3H]acetylcholine release in guinea pig hippocampal synaptosomes is mediated by a 5-hydroxytryptamine1 receptor distinct from 1A, 1B, and 1C subtypes.
    Journal of neurochemistry, 1991, Volume: 56, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Guinea Pigs; Hippocampus; Male; Piperazines; Potassium; Quinoxalines; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Synaptosomes; Tetrahydronaphthalenes

1991
Tolerance to the behavioural effect of serotonergic (5-HT1B) agonists in the isolation-induced social behavioural deficit test.
    Neuropharmacology, 1991, Volume: 30, Issue:6

    Topics: Animals; Behavior, Animal; Drug Tolerance; Indoles; Male; Mice; Piperazines; Quinoxalines; Receptors, N-Methyl-D-Aspartate; Serotonin; Social Isolation

1991
The effects of 5-HT1B characterizing agents in the mouse elevated plus-maze.
    Life sciences, 1990, Volume: 47, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anxiety Disorders; Chlordiazepoxide; Male; Mice; Mice, Inbred Strains; Models, Psychological; Pentylenetetrazole; Piperazines; Quinoxalines; Serotonin

1990
Agonist action at 5-HT1C receptors facilitates 5-HT1A receptor-mediated spontaneous tail-flicks in the rat.
    European journal of pharmacology, 1990, Nov-27, Volume: 191, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Male; Piperazines; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Reflex; Tail; Tetrahydronaphthalenes

1990
Effects of the 5-HT1 receptor agonists DP-5-CT, CGS 12066B, and RU 24969 on plasma adrenaline and glucose levels in the rat.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 342, Issue:4

    Topics: Animals; Blood Glucose; Dose-Response Relationship, Drug; Epinephrine; Indoles; Male; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Tryptamines

1990
Selective reduction by serotonergic agents of hypertonic saline consumption in rats: evidence for possible 5-HT1C receptor mediation.
    Psychopharmacology, 1989, Volume: 99, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Drinking Behavior; Fenfluramine; Fluoxetine; Hypertonic Solutions; Indoles; Male; Piperazines; Pyrazines; Quinoxalines; Quipazine; Rats; Receptors, Serotonin; Serotonin

1989
Electrophysiological evidence for a functional differentiation between subtypes of the 5-HT1 receptor.
    European journal of pharmacology, 1988, Nov-22, Volume: 157, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Animals; Anti-Anxiety Agents; Male; Piperazines; Pyrimidines; Quinoxalines; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Serotonin; Substantia Nigra; Tetrahydronaphthalenes

1988
Biochemical and pharmacological characterization of CGS 12066B, a selective serotonin-1B agonist.
    European journal of pharmacology, 1987, Apr-07, Volume: 136, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Dihydroalprenolol; Electrophysiology; Hypothalamus; In Vitro Techniques; Male; Quinoxalines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Synaptosomes

1987
5-HT1B/1D agonist CGS-12066B attenuates clasp knife reflex in the cat.
    Journal of neurophysiology, 1995, Volume: 74, Issue:1

    Topics: Animals; Cats; Injections, Spinal; Microinjections; Muscle, Skeletal; Quinoxalines; Reflex; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

1995
Differential effects of CGS 12066B and CP-94,253 on murine social and agonistic behaviour.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 52, Issue:1

    Topics: Agonistic Behavior; Animals; Anxiety; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred Strains; Pyridines; Quinoxalines; Serotonin Receptor Agonists; Social Behavior

1995
Cardiovascular effects of intrathecal administration of agents active at 5-hydroxytryptamine1-receptors in the rat: modulation by substance P and a substance P antagonist.
    Journal of neural transmission. General section, 1993, Volume: 93, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Biphenyl Compounds; Blood Pressure; Heart Rate; Hypnotics and Sedatives; Injections, Spinal; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Spinal Cord; Substance P; Tetrahydronaphthalenes; Time Factors

1993
Spinal supersensitivity to 5-HT1, 5-HT2 and 5-HT3 receptor agonists following 5,7-dihydroxytryptamine.
    European journal of pharmacology, 1994, Nov-03, Volume: 264, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Amphetamines; Analgesia; Analgesics; Analysis of Variance; Animals; Binding Sites; Indoles; Injections, Spinal; Male; Pain; Piperazines; Quinoxalines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Up-Regulation

