quinazolines has been researched along with gamma-aminobutyric acid in 15 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (13.33) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 6 (40.00) | 29.6817 |
2010's | 5 (33.33) | 24.3611 |
2020's | 2 (13.33) | 2.80 |
Authors | Studies |
---|---|
Ishida, R; Kudo, Y | 1 |
Ghatak, S; Sen, R; Tekwani, BL; Tripathi, LM | 1 |
Choi, JI; Jeong, SW; Yoon, MH | 1 |
Djahanguiri, B; Massoudi, R; Rezayat, M; Roohbakhsh, A; Zarrindast, MR | 1 |
Iwakura, Y; Jourdi, H; Nagano, T; Namba, H; Nawa, H; Takei, N; Xiong, H | 1 |
Arcella, A; Cantore, G; Di Gennaro, G; Esposito, V; Eusebi, F; Fredholm, BB; Fucile, S; Limatola, C; Manfredi, M; Martinello, K; Mascia, A; Miledi, R; Piccari, V; Quarato, PP; Roseti, C; Simonato, M | 1 |
Cooley-Zgela, T; Gius, D; Morris, JC; Sharp, H; Singh, AK; Van Waes, C | 1 |
Guo, Z; Zhao, H | 1 |
Ali, I; Amir, M; Hassan, MZ | 1 |
Xiao, X; Xu, TL; Zhu, MX | 1 |
Brame, LS; Cao, A; Fang, YT; Fung, KM; Humphreys, MR; Kropp, BP; Lin, HK; Shih, PT; Wu, W; Yang, Q | 1 |
Bastian, G; Bourgoin, S; Hamon, M; Kayser, V; Michot, B | 1 |
Bi, LL; Chen, YH; Gao, TM; Geng, F; Li, XW; Liu, F; Liu, JH; Lu, YS; Mei, L; Sun, XD; Wang, J; Zhang, J; Zhang, M | 1 |
Alex, VV; Anto, RJ; Bava, SV; Chittalakkottu, S; Nisthul A, A; Retnakumari, AP; Shankar G, M; Sundaram, S | 1 |
Crocetti, L; Giovannoni, MP; Guerrini, G; Mascia, MP; Melani, F; Vergelli, C | 1 |
1 review(s) available for quinazolines and gamma-aminobutyric acid
Article | Year |
---|---|
Medicinal chemistry strategies in follow-on drug discovery.
Topics: Animals; Atorvastatin; Bendamustine Hydrochloride; Benzazepines; Chemistry, Pharmaceutical; Clinical Trials as Topic; Drug Delivery Systems; Drug Discovery; gamma-Aminobutyric Acid; Heptanoic Acids; Humans; Lapatinib; Nitrogen Mustard Compounds; Pregabalin; Pyrimidines; Pyrroles; Quinazolines; Sulfonamides | 2009 |
1 trial(s) available for quinazolines and gamma-aminobutyric acid
Article | Year |
---|---|
High incidence of oral dysesthesias on a trial of gefitinib, Paclitaxel, and concurrent external beam radiation for locally advanced head and neck cancers.
Topics: Adult; Aged; Amines; Anticonvulsants; Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Squamous Cell; Combined Modality Therapy; Cyclohexanecarboxylic Acids; Female; Gabapentin; gamma-Aminobutyric Acid; Gefitinib; Head and Neck Neoplasms; Humans; Incidence; Male; Middle Aged; Neoplasm Staging; Paclitaxel; Paresthesia; Prognosis; Quinazolines; Radiation Injuries; Radiotherapy; Stomatitis | 2008 |
13 other study(ies) available for quinazolines and gamma-aminobutyric acid
Article | Year |
---|---|
Effects of afloqualone on vestibular nystagmus and the lateral vestibular nucleus.
Topics: Acetylcholine; Animals; Cats; Dose-Response Relationship, Drug; Female; gamma-Aminobutyric Acid; Histamine H1 Antagonists; Iontophoresis; Male; Muscle Relaxants, Central; Nystagmus, Physiologic; Piperidines; Propiophenones; Quinazolines; Reflex, Monosynaptic; Synaptic Transmission; Vestibular Nuclei | 1989 |
Effect of anticonvulsants, centazolone and centpropazine, on gamma amino butyric acid metabolism in mouse brain.
Topics: 4-Aminobutyrate Transaminase; Animals; Anticonvulsants; Antidepressive Agents; Brain; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Hydrazines; Mice; Piperazines; Quinazolines | 1985 |
Spinal gabapentin and antinociception: mechanisms of action.
Topics: Acetates; Adrenergic alpha-Antagonists; Adrenergic Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amines; Analgesics; Animals; Atropine; Cyclohexanecarboxylic Acids; Dihydroergocristine; Enzyme Inhibitors; Excitatory Amino Acid Agonists; GABA Antagonists; Gabapentin; gamma-Aminobutyric Acid; Injections, Spinal; Leucine; Male; Mecamylamine; Muscarinic Antagonists; N-Methylaspartate; Naloxone; Narcotic Antagonists; Nicotinic Antagonists; Pain Measurement; Quinazolines; Rats; Rats, Sprague-Dawley; Serine; Spinal Cord; Thapsigargin; Triazoles | 2003 |
Cholecystokinin and GABA interaction in the dorsal hippocampus of rats in the elevated plus-maze test of anxiety.
