quinazolines has been researched along with mln8054 in 5 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (20.00) | 29.6817 |
2010's | 4 (80.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bastians, H; Kaestner, P; Stolz, A | 1 |
Deng, X; Gray, N; Huang, HC; Kwiatkowski, N; Mitchison, T; Musacchio, A; Santaguida, S; Tan, L; Villa, F; Wang, J | 1 |
Bartsch, DK; Doll, D; Greene, BH; Hoffmann, S; Khoruzhyk, M; Ramaswamy, A; Roth, S; Wunderlich, A | 1 |
Aguiar, P; Barisic, M; Geley, S; Maiato, H | 1 |
Bastida, CC; Falchook, GS; Kurzrock, R | 1 |
1 review(s) available for quinazolines and mln8054
Article | Year |
---|---|
Aurora Kinase Inhibitors in Oncology Clinical Trials: Current State of the Progress.
Topics: Antineoplastic Agents; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; Benzamides; Benzazepines; Benzimidazoles; Clinical Trials as Topic; Heterocyclic Compounds, 3-Ring; Humans; Molecular Targeted Therapy; Neoplasms; Norbornanes; Organophosphates; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Quinazolines; Urea | 2015 |
4 other study(ies) available for quinazolines and mln8054
Article | Year |
---|---|
Determinants for the efficiency of anticancer drugs targeting either Aurora-A or Aurora-B kinases in human colon carcinoma cells.
Topics: Animals; Apoptosis; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; bcl-2-Associated X Protein; Benzamides; Benzazepines; Blotting, Western; Colonic Neoplasms; Cyclin-Dependent Kinase Inhibitor p21; Drug Synergism; Flow Cytometry; Humans; Mice; Mice, Knockout; Mitosis; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-mdm2; Quinazolines; Spindle Apparatus; Tumor Cells, Cultured; Tumor Suppressor Protein p53 | 2009 |
Selective aurora kinase inhibitors identified using a taxol-induced checkpoint sensitivity screen.
Topics: Animals; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Aurora Kinase B; Aurora Kinases; Benzazepines; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; High-Throughput Screening Assays; Humans; Inhibitory Concentration 50; Isoenzymes; M Phase Cell Cycle Checkpoints; Models, Molecular; Organophosphates; Paclitaxel; Piperazines; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrimidines; Quinazolines; Structure-Activity Relationship; Xenopus laevis | 2012 |
Pretherapeutic drug evaluation by tumor xenografting in anaplastic thyroid cancer.
Topics: Animals; Apoptosis; Benzazepines; Cell Proliferation; Drug Evaluation, Preclinical; Humans; Male; Mice; Mice, Nude; Middle Aged; Neovascularization, Pathologic; Niacinamide; Phenylurea Compounds; Piperidines; Protein Kinase Inhibitors; Quinazolines; Random Allocation; Receptors, Vascular Endothelial Growth Factor; Sorafenib; Thyroid Carcinoma, Anaplastic; Thyroid Neoplasms; Treatment Outcome; Xenograft Model Antitumor Assays | 2013 |
Kinetochore motors drive congression of peripheral polar chromosomes by overcoming random arm-ejection forces.
Topics: Aurora Kinase A; Aurora Kinase B; Benzamides; Benzazepines; Bridged Bicyclo Compounds, Heterocyclic; Cell Division; Cell Line, Tumor; Chromosomal Proteins, Non-Histone; Chromosome Segregation; Cytoplasmic Dyneins; DNA-Binding Proteins; Dyneins; Humans; Kinesins; Kinetochores; Microtubules; Quinazolines; RNA Interference; RNA, Small Interfering; Sarcosine; Spindle Apparatus | 2014 |