Page last updated: 2024-08-17

quinidine and trifluoperazine

quinidine has been researched along with trifluoperazine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19909 (40.91)18.7374
1990's4 (18.18)18.2507
2000's4 (18.18)29.6817
2010's4 (18.18)24.3611
2020's1 (4.55)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Chiang, GH; Unger, SH1
Casciano, CN; Clement, RP; Johnson, WW; Wang, EJ1
Pajeva, IK; Wiese, M1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Abraham, MH; Acree, WE; Ibrahim, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Fisk, L; Greene, N; Naven, RT; Note, RR; Patel, ML; Pelletier, DJ1
Ekins, S; Williams, AJ; Xu, JJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Dranchak, PK; Huang, R; Inglese, J; Lamy, L; Oliphant, E; Queme, B; Tao, D; Wang, Y; Xia, M1
Gottesman, MM; Horio, M; Lovelace, E; Pastan, I1
Hahn, EW; Osswald, H; Pommerenke, EW; Volm, M1
Jørgensen, PL; Karlish, SJ; Klaerke, DA1
Bindslev, N; Demant, EJ; Friche, E; Jensen, PB; Sehested, M; Skovsgaard, T; Vindeløv, L1
Brown, PD; Sepúlveda, FV1
Foskett, JK; Spring, KR1
Bhargava, KP; Dhawan, KN; Kulshrestha, VK; Shamsi, MA1
Hoffman, JF; Yingst, DR1
Kurtzer, RJ; Roberts, ML1
Choe, KJ; Gottesman, MM; Hong, IG; Kim, HS; Kim, WH; Kim, YI; Lee, SK; Lim, KH; Park, JG; Tsuruo, T1
Raderer, M; Scheithauer, W1

Reviews

2 review(s) available for quinidine and trifluoperazine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Clinical trials of agents that reverse multidrug resistance. A literature review.
    Cancer, 1993, Dec-15, Volume: 72, Issue:12

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Clinical Trials as Topic; Cyclosporins; Drug Resistance; Humans; Phenotype; Quinidine; Tamoxifen; Trifluoperazine; Verapamil

1993

Other Studies

20 other study(ies) available for quinidine and trifluoperazine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Octanol-physiological buffer distribution coefficients of lipophilic amines by reversed-phase high-performance liquid chromatography and their correlation with biological activity.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:3

    Topics: Amines; Animals; Buffers; Chromatography, High Pressure Liquid; Histamine Release; Lipid Metabolism; Octanols; Protein Binding; Rats; Serum Albumin, Bovine; Sodium-Potassium-Exchanging ATPase; Solubility; Structure-Activity Relationship

1981
Active transport of fluorescent P-glycoprotein substrates: evaluation as markers and interaction with inhibitors.
    Biochemical and biophysical research communications, 2001, Nov-30, Volume: 289, Issue:2

    Topics: 3T3 Cells; Adrenergic Uptake Inhibitors; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Biological Transport, Active; Cell Line; Cell Separation; Cell Survival; Flow Cytometry; Fluorescent Dyes; Humans; Inhibitory Concentration 50; Mice; Protein Binding; Reserpine; Spectrometry, Fluorescence; Substrate Specificity; Time Factors

2001
Pharmacophore model of drugs involved in P-glycoprotein multidrug resistance: explanation of structural variety (hypothesis).
    Journal of medicinal chemistry, 2002, Dec-19, Volume: 45, Issue:26

    Topics: Adenosine Triphosphatases; Algorithms; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Binding, Competitive; Caco-2 Cells; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Fluoresceins; Humans; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship; Radioligand Assay; Rhodamine 123; Stereoisomerism; Verapamil; Vinblastine

2002
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Air to lung partition coefficients for volatile organic compounds and blood to lung partition coefficients for volatile organic compounds and drugs.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Air; Animals; Humans; Lung; Organic Chemicals; Probability; Rats; Tissue Distribution; Volatilization

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Developing structure-activity relationships for the prediction of hepatotoxicity.
    Chemical research in toxicology, 2010, Jul-19, Volume: 23, Issue:7

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Humans; Structure-Activity Relationship; Tetracyclines; Thiophenes

2010
A predictive ligand-based Bayesian model for human drug-induced liver injury.
    Drug metabolism and disposition: the biological fate of chemicals, 2010, Volume: 38, Issue:12

    Topics: Bayes Theorem; Chemical and Drug Induced Liver Injury; Humans; Ligands

2010
In vivo quantitative high-throughput screening for drug discovery and comparative toxicology.
    Disease models & mechanisms, 2023, 03-01, Volume: 16, Issue:3

    Topics: Animals; Caenorhabditis elegans; Drug Discovery; High-Throughput Screening Assays; Humans; Proteomics; Small Molecule Libraries