1994
Effect of ibogaine on serotonergic and dopaminergic interactions in striatum from mice and rats.
    Neurochemical research, 1994, Volume: 19, Issue:11

    Topics: Animals; Biological Transport; Corpus Striatum; Dopamine; Electric Stimulation; Ibogaine; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Quinoxalines; Rats; Rats, Sprague-Dawley; Reference Values; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sulpiride; Tritium; Tropanes

1994
Endogenous serotonin stimulates striatal dopamine release in conscious rats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:3

    Topics: 5,7-Dihydroxytryptamine; Alanine; Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Male; Microdialysis; Perfusion; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

1994
Hippocampal serotonin 5-HT1A receptor enhances acetylcholine release in conscious rats.
    Journal of neurochemistry, 1994, Volume: 62, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Clomipramine; Hippocampus; Kinetics; Male; Physostigmine; Piperazines; Quinoxalines; Rats; Rats, Inbred F344; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1994
Effect of chronic antidepressant treatment on 5-HT1B presynaptic heteroreceptors inhibiting acetylcholine release.
    Neuropharmacology, 1994, Volume: 33, Issue:1

    Topics: Acetylcholine; Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Citalopram; Hippocampus; In Vitro Techniques; Male; Potassium; Quinoxalines; Rats; Rats, Wistar; Receptors, Presynaptic; Receptors, Serotonin; Synaptosomes; Thiazepines

1994
Antagonism by citalopram and tianeptine of presynaptic 5-HT1B heteroreceptors inhibiting acetylcholine release.
    European journal of pharmacology, 1993, Sep-21, Volume: 242, Issue:1

    Topics: Acetylcholine; Animals; Antidepressive Agents, Tricyclic; Citalopram; Hippocampus; Male; Potassium; Quinoxalines; Rats; Rats, Wistar; Receptors, Serotonin; Synaptosomes; Thiazepines

1993
Evidence that RU 24969-induced locomotor activity in C57/B1/6 mice is specifically mediated by the 5-HT1B receptor.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Biogenic Monoamines; Brain Chemistry; Indoles; Male; Methoxydimethyltryptamines; Mice; Mice, Inbred C57BL; Motor Activity; Prazosin; Quinoxalines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1993
Possible antidepressant dihydroergosine preferentially binds to 5-HT1B receptor sites in the rat hippocampus.
    Journal of neural transmission. General section, 1993, Volume: 92, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antidepressive Agents; Binding, Competitive; Chlorpromazine; Ergotamines; Hippocampus; In Vitro Techniques; Male; Pindolol; Quinoxalines; Rats; Rats, Wistar; Receptors, Serotonin

1993
Withdrawal from continuous or intermittent cocaine: behavioral responsivity to 5-HT1 receptor agonists.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 45, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Cocaine; Drug Tolerance; Male; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Substance Withdrawal Syndrome

1993
Restoration of extensor excitability in the acute spinal cat by the 5-HT2 agonist DOI.
    Journal of neurophysiology, 1996, Volume: 75, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Cats; Decerebrate State; Electromyography; In Vitro Techniques; Quinoxalines; Reflex, Stretch; Serotonin; Serotonin Receptor Agonists

1996
The role of various calcium and potassium channels in the regulation of somatodendritic serotonin release.
    Neurochemical research, 1995, Volume: 20, Issue:12

    Topics: Animals; Axons; Calcium Channels; Dendrites; Hippocampus; Male; Piperazines; Potassium Channels; Quinoxalines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

1995
Effect of ibogaine on cocaine-induced efflux of [3H] dopamine and [3H] serotonin from mouse striatum.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:4

    Topics: Adrenergic beta-Antagonists; Animals; Cocaine; Dopamine; Ibogaine; Male; Mice; Mice, Inbred C57BL; Motor Activity; Narcotics; Neostriatum; Propranolol; Quinoxalines; Receptors, Opioid, kappa; Serotonin; Serotonin Receptor Agonists

1996
Role of 5-HT1b receptor in the pressure-induced behavioral and neurochemical disorders in rats.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:2

    Topics: Adrenergic beta-Agonists; Animals; Atmospheric Pressure; Behavior, Animal; Brain Chemistry; Calibration; Dopamine; Electrochemistry; Electrodes; High Pressure Neurological Syndrome; Isoproterenol; Male; Motor Activity; Neostriatum; Pindolol; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

