Page last updated: 2024-08-21

quinazolines and importazole

quinazolines has been researched along with importazole in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's16 (76.19)24.3611
2020's5 (23.81)2.80

Authors

AuthorsStudies
Bird, SL; Hasegawa, K; Heald, R; Kalab, P; Sampathkumar, Y; Soderholm, JF; Uehara-Bingen, M; Weis, K1
Du, J; Hou, J; Jiang, H; Yan, WQ1
Bird, SL; Heald, R; Weis, K1
Bai, L; Michael, WM; Yan, S1
Brehm, MA; Ehm, P; Kublun, I; Nalaskowski, MM1
Du, J; He, J; Hou, J; Li, R; Yan, W1
Allison, LA; Bondzi, C; Doshi, Y; Dziedzic, RC; McGregor, EL; Parente, LE; Roggero, VR; Schad, SE; Varjabedian, AD; Zhang, J1
Hofmann, WA; Maly, IV1
Bagattin, A; Felix, T; Garbay, S; Heidet, L; Lerner, J; Makinistoglu, MP; Pontoglio, M; Verdeguer, F1
Au, S; Panté, N; Theilmann, DA; Wu, W; Zhou, L1
Noy, N; Vreeland, AC; Zhang, W1
Chao, CY; Chen, WS; Chen, YJ; Chiu, HC; Hsieh, BY; Huang, YA; Hwang, E; Kao, PY1
Bao, L; Cao, Q; Chen, K; Huang, X; Li, X; Liu, L; Lou, N; Qiu, B; Ruan, H; Wang, K; Xiao, W; Xu, G; Yang, H; Yuan, C; Zhang, X1
Asashima, H; Hirota, T; Kondo, Y; Matsumoto, I; Moriyama, M; Nakamura, S; Sumida, T; Takahashi, H; Tsuboi, H1
Chigwechokha, PK; Honda, A; Kamada-Futagami, Y; Komatsu, M; Shiozaki, K1
Chu, CH; Guo, Y; Li, X; Lu, C; Luo, L; Obbad, S; Wang, KJ; Wang, Y; Yan, W; Yang, J; Zhang, R; Zhang, Y1
Mayol, GF; Revuelta, MV; Rópolo, AS; Salusso, A; Touz, MC1
Butler-Browne, G; Coirault, C; Fischer, M; Jabre, S; Mamchaoui, K; Moog, S; Owens, DJ1
Agostini, S; Barbarino, M; Barone, E; Bottaro, M; Catalano, C; Cipollini, M; Corrado, A; Dell'Anno, I; Gemignani, F; Giordano, A; Landi, S; Luzzi, L; Melaiu, O; Melani, A; Migliore, L; Silvestri, R1
Ishikawa, C; Mori, N; Senba, M1
Nakano, M; Sato, Y; Yoshino, H1

Other Studies

21 other study(ies) available for quinazolines and importazole

ArticleYear
Importazole, a small molecule inhibitor of the transport receptor importin-β.
    ACS chemical biology, 2011, Jul-15, Volume: 6, Issue:7

    Topics: Active Transport, Cell Nucleus; Animals; beta Karyopherins; Cell Extracts; Exportin 1 Protein; Female; Fluorescence Resonance Energy Transfer; GTPase-Activating Proteins; HeLa Cells; High-Throughput Screening Assays; Humans; Karyopherins; Mitosis; NFATC Transcription Factors; Ovum; Quinazolines; ran GTP-Binding Protein; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Spindle Apparatus; Xenopus

2011
[Effect of nuclear receptor inhibitor importazole on the proliferation and apoptosis of multiple myeloma cells].
    Zhonghua xue ye xue za zhi = Zhonghua xueyexue zazhi, 2013, Volume: 34, Issue:4

    Topics: Apoptosis; Cell Line, Tumor; Cell Proliferation; Humans; Multiple Myeloma; NF-kappa B; Quinazolines; Signal Transduction

2013
RanGTP and CLASP1 cooperate to position the mitotic spindle.
    Molecular biology of the cell, 2013, Volume: 24, Issue:16

    Topics: Active Transport, Cell Nucleus; beta Karyopherins; Cell Division; Cell Line, Tumor; Cytoplasmic Dyneins; Dyneins; HeLa Cells; Humans; Intracellular Signaling Peptides and Proteins; Microtubule-Associated Proteins; Microtubules; Mitosis; Nocodazole; Nuclear Matrix-Associated Proteins; Quinazolines; ran GTP-Binding Protein; Spindle Apparatus; Tubulin Modulators

2013
Importin β-dependent nuclear import of TopBP1 in ATR-Chk1 checkpoint in Xenopus egg extracts.
    Cellular signalling, 2014, Volume: 26, Issue:5

