Page last updated: 2024-08-17

quinidine and pyrilamine

quinidine has been researched along with pyrilamine in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19903 (27.27)18.7374
1990's2 (18.18)18.2507
2000's3 (27.27)29.6817
2010's2 (18.18)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Nezu, J; Oku, A; Sai, Y; Sakamoto, K; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Nezu, JI; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A; Yabuuchi, H1
Hashimoto, N; Nezu Ji, J; Nikaido, H; Ohashi, R; Oku, A; Sai, Y; Shimane, M; Tamai, I; Tsuji, A1
Ambroso, JL; Ayrton, AD; Baines, IA; Bloomer, JC; Chen, L; Clarke, SE; Ellens, HM; Harrell, AW; Lovatt, CA; Reese, MJ; Sakatis, MZ; Taylor, MA; Yang, EY1
JOHNSON, EA1
JOHNSON, EA; McKINNON, MG1
Chatelain, P; Fuks, B; Gillard, M; Wolff, C1
Irokawa, M; Kobayashi, D; Maeda, T; Tamai, I; Tsuji, A1
Lai, PC; Walters, JD1
Chang, H; Chen, C; Du, H; Guan, C; Li, C; Qiu, L; Wang, S; Wang, T; Wu, Y; Zhang, L; Zhang, S; Zhou, H1

Other Studies

11 other study(ies) available for quinidine and pyrilamine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:2

    Topics: Animals; Biological Transport, Active; Carrier Proteins; Cell Line; Gene Expression; Humans; Hydrogen-Ion Concentration; Membrane Potentials; Membrane Proteins; Membrane Transport Proteins; Oocytes; Organic Cation Transport Proteins; Quinidine; RNA, Messenger; Symporters; Tetraethylammonium Compounds; Xenopus laevis

1999
Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Biological Transport, Active; Carnitine; Carrier Proteins; Cations; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Humans; Hydrogen-Ion Concentration; Kidney; Membrane Proteins; Organic Cation Transport Proteins; Sodium; Solute Carrier Family 22 Member 5; Stereoisomerism

1999
Molecular and physiological evidence for multifunctionality of carnitine/organic cation transporter OCTN2.
    Molecular pharmacology, 2001, Volume: 59, Issue:2

    Topics: Animals; Biological Transport; Carbon Radioisotopes; Carnitine; Carrier Proteins; Cells, Cultured; Embryo, Mammalian; Fibroblasts; Humans; Male; Membrane Proteins; Mice; Mice, Inbred C3H; Organic Cation Transport Proteins; Solute Carrier Family 22 Member 5; Tetraethylammonium; Tissue Distribution; Tritium

2001
Preclinical strategy to reduce clinical hepatotoxicity using in vitro bioactivation data for >200 compounds.
    Chemical research in toxicology, 2012, Oct-15, Volume: 25, Issue:10

    Topics: Chemical and Drug Induced Liver Injury; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Decision Trees; Drug Evaluation, Preclinical; Drug-Related Side Effects and Adverse Reactions; Glutathione; Humans; Liver; Pharmaceutical Preparations; Protein Binding

2012
The effects of quinidine, procaine amide and pyrilamine on the membrane resting and action potential of guinea pig ventricular muscle fibers.
    The Journal of pharmacology and experimental therapeutics, 1956, Volume: 117, Issue:2

    Topics: Action Potentials; Anti-Allergic Agents; Guinea Pigs; Heart; Heart Ventricles; Histamine H1 Antagonists; Myocardium; Procainamide; Pyrilamine; Quinidine

1956
The differential effect of quinidine and pyrilamine on the myocardial action potential at various rates of stimulation.
    The Journal of pharmacology and experimental therapeutics, 1957, Volume: 120, Issue:4

    Topics: Action Potentials; Anti-Allergic Agents; Heart; Histamine H1 Antagonists; Humans; Myocardium; Pyrilamine; Quinidine

1957
[3H]linopirdine binding to rat brain membranes is not relevant for M-channel interaction.
    European journal of pharmacology, 2005, Jul-25, Volume: 518, Issue:1

    Topics: Animals; Anthracenes; Binding, Competitive; Brain; Cell Membrane; Chlorides; CHO Cells; Cricetinae; Cricetulus; Cytochrome P-450 CYP2D6; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Indoles; KCNQ3 Potassium Channel; Ketoconazole; Kinetics; Liver; Male; Miconazole; Potassium Channels, Voltage-Gated; Pyridines; Pyrilamine; Quinidine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Rubidium; Tritium

2005
Carnitine/organic cation transporter OCTN2-mediated transport of carnitine in primary-cultured epididymal epithelial cells.
    Reproduction (Cambridge, England), 2005, Volume: 130, Issue:6

    Topics: Acetylcarnitine; Amino Acid Transport Systems; Animals; Betaine; Biological Transport; Carnitine; Cells, Cultured; Dose-Response Relationship, Drug; Epididymis; Epithelial Cells; Leucine; Lysine; Male; Organic Cation Transport Proteins; Pyrilamine; Quinidine; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA; Sodium; Solute Carrier Family 22 Member 5; Time Factors

2005
Azithromycin kills invasive Aggregatibacter actinomycetemcomitans in gingival epithelial cells.
    Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:3

    Topics: Aggregatibacter actinomycetemcomitans; Anti-Bacterial Agents; Azithromycin; Biological Transport; Carnitine; Cell Line; Dose-Response Relationship, Drug; Epithelial Cells; Gingiva; Humans; Kinetics; Probenecid; Procainamide; Pyrilamine; Quinidine; Time Factors

2013
Effects of membrane transport activity and cell metabolism on the unbound drug concentrations in the skeletal muscle and liver of drugs: A microdialysis study in rats.
    Pharmacology research & perspectives, 2021, Volume: 9, Issue:5

    Topics: Animals; Antipyrine; Atenolol; Carbamazepine; Cell Membrane; Digoxin; Diltiazem; Diphenhydramine; Drug Elimination Routes; Gabapentin; Lamotrigine; Liver; Memantine; Membrane Transport Proteins; Microdialysis; Muscle, Skeletal; Ofloxacin; Pharmaceutical Preparations; Propranolol; Pyrilamine; Quinidine; Rats; Terfenadine

2021