2023
Agents which reverse multidrug-resistance are inhibitors of [3H]vinblastine transport by isolated vesicles.
    Biochimica et biophysica acta, 1991, Jan-09, Volume: 1061, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding, Competitive; Biological Transport, Active; Carcinoma, Squamous Cell; Cell Membrane; Dihydropyridines; Drug Resistance; Humans; Kinetics; Leucine; Membrane Glycoproteins; Phenothiazines; Quinidine; Trifluoperazine; Tumor Cells, Cultured; Verapamil; Vinblastine

1991
Activity of various amphiphilic agents in reversing multidrug resistance of L 1210 cells.
    Cancer letters, 1990, Nov-19, Volume: 55, Issue:1

    Topics: Animals; Drug Resistance; Ethylamines; Hycanthone; Leukemia L1210; Phenotype; Piperidines; Quinidine; Quinine; Tamoxifen; Trifluoperazine; Verapamil

1990
Reconstitution in phospholipid vesicles of calcium-activated potassium channel from outer renal medulla.
    The Journal of membrane biology, 1987, Volume: 95, Issue:2

    Topics: Animals; Calcium; Calmodulin; Imidazoles; Ion Channels; Kidney Medulla; Liposomes; Loop of Henle; Membrane Potentials; Potassium; Quinidine; Rubidium; Swine; Trifluoperazine

1987
Inhibition of vincristine binding to plasma membrane vesicles from daunorubicin-resistant Ehrlich ascites cells by multidrug resistance modulators.
    British journal of cancer, 1989, Volume: 60, Issue:6

    Topics: Animals; Carcinoma, Ehrlich Tumor; Cell Cycle; Cell Membrane; Daunorubicin; Drug Resistance; Polysorbates; Quinidine; Trifluoperazine; Tumor Stem Cell Assay; Verapamil; Vincristine

1989
Potassium movements associated with amino acid and sugar transport in enterocytes isolated from rabbit jejunum.
    The Journal of physiology, 1985, Volume: 363

    Topics: Amino Acids; Animals; Apamin; Barium; Biological Transport, Active; Calcimycin; Cell Membrane Permeability; Female; Furosemide; In Vitro Techniques; Jejunum; Male; Methylglucosides; Methylglycosides; Potassium; Quinidine; Rabbits; Trifluoperazine

1985
Involvement of calcium and cytoskeleton in gallbladder epithelial cell volume regulation.
    The American journal of physiology, 1985, Volume: 248, Issue:1 Pt 1

    Topics: Animals; Calcium; Cytoskeleton; Epithelial Cells; Epithelium; Gallbladder; Gallopamil; Necturus; Osmolar Concentration; Promethazine; Quinidine; Trifluoperazine

1985
Correlation of chemical structure of phenothiazines with their coronary dilator and antiarrhythmic activities.
    Japanese journal of pharmacology, 1971, Volume: 21, Issue:6

    Topics: Alkaloids; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Chlorpromazine; Coronary Vessels; Dogs; In Vitro Techniques; Ligation; Nitroglycerin; Perphenazine; Phenothiazines; Promazine; Promethazine; Quinidine; Rabbits; Strophanthins; Structure-Activity Relationship; Thioridazine; Trifluoperazine; Triflupromazine; Vasodilator Agents

1971
Ca-induced K transport in human red blood cell ghosts containing arsenazo III. Transmembrane interactions of Na, K, and Ca and the relationship to the functioning Na-K pump.
    The Journal of general physiology, 1984, Volume: 83, Issue:1

    Topics: Adenosine Triphosphate; Arsenazo III; Calcimycin; Calcium; Cell Membrane Permeability; Erythrocyte Membrane; Humans; Ion Channels; Potassium; Quinidine; Sodium; Trifluoperazine

1984
Calcium-dependent K+ efflux from rat submandibular gland. The effects of trifluoperazine and quinidine.
    Biochimica et biophysica acta, 1982, Dec-22, Volume: 693, Issue:2

    Topics: Animals; Biological Transport; Calcimycin; Calcium; Epinephrine; Female; Kinetics; Potassium; Quinidine; Rats; Submandibular Gland; Trifluoperazine

1982
MDR1 gene expression: its effect on drug resistance to doxorubicin in human hepatocellular carcinoma cell lines.
    Journal of the National Cancer Institute, 1994, May-04, Volume: 86, Issue:9

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carcinoma, Hepatocellular; Carrier Proteins; Cefoperazone; Ceftriaxone; Doxorubicin; Drug Resistance; Drug Synergism; Gene Expression; Humans; Immunohistochemistry; Liver Neoplasms; Membrane Glycoproteins; Neoplasm Proteins; Quinidine; RNA, Messenger; Trifluoperazine; Tumor Cells, Cultured; Verapamil

1994