1996
Sequential onset of three 5-HT receptors during the 5-hydroxytryptaminergic differentiation of the murine 1C11 cell line.
    British journal of pharmacology, 1996, Volume: 118, Issue:5

    Topics: Animals; Antiparkinson Agents; Cells, Cultured; Colforsin; Cyclic AMP; Ergolines; Gene Expression; Quinoxalines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Time Factors

1996
Serotonin1b receptor stimulation enhances dopamine-mediated reinforcement.
    Psychopharmacology, 1996, Volume: 128, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Narcotics; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Receptor Agonists

1996
5HT1B receptor agonists inhibit light-induced phase shifts of behavioral circadian rhythms and expression of the immediate-early gene c-fos in the suprachiasmatic nucleus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Dec-15, Volume: 16, Issue:24

    Topics: Animals; Behavior, Animal; Circadian Rhythm; Cricetinae; Eye Enucleation; Gene Expression; Genes, fos; Light; Male; Mesocricetus; Piperazines; Quinoxalines; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Superior Colliculi; Suprachiasmatic Nucleus

1996
Antinociception induced by opioid or 5-HT agonists microinjected into the anterior pretectal nucleus of the rat.
    Brain research, 1997, May-16, Volume: 757, Issue:1

    Topics: Analgesics; Animals; Benzomorphans; Brain; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; Male; Microinjections; Pain; Phenazocine; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Serotonin; Serotonin Receptor Agonists

1997
Effects of serotonin 1A or 1B receptor agonists on social aggression in male and female Syrian hamsters.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Cricetinae; Female; Male; Quinoxalines; Serotonin Receptor Agonists; Sex Factors; Social Behavior

1997
Serotonin agonist-induced decreases in intermale aggression are dependent on brain region and receptor subtype.
    Pharmacology, biochemistry, and behavior, 1997, Volume: 58, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Male; Mice; Motor Activity; Preoptic Area; Quinoxalines; Septal Nuclei; Serotonin Receptor Agonists

1997
Modulation of intrinsic circuits by serotonin 5-HT3 receptors in developing ferret visual cortex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Ferrets; gamma-Aminobutyric Acid; Indoles; Ligands; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Pyridinium Compounds; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, GABA-A; Receptors, GABA-B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Tetrodotoxin; Time Factors; Tropisetron; Virulence Factors, Bordetella; Visual Cortex

1997
Characterization of the ethanol-like discriminative stimulus effects of 5-HT receptor agonists as a function of ethanol training dose.
    Psychopharmacology, 1997, Volume: 133, Issue:2

    Topics: Animals; Central Nervous System Depressants; Conditioning, Operant; Discrimination, Psychological; Ethanol; Indoles; Male; Piperazines; Quinoxalines; Rats; Serotonin Receptor Agonists

1997
Repression of the calcitonin gene-related peptide promoter by 5-HT1 receptor activation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-15, Volume: 17, Issue:24

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enhancer Elements, Genetic; Gene Expression Regulation; Genes, Reporter; Neurons; Promoter Regions, Genetic; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; RNA, Messenger; Serotonin Receptor Agonists; Sumatriptan; Thyroid Neoplasms; Time Factors; Transcription, Genetic; Trigeminal Ganglion; Tumor Cells, Cultured

1997
Serotonergic repression of mitogen-activated protein kinase control of the calcitonin gene-related peptide enhancer.
    Molecular endocrinology (Baltimore, Md.), 1998, Volume: 12, Issue:7

    Topics: Animals; Calcitonin Gene-Related Peptide; Calcium-Calmodulin-Dependent Protein Kinases; Carcinoma, Medullary; Cell Cycle Proteins; DNA-Binding Proteins; Dual Specificity Phosphatase 1; Enhancer Elements, Genetic; ets-Domain Protein Elk-1; Genes, jun; Immediate-Early Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinases; Protein Phosphatase 1; Protein Tyrosine Phosphatase, Non-Receptor Type 1; Protein Tyrosine Phosphatases; Proto-Oncogene Proteins; Quinoxalines; Rats; Serotonin; Serotonin Receptor Agonists; Thyroid Neoplasms; Transcription Factors; Transfection; Tumor Cells, Cultured

1998
Endogenous serotonin inhibits epileptiform activity in rat hippocampal CA1 neurons via 5-hydroxytryptamine1A receptor activation.
    Neuroscience, 1998, Volume: 86, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Barium; Epilepsy; Excitatory Postsynaptic Potentials; Fluoxetine; Hippocampus; In Vitro Techniques; Ketanserin; Male; Membrane Potentials; Metergoline; Neurons; Oxadiazoles; Picrotoxin; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Tryptamines

