Page last updated: 2024-08-21

quinazolines and lfm a13

quinazolines has been researched along with lfm a13 in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (75.00)29.6817
2010's0 (0.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Ghosh, S; Liu, XP; Myers, DE; Sudbeck, EA; Uckun, FM; Zheng, Y1
Bartell, S; Mahajan, S; Tibbles, HE; Uckun, FM; Vassilev, A; Zheng, Y1
Cetkovic-Cvrlje, M; Uckun, FM1
Güven, DC; Orhan, C; Şahin, K; Uçkun, FM1

Reviews

2 review(s) available for quinazolines and lfm a13

ArticleYear
Tyrosine kinase inhibitors against EGF receptor-positive malignancies.
    Methods in molecular biology (Clifton, N.J.), 2001, Volume: 166

    Topics: Adenocarcinoma; Amides; Aniline Compounds; Animals; Antineoplastic Agents; Breast Neoplasms; Drug Design; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; Female; Genistein; Humans; Leukemia; Macaca fascicularis; Mice; Mice, Inbred BALB C; Mice, SCID; Models, Molecular; Molecular Structure; Neoplasm Proteins; Neoplasms; Nitriles; Protein Conformation; Protein Structure, Tertiary; Quinazolines; Recombinant Fusion Proteins; Sequence Alignment; Species Specificity; Structure-Activity Relationship; Tumor Cells, Cultured; Tumor Stem Cell Assay; Xenograft Model Antitumor Assays

2001
Data-Driven identification of chemopreventive agents for breast cancer
    Turkish journal of medical sciences, 2020, 11-03, Volume: 50, Issue:SI-2

    Topics: Amides; Animals; Antineoplastic Agents; Breast Neoplasms; Chemoprevention; Female; Humans; Mammary Neoplasms, Experimental; Mice; Nitriles; Protein Kinase Inhibitors; Quinazolines

2020

Other Studies

2 other study(ies) available for quinazolines and lfm a13

ArticleYear
The anti-leukemic Bruton's tyrosine kinase inhibitor alpha-cyano-beta-hydroxy-beta-methyl-N-(2,5-dibromophenyl) propenamide (LFM-A13) prevents fatal thromboembolism.
    Leukemia & lymphoma, 2003, Volume: 44, Issue:9

    Topics: Adenosine Diphosphate; Agammaglobulinaemia Tyrosine Kinase; Amides; Animals; Aspirin; Bleeding Time; Catalytic Domain; Collagen; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Fibrinolytic Agents; Humans; Janus Kinase 3; Male; Mice; Mice, Inbred ICR; Nitriles; Peptide Fragments; Platelet Activation; Platelet Aggregation; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Protein-Tyrosine Kinases; Pulmonary Embolism; Quinazolines; Receptors, Collagen; Signal Transduction; Thrombin; Thromboembolism; Thromboplastin

2003
Dual targeting of Bruton's tyrosine kinase and Janus kinase 3 with rationally designed inhibitors prevents graft-versus-host disease (GVHD) in a murine allogeneic bone marrow transplantation model.
    British journal of haematology, 2004, Volume: 126, Issue:6

    Topics: Acute Disease; Agammaglobulinaemia Tyrosine Kinase; Amides; Animals; Bone Marrow Transplantation; Drug Therapy, Combination; Enzyme Inhibitors; Graft vs Host Disease; Immunosuppressive Agents; Janus Kinase 3; Male; Methotrexate; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Nitriles; Protein-Tyrosine Kinases; Quinazolines; Survival Rate; Treatment Outcome

2004