Page last updated: 2024-08-17

quinidine and amiloride

quinidine has been researched along with amiloride in 39 studies

Research

Studies (39)

TimeframeStudies, this research(%)All Research%
pre-199011 (28.21)18.7374
1990's16 (41.03)18.2507
2000's5 (12.82)29.6817
2010's6 (15.38)24.3611
2020's1 (2.56)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Artursson, P; Bergström, CA; Hoogstraate, J; Matsson, P; Norinder, U; Pedersen, JM1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Du-Cuny, L; Mash, EA; Meuillet, EJ; Moses, S; Powis, G; Song, Z; Zhang, S1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
Campillo, NE; Guerra, A; Páez, JA1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Flatman, PW; Smith, LM1
Günther, T; Höllriegl, V; Vormann, J1
Alvarez, LJ; Candia, OA; Wolosin, JM1
Häussinger, D; Lang, F; Stehle, T1
Abramcheck, FJ; Helman, SI; Van Driessche, W1
Allen, JC; Cragoe, EJ; Kahn, AM; Shelat, H; Zimmer, R1
Civan, MM; Peterson-Yantorno, K; Tang, CS1
Allen, JC; Kahn, AM; Shelat, H1
Insel, PA1
Aronson, PS; Mahnensmith, RL1
Lin, HY; Lowe, A; Warnock, DG; Yee, VJ1
Kuroki, T; Nose, K; Shibanuma, M1
Boullin, DJ; O'Brien, RA1
Arruda, JA1
Fischmeister, R; Mentrard, D; Vassort, G1
Cittadini, A; Di Francesco, A; Wolf, FI1
Diaz, J; Muallem, S; Xu, X; Zhao, H1
Morris, CE; Small, DL1
Bara, M; Guiet-Bara, A1
Günther, T; Vormann, J1
Bendayan, R; Lo, B; Silverman, M1
Chiamvimonvat, N; Duff, HJ; Gillis, AM; Mitchell, LB; Sheldon, RS; Wang, L; Wyse, DG1
Fogelson, BG; Goldstein, JL; Layden, TJ; Mozwecz, H; Schmidt, LN; Snow, JC1
Glaasker, E; Konings, WN; Poolman, B1
Morgan, EH; Savigni, DL1
Geada, MM; Singh, J; Wisdom, DM1
Ebel, H; Günther, T1
Mercure, C; Reudelhuber, TL; Touyz, RM1
Abboud, FM; Chapleau, MW; Lu, Y; Paton, JF; Simms, AE; Tan, ZY; Whiteis, CA1
Cohen, NA; Kreindler, JL; Wilber, M; Xiong, G; Zhao, KQ1
Hotta, K; Oka, K; Shindo, Y; Yamanaka, R1

Reviews

2 review(s) available for quinidine and amiloride

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for quinidine and amiloride

ArticleYear
Amiloride-quinidine interaction: adverse outcomes.
    Clinical pharmacology and therapeutics, 1994, Volume: 56, Issue:6 Pt 1

    Topics: Action Potentials; Aged; Amiloride; Animals; Drug Synergism; Drug Therapy, Combination; Electrocardiography; Female; Guinea Pigs; Humans; Male; Middle Aged; Papillary Muscles; Quinidine; Tachycardia, Ventricular

1994

Other Studies

36 other study(ies) available for quinidine and amiloride

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction and identification of drug interactions with the human ATP-binding cassette transporter multidrug-resistance associated protein 2 (MRP2; ABCC2).
    Journal of medicinal chemistry, 2008, Jun-12, Volume: 51, Issue:11

    Topics: Administration, Oral; Animals; Antineoplastic Agents; Antipsychotic Agents; Antiviral Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Biological Transport; Cell Line; Computer Simulation; Cytochrome P-450 Enzyme System; Drug-Related Side Effects and Adverse Reactions; Estradiol; Humans; Insecta; Liver; Models, Molecular; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Pharmaceutical Preparations; Pharmacology; Structure-Activity Relationship

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Computational modeling of novel inhibitors targeting the Akt pleckstrin homology domain.
    Bioorganic & medicinal chemistry, 2009, Oct-01, Volume: 17, Issue:19

    Topics: Antineoplastic Agents; Blood Proteins; Caco-2 Cells; Cell Membrane Permeability; Computer Simulation; Drug Discovery; Drug Screening Assays, Antitumor; Humans; Models, Molecular; Phosphoproteins; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-akt; Quantitative Structure-Activity Relationship

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
Magnesium transport in ferret red cells.
    The Journal of physiology, 1990, Volume: 431

