quinazolines has been researched along with quinoline in 11 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (9.09) | 29.6817 |
2010's | 6 (54.55) | 24.3611 |
2020's | 4 (36.36) | 2.80 |
Authors | Studies |
---|---|
Chen, Y; Hano, Y; Ma, Z; Nomura, T | 1 |
Cao, R; Mi, N; Zhang, H | 1 |
Nevalainen, T; Saari, R; Törmä, JC | 1 |
Bak-Sypien, II; Dominska, K; Galdyszynska, M; Karwowski, BT; Merecz-Sadowska, A; Piastowska-Ciesielska, AW; Stanczak, A; Szumilak, M | 1 |
Arrowsmith, CH; Babault, N; Brown, PJ; Chen, X; Dong, A; Jin, J; Li, F; Liu, J; Vedadi, M; Wu, H; Xiong, Y; Zeng, H | 1 |
Goto, M; Guo, X; Lee, KH; Li, JC; Liu, YQ; Morris-Natschke, SL; Shang, XF; Xu, XS; Yang, GZ | 1 |
Goto, M; Guo, X; Lee, KH; Li, JC; Liu, YQ; Morris-Natschke, SL; Shang, XF; Xu, XS; Yang, GZ; Zhang, JY | 1 |
Esmaeili, S; Fassihi, A; Fayyazi, N; Ghasemi, JB; Saghaie, L; Taheri, S | 1 |
Charles, MRC; Coumar, MS; Dhayalan, A; Hsieh, HP; Lin, SY; Mahesh, A | 1 |
Damodar, K; Gim, JG; Jeon, SH; Lee, JT; Lee, Y; Nam, KY; Park, JP; Park, LS | 1 |
Astolfi, A; Barreca, ML; Biavasco, F; Cannalire, R; Cecchetti, V; Cedraro, N; Cernicchi, G; Felicetti, T; Manfroni, G; Mangiaterra, G; Massari, S; Sabatini, S; Tabarrini, O; Vaiasicca, S | 1 |
2 review(s) available for quinazolines and quinoline
Article | Year |
---|---|
Biologically active quinoline and quinazoline alkaloids part I.
Topics: Alkaloids; Animals; Humans; Immunologic Factors; Protective Agents; Quinazolines; Quinolines | 2018 |
Biologically active quinoline and quinazoline alkaloids part II.
Topics: Alkaloids; Anti-Inflammatory Agents; Antioxidants; Humans; Protective Agents; Quinazolines; Quinolines | 2018 |
9 other study(ies) available for quinazolines and quinoline
Article | Year |
---|---|
Novel quinazoline-quinoline alkaloids with cytotoxic and DNA topoisomerase II inhibitory activities.
Topics: Alkaloids; Animals; Cell Line, Tumor; DNA Topoisomerases, Type II; Enzyme Inhibitors; Mice; Quinazolines; Quinolines; Topoisomerase II Inhibitors | 2004 |
3D-QSAR study of c-Src kinase inhibitors based on docking.
Topics: Antineoplastic Agents; Computer Simulation; CSK Tyrosine-Protein Kinase; Humans; Nitriles; Protein Binding; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Quantitative Structure-Activity Relationship; Quinazolines; Quinolines; src-Family Kinases | 2010 |
Microwave-assisted synthesis of quinoline, isoquinoline, quinoxaline and quinazoline derivatives as CB2 receptor agonists.
Topics: Isoquinolines; Microwaves; Morpholines; Quinazolines; Quinolines; Quinoxalines; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Structure-Activity Relationship | 2011 |
Synthesis, Biological Activity and Preliminary in Silico ADMET Screening of Polyamine Conjugates with Bicyclic Systems.
Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Cell Survival; DNA; DNA Topoisomerases, Type I; Drug Design; Escherichia coli; Humans; Indoles; Naphthalenes; Nucleic Acid Conformation; Polyamines; Quinazolines; Quinolines; Rats; Structure-Activity Relationship | 2017 |
Structure-activity relationship studies of G9a-like protein (GLP) inhibitors.
Topics: Crystallography, X-Ray; Dose-Response Relationship, Drug; Enzyme Inhibitors; Histone-Lysine N-Methyltransferase; Humans; Models, Molecular; Molecular Structure; Quinazolines; Quinolines; Structure-Activity Relationship | 2017 |
Molecular dynamics simulation and 3D-pharmacophore analysis of new quinoline-based analogues with dual potential against EGFR and VEGFR-2.
Topics: A549 Cells; Aminoquinolines; Antineoplastic Agents; Binding Sites; Cell Line, Tumor; ErbB Receptors; Erlotinib Hydrochloride; Humans; Molecular Docking Simulation; Molecular Dynamics Simulation; Piperidines; Protein Conformation; Quinazolines; Quinolines; Sorafenib; Vascular Endothelial Growth Factor Receptor-2 | 2020 |
Identification of novel quinoline inhibitor for EHMT2/G9a through virtual screening.
Topics: Azepines; Catalytic Domain; Databases, Chemical; Enzyme Inhibitors; HEK293 Cells; Histocompatibility Antigens; Histone-Lysine N-Methyltransferase; Histones; Humans; Methylation; Protein Binding; Quinazolines; Quinolines | 2020 |
Design and Synthesis of π-Extended Resveratrol Analogues and In Vitro Antioxidant and Anti-Inflammatory Activity Evaluation.
Topics: Animals; Anti-Inflammatory Agents; Antioxidants; Cell Survival; Gene Expression Regulation; Interleukin-1beta; Interleukin-6; Isoquinolines; Lipopolysaccharides; Mice; Naphthalenes; Quinazolines; Quinolines; Quinoxalines; RAW 264.7 Cells; Resveratrol; Stilbestrols; Structure-Activity Relationship | 2021 |
From Quinoline to Quinazoline-Based S. aureus NorA Efflux Pump Inhibitors by Coupling a Focused Scaffold Hopping Approach and a Pharmacophore Search.
Topics: Anti-Bacterial Agents; Bacterial Proteins; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Molecular Structure; Multidrug Resistance-Associated Proteins; Quinazolines; Quinolines; Structure-Activity Relationship | 2021 |