    Topics: Active Transport, Cell Nucleus; Amino Acid Motifs; Amino Acid Sequence; Animals; Ataxia Telangiectasia Mutated Proteins; beta Karyopherins; Carrier Proteins; Cell Nucleus; Checkpoint Kinase 1; DNA Repair; DNA-Binding Proteins; Mitomycin; Molecular Sequence Data; Ovum; Phosphorylation; Protein Kinases; Protein Structure, Secondary; Protein Structure, Tertiary; Quinazolines; Signal Transduction; Xenopus laevis; Xenopus Proteins

2014
Efficacious inhibition of Importin α/β-mediated nuclear import of human inositol phosphate multikinase.
    Biochimie, 2014, Volume: 102

    Topics: Active Transport, Cell Nucleus; Cell Nucleus; HeLa Cells; Humans; Hydrogen Peroxide; Inositol Phosphates; Karyopherins; Quinazolines; Signal Transduction

2014
Importin β1 mediates nuclear factor-κB signal transduction into the nuclei of myeloma cells and affects their proliferation and apoptosis.
    Cellular signalling, 2015, Volume: 27, Issue:4

    Topics: Active Transport, Cell Nucleus; Apoptosis; beta Karyopherins; Cell Line, Tumor; Cell Nucleus; Cell Proliferation; Humans; Multiple Myeloma; NF-kappa B; Quinazolines; RNA, Small Interfering; Signal Transduction; Transcription Factor RelA

2015
Nuclear import of the thyroid hormone receptor α1 is mediated by importin 7, importin β1, and adaptor importin α1.
    Molecular and cellular endocrinology, 2016, Jan-05, Volume: 419

    Topics: alpha Karyopherins; beta Karyopherins; Cell Nucleus; HeLa Cells; Humans; Karyopherins; Protein Transport; Quinazolines; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Temperature; Thyroid Hormone Receptors alpha

2016
Calcium-regulated import of myosin IC into the nucleus.
    Cytoskeleton (Hoboken, N.J.), 2016, Volume: 73, Issue:7

    Topics: beta Karyopherins; Calcium Signaling; Cell Line, Tumor; Cell Nucleus; Cytoplasm; Humans; Isoenzymes; Myosin Type I; Quinazolines

2016
Human mutations affect the epigenetic/bookmarking function of HNF1B.
    Nucleic acids research, 2016, 09-30, Volume: 44, Issue:17

    Topics: Animals; Cells, Cultured; Chromatin; Diabetes Mellitus, Type 2; DNA; Dogs; Epigenesis, Genetic; Epithelial Cells; Gene Deletion; Green Fluorescent Proteins; Hepatocyte Nuclear Factor 1-beta; Heterozygote; Humans; Kidney; Madin Darby Canine Kidney Cells; Mitosis; Models, Biological; Mutation; Protein Binding; Protein Domains; Quinazolines; Recombinant Fusion Proteins; Temperature

2016
A new mechanism for nuclear import by actin-based propulsion used by a baculovirus nucleocapsid.
    Journal of cell science, 2016, 08-01, Volume: 129, Issue:15

    Topics: Actin-Related Protein 2-3 Complex; Actins; Active Transport, Cell Nucleus; Baculoviridae; Cell Membrane Permeability; Cell Nucleus; Cytosol; Digitonin; Guanosine 5'-O-(3-Thiotriphosphate); HeLa Cells; Humans; Nuclear Pore; Nucleocapsid; Nucleopolyhedroviruses; Polymerization; Quinazolines; ran GTP-Binding Protein

2016
RNA-binding protein HuR regulates nuclear import of protein.
    Journal of cell science, 2016, 11-01, Volume: 129, Issue:21

    Topics: Active Transport, Cell Nucleus; Animals; Apoproteins; beta Karyopherins; Cell Nucleus; ELAV-Like Protein 1; Endoplasmic Reticulum; HEK293 Cells; Humans; Karyopherins; MCF-7 Cells; Mice; Nuclear Proteins; Quinazolines; Receptors, Retinoic Acid; RNA Stability; RNA, Messenger; Tretinoin

2016
Ran-dependent TPX2 activation promotes acentrosomal microtubule nucleation in neurons.
    Scientific reports, 2017, 02-13, Volume: 7

    Topics: alpha Karyopherins; Animals; beta Karyopherins; Cell Cycle Proteins; Centrosome; Guanosine Triphosphate; Hippocampus; Mice, Inbred C57BL; Microtubule-Associated Proteins; Microtubules; Models, Biological; Morphogenesis; Neurites; Neurons; Nuclear Proteins; Protein Binding; Protein Transport; Quinazolines; ran GTP-Binding Protein