    Topics: Amiloride; Animals; Biological Transport; Cations, Divalent; Choline; Cobalt; Deoxyglucose; Depression, Chemical; Erythrocytes; Ferrets; Imipramine; In Vitro Techniques; Magnesium; Meglumine; Quinidine; Sodium; Temperature

1990
Characterization of Na(+)-dependent Mg2+ efflux from Mg2(+)-loaded rat erythrocytes.
    Biochimica et biophysica acta, 1990, Apr-30, Volume: 1023, Issue:3

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amiloride; Animals; Biological Transport; Erythrocyte Membrane; Erythrocytes; Intracellular Membranes; Kinetics; Magnesium; Quinidine; Rats; Sodium; Spectrophotometry, Atomic

1990
HCO3- transport in the toad lens epithelium is mediated by an electronegative Na(+)-dependent symport.
    The American journal of physiology, 1990, Volume: 258, Issue:5 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Bicarbonates; Biological Transport; Bufo marinus; Chlorides; Cytosol; Epithelium; Hydrogen-Ion Concentration; In Vitro Techniques; Ionophores; Kinetics; Lens, Crystalline; Quinidine; Sodium

1990
Volume regulation in liver: further characterization by inhibitors and ionic substitutions.
    Hepatology (Baltimore, Md.), 1990, Volume: 11, Issue:2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Acetazolamide; Amiloride; Animals; Barium; Chlorides; Hydrogen-Ion Concentration; Liver; Male; Osmolar Concentration; Potassium; Quinidine; Raffinose; Rats; Rats, Inbred Strains; Verapamil; Water-Electrolyte Balance

1990
Autoregulation of apical membrane Na+ permeability of tight epithelia. Noise analysis with amiloride and CGS 4270.
    The Journal of general physiology, 1985, Volume: 85, Issue:4

    Topics: Amiloride; Animals; Cell Membrane Permeability; Electricity; Epithelium; Homeostasis; Ion Channels; Physiology; Pyrazines; Quinidine; Quinine; Rana pipiens; Skin; Sodium

1985
Sodium-lithium exchange in sarcolemmal vesicles from canine superior mesenteric artery.
    Circulation research, 1988, Volume: 62, Issue:3

    Topics: Amiloride; Animals; Biological Transport, Active; Cell Membrane Permeability; Dogs; Female; Ion Channels; Lithium; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Phloretin; Quinidine; Sarcolemma; Sodium

1988
Coupling of volume and Na+ transport in frog skin epithelium.
    Biology of the cell, 1989, Volume: 66, Issue:1-2

    Topics: Amiloride; Animals; Arginine Vasopressin; Cell Membrane; Electric Conductivity; Epithelium; In Vitro Techniques; Kinetics; Membrane Potentials; Models, Biological; Osmolar Concentration; Phlorhizin; Quinidine; Rana pipiens; Skin Physiological Phenomena; Sodium

1989
Na+-Ca2+ exchange in sarcolemmal vesicles from bovine superior mesenteric artery.
    The American journal of physiology, 1988, Volume: 254, Issue:3 Pt 1

    Topics: Amiloride; Animals; Biological Transport; Calcium; Carrier Proteins; Cattle; Electrochemistry; Mesenteric Arteries; Quinidine; Sarcolemma; Sodium; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers

1988
Phenylalkylamines are promiscuous receptor blockers.
    Trends in pharmacological sciences, 1988, Volume: 9, Issue:1

    Topics: Amiloride; Animals; Humans; Phenethylamines; Quinidine; Receptors, Neurotransmitter

1988
Interrelationships among quinidine, amiloride, and lithium as inhibitors of the renal Na+-H+ exchanger.
    The Journal of biological chemistry, 1985, Oct-15, Volume: 260, Issue:23

    Topics: Amiloride; Animals; Binding, Competitive; Carrier Proteins; Kidney; Kinetics; Lithium; Microvilli; Protein Conformation; Quinidine; Rabbits; Sodium-Hydrogen Exchangers

1985
Regulation of the activity of the Na+-H+ antiporter in brush-border membrane vesicles from the proximal tubule.
    Annals of the New York Academy of Sciences, 1985, Volume: 456

    Topics: Amiloride; Animals; Carrier Proteins; Kidney Tubules, Proximal; Kinetics; Lithium; Microvilli; Quaternary Ammonium Compounds; Quinidine; Rabbits; Sodium; Sodium-Hydrogen Exchangers

