Page last updated: 2024-08-21

quinazolines and rucaparib

quinazolines has been researched along with rucaparib in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aherne, W; Anderson, VE; Antoni, L; Boxall, KJ; Caldwell, JJ; Collins, I; Eve, PD; Garrett, MD; Oliver, AW; Pearl, LH; Walton, MI1
Beijnen, JH; Durmus, S; Schellens, JH; Schinkel, AH; Sparidans, RW1
Cupo, M; Mauritz, M; Mitulovic, G; Węsierska-Gądek, J1
Bierbach, U; Ding, S1
Gunn, AR; Kolb, AL; Lakin, ND1

Other Studies

5 other study(ies) available for quinazolines and rucaparib

ArticleYear
CCT241533 is a potent and selective inhibitor of CHK2 that potentiates the cytotoxicity of PARP inhibitors.
    Cancer research, 2011, Jan-15, Volume: 71, Issue:2

    Topics: Antineoplastic Combined Chemotherapy Protocols; Bleomycin; Cell Cycle; Cell Line, Tumor; Checkpoint Kinase 2; Crystallography, X-Ray; Drug Synergism; Enzyme Activation; HCT116 Cells; HeLa Cells; Heterocyclic Compounds, 3-Ring; HT29 Cells; Humans; Models, Molecular; Poly(ADP-ribose) Polymerase Inhibitors; Protein Serine-Threonine Kinases; Quinazolines

2011
Liquid chromatography-tandem mass spectrometric assay for the PARP inhibitor rucaparib in plasma.
    Journal of pharmaceutical and biomedical analysis, 2014, Volume: 88

    Topics: Acetonitriles; Animals; Area Under Curve; Calibration; Chromatography, Liquid; Edetic Acid; Female; Gefitinib; Indoles; Mice; Poly(ADP-ribose) Polymerase Inhibitors; Protein Kinase Inhibitors; Quality Control; Quinazolines; Reproducibility of Results; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry

2014
Differential Potential of Pharmacological PARP Inhibitors for Inhibiting Cell Proliferation and Inducing Apoptosis in Human Breast Cancer Cells.
    Journal of cellular biochemistry, 2015, Volume: 116, Issue:12

    Topics: Apoptosis; Benzamides; BRCA1 Protein; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Female; Gene Expression Regulation, Neoplastic; Humans; Indoles; Phthalazines; Piperazines; Piperidines; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Quinazolines

2015
Linker design for the modular assembly of multifunctional and targeted platinum(ii)-containing anticancer agents.
    Dalton transactions (Cambridge, England : 2003), 2016, Aug-16, Volume: 45, Issue:33

    Topics: Acridines; Amines; Antineoplastic Agents; Dendrimers; Indoles; Organophosphorus Compounds; Platinum; Quinazolines; Tamoxifen

2016
Redundancy between nucleases required for homologous recombination promotes PARP inhibitor resistance in the eukaryotic model organism Dictyostelium.
    Nucleic acids research, 2017, Sep-29, Volume: 45, Issue:17

    Topics: ADP Ribose Transferases; Benzamides; Clone Cells; Cyclin-Dependent Kinase 8; Dictyostelium; DNA Damage; Drug Resistance; Exodeoxyribonucleases; Gene Deletion; Homologous Recombination; Indoles; Phthalazines; Piperazines; Poly(ADP-ribose) Polymerase Inhibitors; Poly(ADP-ribose) Polymerases; Protozoan Proteins; Quinazolines; Rad51 Recombinase; Recombinant Proteins

2017