Page last updated: 2024-08-24

quinelorane and quinpirole

quinelorane has been researched along with quinpirole in 19 studies

Research

Studies (19)

TimeframeStudies, this research(%)All Research%
pre-19902 (10.53)18.7374
1990's11 (57.89)18.2507
2000's6 (31.58)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrieux, M; Besançon, R; Giros, B; Martres, MP; Pilon, C; Schwartz, JC; Sokoloff, P1
Bervoets, K; Brocco, M; Dacquet, C; Girardon, S; Gobert, A; Millan, MJ; Newman-Tancredi, A; Peglion, JL; Rivet, JM; Vian, J1
Doll, MK; Kilts, JD; Lawler, CP; Lewis, MM; Mailman, RB; Nichols, DE; Prioleau, C1
Boeckler, F; Gmeiner, P; Hübner, H; Lehmann, T; Ohnmacht, U; Utz, W1
Berry, SA; Gudelsky, GA1
Evans, AM; Green, KL1
Clemens, JA; Phebus, LA; Roush, ME1
Clemens, JA; Foreman, MM; Fuller, RW; Gidda, JS; Hynes, MD; Kornfeld, EC; Nichols, CL; Schaus, JM1
Fuller, RW; Gust, CM1
Bergstrom, DA; Gonzalez, AM; Huang, KX; Kreiss, DS; Sibley, DR; Walters, JR1
Middlemiss, DN; Reavill, C; Storey, VJ1
Cornish, JL; Head, GA; Morton, SJ; van den Buuse, M1
Ashmeade, T; Routledge, C; Taylor, S; Thorn, L1
Hagan, JJ; Hatcher, JP1
Beardsley, PM; Cook, CD2
Heidbreder, CA; Shilliam, CS1
Beardsley, PM; Cook, CD; Newman, JL; Winfree, JC1
Brooks, JM; Bruno, JP; Sarter, M1

Other Studies

19 other study(ies) available for quinelorane and quinpirole

ArticleYear
Pharmacology of human dopamine D3 receptor expressed in a mammalian cell line: comparison with D2 receptor.
    European journal of pharmacology, 1992, Apr-10, Volume: 225, Issue:4

    Topics: Animals; Chlorides; CHO Cells; Cricetinae; Dopamine; Dopamine Agents; Dopamine Antagonists; Guanylyl Imidodiphosphate; Humans; Lithium; Lithium Chloride; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Sodium Chloride; Sulpiride; Transfection

1992
Functional correlates of dopamine D3 receptor activation in the rat in vivo and their modulation by the selective antagonist, (+)-S 14297: 1. Activation of postsynaptic D3 receptors mediates hypothermia, whereas blockade of D2 receptors elicits prolactin
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:2

    Topics: 2-Naphthylamine; Animals; Body Temperature Regulation; Catalepsy; CHO Cells; Cricetinae; Dopamine Antagonists; Furans; Humans; Male; Prolactin; Rats; Rats, Wistar; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins; Stereoisomerism

1995
Synthesis and dopaminergic properties of benzo-fused analogues of quinpirole and quinelorane.
    Journal of medicinal chemistry, 1999, Mar-11, Volume: 42, Issue:5

    Topics: Animals; Binding, Competitive; Dopamine Agonists; In Vitro Techniques; Isoquinolines; Male; Naphthols; Neostriatum; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Structure-Activity Relationship

1999
CoMFA and CoMSIA investigations revealing novel insights into the binding modes of dopamine D3 receptor agonists.
    Journal of medicinal chemistry, 2005, Apr-07, Volume: 48, Issue:7

    Topics: Animals; Binding Sites; Cattle; CHO Cells; Corpus Striatum; Cricetinae; Cricetulus; Humans; Indolizines; Models, Molecular; Molecular Conformation; Quantitative Structure-Activity Relationship; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Stereoisomerism

2005
Effect of D2 dopamine agonists on tuberoinfundibular dopamine neurons.
    Neuropharmacology, 1991, Volume: 30, Issue:9

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Arcuate Nucleus of Hypothalamus; Benzazepines; Chromatography, High Pressure Liquid; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Ergolines; Haloperidol; Male; Neurons; Quinolines; Quinpirole; Rats; Rats, Inbred Strains

1991
Effects of selective D1 and D2 dopamine agonists on cockroach salivary gland acinar cells in vitro.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Cockroaches; Dopamine Agents; Electrophysiology; Ergolines; Fenoldopam; In Vitro Techniques; Membrane Potentials; Quinolines; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Salivary Glands; Sulpiride

1991
Effect of direct and indirect dopamine agonists on brain extracellular ascorbate levels in the striatum and nucleus accumbens of awake rats.
    Life sciences, 1990, Volume: 47, Issue:15

    Topics: Animals; Ascorbic Acid; Corpus Striatum; Dextroamphetamine; Dopamine Agents; Ergolines; Extracellular Space; Male; Nucleus Accumbens; Phenethylamines; Quinolines; Quinpirole; Rats; Rats, Inbred Strains