1985
Inhibition of proto-oncogene c-fos transcription by inhibitors of protein kinase C and ion transport.
    European journal of biochemistry, 1987, Apr-01, Volume: 164, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 4-Aminopyridine; Amiloride; Aminopyridines; Biological Transport, Active; Calcimycin; Humans; Isoquinolines; Phorbol Esters; Piperazines; Potassium; Protein Kinase C; Proto-Oncogene Mas; Proto-Oncogenes; Quinidine; RNA, Messenger; Sodium; Tetraethylammonium Compounds; Transcription, Genetic

1987
Accumulation, storage and release of adrenergic neuron blocking agents and related drugs by human platelets.
    Biochemical pharmacology, 1972, Jul-01, Volume: 21, Issue:13

    Topics: Amiloride; Binding Sites; Blood Platelets; Carbon Isotopes; Cocaine; Desipramine; Dextroamphetamine; Ethylmaleimide; Guanethidine; Guanidines; Humans; Iodoacetates; Isoquinolines; Ouabain; Parasympatholytics; Quinidine; Reserpine; Serotonin; Tritium

1972
Characterization of the effect of quinidine on Na transport by the toad and turtle bladders.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2

    Topics: Amiloride; Amphotericin B; Animals; Bufo marinus; Calcium; Drug Interactions; Ion Channels; Mitochondria, Liver; Quinidine; Sodium; Turtles; Urinary Bladder

1983
Changes in external Na induce a membrane current related to the Na-Ca exchange in cesium-loaded frog heart cells.
    The Journal of general physiology, 1984, Volume: 84, Issue:2

    Topics: Amiloride; Anesthetics, Local; Animals; Atrial Function; Calcium; Calcium Channel Blockers; Cesium; Doxorubicin; Electric Conductivity; Heart; Hydrogen-Ion Concentration; Ion Exchange; Mathematics; Membrane Potentials; Quinidine; Ranidae; Sodium; Tetrodotoxin; Time Factors

1984
Characterization of magnesium efflux from Ehrlich ascites tumor cells.
    Archives of biochemistry and biophysics, 1994, Feb-01, Volume: 308, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Amiloride; Animals; Antimycin A; Bucladesine; Bumetanide; Calcimycin; Carcinoma, Ehrlich Tumor; Colforsin; Cyclic AMP; Energy Metabolism; Glucose; Homeostasis; Imipramine; Kinetics; Magnesium; Mice; Ouabain; Quinidine; Rotenone; Time Factors; Tumor Cells, Cultured

1994
Regulation of [Na+]i in resting and stimulated submandibular salivary ducts.
    The Journal of biological chemistry, 1995, Aug-18, Volume: 270, Issue:33

    Topics: Amiloride; Animals; Barium Compounds; Carbachol; Ion Transport; Male; Ouabain; Quinidine; Quinine; Rats; Sodium; Submandibular Gland; Tetraethylammonium; Tetraethylammonium Compounds

1995
Pharmacology of stretch-activated K channels in Lymnaea neurones.
    British journal of pharmacology, 1995, Volume: 114, Issue:1

    Topics: Amiloride; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Gadolinium; Lymnaea; Neurons; Patch-Clamp Techniques; Potassium Channels; Quinidine

1995
Inhibitor effects on the ionic exchanges through the human amniotic epithelial cell membranes.
    Cellular and molecular biology (Noisy-le-Grand, France), 1994, Volume: 40, Issue:8

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Amnion; Barium; Cell Membrane; Epithelial Cells; Epithelium; Female; Heterocyclic Compounds; Humans; In Vitro Techniques; Ion Transport; Manganese; Metals; Microvilli; Ouabain; Pregnancy; Quinidine

1994
Reversibility of Na+/Mg2+ antiport in rat erythrocytes.
    Biochimica et biophysica acta, 1995, Mar-08, Volume: 1234, Issue:1

    Topics: Adenosine Triphosphate; Amiloride; Animals; Antiporters; Erythrocytes; Imipramine; In Vitro Techniques; Magnesium; Quinidine; Rats; Sodium

1995
Characterization of cimetidine transport in LLCPK1 cells.
    Journal of the American Society of Nephrology : JASN, 1994, Volume: 5, Issue:1

    Topics: Amiloride; Animals; Anti-Bacterial Agents; Azides; Biological Transport; Carrier Proteins; Cell Line; Cimetidine; Guanidine; Guanidines; Kidney; Macrolides; Microscopy, Fluorescence; Models, Biological; Niacinamide; Proton-Translocating ATPases; Quinidine; Quinine; Sodium Azide; Sodium-Hydrogen Exchangers; Swine; Tetraethylammonium; Tetraethylammonium Compounds