1998
Serotonin reduces polysynaptic inhibition via 5-HT1A receptors in the superficial entorhinal cortex.
    Journal of neurophysiology, 1998, Volume: 80, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Entorhinal Cortex; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Free Radical Scavengers; Membrane Potentials; Neural Inhibition; Organ Culture Techniques; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses

1998
Assessment of the multiple discriminative stimulus effects of ethanol using an ethanol-pentobarbital-water discrimination in rats.
    Behavioural pharmacology, 1997, Volume: 8, Issue:4

    Topics: Animals; Central Nervous System Depressants; Diazepam; Discrimination Learning; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ethanol; GABA Modulators; Hypnotics and Sedatives; Indoles; Male; Midazolam; Morphine; N-Methylaspartate; Narcotics; Pentobarbital; Phencyclidine; Pregnanolone; Quinoxalines; Rats; Rats, Long-Evans; Serotonin Receptor Agonists; Water

1997
Regulation of calcitonin gene-related peptide secretion by a serotonergic antimigraine drug.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, May-01, Volume: 19, Issue:9

    Topics: Animals; Animals, Newborn; Calcitonin Gene-Related Peptide; Cells, Cultured; Colforsin; Cyclic AMP; HeLa Cells; Humans; Inflammation; Kinetics; Models, Neurological; Neurons; Okadaic Acid; Oxadiazoles; Potassium Chloride; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Serotonin Receptor Agonists; Sumatriptan; Transfection; Trigeminal Ganglion; Tryptamines

1999
Serotonergic modulation of neurotransmission in the rat basolateral amygdala.
    Journal of neurophysiology, 1999, Volume: 82, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amygdala; Animals; Bicuculline; Evoked Potentials; Excitatory Postsynaptic Potentials; GABA-A Receptor Antagonists; In Vitro Techniques; Interneurons; Male; Neurons; Patch-Clamp Techniques; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Synaptic Transmission; Tetrodotoxin

1999
Serotonin regulation of aggressive behavior in male golden hamsters (Mesocricetus auratus).
    Behavioral neuroscience, 1999, Volume: 113, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Arginine Vasopressin; Behavior, Animal; Cricetinae; Hypothalamus, Anterior; Male; Mesocricetus; Neural Pathways; Neurotransmitter Agents; Quinoxalines; Raphe Nuclei; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1999
5-HT3 receptor-channels coupled with Na+ influx in human T cells: role in T cell activation.
    Journal of neuroimmunology, 1999, Sep-01, Volume: 99, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Calcium Signaling; Cell Cycle; Enzyme Activation; Granisetron; Humans; Ion Channel Gating; Ion Transport; Jurkat Cells; Lymphocyte Activation; Metoclopramide; Neoplasm Proteins; Phytohemagglutinins; Piperazines; Protein Kinase C; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Ryanodine; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium; Sodium Channels; T-Lymphocytes; Thapsigargin

1999
Effect of 5-HT(1B) receptor ligands on self-administration of ethanol in an operant procedure in rats.
    Pharmacology, biochemistry, and behavior, 2000, Volume: 66, Issue:1

    Topics: Alcohol Drinking; Animals; Conditioning, Operant; Ethanol; Indoles; Male; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration

2000
Serotonin-mediated striatal dopamine release involves the dopamine uptake site and the serotonin receptor.
    Brain research bulletin, 2000, Volume: 53, Issue:3

    Topics: Animals; Bicuculline; Cocaine; Corpus Striatum; Dizocilpine Maleate; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; Ketanserin; Male; Methiothepin; Mice; Mice, Inbred C57BL; Oxymetazoline; Piperazines; Quinoxalines; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Autoregulation of cell-specific MAP kinase control of the tryptophan hydroxylase promoter.
    The Journal of biological chemistry, 2001, Jun-15, Volume: 276, Issue:24

    Topics: Animals; Base Sequence; Butadienes; Cell Line; CHO Cells; Cricetinae; Enzyme Inhibitors; Enzyme Repression; Gene Expression Regulation, Enzymologic; Genes, Reporter; Imidazoles; Kinetics; Luciferases; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Models, Biological; Molecular Sequence Data; Neurons; Nitriles; Promoter Regions, Genetic; Pyridines; Quinoxalines; Recombinant Proteins; Serotonin Receptor Agonists; Transcription, Genetic; Transfection; Tryptophan Hydroxylase

