Page last updated: 2024-08-21

quinazolines and gamma-aminobutyric acid

quinazolines has been researched along with gamma-aminobutyric acid in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19902 (13.33)18.7374
1990's0 (0.00)18.2507
2000's6 (40.00)29.6817
2010's5 (33.33)24.3611
2020's2 (13.33)2.80

Authors

AuthorsStudies
Ishida, R; Kudo, Y1
Ghatak, S; Sen, R; Tekwani, BL; Tripathi, LM1
Choi, JI; Jeong, SW; Yoon, MH1
Djahanguiri, B; Massoudi, R; Rezayat, M; Roohbakhsh, A; Zarrindast, MR1
Iwakura, Y; Jourdi, H; Nagano, T; Namba, H; Nawa, H; Takei, N; Xiong, H1
Arcella, A; Cantore, G; Di Gennaro, G; Esposito, V; Eusebi, F; Fredholm, BB; Fucile, S; Limatola, C; Manfredi, M; Martinello, K; Mascia, A; Miledi, R; Piccari, V; Quarato, PP; Roseti, C; Simonato, M1
Cooley-Zgela, T; Gius, D; Morris, JC; Sharp, H; Singh, AK; Van Waes, C1
Guo, Z; Zhao, H1
Ali, I; Amir, M; Hassan, MZ1
Xiao, X; Xu, TL; Zhu, MX1
Brame, LS; Cao, A; Fang, YT; Fung, KM; Humphreys, MR; Kropp, BP; Lin, HK; Shih, PT; Wu, W; Yang, Q1
Bastian, G; Bourgoin, S; Hamon, M; Kayser, V; Michot, B1
Bi, LL; Chen, YH; Gao, TM; Geng, F; Li, XW; Liu, F; Liu, JH; Lu, YS; Mei, L; Sun, XD; Wang, J; Zhang, J; Zhang, M1
Alex, VV; Anto, RJ; Bava, SV; Chittalakkottu, S; Nisthul A, A; Retnakumari, AP; Shankar G, M; Sundaram, S1
Crocetti, L; Giovannoni, MP; Guerrini, G; Mascia, MP; Melani, F; Vergelli, C1

Reviews

1 review(s) available for quinazolines and gamma-aminobutyric acid

ArticleYear
Medicinal chemistry strategies in follow-on drug discovery.
    Drug discovery today, 2009, Volume: 14, Issue:9-10

    Topics: Animals; Atorvastatin; Bendamustine Hydrochloride; Benzazepines; Chemistry, Pharmaceutical; Clinical Trials as Topic; Drug Delivery Systems; Drug Discovery; gamma-Aminobutyric Acid; Heptanoic Acids; Humans; Lapatinib; Nitrogen Mustard Compounds; Pregabalin; Pyrimidines; Pyrroles; Quinazolines; Sulfonamides

2009

Trials

1 trial(s) available for quinazolines and gamma-aminobutyric acid

ArticleYear
High incidence of oral dysesthesias on a trial of gefitinib, Paclitaxel, and concurrent external beam radiation for locally advanced head and neck cancers.
    American journal of clinical oncology, 2008, Volume: 31, Issue:6

    Topics: Adult; Aged; Amines; Anticonvulsants; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Squamous Cell; Combined Modality Therapy; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Gefitinib; Head and Neck Neoplasms; Humans; Incidence; Male; Middle Aged; Neoplasm Staging; Paclitaxel; Paresthesia; Prognosis; Quinazolines; Radiation Injuries; Radiotherapy; Stomatitis

2008

Other Studies

13 other study(ies) available for quinazolines and gamma-aminobutyric acid

ArticleYear
Effects of afloqualone on vestibular nystagmus and the lateral vestibular nucleus.
    Japanese journal of pharmacology, 1989, Volume: 50, Issue:4

    Topics: Acetylcholine; Animals; Cats; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Histamine H1 Antagonists; Iontophoresis; Male; Muscle Relaxants, Central; Nystagmus, Physiologic; Piperidines; Propiophenones; Quinazolines; Reflex, Monosynaptic; Synaptic Transmission; Vestibular Nuclei

1989
Effect of anticonvulsants, centazolone and centpropazine, on gamma amino butyric acid metabolism in mouse brain.
    Indian journal of experimental biology, 1985, Volume: 23, Issue:8

    Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Antidepressive Agents; Brain; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hydrazines; Mice; Piperazines; Quinazolines

1985
Spinal gabapentin and antinociception: mechanisms of action.
    Journal of Korean medical science, 2003, Volume: 18, Issue:2

    Topics: Acetates; Adrenergic alpha-Antagonists; Adrenergic Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amines; Analgesics; Animals; Atropine; Cyclohexanecarboxylic Acids; Dihydroergocristine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Injections, Spinal; Leucine; Male; Mecamylamine; Muscarinic Antagonists; N-Methylaspartate; Naloxone; Narcotic Antagonists; Nicotinic Antagonists; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Serine; Spinal Cord; Thapsigargin; Triazoles