1994
Rabbit esophageal cells possess K+ channels: effect of hyposmotic stress on channel activity.
    Gastroenterology, 1993, Volume: 104, Issue:2

    Topics: Amiloride; Animals; Barium; Esophagus; In Vitro Techniques; Male; Osmolar Concentration; Potassium Channels; Quinidine; Rabbits; Sodium; Sodium-Potassium-Exchanging ATPase

1993
Glycine betaine fluxes in Lactobacillus plantarum during osmostasis and hyper- and hypo-osmotic shock.
    The Journal of biological chemistry, 1996, Apr-26, Volume: 271, Issue:17

    Topics: Amiloride; Amino Acids; Betaine; Biological Transport, Active; Enzyme Inhibitors; Gadolinium; Hydrogen-Ion Concentration; Lactobacillus; Quinidine; Tetraethylammonium Compounds; Water-Electrolyte Balance

1996
Use of inhibitors of ion transport to differentiate iron transporters in erythroid cells.
    Biochemical pharmacology, 1996, Jul-26, Volume: 52, Issue:2

    Topics: Amiloride; Animals; Erythrocyte Membrane; Hydrogen-Ion Concentration; Ion Transport; Iron; Quinidine; Rabbits; Reticulocytes; Sodium Chloride; Sucrose; Transferrin; Valinomycin

1996
Characterization of a sodium-dependent magnesium efflux from magnesium-loaded rat pancreatic acinar cells.
    Experimental physiology, 1996, Volume: 81, Issue:3

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Amiloride; Animals; Biological Transport; Bumetanide; Choline; Dinitrophenols; Female; In Vitro Techniques; Lidocaine; Magnesium; Male; Ouabain; Pancreas; Quinidine; Rats; Rats, Sprague-Dawley; Time Factors

1996
Characterization of Mg(2+) efflux from rat erythrocytes non-loaded with Mg(2+).
    Biochimica et biophysica acta, 1999, Oct-15, Volume: 1421, Issue:2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Amiloride; Animals; Antiporters; Bucladesine; Cations, Divalent; Cells, Cultured; Choline; Erythrocytes; Furosemide; Gluconates; Magnesium; Male; Quinidine; Rats; Rats, Wistar; Sodium Chloride; Sucrose

1999
Angiotensin II type I receptor modulates intracellular free Mg2+ in renally derived cells via Na+-dependent Ca2+-independent mechanisms.
    The Journal of biological chemistry, 2001, Apr-27, Volume: 276, Issue:17

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Amiloride; Angiotensin II; Animals; Antihypertensive Agents; Benzofurans; Biphenyl Compounds; Calcium; Calcium Channel Agonists; Cell Line; Cells, Cultured; Chelating Agents; Cytosol; Dogs; Dose-Response Relationship, Drug; Egtazic Acid; Ethers, Cyclic; Fluorescent Dyes; Fura-2; Imidazoles; Imipramine; Irbesartan; Kidney; Kinetics; Magnesium; Microscopy, Fluorescence; Peptides; Pyridines; Quinidine; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Angiotensin; Sodium; Tetrazoles; Time Factors

2001
Chemoreceptor hypersensitivity, sympathetic excitation, and overexpression of ASIC and TASK channels before the onset of hypertension in SHR.
    Circulation research, 2010, Feb-19, Volume: 106, Issue:3

    Topics: Acid Sensing Ion Channels; Amiloride; Animals; Carotid Body; Gene Expression Regulation; Hydrogen-Ion Concentration; Hypertension; Nerve Tissue Proteins; Phrenic Nerve; Potassium Channels, Tandem Pore Domain; Quinidine; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Sodium Channels; Sodium Cyanide; Sympathetic Nervous System; Time Factors

2010
A role for two-pore K⁺ channels in modulating Na⁺ absorption and Cl⁻ secretion in normal human bronchial epithelial cells.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Jan-01, Volume: 302, Issue:1

    Topics: Absorption; Amiloride; Bronchi; Bupivacaine; Cell Line; Cell Polarity; Chlorides; Colforsin; Epithelial Cells; Humans; Immunohistochemistry; Ion Transport; Potassium Channel Blockers; Potassium Channels, Tandem Pore Domain; Quinidine; Respiratory Mucosa; Sodium

2012
Inhibition of Mg
    Nutrients, 2020, Sep-10, Volume: 12, Issue:9

    Topics: Amiloride; Animals; Cells, Cultured; Cytosol; Glutamic Acid; Hippocampus; Magnesium; Mitochondria; Neurons; Quinidine; Rats

2020