Page last updated: 2024-08-21

quinazolines and mln8054

quinazolines has been researched along with mln8054 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bastians, H; Kaestner, P; Stolz, A1
Deng, X; Gray, N; Huang, HC; Kwiatkowski, N; Mitchison, T; Musacchio, A; Santaguida, S; Tan, L; Villa, F; Wang, J1
Bartsch, DK; Doll, D; Greene, BH; Hoffmann, S; Khoruzhyk, M; Ramaswamy, A; Roth, S; Wunderlich, A1
Aguiar, P; Barisic, M; Geley, S; Maiato, H1
Bastida, CC; Falchook, GS; Kurzrock, R1

Reviews

1 review(s) available for quinazolines and mln8054

ArticleYear
Aurora Kinase Inhibitors in Oncology Clinical Trials: Current State of the Progress.
    Seminars in oncology, 2015, Volume: 42, Issue:6

    Topics: Antineoplastic Agents; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; Benzamides; Benzazepines; Benzimidazoles; Clinical Trials as Topic; Heterocyclic Compounds, 3-Ring; Humans; Molecular Targeted Therapy; Neoplasms; Norbornanes; Organophosphates; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Quinazolines; Urea

2015

Other Studies

4 other study(ies) available for quinazolines and mln8054

ArticleYear
Determinants for the efficiency of anticancer drugs targeting either Aurora-A or Aurora-B kinases in human colon carcinoma cells.
    Molecular cancer therapeutics, 2009, Volume: 8, Issue:7

    Topics: Animals; Apoptosis; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; bcl-2-Associated X Protein; Benzamides; Benzazepines; Blotting, Western; Colonic Neoplasms; Cyclin-Dependent Kinase Inhibitor p21; Drug Synergism; Flow Cytometry; Humans; Mice; Mice, Knockout; Mitosis; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-mdm2; Quinazolines; Spindle Apparatus; Tumor Cells, Cultured; Tumor Suppressor Protein p53

2009
Selective aurora kinase inhibitors identified using a taxol-induced checkpoint sensitivity screen.
    ACS chemical biology, 2012, Jan-20, Volume: 7, Issue:1

    Topics: Animals; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Aurora Kinase B; Aurora Kinases; Benzazepines; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; High-Throughput Screening Assays; Humans; Inhibitory Concentration 50; Isoenzymes; M Phase Cell Cycle Checkpoints; Models, Molecular; Organophosphates; Paclitaxel; Piperazines; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrimidines; Quinazolines; Structure-Activity Relationship; Xenopus laevis

2012
Pretherapeutic drug evaluation by tumor xenografting in anaplastic thyroid cancer.
    The Journal of surgical research, 2013, Volume: 185, Issue:2

    Topics: Animals; Apoptosis; Benzazepines; Cell Proliferation; Drug Evaluation, Preclinical; Humans; Male; Mice; Mice, Nude; Middle Aged; Neovascularization, Pathologic; Niacinamide; Phenylurea Compounds; Piperidines; Protein Kinase Inhibitors; Quinazolines; Random Allocation; Receptors, Vascular Endothelial Growth Factor; Sorafenib; Thyroid Carcinoma, Anaplastic; Thyroid Neoplasms; Treatment Outcome; Xenograft Model Antitumor Assays

2013
Kinetochore motors drive congression of peripheral polar chromosomes by overcoming random arm-ejection forces.
    Nature cell biology, 2014, Volume: 16, Issue:12

    Topics: Aurora Kinase A; Aurora Kinase B; Benzamides; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cell Division; Cell Line, Tumor; Chromosomal Proteins, Non-Histone; Chromosome Segregation; Cytoplasmic Dyneins; DNA-Binding Proteins; Dyneins; Humans; Kinesins; Kinetochores; Microtubules; Quinazolines; RNA Interference; RNA, Small Interfering; Sarcosine; Spindle Apparatus

2014