2001
The role of 5-hydroxytryptamine1A and 5-hydroxytryptamine1B receptors in modulating spinal nociceptive transmission in normal and carrageenan-injected rats.
    Pain, 2001, Volume: 92, Issue:1-2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Carrageenan; Electric Stimulation; Electrophysiology; Female; Male; Neurons, Afferent; Nociceptors; Pain; Piperazines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

2001
Serotonin increases the incidence of primary afferent-evoked long-term depression in rat deep dorsal horn neurons.
    Journal of neurophysiology, 2001, Volume: 85, Issue:5

    Topics: Afferent Pathways; Amphetamines; Animals; Animals, Newborn; Biguanides; Boron Compounds; Excitatory Postsynaptic Potentials; Long-Term Potentiation; Methacrylates; Methylmethacrylates; Nerve Tissue Proteins; Neuronal Plasticity; Patch-Clamp Techniques; Posterior Horn Cells; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Single-Blind Method; Synaptic Transmission

2001
5-hydroxytryptamine3 (5-HT3) receptors mediate spinal 5-HT antinociception: an antisense approach.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:2

    Topics: Animals; Injections, Spinal; Male; Mice; Nociceptors; Oligodeoxyribonucleotides, Antisense; Pain Measurement; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Agents; Serotonin Receptor Agonists; Spinal Cord

2001
Effects of serotine receptors agonists, TFMPP and CGS12066B, on regional serotonin synthesis in the rat brain: an autoradiographic study.
    Journal of neurochemistry, 2002, Volume: 80, Issue:5

    Topics: Animals; Autoradiography; Body Weight; Brain; Brain Chemistry; Carbon Radioisotopes; Injections, Intraperitoneal; Male; Piperazines; Quinoxalines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Tissue Distribution; Tryptophan

2002
Involvement of the 5-HT(1A) and 5-HT(1B) serotonergic receptor subtypes in sexual arousal in male mice.
    Psychoneuroendocrinology, 2002, Volume: 27, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Female; Male; Mice; Mice, Inbred BALB C; Mice, Inbred CBA; Motivation; Piperazines; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Sexual Behavior, Animal

2002
The effects of 5HT(1) agonists on erection in rats in vivo and rabbit corpus cavernosum in vitro.
    International journal of impotence research, 2002, Volume: 14, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Dopamine Agonists; Male; Muscle, Smooth; Penile Erection; Penis; Pressure; Quinoxalines; Rabbits; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists

2002
Discriminative stimulus effects of ethanol in rats using a three-choice ethanol-midazolam-water discrimination.
    Behavioural pharmacology, 2004, Volume: 15, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Central Nervous System Depressants; Discrimination Learning; Discrimination, Psychological; Dizocilpine Maleate; Dose-Response Relationship, Drug; Ethanol; Excitatory Amino Acid Antagonists; Hypnotics and Sedatives; Indoles; Midazolam; Pentobarbital; Phencyclidine; Piperazines; Pregnanolone; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Serotonin Receptor Agonists

2004
Effects of CGS-12066A on medial vestibular nuclear neurons.
    Brain research, 2005, Mar-15, Volume: 1038, Issue:1

    Topics: Action Potentials; Animals; Calcium; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Potassium Channels; Quinoxalines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists; Vestibular Nuclei

2005
The serotonergic agonists quipazine, CGS-12066A, and alpha-methylserotonin alter motor activity and induce hindlimb stepping in the intact and spinal rat fetus.
    Behavioral neuroscience, 2005, Volume: 119, Issue:3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Embryo, Mammalian; Female; Hindlimb; Male; Motor Activity; Pregnancy; Psychomotor Performance; Quinoxalines; Quipazine; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Receptor Agonists; Spinal Cord Injuries

2005
Acute and long-term effects of a single dose of MDMA on aggression in Dark Agouti rats.
    The international journal of neuropsychopharmacology, 2006, Volume: 9, Issue:1

    Topics: Adrenergic Uptake Inhibitors; Aggression; Animals; Brain; Glucose; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Pyridines; Quinoxalines; Rats; Receptors, Serotonin, 5-HT1; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Time Factors

