Page last updated: 2024-08-21

quinazolines and hoe 33342

quinazolines has been researched along with hoe 33342 in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (11.11)29.6817
2010's7 (77.78)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Higgins, CF; Konings, WN; Margolles, A; Müller, M; van Veen, HW1
Chiba, M; Fujiwara, M; Goya, T; Kishino, T; Matsushima, S; Morii, T; Ogura, W; Ohnishi, H; Ohtsuka, K; Watanabe, T1
Baker, LC; Boult, JK; Burrell, JS; Halliday, J; Jamin, Y; Robinson, SP; Ryan, AJ; Walker-Samuel, S; Waterton, JC1
Pick, A; Wiese, M1
Chen, FH; Chiang, CS; Fu, SY; Hong, JH; Wang, CC; Yang, YC1
Du, J; Kang, Y; Lin, Y; Luo, Q; Wang, F; Wang, Y; Wang, Z; Wu, K; Zhang, Y; Zhao, Y; Zheng, W1
Ambudkar, SV; Chen, ZS; Liu, L; Shukla, S; Wang, YJ; Xu, H; Yang, DH; Zhang, D; Zhang, GN; Zhang, XY; Zhang, YK1
Gallus, J; Krapf, MK; Namasivayam, V; Wiese, M1
Chen, R; Jing, W; Li, W; Luo, J; Peng, S; Su, X; Wang, Z; Ye, X; Zhou, M1

Other Studies

9 other study(ies) available for quinazolines and hoe 33342

ArticleYear
The homodimeric ATP-binding cassette transporter LmrA mediates multidrug transport by an alternating two-site (two-cylinder engine) mechanism.
    The EMBO journal, 2000, Jun-01, Volume: 19, Issue:11

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Allosteric Regulation; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Bacterial Proteins; Benzimidazoles; Binding Sites; Biological Transport, Active; Calcium Channel Blockers; Catalysis; Cell Membrane; Dimerization; Drug Resistance, Multiple; Isoquinolines; Lactococcus lactis; Liposomes; Models, Molecular; Multidrug Resistance-Associated Proteins; Mutagenesis, Site-Directed; Photoaffinity Labels; Protein Structure, Tertiary; Quinazolines; Recombinant Fusion Proteins; Vanadates; Vinblastine

2000
Downregulated ABCG2 enhances sensitivity to topoisomerase I inhibitor in epidermal growth factor receptor tyrosine kinase inhibitor-resistant non-small cell lung cancer.
    Journal of thoracic oncology : official publication of the International Association for the Study of Lung Cancer, 2010, Volume: 5, Issue:11

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzimidazoles; Carcinoma, Non-Small-Cell Lung; Cell Proliferation; DNA Topoisomerases, Type I; DNA, Neoplasm; Down-Regulation; Drug Resistance, Neoplasm; Enzyme Inhibitors; ErbB Receptors; Genotype; Humans; Lung Neoplasms; Mutation; Neoplasm Proteins; Polymerase Chain Reaction; Protein Tyrosine Phosphatases; Quinazolines; Radiation-Sensitizing Agents; Tumor Cells, Cultured; Tyrphostins

2010
Evaluation of novel combined carbogen USPIO (CUSPIO) imaging biomarkers in assessing the antiangiogenic effects of cediranib (AZD2171) in rat C6 gliomas.
    International journal of cancer, 2012, Oct-15, Volume: 131, Issue:8

    Topics: Angiogenesis Inhibitors; Animals; Benzimidazoles; Biomarkers, Tumor; Contrast Media; Dextrans; Fluorescent Dyes; Glioma; Magnetic Resonance Imaging; Magnetite Nanoparticles; Male; Nitroimidazoles; Quinazolines; Radiation-Sensitizing Agents; Rats; Rats, Nude; Tumor Cells, Cultured

2012
Tyrosine kinase inhibitors influence ABCG2 expression in EGFR-positive MDCK BCRP cells via the PI3K/Akt signaling pathway.
    ChemMedChem, 2012, Volume: 7, Issue:4

    Topics: Animals; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP Binding Cassette Transporter, Subfamily G, Member 2; ATP-Binding Cassette Transporters; Benzamides; Benzimidazoles; Cell Line; Cetuximab; Chromones; Dose-Response Relationship, Drug; Drug Resistance, Multiple; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; Humans; Imatinib Mesylate; Morpholines; Multidrug Resistance-Associated Proteins; Neoplasm Proteins; Phosphatidylinositol 3-Kinases; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyrimidines; Quinazolines; Signal Transduction; Tyrphostins

2012
Combination of vessel-targeting agents and fractionated radiation therapy: the role of the SDF-1/CXCR4 pathway.
    International journal of radiation oncology, biology, physics, 2013, Jul-15, Volume: 86, Issue:4

    Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Benzimidazoles; Benzylamines; Bone Marrow Cells; Chemokine CXCL12; Combined Modality Therapy; Cyclams; Dose Fractionation, Radiation; ErbB Receptors; Gefitinib; Green Fluorescent Proteins; Heterocyclic Compounds; Luminescent Agents; Male; Mice; Mice, Inbred C57BL; Neovascularization, Pathologic; Pericytes; Prostatic Neoplasms; Quinazolines; Receptors, CXCR4; Tumor Microenvironment

2013
Synthesis, Characterization, and in Vitro Antitumor Activity of Ruthenium(II) Polypyridyl Complexes Tethering EGFR-Inhibiting 4-Anilinoquinazolines.
    Inorganic chemistry, 2016, 05-02, Volume: 55, Issue:9

    Topics: 2,2'-Dipyridyl; Aniline Compounds; Antineoplastic Agents; Apoptosis; Benzimidazoles; Cell Line, Tumor; Cisplatin; Coordination Complexes; DNA; ErbB Receptors; Fluorescent Dyes; Gefitinib; Humans; Hydrolysis; Ligands; Membrane Proteins; Phenanthrolines; Quinazolines; Ruthenium

2016
Selective reversal of BCRP-mediated MDR by VEGFR-2 inhibitor ZM323881.
    Biochemical pharmacology, 2017, 05-15, Volume: 132

    Topics: ATP Binding Cassette Transporter, Subfamily G, Member 2; Benzimidazoles; Cell Line, Tumor; Doxorubicin; Drug Resistance, Multiple; HEK293 Cells; Humans; Mitoxantrone; Molecular Dynamics Simulation; Neoplasm Proteins; Quinazolines; Vascular Endothelial Growth Factor Receptor-2

2017
2,4,6-Substituted Quinazolines with Extraordinary Inhibitory Potency toward ABCG2.
    Journal of medicinal chemistry, 2018, 09-13, Volume: 61, Issue:17

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Benzimidazoles; Cell Proliferation; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Humans; Molecular Structure; Neoplasm Proteins; Neoplasms; Protein Conformation; Quinazolines; Structure-Activity Relationship; Tumor Cells, Cultured

2018
In vitro and ex vivo anti‑tumor effect and mechanism of Tucatinib in leukemia stem cells and ABCG2‑overexpressing leukemia cells.
    Oncology reports, 2021, Volume: 45, Issue:3

    Topics: Adenosine Triphosphatases; Adult; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily G, Member 2; Benzimidazoles; Cell Survival; Drug Resistance, Neoplasm; Female; Humans; Leukemia; Male; Mitoxantrone; Neoplasm Proteins; Neoplastic Stem Cells; Oxazoles; Pyridines; Quinazolines; Side-Population Cells; Tumor Cells, Cultured

2021