Page last updated: 2024-08-21

quinazolines and pyrazole

quinazolines has been researched along with pyrazole in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (57.14)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abdel-Gawad, SM; El-Gaby, MS; Ghorab, MM1
Catarzi, D; Colotta, V; Costagli, C; Filacchioni, G; Galli, A; Lenzi, O; Varano, F1
McLaughlin, ML; Talele, TT1
Beijnen, JH; Pluim, D; Schellens, JH; van Tellingen, O1
Gangarajula, S; Ghosh, AK; Huang, X; Kulkarni, S; Pandey, S; Rao, KV; Tang, J; Xu, X1
Li, QS; Sun, S; Tang, JF; Wang, XL; Yang, YS; Zhang, F; Zhang, YB; Zhu, HL1
Hu, C; Hu, J; Jin, Z; Ke, J; Lu, Q; Sun, R; Wan, DC; Wang, X; Zhan, X1

Other Studies

7 other study(ies) available for quinazolines and pyrazole

ArticleYear
Synthesis and antifungal activity of novel pyrano[2',3':4,5]thiazolo[2,3-b]quinazolines, pyrido[2',3':4,5]thiazolo[2,3-b]quinazolines and pyrazolo[2',3':4,5]thiazolo[2,3-b]quinazolines.
    Farmaco (Societa chimica italiana : 1989), 2000, Volume: 55, Issue:4

    Topics: Antifungal Agents; Aspergillus flavus; Aspergillus ochraceus; Candida albicans; Microbial Sensitivity Tests; Molecular Structure; Penicillium chrysogenum; Pyrans; Pyrazoles; Pyridines; Quinazolines; Thiazoles

2000
Novel AMPA and kainate receptor antagonists containing the pyrazolo[1,5-c]quinazoline ring system: Synthesis and structure-activity relationships.
    Bioorganic & medicinal chemistry, 2008, Mar-01, Volume: 16, Issue:5

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Molecular Structure; N-Methylaspartate; Pyrazoles; Quinazolines; Receptors, Kainic Acid; Structure-Activity Relationship

2008
Molecular docking/dynamics studies of Aurora A kinase inhibitors.
    Journal of molecular graphics & modelling, 2008, Volume: 26, Issue:8

    Topics: Aurora Kinases; Binding Sites; Computer Simulation; Hydrogen Bonding; Indoles; Inhibitory Concentration 50; Models, Molecular; Molecular Conformation; Molecular Structure; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrazoles; Pyrimidines; Quinazolines; Structure-Activity Relationship; Sulfonamides

2008
Simultaneous determination of AZD1152 (prodrug) and AZD1152-hydroxyquinazoline pyrazol anilide by reversed phase liquid chromatography.
    Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2009, Nov-01, Volume: 877, Issue:29

    Topics: Animals; Chromatography, High Pressure Liquid; Humans; Hydroxyquinolines; Mice; Molecular Structure; Organophosphates; Pyrazoles; Quinazolines; Reproducibility of Results

2009
Structure-based design, synthesis, and biological evaluation of dihydroquinazoline-derived potent β-secretase inhibitors.
    Bioorganic & medicinal chemistry letters, 2012, Sep-01, Volume: 22, Issue:17

    Topics: Alzheimer Disease; Amyloid Precursor Protein Secretases; Catalytic Domain; Cell Line, Tumor; Crystallography, X-Ray; Drug Design; Enzyme Inhibitors; Humans; Models, Molecular; Pyrazoles; Quinazolines; Structure-Activity Relationship; Thiazoles

2012
Design, modification and 3D QSAR studies of novel 2,3-dihydrobenzo[b][1,4]dioxin-containing 4,5-dihydro-1H-pyrazole derivatives as inhibitors of B-Raf kinase.
    Bioorganic & medicinal chemistry, 2012, Oct-15, Volume: 20, Issue:20

    Topics: Binding Sites; Cell Line, Tumor; Cell Proliferation; Dioxanes; Dioxins; Drug Design; Erlotinib Hydrochloride; Humans; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins B-raf; Pyrazoles; Quantitative Structure-Activity Relationship; Quinazolines; Thermodynamics

2012
Discovery of 4,5-Dihydro-1
    Molecules (Basel, Switzerland), 2018, Aug-08, Volume: 23, Issue:8

    Topics: A549 Cells; ErbB Receptors; Gefitinib; Hep G2 Cells; Humans; Inhibitory Concentration 50; Molecular Docking Simulation; Protein Kinase Inhibitors; Pyrazoles; Quinazolines

2018