2003
Cholecystokinin and GABA interaction in the dorsal hippocampus of rats in the elevated plus-maze test of anxiety.
    Physiology & behavior, 2005, Apr-13, Volume: 84, Issue:5

    Topics: Animals; Anxiety; Bicuculline; Cholecystokinin; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Microinjections; Quinazolines; Quinazolinones; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stereotaxic Techniques

2005
Transforming growth factor alpha attenuates the functional expression of AMPA receptors in cortical GABAergic neurons.
    Molecular and cellular neurosciences, 2006, Volume: 31, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Brain-Derived Neurotrophic Factor; Cells, Cultured; Cerebral Cortex; Culture Media, Serum-Free; Electrophysiology; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; gamma-Aminobutyric Acid; Heparin-binding EGF-like Growth Factor; Intercellular Signaling Peptides and Proteins; Ligands; Neurons; Protein Subunits; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Transforming Growth Factor alpha

2006
Adenosine receptor antagonists alter the stability of human epileptic GABAA receptors.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Sep-30, Volume: 105, Issue:39

    Topics: Adenosine; Adenosine Deaminase; Adult; Animals; Anticonvulsants; Cerebral Cortex; Epilepsy; Female; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Male; Neurons; Oocytes; Purinergic P1 Receptor Antagonists; Pyramidal Tracts; Pyrimidines; Quinazolines; Rats; Receptors, GABA-A; Triazoles; Xanthines; Xenopus

2008
Design and synthesis of some new quinazolin-4-(3H)-ones as anticonvulsant and antidepressant agents.
    Archives of pharmacal research, 2013, Volume: 36, Issue:1

    Topics: Animals; Anticonvulsants; Antidepressive Agents; Brain; Disease Models, Animal; Drug Design; gamma-Aminobutyric Acid; Mice; Molecular Structure; Quinazolines; Seizures; Structure-Activity Relationship; Swimming

2013
2-Guanidine-4-methylquinazoline acts as a novel competitive antagonist of A type γ-aminobutyric acid receptors.
    Neuropharmacology, 2013, Volume: 75

    Topics: Acetylcholine; Action Potentials; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Excitatory Amino Acid Agents; GABA Agents; gamma-Aminobutyric Acid; Glycine; Guanidines; Hippocampus; Humans; In Vitro Techniques; Mutation; Neurons; Protein Subunits; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A

2013
Linking γ-aminobutyric acid A receptor to epidermal growth factor receptor pathways activation in human prostate cancer.
    Molecular and cellular endocrinology, 2014, Mar-05, Volume: 383, Issue:1-2

    Topics: Autocrine Communication; Cell Line, Tumor; Cell Proliferation; ErbB Receptors; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gefitinib; Gene Expression Regulation, Neoplastic; Humans; Isonicotinic Acids; Male; Paracrine Communication; Phosphorylation; Picrotoxin; Prostate; Prostatic Neoplasms; Protein Kinase Inhibitors; Quinazolines; Receptors, GABA-A; Signal Transduction; src-Family Kinases

2014
Differential pharmacological alleviation of oxaliplatin-induced hyperalgesia/allodynia at cephalic versus extra-cephalic level in rodents.
    Neuropharmacology, 2014, Volume: 79

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amines; Analgesics; Animals; Cold Temperature; Cyclohexanecarboxylic Acids; Dipeptides; Formaldehyde; Gabapentin; gamma-Aminobutyric Acid; Ganglia, Spinal; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Organoplatinum Compounds; Oxaliplatin; Piperazines; Piperidines; Quinazolines; Rats; Rats, Sprague-Dawley; Spinal Cord; Touch; TRPA1 Cation Channel; TRPC Cation Channels; Tryptamines

2014
Amygdala NRG1-ErbB4 is critical for the modulation of anxiety-like behaviors.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2015, Volume: 40, Issue:4

    Topics: Amygdala; Animals; Anxiety; Disease Models, Animal; Enzyme Inhibitors; Exploratory Behavior; Feeding Behavior; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; GPI-Linked Proteins; In Vitro Techniques; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myelin Proteins; Nogo Receptor 1; Pyrimidines; Quinazolines; Reaction Time; Receptor, ErbB-4; Receptors, Cell Surface; Signal Transduction; Tyrphostins

2015
Pre-clinical evidences for the efficacy of tryptanthrin as a potent suppressor of skin cancer.
    Cell proliferation, 2020, Volume: 53, Issue:1

    Topics: Animals; Drug Screening Assays, Antitumor; gamma-Aminobutyric Acid; Ki-67 Antigen; Mice; Neoplasm Proteins; Proliferating Cell Nuclear Antigen; Quinazolines; Skin Neoplasms; Tetradecanoylphorbol Acetate

2020
GABA
    International journal of molecular sciences, 2022, Oct-27, Volume: 23, Issue:21

    Topics: Animals; gamma-Aminobutyric Acid; Molecular Docking Simulation; Oocytes; Quinazolines; Receptors, GABA-A; Xenopus laevis

2022