Topics: Animals; Anxiety; Bicuculline; Cholecystokinin; Dose-Response Relationship, Drug; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Male; Microinjections; Quinazolines; Quinazolinones; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stereotaxic Techniques | 2005 |
Transforming growth factor alpha attenuates the functional expression of AMPA receptors in cortical GABAergic neurons.
Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Brain-Derived Neurotrophic Factor; Cells, Cultured; Cerebral Cortex; Culture Media, Serum-Free; Electrophysiology; Enzyme Inhibitors; Epidermal Growth Factor; ErbB Receptors; gamma-Aminobutyric Acid; Heparin-binding EGF-like Growth Factor; Intercellular Signaling Peptides and Proteins; Ligands; Neurons; Protein Subunits; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Transforming Growth Factor alpha | 2006 |
Adenosine receptor antagonists alter the stability of human epileptic GABAA receptors.
Topics: Adenosine; Adenosine Deaminase; Adult; Animals; Anticonvulsants; Cerebral Cortex; Epilepsy; Female; GABA-A Receptor Agonists; gamma-Aminobutyric Acid; Humans; Male; Neurons; Oocytes; Purinergic P1 Receptor Antagonists; Pyramidal Tracts; Pyrimidines; Quinazolines; Rats; Receptors, GABA-A; Triazoles; Xanthines; Xenopus | 2008 |
Design and synthesis of some new quinazolin-4-(3H)-ones as anticonvulsant and antidepressant agents.
Topics: Animals; Anticonvulsants; Antidepressive Agents; Brain; Disease Models, Animal; Drug Design; gamma-Aminobutyric Acid; Mice; Molecular Structure; Quinazolines; Seizures; Structure-Activity Relationship; Swimming | 2013 |
2-Guanidine-4-methylquinazoline acts as a novel competitive antagonist of A type γ-aminobutyric acid receptors.
Topics: Acetylcholine; Action Potentials; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Embryo, Mammalian; Excitatory Amino Acid Agents; GABA Agents; gamma-Aminobutyric Acid; Glycine; Guanidines; Hippocampus; Humans; In Vitro Techniques; Mutation; Neurons; Protein Subunits; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A | 2013 |
Linking γ-aminobutyric acid A receptor to epidermal growth factor receptor pathways activation in human prostate cancer.
Topics: Autocrine Communication; Cell Line, Tumor; Cell Proliferation; ErbB Receptors; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gefitinib; Gene Expression Regulation, Neoplastic; Humans; Isonicotinic Acids; Male; Paracrine Communication; Phosphorylation; Picrotoxin; Prostate; Prostatic Neoplasms; Protein Kinase Inhibitors; Quinazolines; Receptors, GABA-A; Signal Transduction; src-Family Kinases | 2014 |
Differential pharmacological alleviation of oxaliplatin-induced hyperalgesia/allodynia at cephalic versus extra-cephalic level in rodents.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amines; Analgesics; Animals; Cold Temperature; Cyclohexanecarboxylic Acids; Dipeptides; Formaldehyde; Gabapentin; gamma-Aminobutyric Acid; Ganglia, Spinal; Hyperalgesia; Male; Mice; Mice, Inbred C57BL; Morphine; Organoplatinum Compounds; Oxaliplatin; Piperazines; Piperidines; Quinazolines; Rats; Rats, Sprague-Dawley; Spinal Cord; Touch; TRPA1 Cation Channel; TRPC Cation Channels; Tryptamines | 2014 |
Amygdala NRG1-ErbB4 is critical for the modulation of anxiety-like behaviors.
Topics: Amygdala; Animals; Anxiety; Disease Models, Animal; Enzyme Inhibitors; Exploratory Behavior; Feeding Behavior; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; GPI-Linked Proteins; In Vitro Techniques; Male; Maze Learning; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myelin Proteins; Nogo Receptor 1; Pyrimidines; Quinazolines; Reaction Time; Receptor, ErbB-4; Receptors, Cell Surface; Signal Transduction; Tyrphostins | 2015 |
Pre-clinical evidences for the efficacy of tryptanthrin as a potent suppressor of skin cancer.
Topics: Animals; Drug Screening Assays, Antitumor; gamma-Aminobutyric Acid; Ki-67 Antigen; Mice; Neoplasm Proteins; Proliferating Cell Nuclear Antigen; Quinazolines; Skin Neoplasms; Tetradecanoylphorbol Acetate | 2020 |
GABA
Topics: Animals; gamma-Aminobutyric Acid; Molecular Docking Simulation; Oocytes; Quinazolines; Receptors, GABA-A; Xenopus laevis | 2022 |