1990
Preclinical studies on quinelorane, a potent and highly selective D2-dopaminergic agonist.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: Acetylcholine; Animals; Biogenic Amines; Brain; Corticosterone; Dopamine; Dose-Response Relationship, Drug; Emetics; Ergolines; Male; Motor Activity; Pergolide; Prolactin; Quinolines; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Reference Values; Stereotyped Behavior

1989
Further characterization of tolerance to the corticosterone-elevating effect of pergolide in rats.
    Neuroscience letters, 1988, Nov-11, Volume: 93, Issue:2-3

    Topics: Animals; Corticosterone; Dopamine; Dopamine Agents; Ergolines; Male; Oxazines; Pergolide; Pharmaceutical Vehicles; Quinolines; Quinpirole; Rats; Rats, Inbred Strains

1988
Dopamine receptor agonist potencies for inhibition of cell firing correlate with dopamine D3 receptor binding affinities.
    European journal of pharmacology, 1995, Apr-24, Volume: 277, Issue:2-3

    Topics: Aminoquinolines; Animals; Apomorphine; Azepines; Benzothiazoles; Binding, Competitive; CHO Cells; Cricetinae; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Imidazoles; Male; Neurons; Phenethylamines; Piperidines; Pramipexole; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3; Structure-Activity Relationship; Substantia Nigra; Tetrahydronaphthalenes; Thiazoles; Thiophenes; Transfection

1995
Effect of haloperidol and (-)-sulpiride on dopamine agonist-induced hypoactivity.
    Neuropharmacology, 1995, Volume: 34, Issue:4

    Topics: Animals; Apomorphine; Benzopyrans; Dopamine Agonists; Dose-Response Relationship, Drug; Ergolines; Haloperidol; Male; Motor Activity; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Sulpiride; Tetrahydronaphthalenes

1995
Prolonged central effects of quinpirole on cardiovascular regulation.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 277, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzazepines; Blood Pressure; Brain; Clonidine; Dopamine Agonists; Ergolines; Heart Rate; Male; Quinolines; Quinpirole; Raclopride; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley; Salicylamides; Species Specificity

1996
Elucidation of D3 receptor function in vivo: do D3 receptors mediate inhibition of dopamine neuronal activity?
    Biochemical Society transactions, 1996, Volume: 24, Issue:1

    Topics: Animals; Apomorphine; Corpus Striatum; Dopamine; Dopamine Agonists; Ergolines; Male; Mice; Mice, Inbred Strains; Microdialysis; Neurons; Nucleus Accumbens; Oxazines; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes

1996
The effects of dopamine D3/D2 receptor agonists on intracranial self stimulation in the rat.
    Psychopharmacology, 1998, Volume: 140, Issue:4

    Topics: Animals; Area Under Curve; Brain; Dopamine Agonists; Injections, Subcutaneous; Male; Quinolines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Stimulation; Tetrahydronaphthalenes

1998
The modulatory actions of dopamine D2/3 agonists and antagonists on the locomotor-activating effects of morphine and caffeine in mice.
    Pharmacology, biochemistry, and behavior, 2003, Volume: 75, Issue:2

    Topics: Animals; Caffeine; Central Nervous System Stimulants; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Mice; Morphine; Motor Activity; Naphthalenes; Narcotic Antagonists; Narcotics; Pyrrolidines; Quinolines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Salicylamides; Water

2003
Gradient of dopamine responsiveness to dopamine receptor agonists in subregions of the rat nucleus accumbens.
    European journal of pharmacology, 2003, Sep-12, Volume: 477, Issue:2

    Topics: Animals; Apomorphine; Chromatography, High Pressure Liquid; Dopamine; Dose-Response Relationship, Drug; Male; Microdialysis; Nucleus Accumbens; Quinolines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Tetrahydronaphthalenes; Time Factors

2003
Modulation of the locomotor activating effects of the noncompetitive NMDA receptor antagonist MK801 by dopamine D2/3 receptor agonists in mice.
    Pharmacology, biochemistry, and behavior, 2004, Volume: 77, Issue:2

    Topics: Animals; Dizocilpine Maleate; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Mice; Motor Activity; Naphthalenes; Piperazines; Pyrrolidines; Quinolines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, N-Methyl-D-Aspartate; Salicylamides; Stereotyped Behavior

2004
Modulation of the discriminative stimulus effects of mu opioid agonists in rats: II. Effects of dopamine D2/3 agonists.
    Behavioural pharmacology, 2004, Volume: 15, Issue:1

    Topics: Animals; Appetitive Behavior; Brain; Discrimination Learning; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Heroin; Male; Methadone; Morphine; Motivation; Nalbuphine; Quinolines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, mu; Tetrahydronaphthalenes

2004
D2-like receptors in nucleus accumbens negatively modulate acetylcholine release in prefrontal cortex.
    Neuropharmacology, 2007, Volume: 53, Issue:3

    Topics: Acetylcholine; Analysis of Variance; Animals; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Male; Microdialysis; N-Methylaspartate; Nucleus Accumbens; Prefrontal Cortex; Quinolines; Quinpirole; Rats; Rats, Inbred F344; Receptors, Dopamine D2

2007