2017
Calpain and AR-V7: Two potential therapeutic targets to overcome acquired docetaxel resistance in castration-resistant prostate cancer cells.
    Oncology reports, 2017, Volume: 37, Issue:6

    Topics: Androgens; Calpain; Cell Line, Tumor; Docetaxel; Drug Resistance, Neoplasm; Gene Expression Regulation, Neoplastic; Humans; Male; Prostatic Neoplasms, Castration-Resistant; Protein Isoforms; Quinazolines; Receptors, Androgen; Signal Transduction; Taxoids

2017
cDNA microarray analysis identifies NR4A2 as a novel molecule involved in the pathogenesis of Sjögren's syndrome.
    Clinical and experimental immunology, 2017, Volume: 190, Issue:1

    Topics: Active Transport, Cell Nucleus; Adult; Aged; beta Karyopherins; Cell Differentiation; Cells, Cultured; DNA, Complementary; Female; Gene Expression Profiling; Humans; Immune System Diseases; Immunoglobulin G; Interleukins; Middle Aged; Nuclear Receptor Subfamily 4, Group A, Member 2; Quinazolines; Salivary Glands; Sjogren's Syndrome; Th17 Cells; Tissue Array Analysis

2017
Unique nuclear localization of Nile tilapia (Oreochromis niloticus) Neu4 sialidase is regulated by nuclear transport receptor importin α/β.
    Biochimie, 2018, Volume: 149

    Topics: Active Transport, Cell Nucleus; Animals; beta Karyopherins; Cichlids; Neuraminidase; Nuclear Localization Signals; Oryzias; Peptides; Protein Binding; Quinazolines; Sialic Acids; Substrate Specificity; Zebrafish

2018
Inhibition of Karyopherin beta 1 suppresses prostate cancer growth.
    Oncogene, 2019, Volume: 38, Issue:24

    Topics: Animals; beta Karyopherins; Cell Line, Tumor; Cell Proliferation; Down-Regulation; Gene Expression Regulation, Neoplastic; Humans; Male; Mice; Mice, Nude; PC-3 Cells; Prostatic Neoplasms; Quinazolines; RNA, Small Interfering; Xenograft Model Antitumor Assays

2019
Evidence of nuclear transport mechanisms in the protozoan parasite Giardia lamblia.
    Biochimica et biophysica acta. Molecular cell research, 2020, Volume: 1867, Issue:1

    Topics: Active Transport, Cell Nucleus; alpha Karyopherins; Animals; Antiparasitic Agents; beta Karyopherins; Cell Nucleus; Computational Biology; Giardia lamblia; Hydrolases; Ivermectin; Parasite Encystment; Protein Transport; Protozoan Proteins; Quinazolines

2020
Lamin Mutations Cause Increased YAP Nuclear Entry in Muscle Stem Cells.
    Cells, 2020, 03-27, Volume: 9, Issue:4

    Topics: Active Transport, Cell Nucleus; Adaptor Proteins, Signal Transducing; Cell Nucleus; Humans; Lamin Type A; Muscles; Mutation; Phosphorylation; Phosphoserine; Quinazolines; Stem Cells; Transcription Factors; Transcription, Genetic; YAP-Signaling Proteins

2020
    International journal of molecular sciences, 2020, Jul-09, Volume: 21, Issue:14

    Topics: beta Karyopherins; Carcinogenesis; Cell Line, Tumor; Cell Proliferation; Epithelium; Eukaryotic Initiation Factor-4G; Gene Expression Regulation, Neoplastic; Humans; Mesothelioma, Malignant; Pleural Neoplasms; Quinazolines; ran GTP-Binding Protein; RNA, Small Interfering; Small Molecule Libraries

2020
Importin β1 regulates cell growth and survival during adult T cell leukemia/lymphoma therapy.
    Investigational new drugs, 2021, Volume: 39, Issue:2

    Topics: Animals; Apoptosis; beta Karyopherins; Cell Cycle; Cell Survival; Female; Human T-lymphotropic virus 1; Humans; Leukemia-Lymphoma, Adult T-Cell; Mice; Mice, SCID; NF-kappa B; Quinazolines; Signal Transduction; T-Lymphocytes; Transcription Factor AP-1; Xenograft Model Antitumor Assays

2021
KPNB1 Inhibitor Importazole Reduces Ionizing Radiation-Increased Cell Surface PD-L1 Expression by Modulating Expression and Nuclear Import of IRF1.
    Current issues in molecular biology, 2021, May-19, Volume: 43, Issue:1

    Topics: Active Transport, Cell Nucleus; B7-H1 Antigen; beta Karyopherins; Cell Line, Tumor; Gene Expression Regulation, Neoplastic; Humans; Immunotherapy; Interferon Regulatory Factor-1; Lung Neoplasms; Quinazolines; Radiation, Ionizing

2021