2006
Effect of 5-hydroxytryptamine on neurogenic vasoconstriction in the isolated, autoperfused hindquarters of the rat.
    Clinical and experimental pharmacology & physiology, 2005, Volume: 32, Issue:10

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Biguanides; Biphenyl Compounds; Dose-Response Relationship, Drug; Electric Stimulation; Hindlimb; In Vitro Techniques; Infusions, Intravenous; Male; Methiothepin; Oxadiazoles; Perfusion; Piperazines; Pressure; Quinoxalines; Rats; Rats, Wistar; Ritanserin; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Agonists; Serotonin 5-HT3 Receptor Agonists; Serotonin Agents; Serotonin Antagonists; Serotonin Receptor Agonists; Tryptamines; Vasoconstriction

2005
5-HT1A receptor-mediated G protein activation assessed by [35S]GTPgammaS binding in rat cerebral cortex.
    European journal of pharmacology, 2005, Oct-03, Volume: 521, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; Dose-Response Relationship, Drug; Enzyme Activation; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Hippocampus; Magnesium Chloride; Male; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride; Sulfur Radioisotopes

2005
Evidence that the deficit in sexual behavior in adult rats neonatally exposed to citalopram is a consequence of 5-HT1 receptor stimulation during development.
    Brain research, 2006, Dec-13, Volume: 1125, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Age Factors; Analysis of Variance; Animals; Animals, Newborn; Behavior, Animal; Citalopram; Female; Male; Pregnancy; Quinoxalines; Rats; Rats, Long-Evans; Reaction Time; Receptors, Serotonin, 5-HT1; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Sexual Behavior, Animal; Sexual Dysfunction, Physiological

2006
Rikkunshito and 5-HT2C receptor antagonist improve cisplatin-induced anorexia via hypothalamic ghrelin interaction.
    Regulatory peptides, 2010, Apr-09, Volume: 161, Issue:1-3

    Topics: Animals; Anorexia; Cisplatin; Drugs, Chinese Herbal; Eating; Gastric Mucosa; Ghrelin; Granisetron; Hypothalamus; Male; Oligopeptides; Ondansetron; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, Ghrelin; Reverse Transcriptase Polymerase Chain Reaction; Serotonin 5-HT2 Receptor Antagonists; Stomach

2010
Differential involvement of 5-HT(1A) and 5-HT(1B/1D) receptors in human interferon-alpha-induced immobility in the mouse forced swimming test.
    Arzneimittel-Forschung, 2010, Volume: 60, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Buspirone; Depression; Fluoxetine; Interferon-alpha; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2010
5HT(1A) and 5HT(1B) receptors of medial prefrontal cortex modulate anxiogenic-like behaviors in rats.
    Neuroscience letters, 2011, Oct-31, Volume: 504, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Anti-Anxiety Agents; Anxiety; Exploratory Behavior; Male; Microinjections; Piperazines; Piperidones; Prefrontal Cortex; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds

2011
Lasting neurobehavioral abnormalities in rats after neonatal activation of serotonin 1A and 1B receptors: possible mechanisms for serotonin dysfunction in autistic spectrum disorders.
    Psychopharmacology, 2014, Volume: 231, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Animals, Newborn; Brain; Citalopram; Exploratory Behavior; Female; Freezing Reaction, Cataleptic; Locomotion; Male; Oxadiazoles; Piperazines; Pyridines; Quinoxalines; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Receptor Agonists; Social Behavior

2014
5-HT1D receptor inhibits renal sympathetic neurotransmission by nitric oxide pathway in anesthetized rats.
    Vascular pharmacology, 2015, Volume: 72

    Topics: Animals; Blood Pressure; Heart Rate; Kidney; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; Oxadiazoles; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin 5-HT1 Receptor Antagonists; Sympathetic Nervous System; Synaptic Transmission; Tryptamines

2015
Enhancement by Hydrogen Peroxide of Calcium Signals in Endothelial Cells Induced by 5-HT1B and 5-HT2B Receptor Agonists.
    Oxidative medicine and cellular longevity, 2019, Volume: 2019

    Topics: Acetylcysteine; Benzoxazoles; Calcium; Calcium Signaling; Fluorescence; Human Umbilical Vein Endothelial Cells; Humans; Hydrogen Peroxide; Indoles; Quinoxalines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2B; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT2 Receptor Agonists; Thiophenes; Triazoles; Vanadates

2019